Cell Line ID	CL000011
Cell Line Name	CHO
Synonyms	Chinese Hamster Ovary CHO-ori
Category	Spontaneously immortalized cell line
Organism	Cricetulus griseus (Chinese hamster)
Cellosaurus ID	CVCL_0213
Tissue Information	Ovary
Disease	None

Map of Molecular Bioactivity Related to the Cell Line Cell Line Protein Compound Bioactivity Value: <= 0.1 μM > 0.1 μM and <= 10 μM > 10 μM Imprecise Activity

Compound ID	Compound Name	Compound Formula
CP0861283  Compound Info	US9163012, 68    Show/Hide	C23H27ClN4O4	1
1	IC50 = 0.46 nM  Bioactivity Info	TI    LI    LO    TS
CP0521496  Compound Info	US9163012, 53    Show/Hide	C24H29N3O3S	1
1	IC50 = 0.47 nM  Bioactivity Info	TI    LI    LO    TS
CP0214912  Compound Info	N-(2-adamantyl)-1-(2-amino-2-oxoethyl)-4-bromospiro[1,2-dihydroindene-3,4'-piperidine]-1'-carboxamide    Show/Hide	C26H34BrN3O2	1
1	IC50 = 0.5 nM  Bioactivity Info	TI    LI    LO    TS
CP0064790  Compound Info	(6S)-6-(4-fluorophenyl)-3-[(1S)-1-[4-(4-fluorophenyl)phenyl]ethyl]-6-(2-hydroxyethyl)-1,3-oxazinan-2-one    Show/Hide	C26H25F2NO3	2
1	IC50 = 0.5 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 18.5 nM  Bioactivity Info	TI    LI    LO    TS
CP0509094  Compound Info	(6S)-3-[(1S)-1-[4-(4-fluorophenyl)phenyl]ethyl]-6-(2-hydroxyethyl)-6-phenyl-1,3-oxazinan-2-one    Show/Hide	C26H26FNO3	2
1	IC50 = 0.5 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 5.7 nM  Bioactivity Info	TI    LI    LO    TS
CP0483002  Compound Info	US9163012, 34    Show/Hide	C19H24ClN3O2	1
1	IC50 = 0.52 nM  Bioactivity Info	TI    LI    LO    TS
CP0478264  Compound Info	US9163012, 1    Show/Hide	C21H25F2N3O4	1
1	IC50 = 0.54 nM  Bioactivity Info	TI    LI    LO    TS
CP0478265  Compound Info	US9163012, 6    Show/Hide	C22H26F3N3O4	1
1	IC50 = 0.54 nM  Bioactivity Info	TI    LI    LO    TS
CP0072901  Compound Info	(R)-3-(3-Trifluoromethyl-pyridin-2-ylamino)-pyrrolidine-1-carboxylic acid 5-carbamoyl-adamantan-2-yl ester    Show/Hide	C22H27F3N4O3	1
1	IC50 = 0.55 nM  Bioactivity Info	TI    LI    LO    TS
CP0064791  Compound Info	(6R)-3-[(1S)-1-[4-(4-fluorophenyl)phenyl]ethyl]-6-(3-hydroxypropyl)-6-phenyl-1,3-oxazinan-2-one    Show/Hide	C27H28FNO3	2
1	IC50 = 0.6 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 11.9 nM  Bioactivity Info	TI    LI    LO    TS
CP0227029  Compound Info	(6R)-3-[(1S)-1-[4-(2,4-difluorophenyl)phenyl]ethyl]-6-(3-hydroxypropyl)-6-phenyl-1,3-oxazinan-2-one    Show/Hide	C27H27F2NO3	2
1	IC50 = 0.6 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 17.9 nM  Bioactivity Info	TI    LI    LO    TS
CP0313822  Compound Info	(6R)-6-(4-fluorophenyl)-3-[(1S)-1-[4-(4-fluorophenyl)phenyl]ethyl]-6-(3-hydroxypropyl)-1,3-oxazinan-2-one    Show/Hide	C27H27F2NO3	2
1	IC50 = 0.6 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 14.7 nM  Bioactivity Info	TI    LI    LO    TS
CP0342700  Compound Info	(6R)-3-[(1S)-1-[4-(4-fluorophenyl)phenyl]propyl]-6-(3-hydroxypropyl)-6-phenyl-1,3-oxazinan-2-one    Show/Hide	C28H30FNO3	2
1	IC50 = 0.6 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 18.7 nM  Bioactivity Info	TI    LI    LO    TS
CP0309631  Compound Info	(S)-3-(3-Trifluoromethyl-pyridin-2-ylamino)-pyrrolidine-1-carboxylic acid 5-carbamoyl-adamantan-2-yl ester    Show/Hide	C22H27F3N4O3	1
1	IC50 = 0.63 nM  Bioactivity Info	TI    LI    LO    TS
CP0060924  Compound Info	(R)-3-(6-Trifluoromethyl-pyridin-2-ylamino)-pyrrolidine-1-carboxylic acid 5-carbamoyl-adamantan-2-yl ester    Show/Hide	C22H27F3N4O3	1
1	IC50 = 0.67 nM  Bioactivity Info	TI    LI    LO    TS
CP0577337  Compound Info	US9163012, 71    Show/Hide	C24H29ClN4O4	1
1	IC50 = 0.67 nM  Bioactivity Info	TI    LI    LO    TS
CP0525176  Compound Info	US9163012, 2    Show/Hide	C21H25F2N3O4	1
1	IC50 = 0.68 nM  Bioactivity Info	TI    LI    LO    TS
CP0909883  Compound Info	US9163012, 67    Show/Hide	C23H27ClN4O4	1
1	IC50 = 0.68 nM  Bioactivity Info	TI    LI    LO    TS
CP0421759  Compound Info	N-(2-adamantyl)spiro[1,3-dihydroindene-2,3'-piperidine]-1'-carboxamide    Show/Hide	C24H32N2O	1
1	IC50 = 0.7 nM  Bioactivity Info	TI    LI    LO    TS
CP0476378  Compound Info	(6S)-3-[(1S)-1-[4-(2,4-difluorophenyl)phenyl]ethyl]-6-(2-hydroxyethyl)-6-phenyl-1,3-oxazinan-2-one    Show/Hide	C26H25F2NO3	2
1	IC50 = 0.7 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 8.4 nM  Bioactivity Info	TI    LI    LO    TS
CP0570634  Compound Info	US9163012, 51    Show/Hide	C23H27N3O2S	1
1	IC50 = 0.7 nM  Bioactivity Info	TI    LI    LO    TS
CP0243879  Compound Info	(S)-3-(5-Trifluoromethyl-pyridin-2-ylamino)-pyrrolidine-1-carboxylic acid 5-carbamoyl-adamantan-2-yl ester    Show/Hide	C22H27F3N4O3	1
1	IC50 = 0.74 nM  Bioactivity Info	TI    LI    LO    TS
CP0927520  Compound Info	US9163012, 60    Show/Hide	C23H28N4O4	1
1	IC50 = 0.76 nM  Bioactivity Info	TI    LI    LO    TS
CP0166399  Compound Info	N-(2-adamantyl)spiro[1,2-dihydroindene-3,4'-piperidine]-1'-carboxamide    Show/Hide	C24H32N2O	1
1	IC50 = 0.8 nM  Bioactivity Info	TI    LI    LO    TS
CP0506313  Compound Info	3-Phenyl-piperidine-1-carboxylic acid adamantan-2-ylamide    Show/Hide	C22H30N2O	1
1	IC50 = 0.8 nM  Bioactivity Info	TI    LI    LO    TS
CP0093362  Compound Info	(6S)-3-[(1S)-1-[4-(2,4-difluorophenyl)phenyl]ethyl]-6-(4-fluorophenyl)-6-(2-hydroxyethyl)-1,3-oxazinan-2-one    Show/Hide	C26H24F3NO3	2
1	IC50 = 0.8 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 17.5 nM  Bioactivity Info	TI    LI    LO    TS
CP0305091  Compound Info	2-[(6R)-3-[(1S)-1-[4-(2,4-difluorophenyl)phenyl]ethyl]-6-(4-fluorophenyl)-2-oxo-1,3-oxazinan-6-yl]ethylurea    Show/Hide	C27H26F3N3O3	2
1	IC50 = 0.8 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 29 nM  Bioactivity Info	TI    LI    LO    TS
CP0038293  Compound Info	(R)-3-(5-Trifluoromethyl-pyridin-2-ylamino)-pyrrolidine-1-carboxylic acid 5-carbamoyl-adamantan-2-yl ester    Show/Hide	C22H27F3N4O3	1
1	IC50 = 0.82 nM  Bioactivity Info	TI    LI    LO    TS
CP0038295  Compound Info	(R)-3-(3-Cyano-pyridin-2-ylamino)-pyrrolidine-1-carboxylic acid 5-carbamoyl-adamantan-2-yl ester    Show/Hide	C22H27N5O3	2
1	IC50 = 0.87 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 2.4 nM  Bioactivity Info	TI    LI    LO    TS
CP0514308  Compound Info	3-Benzyl-piperidine-1-carboxylic acid adamantan-2-ylamide    Show/Hide	C23H32N2O	1
1	IC50 = 0.9 nM  Bioactivity Info	TI    LI    LO    TS
CP0514311  Compound Info	4-Phenyl-piperidine-1-carboxylic acid adamantan-2-ylamide    Show/Hide	C22H30N2O	1
1	IC50 = 0.9 nM  Bioactivity Info	TI    LI    LO    TS
CP0086590  Compound Info	(6R)-6-(2-fluorophenyl)-3-[(1S)-1-[4-(4-fluorophenyl)phenyl]ethyl]-6-(3-hydroxypropyl)-1,3-oxazinan-2-one    Show/Hide	C27H27F2NO3	2
1	IC50 = 0.9 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 8.6 nM  Bioactivity Info	TI    LI    LO    TS
CP0238173  Compound Info	(6R)-6-(3-fluorophenyl)-3-[(1S)-1-[4-(4-fluorophenyl)phenyl]ethyl]-6-(3-hydroxypropyl)-1,3-oxazinan-2-one    Show/Hide	C27H27F2NO3	2
1	IC50 = 0.9 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 11.8 nM  Bioactivity Info	TI    LI    LO    TS
CP0577336  Compound Info	US9163012, 50    Show/Hide	C23H27N3O2S	1
1	IC50 = 0.91 nM  Bioactivity Info	TI    LI    LO    TS
CP0539983  Compound Info	US9163012, 5    Show/Hide	C22H26F3N3O4	1
1	IC50 = 0.99 nM  Bioactivity Info	TI    LI    LO    TS
CP0238172  Compound Info	N-[2-[(6S)-3-[(1S)-1-[4-(2,4-difluorophenyl)phenyl]ethyl]-6-(4-fluorophenyl)-2-oxo-1,3-oxazinan-6-yl]ethyl]methanesulfonamide    Show/Hide	C27H27F3N2O4S	2
1	IC50 = 1 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 45 nM  Bioactivity Info	TI    LI    LO    TS
CP0297084  Compound Info	3-[(6R)-3-[(1S)-1-[4-(2,4-difluorophenyl)phenyl]ethyl]-6-(4-fluorophenyl)-2-oxo-1,3-oxazinan-6-yl]propanamide    Show/Hide	C27H25F3N2O3	2
1	IC50 = 1 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 42 nM  Bioactivity Info	TI    LI    LO    TS
CP0934304  Compound Info	US9163012, 63    Show/Hide	C23H27FN4O4	1
1	IC50 = 1.01 nM  Bioactivity Info	TI    LI    LO    TS
CP0966864  Compound Info	US9163012, 69    Show/Hide	C22H26ClN5O4	1
1	IC50 = 1.04 nM  Bioactivity Info	TI    LI    LO    TS
CP0573358  Compound Info	US9163012, 32    Show/Hide	C24H30N4O3	1
1	IC50 = 1.08 nM  Bioactivity Info	TI    LI    LO    TS
CP0214910  Compound Info	2-[(3R)-1'-[(adamantan-2-yl)carbamoyl]-7-bromo-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetic acid    Show/Hide	C26H33BrN2O3	1
1	IC50 = 1.1 nM  Bioactivity Info	TI    LI    LO    TS
CP0506249  Compound Info	4-Benzyl-piperidine-1-carboxylic acid adamantan-2-ylamide    Show/Hide	C23H32N2O	1
1	IC50 = 1.1 nM  Bioactivity Info	TI    LI    LO    TS
CP0341245  Compound Info	(6R)-3-[(1S)-1-[4-(2,4-difluorophenyl)phenyl]ethyl]-6-(4-fluorophenyl)-6-(3-hydroxypropyl)-1,3-oxazinan-2-one    Show/Hide	C27H26F3NO3	2
1	IC50 = 1.1 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 18 nM  Bioactivity Info	TI    LI    LO    TS
CP0570743  Compound Info	US9163012, 76    Show/Hide	C24H29ClN4O3	1
1	IC50 = 1.11 nM  Bioactivity Info	TI    LI    LO    TS
CP0529503  Compound Info	US9163012, 26    Show/Hide	C20H25ClN4O3	1
1	IC50 = 1.12 nM  Bioactivity Info	TI    LI    LO    TS
CP0521495  Compound Info	US9163012, 52    Show/Hide	C23H27N3O3S	1
1	IC50 = 1.19 nM  Bioactivity Info	TI    LI    LO    TS
CP0502290  Compound Info	2-Benzyl-piperidine-1-carboxylic acid adamantan-2-ylamide    Show/Hide	C23H32N2O	1
1	IC50 = 1.4 nM  Bioactivity Info	TI    LI    LO    TS
CP0238174  Compound Info	3-[(6R)-3-[(1S)-1-[4-(2,4-difluorophenyl)phenyl]ethyl]-6-(4-fluorophenyl)-2-oxo-1,3-oxazinan-6-yl]propylurea    Show/Hide	C28H28F3N3O3	2
1	IC50 = 1.4 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 53 nM  Bioactivity Info	TI    LI    LO    TS
CP0060925  Compound Info	(R)-3-(5-Cyano-pyridin-2-ylamino)-pyrrolidine-1-carboxylic acid 5-carbamoyl-adamantan-2-yl ester    Show/Hide	C22H27N5O3	2
1	IC50 = 1.5 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 3.2 nM  Bioactivity Info	TI    LI    LO    TS
CP0236094  Compound Info	2-{1'-[(adamantan-2-yl)carbamoyl]-7-bromo-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl}acetic acid    Show/Hide	C26H33BrN2O3	1
1	IC50 = 1.6 nM  Bioactivity Info	TI    LI    LO    TS
CP0468486  Compound Info	3-[3-(2,4-difluorophenyl)phenyl]-6-methyl-6-phenyl-1,3-oxazinan-2-one    Show/Hide	C23H19F2NO2	1
1	IC50 = 1.6 nM  Bioactivity Info	TI    LI    LO    TS
CP0265676  Compound Info	N-(2-adamantyl)-4-bromo-1-(2-hydroxyethyl)spiro[1,2-dihydroindene-3,4'-piperidine]-1'-carboxamide    Show/Hide	C26H35BrN2O2	1
1	IC50 = 1.7 nM  Bioactivity Info	TI    LI    LO    TS
CP0342446  Compound Info	(S)-3-(5-Cyano-pyridin-2-ylamino)-pyrrolidine-1-carboxylic acid 5-carbamoyl-adamantan-2-yl ester    Show/Hide	C22H27N5O3	1
1	IC50 = 1.7 nM  Bioactivity Info	TI    LI    LO    TS
CP0926673  Compound Info	US9163012, 64    Show/Hide	C24H27N5O4	1
1	IC50 = 1.71 nM  Bioactivity Info	TI    LI    LO    TS
CP0316007  Compound Info	N-[3-[(6R)-3-[(1S)-1-[4-(2,4-difluorophenyl)phenyl]ethyl]-6-(4-fluorophenyl)-2-oxo-1,3-oxazinan-6-yl]propyl]methanesulfonamide    Show/Hide	C28H29F3N2O4S	2
1	IC50 = 1.8 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 32 nM  Bioactivity Info	TI    LI    LO    TS
CP0523675  Compound Info	(R)-3-(2-Trifluoromethyl-pyrimidin-4-ylamino)-pyrrolidine-1-carboxylic acid 5-carbamoyl-adamantan-2-yl ester    Show/Hide	C21H26F3N5O3	1
1	IC50 = 1.9 nM  Bioactivity Info	TI    LI    LO    TS
CP0573279  Compound Info	US9163012, 59    Show/Hide	C24H29ClN4O3	1
1	IC50 = 1.92 nM  Bioactivity Info	TI    LI    LO    TS
CP0521497  Compound Info	US9163012, 56    Show/Hide	C25H30N4O4S	1
1	IC50 = 1.95 nM  Bioactivity Info	TI    LI    LO    TS
CP0478267  Compound Info	US9163012, 17    Show/Hide	C25H30N2O3	1
1	IC50 = 1.96 nM  Bioactivity Info	TI    LI    LO    TS
CP0316539  Compound Info	N-(2-adamantyl)-4-bromo-1-[2-(methanesulfonamido)-2-oxoethyl]spiro[1,2-dihydroindene-3,4'-piperidine]-1'-carboxamide    Show/Hide	C27H36BrN3O4S	1
1	IC50 = 2 nM  Bioactivity Info	TI    LI    LO    TS
CP0323223  Compound Info	2-[(3S)-1'-[(adamantan-2-yl)carbamoyl]-7-bromo-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetic acid    Show/Hide	C26H33BrN2O3	1
1	IC50 = 2 nM  Bioactivity Info	TI    LI    LO    TS
CP0427990  Compound Info	(R)-3-Isobutoxycarbonylamino-pyrrolidine-1-carboxylic acid adamantan-2-yl ester    Show/Hide	C20H32N2O4	1
1	IC50 = 2 nM  Bioactivity Info	TI    LI    LO    TS
CP0224277  Compound Info	(6S)-3-[(1S)-1-[4-(2,4-difluorophenyl)phenyl]ethyl]-6-(4-fluorophenyl)-2-oxo-6-[2-(sulfamoylamino)ethyl]-1,3-oxazinane    Show/Hide	C26H26F3N3O4S	2
1	IC50 = 2 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 37 nM  Bioactivity Info	TI    LI    LO    TS
CP0259350  Compound Info	4-[(3R)-3-methyl-4-[5-[(2R)-1,1,1-trifluoro-2-hydroxypropan-2-yl]thiophen-2-yl]sulfonylpiperazin-1-yl]-3-(trifluoromethyl)benzamide    Show/Hide	C20H21F6N3O4S2	1
1	IC50 = 2 nM  Bioactivity Info	TI    LI    LO    TS
CP0425546  Compound Info	US9163012, 55    Show/Hide	C25H30N4O4S	1
1	IC50 = 2.07 nM  Bioactivity Info	TI    LI    LO    TS
CP0521494  Compound Info	US9163012, 49    Show/Hide	C26H36N2O4	1
1	IC50 = 2.07 nM  Bioactivity Info	TI    LI    LO    TS
CP0214909  Compound Info	2-{1'-[(adamantan-2-yl)carbamoyl]-7-chloro-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl}acetic acid    Show/Hide	C26H33ClN2O3	1
1	IC50 = 2.2 nM  Bioactivity Info	TI    LI    LO    TS
CP0514309  Compound Info	2-Phenyl-piperidine-1-carboxylic acid adamantan-2-ylamide    Show/Hide	C22H30N2O	1
1	IC50 = 2.2 nM  Bioactivity Info	TI    LI    LO    TS
CP0572356  Compound Info	US9163012, 15    Show/Hide	C26H35NO5	1
1	IC50 = 2.39 nM  Bioactivity Info	TI    LI    LO    TS
CP0962346  Compound Info	US9163012, 66    Show/Hide	C24H27N5O4	1
1	IC50 = 2.48 nM  Bioactivity Info	TI    LI    LO    TS
CP0060926  Compound Info	(S)-3-(3-Cyano-pyridin-2-ylamino)-pyrrolidine-1-carboxylic acid 5-carbamoyl-adamantan-2-yl ester    Show/Hide	C22H27N5O3	1
1	IC50 = 2.6 nM  Bioactivity Info	TI    LI    LO    TS
CP0406767  Compound Info	US9163012, 4    Show/Hide	C21H25F3N2O4	1
1	IC50 = 2.63 nM  Bioactivity Info	TI    LI    LO    TS
CP0902143  Compound Info	US9163012, 54    Show/Hide	C24H28N4O4S	1
1	IC50 = 2.67 nM  Bioactivity Info	TI    LI    LO    TS
CP0243880  Compound Info	(R)-3-tert-Butoxycarbonylamino-pyrrolidine-1-carboxylic acid adamantan-2-yl ester    Show/Hide	C20H32N2O4	1
1	IC50 = 2.7 nM  Bioactivity Info	TI    LI    LO    TS
CP0305088  Compound Info	(6R)-6-(2-aminoethyl)-3-[(1S)-1-[4-(2,4-difluorophenyl)phenyl]ethyl]-6-(4-fluorophenyl)-1,3-oxazinan-2-one    Show/Hide	C26H25F3N2O2	1
1	IC50 = 2.7 nM  Bioactivity Info	TI    LI    LO    TS
CP0297085  Compound Info	2-[(6S)-3-[(1S)-1-[4-(2,4-difluorophenyl)phenyl]ethyl]-6-(4-fluorophenyl)-2-oxo-1,3-oxazinan-6-yl]acetamide    Show/Hide	C26H23F3N2O3	2
1	IC50 = 2.8 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 62 nM  Bioactivity Info	TI    LI    LO    TS
CP0506527  Compound Info	(R)-3-(tert-Butoxycarbonyl-methyl-amino)-pyrrolidine-1-carboxylic acid adamantan-2-yl ester    Show/Hide	C21H34N2O4	1
1	IC50 = 2.9 nM  Bioactivity Info	TI    LI    LO    TS
CP0522216  Compound Info	US9163012, 62    Show/Hide	C24H30N4O4	1
1	IC50 = 3.07 nM  Bioactivity Info	TI    LI    LO    TS
CP0427992  Compound Info	(R)-3-(4-Trifluoromethyl-pyridin-2-ylamino)-pyrrolidine-1-carboxylic acid 5-carbamoyl-adamantan-2-yl ester    Show/Hide	C22H27F3N4O3	1
1	IC50 = 3.1 nM  Bioactivity Info	TI    LI    LO    TS
CP0070037  Compound Info	1-[2-[(6R)-3-[(1S)-1-[4-(2,4-difluorophenyl)phenyl]ethyl]-6-(4-fluorophenyl)-2-oxo-1,3-oxazinan-6-yl]ethyl]-3-methylurea    Show/Hide	C28H28F3N3O3	1
1	IC50 = 3.1 nM  Bioactivity Info	TI    LI    LO    TS
CP0406768  Compound Info	US9163012, 70    Show/Hide	C25H29N5O4	1
1	IC50 = 3.14 nM  Bioactivity Info	TI    LI    LO    TS
CP0396748  Compound Info	3-[3-(2,4-difluorophenyl)phenyl]-6-phenyl-6-prop-2-enyl-1,3-oxazinan-2-one    Show/Hide	C25H21F2NO2	1
1	IC50 = 3.2 nM  Bioactivity Info	TI    LI    LO    TS
CP0268759  Compound Info	2-{1'-[(adamantan-2-yl)carbamoyl]-5-chloro-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl}acetic acid    Show/Hide	C26H33ClN2O3	1
1	IC50 = 3.4 nM  Bioactivity Info	TI    LI    LO    TS
CP0290311  Compound Info	2-{1'-[(adamantan-2-yl)carbamoyl]-6-chloro-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl}acetic acid    Show/Hide	C26H33ClN2O3	1
1	IC50 = 3.4 nM  Bioactivity Info	TI    LI    LO    TS
CP0316537  Compound Info	2-{1'-[(adamantan-2-yl)carbamoyl]-4-methyl-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl}acetic acid    Show/Hide	C27H36N2O3	1
1	IC50 = 3.4 nM  Bioactivity Info	TI    LI    LO    TS
CP0038296  Compound Info	(R)-3-tert-Butoxycarbonylamino-pyrrolidine-1-carboxylic acid 5-carbamoyl-adamantan-2-yl ester    Show/Hide	C21H33N3O5	1
1	IC50 = 3.4 nM  Bioactivity Info	TI    LI    LO    TS
CP0478269  Compound Info	US9163012, 28    Show/Hide	C20H25ClN4O5	1
1	IC50 = 3.69 nM  Bioactivity Info	TI    LI    LO    TS
CP0424131  Compound Info	US8927539, 1    Show/Hide	C25H26FNO2	1
1	IC50 = 3.7 nM  Bioactivity Info	TI    LI    LO    TS
CP0504569  Compound Info	(R)-3-tert-Butoxycarbonylamino-pyrrolidine-1-carboxylic acid 5-hydroxy-adamantan-2-yl ester    Show/Hide	C20H32N2O5	1
1	IC50 = 3.8 nM  Bioactivity Info	TI    LI    LO    TS
CP0483620  Compound Info	(5S)-2-{[(1S)-1-(2-fluorophenyl)ethyl]amino}-5-methyl-5-(propan-2-yl)-4,5-dihydro-1,3-thiazol-4-one    Show/Hide	C15H19FN2OS	1
1	IC50 = 4 nM  Bioactivity Info	TI    LI    LO    TS
CP0311008  Compound Info	1-[3-[(6R)-3-[(1S)-1-[4-(2,4-difluorophenyl)phenyl]ethyl]-6-(4-fluorophenyl)-2-oxo-1,3-oxazinan-6-yl]propyl]-3-methylurea    Show/Hide	C29H30F3N3O3	1
1	IC50 = 4.1 nM  Bioactivity Info	TI    LI    LO    TS
CP0966863  Compound Info	US9163012, 61    Show/Hide	C23H28N4O4	1
1	IC50 = 4.17 nM  Bioactivity Info	TI    LI    LO    TS
CP0468485  Compound Info	3-[3-(3-fluorophenyl)phenyl]-6-methyl-6-phenyl-1,3-oxazinan-2-one    Show/Hide	C23H20FNO2	1
1	IC50 = 4.2 nM  Bioactivity Info	TI    LI    LO    TS
CP0523674  Compound Info	(S)-3-tert-Butoxycarbonylamino-pyrrolidine-1-carboxylic acid 5-carbamoyl-adamantan-2-yl ester    Show/Hide	C21H33N3O5	1
1	IC50 = 4.4 nM  Bioactivity Info	TI    LI    LO    TS
CP0473572  Compound Info	3-[3-(2,4-difluorophenyl)phenyl]-6-(3-hydroxypropyl)-6-phenyl-1,3-oxazinan-2-one    Show/Hide	C25H23F2NO3	1
1	IC50 = 4.4 nM  Bioactivity Info	TI    LI    LO    TS
CP0396747  Compound Info	6-methyl-6-phenyl-3-(3-phenylphenyl)-1,3-oxazinan-2-one    Show/Hide	C23H21NO2	1
1	IC50 = 4.7 nM  Bioactivity Info	TI    LI    LO    TS
CP0554136  Compound Info	US8927539, 3    Show/Hide	C29H30N2O3	1
1	IC50 = 4.9 nM  Bioactivity Info	TI    LI    LO    TS
CP0045322  Compound Info	N-(5-hydroxy-2-adamantyl)-2-[4-[5-(trifluoromethyl)pyridin-2-yl]piperazin-1-yl]propanamide    Show/Hide	C23H31F3N4O2	1
1	IC50 = 5 nM  Bioactivity Info	TI    LI    LO    TS
CP0541915  Compound Info	N-(5-hydroxy-2-adamantyl)-2-methyl-2-(3-methylphenyl)propanamide    Show/Hide	C21H29NO2	1
1	IC50 = 5 nM  Bioactivity Info	TI    LI    LO    TS
CP0479531  Compound Info	2-adamantyl piperidine-1-carboxylate    Show/Hide	C16H25NO2	1
1	IC50 = 5 nM  Bioactivity Info	TI    LI    LO    TS
CP0408902  Compound Info	3-(3,4-Dichloro-benzenesulfonyl)-thiazolidine-2-carboxylic acid(5-carbamoyl-adamantan-2-yl)-amide    Show/Hide	C21H25Cl2N3O4S2	1
1	IC50 = 5 nM  Bioactivity Info	TI    LI    LO    TS
CP0546119  Compound Info	US9163012, 75    Show/Hide	C25H29N5O3	1
1	IC50 = 5.03 nM  Bioactivity Info	TI    LI    LO    TS
CP0479548  Compound Info	(R)-3-(4-Trifluoromethyl-pyrimidin-2-ylamino)-pyrrolidine-1-carboxylic acid 5-carbamoyl-adamantan-2-yl ester    Show/Hide	C21H26F3N5O3	1
1	IC50 = 5.2 nM  Bioactivity Info	TI    LI    LO    TS
CP0557072  Compound Info	US8927539, 8    Show/Hide	C23H28BrNO3	1
1	IC50 = 5.3 nM  Bioactivity Info	TI    LI    LO    TS
CP0522117  Compound Info	(R)-3-Propoxycarbonylamino-pyrrolidine-1-carboxylic acid adamantan-2-yl ester    Show/Hide	C19H30N2O4	1
1	IC50 = 5.4 nM  Bioactivity Info	TI    LI    LO    TS
CP0553805  Compound Info	US8927539, 2    Show/Hide	C25H28FNO3	1
1	IC50 = 5.6 nM  Bioactivity Info	TI    LI    LO    TS
CP0282222  Compound Info	(6R)-6-(3-aminopropyl)-3-[(1S)-1-[4-(2,4-difluorophenyl)phenyl]ethyl]-6-(4-fluorophenyl)-1,3-oxazinan-2-one    Show/Hide	C27H27F3N2O2	1
1	IC50 = 5.7 nM  Bioactivity Info	TI    LI    LO    TS
CP0504571  Compound Info	(R)-3-tert-Butoxycarbonylamino-pyrrolidine-1-carboxylic acid 5-hydroxymethyl-adamantan-2-yl ester    Show/Hide	C21H34N2O5	1
1	IC50 = 5.8 nM  Bioactivity Info	TI    LI    LO    TS
CP0522211  Compound Info	US9163012, 3    Show/Hide	C22H27N5O4	1
1	IC50 = 6.39 nM  Bioactivity Info	TI    LI    LO    TS
CP0533455  Compound Info	(R)-3-Isopropoxycarbonylamino-pyrrolidine-1-carboxylic acid adamantan-2-yl ester    Show/Hide	C19H30N2O4	1
1	IC50 = 6.4 nM  Bioactivity Info	TI    LI    LO    TS
CP0469976  Compound Info	US9163012, 11    Show/Hide	C24H31NO4	1
1	IC50 = 6.65 nM  Bioactivity Info	TI    LI    LO    TS
CP0268757  Compound Info	2-{1'-[(adamantan-2-yl)carbamoyl]-5-methyl-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl}acetic acid    Show/Hide	C27H36N2O3	1
1	IC50 = 6.7 nM  Bioactivity Info	TI    LI    LO    TS
CP0516266  Compound Info	US9163012, 19    Show/Hide	C21H26N2O4	1
1	IC50 = 6.74 nM  Bioactivity Info	TI    LI    LO    TS
CP0468483  Compound Info	N-[2-[(6R)-3-[(1S)-1-[4-(2,4-difluorophenyl)phenyl]ethyl]-6-(4-fluorophenyl)-2-oxo-1,3-oxazinan-6-yl]ethyl]acetamide    Show/Hide	C28H27F3N2O3	2
1	IC50 = 7.1 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 164 nM  Bioactivity Info	TI    LI    LO    TS
CP0522212  Compound Info	US9163012, 14    Show/Hide	C27H37NO5	1
1	IC50 = 7.15 nM  Bioactivity Info	TI    LI    LO    TS
CP0526509  Compound Info	(R)-3-tert-Butoxycarbonylamino-pyrrolidine-1-carboxylic acid 5-cyano-adamantan-2-yl ester    Show/Hide	C21H31N3O4	1
1	IC50 = 7.4 nM  Bioactivity Info	TI    LI    LO    TS
CP0573359  Compound Info	US9163012, 33    Show/Hide	C23H27N3O3S	1
1	IC50 = 7.46 nM  Bioactivity Info	TI    LI    LO    TS
CP0316538  Compound Info	2-{1'-[(adamantan-2-yl)carbamoyl]-7-methyl-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl}acetic acid    Show/Hide	C27H36N2O3	1
1	IC50 = 7.6 nM  Bioactivity Info	TI    LI    LO    TS
CP0054287  Compound Info	3-(Toluene-4-sulfonyl)-thiazolidine-2-carboxylic acid(5-carbamoyl-adamantan-2-yl)-amide    Show/Hide	C22H29N3O4S2	1
1	IC50 = 8 nM  Bioactivity Info	TI    LI    LO    TS
CP0290309  Compound Info	2-{1'-[(adamantan-2-yl)carbamoyl]-6-methyl-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl}acetic acid    Show/Hide	C27H36N2O3	1
1	IC50 = 8.9 nM  Bioactivity Info	TI    LI    LO    TS
CP0533456  Compound Info	(R)-3-Benzyloxycarbonylamino-pyrrolidine-1-carboxylic acid adamantan-2-yl ester    Show/Hide	C23H30N2O4	1
1	IC50 = 9 nM  Bioactivity Info	TI    LI    LO    TS
CP0784545  Compound Info	2-(2-chlorophenylamino)-5-isopropylthiazol-4(5H)-one    Show/Hide	C12H13ClN2OS	1
1	IC50 = 10 nM  Bioactivity Info	TI    LI    LO    TS
CP0343983  Compound Info	2-((S)-1-(2-chlorophenyl)ethylamino)-5-isopropyl-5-methylthiazol-4(5H)-one    Show/Hide	C15H19ClN2OS	1
1	IC50 = 10 nM  Bioactivity Info	TI    LI    LO    TS
CP0397022  Compound Info	(2R)-1-(3-Chloro-4-(4-(4-fluoro-2-(trifluoromethyl)phenyl)-2-methylpiperazin-1-ylsulfonyl)phenyl)piperidine-4-carboxylic Acid    Show/Hide	C24H26ClF4N3O4S	1
1	IC50 = 10 nM  Bioactivity Info	TI    LI    LO    TS
CP0397023  Compound Info	(2R)-1-{[2-Chloro-4-(1H-1,2,4-triazol-1-yl)phenyl]sulfonyl}-4-[4-fluoro-2-(trifluoromethyl)phenyl]-2-methylpiperazine    Show/Hide	C20H18ClF4N5O2S	1
1	IC50 = 10 nM  Bioactivity Info	TI    LI    LO    TS
CP0397024  Compound Info	(2R)-3-Chloro-4-({(2R)-4-[4-fluoro-2-(trifluoromethyl)phenyl]-2-methylpiperazin-1-yl}sulfonyl)benzamide    Show/Hide	C19H18ClF4N3O3S	1
1	IC50 = 10 nM  Bioactivity Info	TI    LI    LO    TS
CP0410561  Compound Info	(2R)-1-(3-Chloro-4-(2-fluoro-4-(4-fluoro-2-(trifluoromethyl)-phenyl)piperazin-1-ylsulfonyl)phenyl)piperidin-4-ol    Show/Hide	C23H26ClF4N3O3S	1
1	IC50 = 10 nM  Bioactivity Info	TI    LI    LO    TS
CP0410567  Compound Info	(2R)-4-[3-Chloro-4-({(2R)-4-[4-fluoro-2-(trifluoromethyl)phenyl]-2-methylpiperazin-1-yl}sulfonyl)phenyl]piperazin-2-one    Show/Hide	C22H23ClF4N4O3S	1
1	IC50 = 10 nM  Bioactivity Info	TI    LI    LO    TS
CP0427273  Compound Info	(2R)-4-[3-Chloro-4-({(2R)-4-[4-fluoro-2-(trifluoromethyl)phenyl]-2-methylpiperazin-1-yl}sulfonyl)phenyl]morpholine    Show/Hide	C22H24ClF4N3O3S	1
1	IC50 = 10 nM  Bioactivity Info	TI    LI    LO    TS
CP0429625  Compound Info	(2R)-1-(4-Bromo-2-chlorophenylsulfonyl)-4-(4-fluoro-2-(trifluoromethyl)phenyl)-2-methylpiperazine    Show/Hide	C18H16BrClF4N2O2S	1
1	IC50 = 10 nM  Bioactivity Info	TI    LI    LO    TS
CP0457493  Compound Info	(2R)-4-[3-Chloro-4-({(2R)-4-[4-fluoro-2-(trifluoromethyl)phenyl]-2-methylpiperazin-1-yl}sulfonyl)phenyl]thiomorpholine-1,1-dioxide    Show/Hide	C22H24ClF4N3O4S2	1
1	IC50 = 10 nM  Bioactivity Info	TI    LI    LO    TS
CP0506354  Compound Info	(2R)-4-(4-(4-Fluoro-2-(trifluoromethyl)phenyl)-2-methylpiperazin-1-ylsulfonyl)benzonitrile    Show/Hide	C19H17F4N3O2S	1
1	IC50 = 10 nM  Bioactivity Info	TI    LI    LO    TS
CP0138700  Compound Info	1-[3-({(2R)-4-[4-fluoro-2-(trifluoromethyl)phenyl]-2-methylpiperazin-1-yl}sulfonyl)phenyl]pyrrolidin-3-ol    Show/Hide	C22H25F4N3O3S	1
1	IC50 = 10 nM  Bioactivity Info	TI    LI    LO    TS
CP0218773  Compound Info	(3R)-1-[3-({(2R)-4-[4-fluoro-2-(trifluoromethyl)phenyl]-2-methylpiperazin-1-yl}sulfonyl)phenyl]pyrrolidin-3-ol    Show/Hide	C22H25F4N3O3S	1
1	IC50 = 10 nM  Bioactivity Info	TI    LI    LO    TS
CP0374510  Compound Info	(2R)-1-[(3,4-dichlorophenyl)sulfonyl]-2-methyl-4-[2-(trifluoromethyl)phenyl]piperazine    Show/Hide	C18H17Cl2F3N2O2S	1
1	IC50 = 10 nM  Bioactivity Info	TI    LI    LO    TS
CP0407969  Compound Info	3-Benzenesulfonyl-thiazolidine-2-carboxylic acid adamantan-2-ylamide    Show/Hide	C20H26N2O3S2	1
1	IC50 = 10 nM  Bioactivity Info	TI    LI    LO    TS
CP0407975  Compound Info	(R)-1-(2-Fluoro-benzenesulfonyl)-pyrrolidine-2-carboxylic acid(5-carbamoyl-adamantan-2-yl)-amide    Show/Hide	C22H28FN3O4S	1
1	IC50 = 10 nM  Bioactivity Info	TI    LI    LO    TS
CP0466786  Compound Info	3-(4-Chloro-benzenesulfonyl)-thiazolidine-2-carboxylic acid adamantan-2-ylamide    Show/Hide	C20H25ClN2O3S2	1
1	IC50 = 10 nM  Bioactivity Info	TI    LI    LO    TS
CP0466787  Compound Info	3-(3,4-Dichloro-benzenesulfonyl)-thiazolidine-2-carboxylic acid adamantan-2-ylamide    Show/Hide	C20H24Cl2N2O3S2	1
1	IC50 = 10 nM  Bioactivity Info	TI    LI    LO    TS
CP0499751  Compound Info	3-(2-Fluoro-benzenesulfonyl)-thiazolidine-2-carboxylic acid adamantan-2-ylamide    Show/Hide	C20H25FN2O3S2	1
1	IC50 = 10 nM  Bioactivity Info	TI    LI    LO    TS
CP0067583  Compound Info	(2R)-3,3,3-trifluoro-2-[5-[(2R)-4-[4-fluoro-2-(trifluoromethyl)phenyl]-2-methylpiperazin-1-yl]sulfonylthiophen-2-yl]-2-hydroxypropanamide    Show/Hide	C19H18F7N3O4S2	1
1	IC50 = 10 nM  Bioactivity Info	TI    LI    LO    TS
CP0128863  Compound Info	4-[(3R)-3-methyl-4-[5-[(2S)-1,1,1-trifluoro-2-hydroxypropan-2-yl]thiophen-2-yl]sulfonylpiperazin-1-yl]-3-(trifluoromethyl)benzamide    Show/Hide	C20H21F6N3O4S2	1
1	IC50 = 10 nM  Bioactivity Info	TI    LI    LO    TS
CP0450265  Compound Info	(2R)-1,1,1-trifluoro-2-[5-[(2R)-4-[4-fluoro-2-(trifluoromethyl)phenyl]-2-methylpiperazin-1-yl]sulfonylthiophen-2-yl]propan-2-ol    Show/Hide	C19H19F7N2O3S2	1
1	IC50 = 10 nM  Bioactivity Info	TI    LI    LO    TS
CP0483436  Compound Info	2,2,2-trifluoro-1-[5-[(2R)-4-[4-fluoro-2-(trifluoromethyl)phenyl]-2-methylpiperazin-1-yl]sulfonylthiophen-2-yl]-1-(1H-1,2,4-triazol-5-yl)ethanol    Show/Hide	C20H18F7N5O3S2	1
1	IC50 = 10 nM  Bioactivity Info	TI    LI    LO    TS
CP0135762  Compound Info	(S)-2-((1S,2S,4R)-Bicyclo[2.2.1]heptan-2-ylamino)-5-isopropyl-5-methylthiazol-4(5H)-one    Show/Hide	C14H22N2OS	1
1	IC50 = 10.1 nM  Bioactivity Info	TI    LI    LO    TS
CP0454886  Compound Info	(5S)-5-methyl-2-[[(1R,2S,4R)-5-oxo-2-bicyclo[2.2.1]heptanyl]imino]-5-propan-2-yl-1,3-thiazolidin-4-one    Show/Hide	C14H20N2O2S	1
1	IC50 = 10.2 nM  Bioactivity Info	TI    LI    LO    TS
CP0423421  Compound Info	2-[(S)-1-(4-Fluorophenyl)ethylamino]-5-(1-hydroxycyclopentyl)-5-methylthiazol-4(5H)-one    Show/Hide	C17H21FN2O2S	1
1	IC50 = 11 nM  Bioactivity Info	TI    LI    LO    TS
CP0410566  Compound Info	(2R)-4-(3-Fluoro-4-(4-(4-fluoro-2-(trifluoromethyl)phenyl)-2-methylpiperazin-1-ylsulfonyl)phenyl)morpholine    Show/Hide	C22H24F5N3O3S	1
1	IC50 = 11 nM  Bioactivity Info	TI    LI    LO    TS
CP0498950  Compound Info	(2R)-1-[(2-Chloro-4-pyrrolidin-1-ylphenyl)sulfonyl]-4-[4-fluoro-2-(trifluoromethyl)phenyl]-2-methylpiperazine    Show/Hide	C22H24ClF4N3O2S	1
1	IC50 = 11 nM  Bioactivity Info	TI    LI    LO    TS
CP0256078  Compound Info	methyl 1-[3-[(2R)-4-[4-fluoro-2-(trifluoromethyl)phenyl]-2-methylpiperazin-1-yl]sulfonylphenyl]pyrrolidine-3-carboxylate    Show/Hide	C24H27F4N3O4S	1
1	IC50 = 11 nM  Bioactivity Info	TI    LI    LO    TS
CP0379968  Compound Info	3-(3-Fluoro-benzenesulfonyl)-thiazolidine-2-carboxylic acid(5-carbamoyl-adamantan-2-yl)-amide    Show/Hide	C21H26FN3O4S2	1
1	IC50 = 11 nM  Bioactivity Info	TI    LI    LO    TS
CP0407976  Compound Info	3-(4-Fluoro-benzenesulfonyl)-thiazolidine-2-carboxylic acid(5-carbamoyl-adamantan-2-yl)-amide    Show/Hide	C21H26FN3O4S2	1
1	IC50 = 11 nM  Bioactivity Info	TI    LI    LO    TS
CP0533454  Compound Info	(R)-3-Ethoxycarbonylamino-pyrrolidine-1-carboxylic acid adamantan-2-ylester    Show/Hide	C18H28N2O4	1
1	IC50 = 12 nM  Bioactivity Info	TI    LI    LO    TS
CP0494288  Compound Info	3-[3-(2-fluorophenyl)phenyl]-6-methyl-6-phenyl-1,3-oxazinan-2-one    Show/Hide	C23H20FNO2	1
1	IC50 = 12 nM  Bioactivity Info	TI    LI    LO    TS
CP0389761  Compound Info	(5S)-2-[[(1R,2S,4R,5S)-5-hydroxy-2-bicyclo[2.2.1]heptanyl]imino]-5-methyl-5-propan-2-yl-1,3-thiazolidin-4-one    Show/Hide	C14H22N2O2S	1
1	IC50 = 12.7 nM  Bioactivity Info	TI    LI    LO    TS
CP0213664  Compound Info	(2R)-4-[4-fluoro-2-(trifluoromethyl)phenyl]-2-methyl-1-{[3-(1H-pyrazol-1-yl)phenyl]sulfonyl}piperazine    Show/Hide	C21H20F4N4O2S	1
1	IC50 = 13 nM  Bioactivity Info	TI    LI    LO    TS
CP0256079  Compound Info	4-[3-({(2R)-4-[4-fluoro-2-(trifluoromethyl)phenyl]-2-methylpiperazin-1-yl}sulfonyl)phenyl]morpholine    Show/Hide	C22H25F4N3O3S	1
1	IC50 = 13 nM  Bioactivity Info	TI    LI    LO    TS
CP0433330  Compound Info	(2S)-3,3,3-trifluoro-2-[4-[(2R)-4-[4-fluoro-2-(trifluoromethyl)phenyl]-2-methylpiperazin-1-yl]sulfonylphenyl]-2-hydroxypropanamide    Show/Hide	C21H20F7N3O4S	1
1	IC50 = 13 nM  Bioactivity Info	TI    LI    LO    TS
CP0516269  Compound Info	US9163012, 45    Show/Hide	C20H25ClN4O3	1
1	IC50 = 13.49 nM  Bioactivity Info	TI    LI    LO    TS
CP0535213  Compound Info	N-[3-[(4aS,8aR)-3,4,4a,5,6,7,8,8a-octahydro-2H-quinoline-1-carbonyl]phenyl]benzamide    Show/Hide	C23H26N2O2	1
1	IC50 = 14 nM  Bioactivity Info	TI    LI    LO    TS
CP0778552  Compound Info	(R)-2-(2-fluorophenylamino)-5-isopropylthiazol-4(5H)-one    Show/Hide	C12H13FN2OS	1
1	IC50 = 15 nM  Bioactivity Info	TI    LI    LO    TS
CP0372511  Compound Info	(2R)-3-Chloro-4-(4-(4-fluoro-2-(trifluoromethyl)phenyl)-2-methylpiperazin-1-ylsulfonyl)-N,N-dimethylaniline    Show/Hide	C20H22ClF4N3O2S	1
1	IC50 = 15 nM  Bioactivity Info	TI    LI    LO    TS
CP0410549  Compound Info	(2R)-1-[3-Chloro-4-({(2R)-4-[4-fluoro-2-(trifluoromethyl)phenyl]-2-methylpiperazin-1-yl}sulfonyl)phenyl]-N,N-dimethylpiperidin-4-amine    Show/Hide	C25H31ClF4N4O2S	1
1	IC50 = 15 nM  Bioactivity Info	TI    LI    LO    TS
CP0333759  Compound Info	(2R)-4-[4-fluoro-2-(trifluoromethyl)phenyl]-2-methyl-1-[(3-piperidin-1-ylphenyl)sulfonyl]piperazine    Show/Hide	C23H27F4N3O2S	1
1	IC50 = 15 nM  Bioactivity Info	TI    LI    LO    TS
CP0517484  Compound Info	(5S)-2-[[(1R,2S,4R,5R)-5-hydroxy-2-bicyclo[2.2.1]heptanyl]imino]-5-methyl-5-propan-2-yl-1,3-thiazolidin-4-one    Show/Hide	C14H22N2O2S	1
1	IC50 = 15 nM  Bioactivity Info	TI    LI    LO    TS
CP0908163  Compound Info	1,1,1-trifluoro-2-(5-((R)-4-(4-fluoro-2-(trifluoromethyl)phenyl)-2-methylpiperazin-1-ylsulfonyl)thiophen-2-yl)propan-2-ol    Show/Hide	C19H19F7N2O3S2	1
1	IC50 = 15 nM  Bioactivity Info	TI    LI    LO    TS
CP0373288  Compound Info	(R)-3-(Benzyl-tert-butoxycarbonyl-amino)-pyrrolidine-1-carboxylic acid adamantan-2-yl ester    Show/Hide	C27H38N2O4	1
1	IC50 = 15.3 nM  Bioactivity Info	TI    LI    LO    TS
CP0526508  Compound Info	(R)-3-tert-Butoxycarbonylamino-pyrrolidine-1-carboxylic acid 5-acetylamino-adamantan-2-yl ester    Show/Hide	C22H35N3O5	1
1	IC50 = 15.7 nM  Bioactivity Info	TI    LI    LO    TS
CP0496339  Compound Info	(2R)-3-Chloro-4-(4-(4-fluoro-2-(trifluoromethyl)phenyl)-2-methylpiperazin-1-ylsulfonyl)benzonitrile    Show/Hide	C19H16ClF4N3O2S	1
1	IC50 = 16 nM  Bioactivity Info	TI    LI    LO    TS
CP0479530  Compound Info	N-(2-adamantyl)piperidine-1-carboxamide    Show/Hide	C16H26N2O	2
1	IC50 = 16 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 16.1 nM  Bioactivity Info	TI    LI    LO    TS
CP0379969  Compound Info	3-(4-Methoxy-benzenesulfonyl)-thiazolidine-2-carboxylic acid(5-carbamoyl-adamantan-2-yl)-amide    Show/Hide	C22H29N3O5S2	1
1	IC50 = 16 nM  Bioactivity Info	TI    LI    LO    TS
CP0414447  Compound Info	(5S)-2-[[(1S,2S,4R)-2-bicyclo[2.2.1]heptanyl]imino]-5-methyl-5-prop-1-en-2-yl-1,3-thiazolidin-4-one    Show/Hide	C14H20N2OS	1
1	IC50 = 16 nM  Bioactivity Info	TI    LI    LO    TS
CP0778563  Compound Info	2-(2-chlorophenylamino)-5-cyclopentylthiazol-4(5H)-one    Show/Hide	C14H15ClN2OS	1
1	IC50 = 17 nM  Bioactivity Info	TI    LI    LO    TS
CP0462630  Compound Info	(2R)-1-(3-Chloro-4-(4-(4-fluoro-2-(trifluoromethyl)phenyl)-2-methylpiperazin-1-ylsulfonyl)phenyl)piperidine-4-carboxamide    Show/Hide	C24H27ClF4N4O3S	1
1	IC50 = 17 nM  Bioactivity Info	TI    LI    LO    TS
CP0483438  Compound Info	(2S)-1,1,1-trifluoro-2-[5-[(2R)-4-[4-fluoro-2-(trifluoromethyl)phenyl]-2-methylpiperazin-1-yl]sulfonylthiophen-2-yl]propan-2-ol    Show/Hide	C19H19F7N2O3S2	1
1	IC50 = 17 nM  Bioactivity Info	TI    LI    LO    TS
CP0529502  Compound Info	US9163012, 23    Show/Hide	C19H26N4O4	1
1	IC50 = 17.62 nM  Bioactivity Info	TI    LI    LO    TS
CP0192853  Compound Info	2- ((S)-1-(2-fluorophenyl)ethylamino)-5-(2-fluoropropan-2-yl)-5-methylthiazol-5H)-one    Show/Hide	C15H18F2N2OS	1
1	IC50 = 18 nM  Bioactivity Info	TI    LI    LO    TS
CP0215290  Compound Info	(5R)-2-{[(1S)-1-(2-fluorophenyl)ethyl]amino}-5-methyl-5-(propan-2-yl)-4,5-dihydro-1,3-thiazol-4-one    Show/Hide	C15H19FN2OS	1
1	IC50 = 18 nM  Bioactivity Info	TI    LI    LO    TS
CP0221125  Compound Info	2-((S)-1-(2-fluorophenyl)ethylamino)-5-isopropyl-5-methylthiazol-4(5H)-one    Show/Hide	C15H19FN2OS	1
1	IC50 = 18 nM  Bioactivity Info	TI    LI    LO    TS
CP0284957  Compound Info	2-((S)-1-(2-bromophenyl)ethylamino)-5-isopropyl-5-methylthiazol-4(5H)-one    Show/Hide	C15H19BrN2OS	1
1	IC50 = 18 nM  Bioactivity Info	TI    LI    LO    TS
CP0452528  Compound Info	2-[(S)-1-(2-Chlorophenyl)ethylamino]-5-(2-hydroxypropan-2-yl)-5-methylthiazol-4(5H)-one    Show/Hide	C15H19ClN2O2S	1
1	IC50 = 18 nM  Bioactivity Info	TI    LI    LO    TS
CP0506073  Compound Info	(2R)-1-[3-Chloro-4-({(2R)-4-[4-fluoro-2-(trifluoromethyl)phenyl]-2-methylpiperazin-1-yl}sulfonyl)phenyl]piperazin-2-one    Show/Hide	C22H23ClF4N4O3S	1
1	IC50 = 18 nM  Bioactivity Info	TI    LI    LO    TS
CP0506075  Compound Info	(2R)-1-(2-Chloro-4-(difluoromethoxy)phenylsulfonyl)-4-(4-fluoro-2-(trifluoromethyl)phenyl)-2-methylpiperazine    Show/Hide	C19H17ClF6N2O3S	1
1	IC50 = 18 nM  Bioactivity Info	TI    LI    LO    TS
CP0739802  Compound Info	5-cyclopentyl-2-(2-fluorophenylamino)thiazol-4(5H)-one    Show/Hide	C14H15FN2OS	1
1	IC50 = 19 nM  Bioactivity Info	TI    LI    LO    TS
CP0284960  Compound Info	2-Benzylamine analog 3    Show/Hide	C15H20N2OS	1
1	IC50 = 20 nM  Bioactivity Info	TI    LI    LO    TS
CP0498946  Compound Info	(2R)-4-(4-Fluoro-2-(trifluoromethyl)phenyl)-1-(4-methoxyphenylsulfonyl)-2-methylpiperazine    Show/Hide	C19H20F4N2O3S	1
1	IC50 = 20 nM  Bioactivity Info	TI    LI    LO    TS
CP0379967  Compound Info	3-(Toluene-4-sulfonyl)-thiazolidine-2-carboxylic acid adamantan-2-ylamide    Show/Hide	C21H28N2O3S2	1
1	IC50 = 20 nM  Bioactivity Info	TI    LI    LO    TS
CP0499750  Compound Info	3-(4-Fluoro-benzenesulfonyl)-thiazolidine-2-carboxylic acid adamantan-2-ylamide    Show/Hide	C20H25FN2O3S2	1
1	IC50 = 20 nM  Bioactivity Info	TI    LI    LO    TS
CP0504023  Compound Info	3-Benzyl-thiazolidine-2-carboxylic acid adamantan-2-ylamide    Show/Hide	C21H28N2OS	1
1	IC50 = 20 nM  Bioactivity Info	TI    LI    LO    TS
CP0386207  Compound Info	(2R)-3,3,3-trifluoro-2-[2-[(2R)-4-[4-fluoro-2-(trifluoromethyl)phenyl]-2-methylpiperazin-1-yl]sulfonyl-1,3-thiazol-5-yl]-2-hydroxypropanamide    Show/Hide	C18H17F7N4O4S2	1
1	IC50 = 20 nM  Bioactivity Info	TI    LI    LO    TS
CP0533457  Compound Info	(R)-3-(2,6-Dimethyl-pyrimidin-4-ylamino)-pyrrolidine-1-carboxylic acid 5-carbamoyl-adamantan-2-yl ester    Show/Hide	C22H31N5O3	1
1	IC50 = 20.7 nM  Bioactivity Info	TI    LI    LO    TS
CP0425543  Compound Info	US9163012, 21    Show/Hide	C20H26N2O3	1
1	IC50 = 20.78 nM  Bioactivity Info	TI    LI    LO    TS
CP0918464  Compound Info	2-(2,6-dichlorophenylamino)-5-isopropylthiazol-4(5H)-one    Show/Hide	C12H12Cl2N2OS	1
1	IC50 = 21 nM  Bioactivity Info	TI    LI    LO    TS
CP0138702  Compound Info	(2R)-4-[4-fluoro-2-(trifluoromethyl)phenyl]-2-methyl-1-{[3-(4-methylpiperazin-1-yl)phenyl]sulfonyl}piperazine    Show/Hide	C23H28F4N4O2S	1
1	IC50 = 21 nM  Bioactivity Info	TI    LI    LO    TS
CP0533458  Compound Info	(R)-3-(5-Trifluoromethyl-[1,3,4]thiadiazol-2-ylamino)-pyrrolidine-1-carboxylic acid 5-carbamoyl-adamantan-2-yl ester    Show/Hide	C19H24F3N5O3S	1
1	IC50 = 21.3 nM  Bioactivity Info	TI    LI    LO    TS
CP0432930  Compound Info	(5S)-2-[[(1S,2S,4R)-2-bicyclo[2.2.1]heptanyl]imino]-5-(1,1-dihydroxyethyl)-5-methyl-1,3-thiazolidin-4-one    Show/Hide	C13H20N2O3S	1
1	IC50 = 21.3 nM  Bioactivity Info	TI    LI    LO    TS
CP0501566  Compound Info	3-[(6R)-3-[(1S)-1-[4-(2,4-difluorophenyl)phenyl]ethyl]-6-(4-fluorophenyl)-2-oxo-1,3-oxazinan-6-yl]-N-methylpropanamide    Show/Hide	C28H27F3N2O3	1
1	IC50 = 22 nM  Bioactivity Info	TI    LI    LO    TS
CP0503523  Compound Info	1-[2-[(6R)-3-[(1S)-1-[4-(2,4-difluorophenyl)phenyl]ethyl]-6-(4-fluorophenyl)-2-oxo-1,3-oxazinan-6-yl]ethyl]-3-ethylurea    Show/Hide	C29H30F3N3O3	1
1	IC50 = 22 nM  Bioactivity Info	TI    LI    LO    TS
CP0548647  Compound Info	3-(3-bromophenyl)-6-methyl-6-phenyl-1,3-oxazinan-2-one    Show/Hide	C17H16BrNO2	1
1	IC50 = 23 nM  Bioactivity Info	TI    LI    LO    TS
CP0450251  Compound Info	(2R)-3,3,3-trifluoro-2-[3-[(2R)-4-[4-fluoro-2-(trifluoromethyl)phenyl]-2-methylpiperazin-1-yl]sulfonylphenyl]-2-hydroxypropanamide    Show/Hide	C21H20F7N3O4S	1
1	IC50 = 23 nM  Bioactivity Info	TI    LI    LO    TS
CP0550183  Compound Info	US8927539, 4    Show/Hide	C25H28N4O2	1
1	IC50 = 23 nM  Bioactivity Info	TI    LI    LO    TS
CP0040668  Compound Info	(2R)-4-[4-fluoro-2-(trifluoromethyl)phenyl]-2-methyl-1-{[3-(1H-1,2,4-triazol-1-yl)phenyl]sulfonyl}piperazine    Show/Hide	C20H19F4N5O2S	1
1	IC50 = 26 nM  Bioactivity Info	TI    LI    LO    TS
CP0523904  Compound Info	US9163012, 18    Show/Hide	C23H29NO4	1
1	IC50 = 27.79 nM  Bioactivity Info	TI    LI    LO    TS
CP0789330  Compound Info	5-isopropyl-2-(2-(trifluoromethyl)phenylamino)thiazol-4(5H)-one    Show/Hide	C13H13F3N2OS	1
1	IC50 = 28 nM  Bioactivity Info	TI    LI    LO    TS
CP0830832  Compound Info	2-(2,5-difluorophenylamino)-5-isopropylthiazol-4(5H)-one    Show/Hide	C12H12F2N2OS	1
1	IC50 = 28 nM  Bioactivity Info	TI    LI    LO    TS
CP0505015  Compound Info	(2R)-1-(4-Bromophenylsulfonyl)-4-(4-fluoro-2-(trifluoromethyl)-phenyl)-2-methylpiperazine    Show/Hide	C18H17BrF4N2O2S	1
1	IC50 = 28 nM  Bioactivity Info	TI    LI    LO    TS
CP0302962  Compound Info	(3S)-1-[3-({(2R)-4-[4-fluoro-2-(trifluoromethyl)phenyl]-2-methylpiperazin-1-yl}sulfonyl)phenyl]pyrrolidin-3-ol    Show/Hide	C22H25F4N3O3S	1
1	IC50 = 28 nM  Bioactivity Info	TI    LI    LO    TS
CP0346551  Compound Info	(2R)-1-{[3-(4-ethylpiperazin-1-yl)phenyl]sulfonyl}-4-[4-fluoro-2-(trifluoromethyl)phenyl]-2-methylpiperazine    Show/Hide	C24H30F4N4O2S	1
1	IC50 = 30 nM  Bioactivity Info	TI    LI    LO    TS
CP0452461  Compound Info	(2R)-1-(2-Chloro-4-(2-methoxyethoxy)phenylsulfonyl)-4-(4-fluoro-2-(trifluoromethyl)phenyl)-2-methylpiperazine    Show/Hide	C21H23ClF4N2O4S	1
1	IC50 = 31 nM  Bioactivity Info	TI    LI    LO    TS
CP0450736  Compound Info	2-[(S)-1-(4-Fluorophenyl)ethylamino]-5-(1-hydroxycyclobutyl)-5-methylthiazol-4(5H)-one    Show/Hide	C16H19FN2O2S	1
1	IC50 = 32 nM  Bioactivity Info	TI    LI    LO    TS
CP0346549  Compound Info	1-[3-({(2R)-4-[4-fluoro-2-(trifluoromethyl)phenyl]-2-methylpiperazin-1-yl}sulfonyl)phenyl]pyrrolidine-3-carboxamide    Show/Hide	C23H26F4N4O3S	1
1	IC50 = 32 nM  Bioactivity Info	TI    LI    LO    TS
CP0739803  Compound Info	2-(2-chlorophenylamino)-5-cyclohexylthiazol-4(5H)-one    Show/Hide	C15H17ClN2OS	1
1	IC50 = 33 nM  Bioactivity Info	TI    LI    LO    TS
CP0132363  Compound Info	(5S)-2-{[(1S)-1-(2-fluorophenyl)ethyl]amino}-5-methyl-5-(trifluoromethyl)-4,5-dihydro-1,3-thiazol-4-one    Show/Hide	C13H12F4N2OS	1
1	IC50 = 33 nM  Bioactivity Info	TI    LI    LO    TS
CP0957878  Compound Info	US9163012, 65    Show/Hide	C24H27N5O4	1
1	IC50 = 33.3 nM  Bioactivity Info	TI    LI    LO    TS
CP0450737  Compound Info	(5S)-2-{[(1S)-1-(4-fluorophenyl)ethyl]amino}-5-(1-hydroxy-1-methylethyl)-5-methyl-1,3-thiazol-4(5H)-one    Show/Hide	C15H19FN2O2S	1
1	IC50 = 34 nM  Bioactivity Info	TI    LI    LO    TS
CP0407974  Compound Info	(S)-1-(2-Fluoro-benzenesulfonyl)-pyrrolidine-2-carboxylic acid(5-carbamoyl-adamantan-2-yl)-amide    Show/Hide	C22H28FN3O4S	1
1	IC50 = 37 nM  Bioactivity Info	TI    LI    LO    TS
CP0491354  Compound Info	US8927539, 9    Show/Hide	C29H34N2O4	1
1	IC50 = 37 nM  Bioactivity Info	TI    LI    LO    TS
CP0491355  Compound Info	US8927539, 10    Show/Hide	C31H36N2O4	1
1	IC50 = 38 nM  Bioactivity Info	TI    LI    LO    TS
CP0532681  Compound Info	US8927539, 5    Show/Hide	C26H32N4O2	1
1	IC50 = 39 nM  Bioactivity Info	TI    LI    LO    TS
CP0523905  Compound Info	US9163012, 25    Show/Hide	C19H27N3O4	1
1	IC50 = 39.46 nM  Bioactivity Info	TI    LI    LO    TS
CP0803239  Compound Info	2-(2,4-dichlorophenylamino)-5-isopropylthiazol-4(5H)-one    Show/Hide	C12H12Cl2N2OS	1
1	IC50 = 40 nM  Bioactivity Info	TI    LI    LO    TS
CP0442432  Compound Info	2-(S)-Phenethylamine analog 6    Show/Hide	C16H19F3N2OS	1
1	IC50 = 40 nM  Bioactivity Info	TI    LI    LO    TS
CP0506074  Compound Info	(2R)-1-(4-tert-Butoxy-2-chlorophenylsulfonyl)-4-(4-fluoro-2-(trifluoromethyl)phenyl)-2-methylpiperazine    Show/Hide	C22H25ClF4N2O3S	1
1	IC50 = 40 nM  Bioactivity Info	TI    LI    LO    TS
CP0468488  Compound Info	3-(2-chlorophenyl)-6-methyl-6-phenyl-1,3-oxazinan-2-one    Show/Hide	C17H16ClNO2	1
1	IC50 = 40 nM  Bioactivity Info	TI    LI    LO    TS
CP0284958  Compound Info	2-(S)-Phenethylamine analog 7    Show/Hide	C16H19F3N2OS	1
1	IC50 = 41 nM  Bioactivity Info	TI    LI    LO    TS
CP0491241  Compound Info	4-Phenyl-piperidine-1,4-dicarboxylic acid 1-adamantan-2-ylamide 4-amide    Show/Hide	C23H31N3O2	1
1	IC50 = 41.6 nM  Bioactivity Info	TI    LI    LO    TS
CP0778554  Compound Info	5-cyclohexyl-2-(2-fluorophenylamino)thiazol-4(5H)-one    Show/Hide	C15H17FN2OS	1
1	IC50 = 43 nM  Bioactivity Info	TI    LI    LO    TS
CP0498890  Compound Info	(S)-5-(2-Hydroxypropan-2-yl)-5-methyl-2-{1-[2-(trifluoromethyl)-phenyl]ethylamino}thiazol-4(5H)-one    Show/Hide	C16H19F3N2O2S	1
1	IC50 = 43 nM  Bioactivity Info	TI    LI    LO    TS
CP0386208  Compound Info	1,1,1-trifluoro-2-[4-[(2R)-4-[4-fluoro-2-(trifluoromethyl)phenyl]-2-methylpiperazin-1-yl]sulfonyl-1-methylimidazol-2-yl]propan-2-ol    Show/Hide	C19H21F7N4O3S	1
1	IC50 = 43 nM  Bioactivity Info	TI    LI    LO    TS
CP0556157  Compound Info	US9163012, 16    Show/Hide	C25H33NO5	1
1	IC50 = 43.78 nM  Bioactivity Info	TI    LI    LO    TS
CP0830831  Compound Info	2-(2,4-difluorophenylamino)-5-isopropylthiazol-4(5H)-one    Show/Hide	C12H12F2N2OS	1
1	IC50 = 45 nM  Bioactivity Info	TI    LI    LO    TS
CP0803240  Compound Info	2-(2-fluorophenylamino)-5-isopropylthiazol-4(5H)-one    Show/Hide	C12H13FN2OS	1
1	IC50 = 50 nM  Bioactivity Info	TI    LI    LO    TS
CP0397021  Compound Info	(2R)-1-{[2-Chloro-4-(4-fluoropiperidin-1-yl)phenyl]sulfonyl}-4-[4-fluoro-2-(trifluoromethyl)phenyl]-2-methylpiperazine    Show/Hide	C23H25ClF5N3O2S	1
1	IC50 = 50 nM  Bioactivity Info	TI    LI    LO    TS
CP0410568  Compound Info	(2R)-3-Chloro-4-(4-(4-fluoro-2-(trifluoromethyl)phenyl)-2-methylpiperazin-1-ylsulfonyl)phenol    Show/Hide	C18H17ClF4N2O3S	1
1	IC50 = 50 nM  Bioactivity Info	TI    LI    LO    TS
CP0459919  Compound Info	(2S)-3,3,3-trifluoro-2-[2-[(2R)-4-[4-fluoro-2-(trifluoromethyl)phenyl]-2-methylpiperazin-1-yl]sulfonyl-1,3-thiazol-5-yl]-2-hydroxypropanamide    Show/Hide	C18H17F7N4O4S2	1
1	IC50 = 50 nM  Bioactivity Info	TI    LI    LO    TS
CP0535206  Compound Info	2-((S)-1-(4-fluorophenyl)ethylamino)-5-(2-hydroxypropan-2-yl)-5-methylthiazol-4(5H)-one    Show/Hide	C15H19FN2O2S	1
1	IC50 = 51 nM  Bioactivity Info	TI    LI    LO    TS
CP0418049  Compound Info	(2S)-3,3,3-trifluoro-2-[3-[(2R)-4-[4-fluoro-2-(trifluoromethyl)phenyl]-2-methylpiperazin-1-yl]sulfonylphenyl]-2-hydroxypropanamide    Show/Hide	C21H20F7N3O4S	1
1	IC50 = 51 nM  Bioactivity Info	TI    LI    LO    TS
CP0379070  Compound Info	1-[(3,4-dichlorophenyl)sulfonyl]-4-[2-(trifluoromethyl)phenyl]piperazine    Show/Hide	C17H15Cl2F3N2O2S	1
1	IC50 = 52 nM  Bioactivity Info	TI    LI    LO    TS
CP0172645  Compound Info	2-(benzylamino)-5-isopropyl-5-methylthiazol-4(5H)-one    Show/Hide	C14H18N2OS	1
1	IC50 = 53 nM  Bioactivity Info	TI    LI    LO    TS
CP0450726  Compound Info	5-(4-Fluorophenyl)-2-[(S)-1-(4-fluorophenyl)ethylamino]-5-methylthiazol-4(5H)-one    Show/Hide	C18H16F2N2OS	1
1	IC50 = 53 nM  Bioactivity Info	TI    LI    LO    TS
CP0527657  Compound Info	3-(4-Methoxy-benzenesulfonyl)-thiazolidine-2-carboxylic acid adamantan-2-ylamide    Show/Hide	C21H28N2O4S2	1
1	IC50 = 55 nM  Bioactivity Info	TI    LI    LO    TS
CP0250945  Compound Info	2-(S)-Phenethylamine analog 15    Show/Hide	C13H12F4N2OS	1
1	IC50 = 56 nM  Bioactivity Info	TI    LI    LO    TS
CP0452742  Compound Info	4-Hydroxy-4-phenyl-piperidine-1-carboxylic acid adamantan-2-ylamide    Show/Hide	C22H30N2O2	1
1	IC50 = 56.8 nM  Bioactivity Info	TI    LI    LO    TS
CP0399401  Compound Info	1-(3-methoxyphenyl)-2-(phenylsulfonyl)ethanone    Show/Hide	C15H14O4S	1
1	IC50 = 60 nM  Bioactivity Info	TI    LI    LO    TS
CP0236339  Compound Info	(2R)-4-[4-fluoro-2-(trifluoromethyl)phenyl]-2-methyl-1-[(3-pyrrolidin-1-ylphenyl)sulfonyl]piperazine    Show/Hide	C22H25F4N3O2S	1
1	IC50 = 61 nM  Bioactivity Info	TI    LI    LO    TS
CP0423404  Compound Info	1-[(3,4-dichlorophenyl)sulfonyl]-4-[3-(trifluoromethyl)pyridin-2-yl]piperazine    Show/Hide	C16H14Cl2F3N3O2S	1
1	IC50 = 61 nM  Bioactivity Info	TI    LI    LO    TS
CP0506076  Compound Info	(2R)-1-(2-Chloro-4-ethoxyphenylsulfonyl)-4-(4-fluoro-2-(trifluoromethyl)phenyl)-2-methylpiperazine    Show/Hide	C20H21ClF4N2O3S	1
1	IC50 = 63 nM  Bioactivity Info	TI    LI    LO    TS
CP0498348  Compound Info	3-Benzoyl-thiazolidine-2-carboxylic acid adamantan-2-ylamide    Show/Hide	C21H26N2O2S	1
1	IC50 = 63 nM  Bioactivity Info	TI    LI    LO    TS
CP0386206  Compound Info	(2R)-3,3,3-trifluoro-2-[4-[(2R)-4-[4-fluoro-2-(trifluoromethyl)phenyl]-2-methylpiperazin-1-yl]sulfonylphenyl]-2-hydroxypropanamide    Show/Hide	C21H20F7N3O4S	1
1	IC50 = 64 nM  Bioactivity Info	TI    LI    LO    TS
CP0381219  Compound Info	3-Benzenesulfonyl-thiazolidine-2-carboxylic acid(5-carbamoyl-adamantan-2-yl)-amide    Show/Hide	C21H27N3O4S2	1
1	IC50 = 67 nM  Bioactivity Info	TI    LI    LO    TS
CP0384638  Compound Info	1-[(3,4-dichlorophenyl)sulfonyl]-4-[4-fluoro-2-trifluoromethyl)phenyl]piperazine    Show/Hide	C17H14Cl2F4N2O2S	1
1	IC50 = 68 nM  Bioactivity Info	TI    LI    LO    TS
CP0504568  Compound Info	(R)-3-(3,3-Dimethyl-butyrylamino)-pyrrolidine-1-carboxylic acid adamantan-2-yl ester    Show/Hide	C21H34N2O3	1
1	IC50 = 68 nM  Bioactivity Info	TI    LI    LO    TS
CP0298969  Compound Info	1'-[(adamantan-2-yl)carbamoyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-carboxylic acid    Show/Hide	C25H32N2O3	1
1	IC50 = 68.6 nM  Bioactivity Info	TI    LI    LO    TS
CP0346548  Compound Info	1-(3-((R)-4-(4-fluoro-2-(trifluoromethyl)phenyl)-2-methylpiperazin-1-ylsulfonyl)phenyl)pyrrolidine-2-carboxylic acid    Show/Hide	C23H25F4N3O4S	1
1	IC50 = 69 nM  Bioactivity Info	TI    LI    LO    TS
CP0461516  Compound Info	2-[(S)-1-(2-Fluorophenyl)ethylamino]-5-(2-hydroxypropan-2-yl)-5-methylthiazol-4(5H)-one    Show/Hide	C15H19FN2O2S	1
1	IC50 = 70 nM  Bioactivity Info	TI    LI    LO    TS
CP0566109  Compound Info	(5S)-2-[[(1S,2S,4R)-2-bicyclo[2.2.1]heptanyl]imino]-5-[(1S)-1,2-dihydroxyethyl]-5-methyl-1,3-thiazolidin-4-one    Show/Hide	C13H20N2O3S	1
1	IC50 = 71.6 nM  Bioactivity Info	TI    LI    LO    TS
CP0429626  Compound Info	(2R)-1-{[2-Chloro-4-(4,4-difluoropiperidin-1-yl)phenyl]sulfonyl}-4-[4-fluoro-2-(trifluoromethyl)phenyl]-2-methylpiperazine    Show/Hide	C23H24ClF6N3O2S	1
1	IC50 = 74 nM  Bioactivity Info	TI    LI    LO    TS
CP0158847  Compound Info	(2R)-4-[4-fluoro-2-(trifluoromethyl)phenyl]-2-methyl-1-{[3-(1H-pyrazol-1-yl)phenyl]sulfonyl}piperazine    Show/Hide	C21H20F4N4O2S	1
1	IC50 = 74 nM  Bioactivity Info	TI    LI    LO    TS
CP0565579  Compound Info	US8927539, 6    Show/Hide	C29H30N2O3	1
1	IC50 = 74 nM  Bioactivity Info	TI    LI    LO    TS
CP0490318  Compound Info	1-(4-methoxyphenyl)-2-(phenylsulfonyl)ethanone    Show/Hide	C15H14O4S	1
1	IC50 = 75 nM  Bioactivity Info	TI    LI    LO    TS
CP0547166  Compound Info	2-[(S)-1-(4-Chlorophenyl)ethylamino]-5-(3-hydroxypropan-2-yl)-5-methylthiazol-4(5H)-one    Show/Hide	C15H19ClN2O2S	1
1	IC50 = 78 nM  Bioactivity Info	TI    LI    LO    TS
CP0472064  Compound Info	4-{2-[(S)-1-(4-Fluorophenyl)ethylamino]-5-methyl-4-oxo-4,5-dihydrothiazol-5-yl}benzamide    Show/Hide	C19H18FN3O2S	1
1	IC50 = 79 nM  Bioactivity Info	TI    LI    LO    TS
CP0452479  Compound Info	(5S)-2-[[(1S,2S,4R)-2-bicyclo[2.2.1]heptanyl]imino]-5-[(1R)-1,2-dihydroxyethyl]-5-methyl-1,3-thiazolidin-4-one    Show/Hide	C13H20N2O3S	1
1	IC50 = 87 nM  Bioactivity Info	TI    LI    LO    TS
CP0461730  Compound Info	1-(4-fluorophenyl)-2-(phenylsulfonyl)ethanone    Show/Hide	C14H11FO3S	1
1	IC50 = 90 nM  Bioactivity Info	TI    LI    LO    TS
CP0512036  Compound Info	US9163012, 31    Show/Hide	C24H30N4O3	1
1	IC50 = 91.7 nM  Bioactivity Info	TI    LI    LO    TS
CP0410570  Compound Info	(2R)-2-(3-Chloro-4-(4-(4-fluoro-2-(trifluoromethyl)phenyl)-2-methylpiperazin-1-ylsulfonyl)phenoxy)-N,N-dimethylethanamine    Show/Hide	C22H26ClF4N3O3S	1
1	IC50 = 92 nM  Bioactivity Info	TI    LI    LO    TS
CP0499239  Compound Info	(6S)-3-[(1R)-1-[4-(2,4-difluorophenyl)phenyl]ethyl]-6-(4-fluorophenyl)-6-(2-hydroxyethyl)-1,3-oxazinan-2-one    Show/Hide	C26H24F3NO3	1
1	IC50 = 92 nM  Bioactivity Info	TI    LI    LO    TS
CP0215289  Compound Info	(5R)-2-{[(1S)-1-(2-fluorophenyl)ethyl]amino}-5-methyl-5-(trifluoromethyl)-4,5-dihydro-1,3-thiazol-4-one    Show/Hide	C13H12F4N2OS	1
1	IC50 = 96 nM  Bioactivity Info	TI    LI    LO    TS
CP0841218  Compound Info	(S)-2-(2-fluorophenylamino)-5-isopropylthiazol-4(5H)-one    Show/Hide	C12H13FN2OS	1
1	IC50 = 97 nM  Bioactivity Info	TI    LI    LO    TS
CP0507956  Compound Info	(2R)-1-[(2-Chloro-4-piperidin-1-ylphenyl)sulfonyl]-4-[4-fluoro-2-(trifluoromethyl)phenyl]-2-methylpiperazine    Show/Hide	C23H26ClF4N3O2S	1
1	IC50 = 97 nM  Bioactivity Info	TI    LI    LO    TS
CP0527229  Compound Info	(R)-3-tert-Butoxycarbonylamino-pyrrolidine-1-carboxylic acid 5-(1-hydroxy-1-methyl-ethyl)-adamantan-2-yl ester    Show/Hide	C23H38N2O5	1
1	IC50 = 98 nM  Bioactivity Info	TI    LI    LO    TS
CP0492243  Compound Info	4-[4-({(2R)-4-[4-Fluoro-2-(trifluoromethyl)phenyl]-2-methylpiperazin-1-yl}sulfonyl)phenyl]morpholine    Show/Hide	C22H25F4N3O3S	1
1	IC50 = 100 nM  Bioactivity Info	TI    LI    LO    TS
CP0478268  Compound Info	US9163012, 22    Show/Hide	C20H26N2O4	1
1	IC50 = 100 nM  Bioactivity Info	TI    LI    LO    TS
CP0529501  Compound Info	US9163012, 20    Show/Hide	C24H27ClN4O4	1
1	IC50 = 100 nM  Bioactivity Info	TI    LI    LO    TS
CP0572357  Compound Info	US9163012, 29    Show/Hide	C23H28ClN5O4	1
1	IC50 = 100 nM  Bioactivity Info	TI    LI    LO    TS
CP0399403  Compound Info	1-(3,4-dichlorophenyl)-2-(phenylsulfonyl)ethanone    Show/Hide	C14H10Cl2O3S	1
1	IC50 = 101 nM  Bioactivity Info	TI    LI    LO    TS
CP0485315  Compound Info	2-(phenylsulfonyl)-1-p-tolylethanone    Show/Hide	C15H14O3S	1
1	IC50 = 102 nM  Bioactivity Info	TI    LI    LO    TS
CP0476379  Compound Info	3-(3-chlorophenyl)-6-methyl-6-phenyl-1,3-oxazinan-2-one    Show/Hide	C17H16ClNO2	1
1	IC50 = 103 nM  Bioactivity Info	TI    LI    LO    TS
CP0483439  Compound Info	1,1,1-trifluoro-2-[5-[(2R)-4-[4-fluoro-2-(trifluoromethyl)phenyl]-2-methylpiperazin-1-yl]sulfonyl-2-methyl-1,2,4-triazol-3-yl]propan-2-ol    Show/Hide	C18H20F7N5O3S	1
1	IC50 = 104 nM  Bioactivity Info	TI    LI    LO    TS
CP0423419  Compound Info	1-(4-{2-[(S)-1-(4-Fluorophenyl)ethylamino]-5-methyl-4-oxo-4,5-dihydrothiazol-5-yl}phenyl)cyclopropanecarboxamide    Show/Hide	C22H22FN3O2S	1
1	IC50 = 110 nM  Bioactivity Info	TI    LI    LO    TS
CP0493905  Compound Info	2-[(S)-1-(4-Fluorophenyl)ethylamino]-5-[4-(hydroxymethyl)phenyl]-5-methylthiazol-4(5H)-one    Show/Hide	C19H19FN2O2S	1
1	IC50 = 110 nM  Bioactivity Info	TI    LI    LO    TS
CP0439669  Compound Info	(2R)-N-[3-Chloro-4-({4-[4-fluoro-2-(trifluoromethyl)phenyl]-piperazin-1-yl}sulfonyl)phenyl]morpholine-4-carboxamide    Show/Hide	C23H25ClF4N4O4S	1
1	IC50 = 115 nM  Bioactivity Info	TI    LI    LO    TS
CP0764930  Compound Info	2-(o-toluidino)-5-isopropylthiazol-4(5H)-one    Show/Hide	C13H16N2OS	1
1	IC50 = 120 nM  Bioactivity Info	TI    LI    LO    TS
CP0346546  Compound Info	(2R)-4-[4-fluoro-2-(trifluoromethyl)phenyl]-2-methyl-1-{[3-(4H-1,2,4-triazol-4-yl)phenyl]sulfonyl}piperazine    Show/Hide	C20H19F4N5O2S	1
1	IC50 = 120 nM  Bioactivity Info	TI    LI    LO    TS
CP0472063  Compound Info	2-{(S)-[1-(4-fluorophenyl)ethyl]amino}-5-[4-(2-hydroxyethyl)phenyl]-5-methyl-1,3-thiazol-4(5H)-one    Show/Hide	C20H21FN2O2S	1
1	IC50 = 130 nM  Bioactivity Info	TI    LI    LO    TS
CP0441476  Compound Info	2-(phenylsulfonyl)-1-(5-phenylthiophen-2-yl)ethanone    Show/Hide	C18H14O3S2	1
1	IC50 = 134 nM  Bioactivity Info	TI    LI    LO    TS
CP0457492  Compound Info	(2R)-1-{[2-Chloro-4-(4-methylpiperazin-1-yl)phenyl]sulfonyl}-4-[4-fluoro-2-(trifluoromethyl)phenyl]-2-methylpiperazine    Show/Hide	C23H27ClF4N4O2S	1
1	IC50 = 136 nM  Bioactivity Info	TI    LI    LO    TS
CP0418046  Compound Info	(2S)-3,3,3-trifluoro-2-[5-[(2R)-4-[4-fluoro-2-(trifluoromethyl)phenyl]-2-methylpiperazin-1-yl]sulfonylthiophen-2-yl]-2-hydroxypropanamide    Show/Hide	C19H18F7N3O4S2	1
1	IC50 = 145 nM  Bioactivity Info	TI    LI    LO    TS
CP0527658  Compound Info	3-(4-tert-Butyl-benzenesulfonyl)-thiazolidine-2-carboxylic acid adamantan-2-ylamide    Show/Hide	C24H34N2O3S2	1
1	IC50 = 149 nM  Bioactivity Info	TI    LI    LO    TS
CP0166536  Compound Info	1-[3-({(2R)-4-[4-fluoro-2-(trifluoromethyl)phenyl]-2-methylpiperazin-1-yl}sulfonyl)phenyl]pyrrolidine-3-carboxylic acid    Show/Hide	C23H25F4N3O4S	1
1	IC50 = 160 nM  Bioactivity Info	TI    LI    LO    TS
CP0471082  Compound Info	6-methyl-3,6-diphenyl-1,3-oxazinan-2-one    Show/Hide	C17H17NO2	1
1	IC50 = 160 nM  Bioactivity Info	TI    LI    LO    TS
CP0441475  Compound Info	1-(5-(2,4-dichlorophenyl)furan-2-yl)-2-(phenylsulfonyl)ethanone    Show/Hide	C18H12Cl2O4S	1
1	IC50 = 169 nM  Bioactivity Info	TI    LI    LO    TS
CP0051751  Compound Info	2-(S)-Phenethylamine analog 5    Show/Hide	C16H19F3N2OS	1
1	IC50 = 170 nM  Bioactivity Info	TI    LI    LO    TS
CP0508674  Compound Info	4-{[3-(3,4-Dichloro-benzenesulfonyl)-thiazolidine-2-carbonyl]-amino}-adamantane-1-carboxylic acid methyl ester    Show/Hide	C22H26Cl2N2O5S2	1
1	IC50 = 170 nM  Bioactivity Info	TI    LI    LO    TS
CP0506371  Compound Info	2-[(S)-1-(3-Fluorophenyl)ethylamino]-5-(2-hydroxypropan-2-yl)-5-methylthiazol-4(5H)-one    Show/Hide	C15H19FN2O2S	1
1	IC50 = 180 nM  Bioactivity Info	TI    LI    LO    TS
CP0050141  Compound Info	2-(phenylsulfonyl)-1-(4-(trifluoromethyl)phenyl)ethanone    Show/Hide	C15H11F3O3S	2
1	IC50 = 187 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 190 nM  Bioactivity Info	TI    LI    LO    TS
CP0471998  Compound Info	(2R)-4-[4-Fluoro-2-(trifluoromethyl)phenyl]-2-methyl-1-[(4-piperidin-1-ylphenyl)sulfonyl]piperazine    Show/Hide	C23H27F4N3O2S	1
1	IC50 = 190 nM  Bioactivity Info	TI    LI    LO    TS
CP0837725  Compound Info	5-isopropyl-2-(isoquinolin-5-ylamino)thiazol-4(5H)-one    Show/Hide	C15H15N3OS	1
1	IC50 = 200 nM  Bioactivity Info	TI    LI    LO    TS
CP0501261  Compound Info	1-(4-chlorophenyl)-2-(phenylsulfonyl)ethanone    Show/Hide	C14H11ClO3S	1
1	IC50 = 200 nM  Bioactivity Info	TI    LI    LO    TS
CP0439668  Compound Info	(2R)-4-(4-Fluoro-2-(trifluoromethyl)phenyl)-2-methyl-1-(4-(trifluoromethoxy)-phenylsulfonyl)-piperazine    Show/Hide	C19H17F7N2O3S	1
1	IC50 = 200 nM  Bioactivity Info	TI    LI    LO    TS
CP0531000  Compound Info	3-(4-chlorophenyl)-6-methyl-6-phenyl-1,3-oxazinan-2-one    Show/Hide	C17H16ClNO2	1
1	IC50 = 229 nM  Bioactivity Info	TI    LI    LO    TS
CP0830643  Compound Info	2-(4-fluorophenylamino)-5-isopropylthiazol-4(5H)-one    Show/Hide	C12H13FN2OS	1
1	IC50 = 230 nM  Bioactivity Info	TI    LI    LO    TS
CP0526205  Compound Info	(5S)-2-[[(1S,2S,4R,6R)-6-hydroxy-2-bicyclo[2.2.1]heptanyl]imino]-5-methyl-5-propan-2-yl-1,3-thiazolidin-4-one    Show/Hide	C14H22N2O2S	1
1	IC50 = 237 nM  Bioactivity Info	TI    LI    LO    TS
CP0284959  Compound Info	2-Benzylamine analog 4    Show/Hide	C15H20N2OS	1
1	IC50 = 268 nM  Bioactivity Info	TI    LI    LO    TS
CP0504570  Compound Info	(R)-3-tert-Butoxycarbonylamino-pyrrolidine-1-carboxylic acid 5-methoxycarbonyl-adamantan-2-yl ester    Show/Hide	C22H34N2O6	1
1	IC50 = 289 nM  Bioactivity Info	TI    LI    LO    TS
CP0522190  Compound Info	(R)-2-[(S)-1-(4-Fluorophenyl)ethylamino]-5-(2-hydroxypropan-2-yl)-5-methylthiazol-4(5H)-one    Show/Hide	C15H19FN2O2S	1
1	IC50 = 300 nM  Bioactivity Info	TI    LI    LO    TS
CP0138630  Compound Info	2-[3-({(2R)-4-[4-fluoro-2-(trifluoromethyl)phenyl]-2-methylpiperazin-1-yl}sulfonyl)phenoxy]-2-methylpropanoic acid    Show/Hide	C22H24F4N2O5S	1
1	IC50 = 300 nM  Bioactivity Info	TI    LI    LO    TS
CP0803238  Compound Info	5-isopropyl-2-(phenylamino)thiazol-4(5H)-one    Show/Hide	C12H14N2OS	1
1	IC50 = 310 nM  Bioactivity Info	TI    LI    LO    TS
CP0535208  Compound Info	2-[(S)-1-(4-Fluorophenyl)ethylamino]-5-(2-hydroxy-2-methylpropyl)-5-methylthiazol-4(5H)-one    Show/Hide	C16H21FN2O2S	1
1	IC50 = 310 nM  Bioactivity Info	TI    LI    LO    TS
CP0166537  Compound Info	methyl 4-[3-[(2R)-4-[4-fluoro-2-(trifluoromethyl)phenyl]-2-methylpiperazin-1-yl]sulfonylphenyl]piperazine-1-carboxylate    Show/Hide	C24H28F4N4O4S	1
1	IC50 = 330 nM  Bioactivity Info	TI    LI    LO    TS
CP0457467  Compound Info	2-(phenylsulfonyl)-1-(thiophen-3-yl)ethanone    Show/Hide	C12H10O3S2	1
1	IC50 = 345 nM  Bioactivity Info	TI    LI    LO    TS
CP0502502  Compound Info	(6S)-3-(3-methylphenyl)-6-phenyl-1,3-oxazinan-2-one    Show/Hide	C17H17NO2	1
1	IC50 = 353 nM  Bioactivity Info	TI    LI    LO    TS
CP0783486  Compound Info	2-(1H-indol-4-ylamino)-5-isopropylthiazol-4(5H)-one    Show/Hide	C14H15N3OS	1
1	IC50 = 360 nM  Bioactivity Info	TI    LI    LO    TS
CP0236340  Compound Info	N-ethyl-4-[3-[(2R)-4-[4-fluoro-2-(trifluoromethyl)phenyl]-2-methylpiperazin-1-yl]sulfonylphenyl]piperazine-1-carboxamide    Show/Hide	C25H31F4N5O3S	1
1	IC50 = 370 nM  Bioactivity Info	TI    LI    LO    TS
CP0166538  Compound Info	(2R)-4-[4-fluoro-2-(trifluoromethyl)phenyl]-1-{[3-(4-isopropylpiperazin-1-yl)phenyl]sulfonyl}-2-methylpiperazine    Show/Hide	C25H32F4N4O2S	1
1	IC50 = 490 nM  Bioactivity Info	TI    LI    LO    TS
CP0423433  Compound Info	1-[(3,4-dichlorophenyl)sulfonyl]-4-[3-(trifluoromethyl)pyridin-2-yl]piperazin-2-one    Show/Hide	C16H12Cl2F3N3O3S	1
1	IC50 = 500 nM  Bioactivity Info	TI    LI    LO    TS
CP0062733  Compound Info	3beta-O-Succinyl-18-beta-glycyrrhetinic acid    Show/Hide	C34H50O7	1
1	IC50 = 500 nM  Bioactivity Info	TI    LI    LO    TS
CP0538620  Compound Info	1-(3-methylbenzo[b]thiophen-2-yl)-2-(phenylsulfonyl)ethanone    Show/Hide	C17H14O3S2	1
1	IC50 = 525 nM  Bioactivity Info	TI    LI    LO    TS
CP0511682  Compound Info	2-(Adamantan-2-ylcarbamoyl)-thiazolidine-3-carboxylic acid tert-butyl ester    Show/Hide	C19H30N2O3S	1
1	IC50 = 554 nM  Bioactivity Info	TI    LI    LO    TS
CP0455268  Compound Info	(2R)-4-(4-(4-Fluoro-2-(trifluoromethyl)phenyl)-2-methylpiperazin-1-ylsulfonyl)benzamide    Show/Hide	C19H19F4N3O3S	1
1	IC50 = 630 nM  Bioactivity Info	TI    LI    LO    TS
CP0396753  Compound Info	3-[(4-bromophenyl)methyl]-6-methyl-6-phenyl-1,3-oxazinan-2-one    Show/Hide	C18H18BrNO2	1
1	IC50 = 631 nM  Bioactivity Info	TI    LI    LO    TS
CP0492245  Compound Info	(2R)-1-({2-Chloro-4-[(3S)-3-methylpiperazin-1-yl]phenyl}sulfonyl)-4-[4-fluoro-2-(trifluoromethyl)phenyl]-2-methylpiperazine    Show/Hide	C23H27ClF4N4O2S	1
1	IC50 = 639 nM  Bioactivity Info	TI    LI    LO    TS
CP0427271  Compound Info	(2R)-4-[4-Fluoro-2-(trifluoromethyl)phenyl]-2-methyl-1-{[4-(1Htetrazol-5-yl)phenyl]sulfonyl}piperazine    Show/Hide	C19H18F4N6O2S	1
1	IC50 = 674 nM  Bioactivity Info	TI    LI    LO    TS
CP0393207  Compound Info	3-(4-{2-[(S)-1-(4-Fluorophenyl)ethylamino]-5-methyl-4-oxo-4,5-dihydrothiazol-5-yl}phenyl)propanamide    Show/Hide	C21H22FN3O2S	1
1	IC50 = 680 nM  Bioactivity Info	TI    LI    LO    TS
CP0504022  Compound Info	3-(3,4-Dichloro-benzenesulfonyl)-thiazolidine-2-carboxylic acid(5-hydroxy-adamantan-2-yl)-amide    Show/Hide	C20H24Cl2N2O4S2	1
1	IC50 = 683 nM  Bioactivity Info	TI    LI    LO    TS
CP0396751  Compound Info	6-methyl-6-phenyl-3-[4-(trifluoromethyl)phenyl]-1,3-oxazinan-2-one    Show/Hide	C18H16F3NO2	1
1	IC50 = 805 nM  Bioactivity Info	TI    LI    LO    TS
CP0398796  Compound Info	2-N-(2-adamantyl)-3-N-phenyl-1,3-thiazolidine-2,3-dicarboxamide    Show/Hide	C21H27N3O2S	1
1	IC50 = 945 nM  Bioactivity Info	TI    LI    LO    TS
CP0396750  Compound Info	(6R)-3-(3-methylphenyl)-6-phenyl-1,3-oxazinan-2-one    Show/Hide	C17H17NO2	1
1	IC50 = 999 nM  Bioactivity Info	TI    LI    LO    TS
CP0538621  Compound Info	1-(3,5-dimethylphenyl)-2-(phenylsulfonyl)ethanone    Show/Hide	C16H16O3S	1
1	IC50 = 1200 nM  Bioactivity Info	TI    LI    LO    TS
CP0372432  Compound Info	(2R,6S)-4-(3-chloropyridin-2-yl)-1-(3,4-dichlorophenyl)sulfonyl-2,6-dimethylpiperazine    Show/Hide	C17H18Cl3N3O2S	1
1	IC50 = 1300 nM  Bioactivity Info	TI    LI    LO    TS
CP0501262  Compound Info	1-(4-nitrophenyl)-2-(phenylsulfonyl)ethanone    Show/Hide	C14H11NO5S	1
1	IC50 = 1310 nM  Bioactivity Info	TI    LI    LO    TS
CP0881783  Compound Info	5-isopropyl-2-(pyridin-2-ylamino)thiazol-4(5H)-one    Show/Hide	C11H13N3OS	1
1	IC50 = 1400 nM  Bioactivity Info	TI    LI    LO    TS
CP0739806  Compound Info	5-isopropyl-2-(2-methoxyphenylamino)thiazol-4(5H)-one    Show/Hide	C13H16N2O2S	1
1	IC50 = 1500 nM  Bioactivity Info	TI    LI    LO    TS
CP0841219  Compound Info	2-(1H-indazol-5-ylamino)-5-isopropylthiazol-4(5H)-one    Show/Hide	C13H14N4OS	1
1	IC50 = 1500 nM  Bioactivity Info	TI    LI    LO    TS
CP0036916  Compound Info	2-(2-(3-chloro-2-methylphenylsulfonamido)thiazol-4-yl)-N,N-diethylacetamide    Show/Hide	C16H20ClN3O3S2	1
1	IC50 = 1500 nM  Bioactivity Info	TI    LI    LO    TS
CP0372439  Compound Info	(2S,5R)-1-(3-chloropyridin-2-yl)-4-(3,4-dichlorophenyl)sulfonyl-2,5-dimethylpiperazine    Show/Hide	C17H18Cl3N3O2S	1
1	IC50 = 1600 nM  Bioactivity Info	TI    LI    LO    TS
CP0848231  Compound Info	Thiazolidine-2-carboxylic acid adamantan-2-ylamide hydrochloride    Show/Hide	C14H23ClN2OS	1
1	IC50 = 2130 nM  Bioactivity Info	TI    LI    LO    TS
CP0464514  Compound Info	1,1-diphenyl-3-(phenylsulfonyl)propan-2-one    Show/Hide	C21H18O3S	1
1	IC50 = 2900 nM  Bioactivity Info	TI    LI    LO    TS
CP0739804  Compound Info	2-(4-cyclohexylphenylamino)-5-isopropylthiazol-4(5H)-one    Show/Hide	C18H24N2OS	1
1	IC50 = 3300 nM  Bioactivity Info	TI    LI    LO    TS
CP0441479  Compound Info	1-(4-(diethylamino)phenyl)-2-(phenylsulfonyl)ethanone    Show/Hide	C18H21NO3S	1
1	IC50 = 4400 nM  Bioactivity Info	TI    LI    LO    TS
CP0461728  Compound Info	ethyl 5-(benzenesulfonyl)-3,3-dimethyl-4-oxopentanoate    Show/Hide	C15H20O5S	1
1	IC50 = 5000 nM  Bioactivity Info	TI    LI    LO    TS
CP0530862  Compound Info	N-(benzenesulfonyl)-N-benzylbenzamide    Show/Hide	C20H17NO3S	1
1	IC50 = 5700 nM  Bioactivity Info	TI    LI    LO    TS
CP0399402  Compound Info	1-(2,5-dimethoxyphenyl)-2-(phenylsulfonyl)ethanone    Show/Hide	C16H16O5S	1
1	IC50 = 9300 nM  Bioactivity Info	TI    LI    LO    TS
CP0463476  Compound Info	4-(3,4-dichloro-benzenesulfonyl)-1-(3-trifluoromethyl-pyridin-2-yl)-piperazin-2-one    Show/Hide	C16H12Cl2F3N3O3S	1
1	IC50 = 9900 nM  Bioactivity Info	TI    LI    LO    TS
CP0138701  Compound Info	(2R)-4-[4-fluoro-2-(trifluoromethyl)phenyl]-2-methyl-1-[(3-piperazin-1-ylphenyl)sulfonyl]piperazine    Show/Hide	C22H26F4N4O2S	1
1	IC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0520177  Compound Info	1-(phenylsulfonyl)butan-2-one    Show/Hide	C10H12O3S	1
1	IC50 = 15000 nM  Bioactivity Info	TI    LI    LO    TS
CP0501263  Compound Info	1-phenyl-3-(phenylsulfonyl)propan-1-one    Show/Hide	C15H14O3S	1
1	IC50 = 17400 nM  Bioactivity Info	TI    LI    LO    TS
CP0490320  Compound Info	1-(4-fluorophenyl)-3-(phenylsulfonyl)propan-1-one    Show/Hide	C15H13FO3S	1
1	IC50 = 19600 nM  Bioactivity Info	TI    LI    LO    TS
CP0399404  Compound Info	1-(4-chlorophenyl)-3-(phenylsulfonyl)propan-1-one    Show/Hide	C15H13ClO3S	1
1	IC50 = 24000 nM  Bioactivity Info	TI    LI    LO    TS
CP0501264  Compound Info	1-(4-bromophenyl)-3-(phenylsulfonyl)propan-1-one    Show/Hide	C15H13BrO3S	1
1	IC50 = 25000 nM  Bioactivity Info	TI    LI    LO    TS
CP0485316  Compound Info	N-(benzenesulfonyl)-N-methylbenzamide    Show/Hide	C14H13NO3S	1
1	IC50 = 35500 nM  Bioactivity Info	TI    LI    LO    TS
CP0441477  Compound Info	3,3-dimethyl-1-(phenylsulfonyl)butan-2-one    Show/Hide	C12H16O3S	1
1	IC50 = 90000 nM  Bioactivity Info	TI    LI    LO    TS
CP0211666  Compound Info	N-(benzenesulfonyl)benzamide    Show/Hide	C13H11NO3S	1
1	IC50 > 100000 nM  Bioactivity Info	TI    LI    LO    TS
CP0441182  Compound Info	2-(phenylsulfonyl)-1-(4-(trifluoromethyl)phenyl)ethanol    Show/Hide	C15H13F3O3S	1
1	IC50 = 100000 nM  Bioactivity Info	TI    LI    LO    TS
CP0457468  Compound Info	3-chloro-N-(phenylsulfonyl)benzamide    Show/Hide	C13H10ClNO3S	1
1	IC50 > 100000 nM  Bioactivity Info	TI    LI    LO    TS
CP0461731  Compound Info	N-(4-methylphenyl)sulfonylbenzamide    Show/Hide	C14H13NO3S	1
1	IC50 > 100000 nM  Bioactivity Info	TI    LI    LO    TS
CP0461732  Compound Info	N-(4-chlorophenyl)sulfonylbenzamide    Show/Hide	C13H10ClNO3S	1
1	IC50 > 100000 nM  Bioactivity Info	TI    LI    LO    TS
CP0510061  Compound Info	N-(benzenesulfonyl)-4-(trifluoromethyl)benzamide    Show/Hide	C14H10F3NO3S	1
1	IC50 > 100000 nM  Bioactivity Info	TI    LI    LO    TS
CP0501653  Compound Info	(6R)-3-[(1R)-1-[4-(2,4-difluorophenyl)phenyl]ethyl]-6-(4-fluorophenyl)-6-(2-hydroxyethyl)-1,3-oxazinan-2-one    Show/Hide	C26H24F3NO3	1
1	IC50 > 100 nM  Bioactivity Info	TI    LI    LO    TS
CP0501654  Compound Info	(6R)-3-[(1S)-1-[4-(2,4-difluorophenyl)phenyl]ethyl]-6-(4-fluorophenyl)-6-(2-hydroxyethyl)-1,3-oxazinan-2-one    Show/Hide	C26H24F3NO3	1
1	IC50 > 100 nM  Bioactivity Info	TI    LI    LO    TS
CP0450217  Compound Info	US8927539, 7    Show/Hide	C29H32N2O4	1
1	IC50 > 100 nM  Bioactivity Info	TI    LI    LO    TS

Compound ID	Compound Name	Compound Formula
CP0002778  Compound Info	4-[(4-methylpiperazin-1-yl)methyl]-N-[4-methyl-3-[(4-pyridin-3-ylpyrimidin-2-yl)amino]phenyl]benzamide    Show/Hide	C29H31N7O	1
1	GI50 > 10000 nM	TI    LI    LO    TS
CP0031719  Compound Info	(R)-3-(1-(2,6-dichloro-3-fluorophenyl)ethoxy)-5-(1-(piperidin-4-yl)-1H-pyrazol-4-yl)pyridin-2-amine    Show/Hide	C21H22Cl2FN5O	1
1	GI50 = 3200 nM	TI    LI    LO    TS
CP0036865  Compound Info	Atripla    Show/Hide	C9H14N5O4P	1
1	CC50 = 435000 nM	TI    LI    LO    TS
CP0059062  Compound Info	N-[3-[5-chloro-2-[2-methoxy-4-(4-methylpiperazin-1-yl)anilino]pyrimidin-4-yl]oxyphenyl]prop-2-enamide    Show/Hide	C25H27ClN6O3	1
1	GI50 = 3900 nM	TI    LI    LO    TS
CP0175008  Compound Info	2-amino-1-[3-(4-fluoroanilino)-2-(4-fluorophenyl)-8,8-dimethyl-5,6-dihydroimidazo[1,2-a]pyrazin-7-yl]ethanone    Show/Hide	C22H23F2N5O	1
1	CC50 > 12000 nM	TI    LI    LO    TS
CP0224766  Compound Info	4-(methylamino)-2-[4-methyl-3-(prop-2-enoylamino)anilino]-N-[2-methyl-5-[(3,4,5-trimethoxybenzoyl)amino]phenyl]pyrimidine-5-carboxamide    Show/Hide	C33H35N7O6	1
1	GI50 > 10000 nM	TI    LI    LO    TS
CP0225649  Compound Info	2-amino-1-[3-(4-fluoroanilino)-2-(4-fluorophenyl)-6,8-dihydro-5H-imidazo[1,2-a]pyrazin-7-yl]-2-methylpropan-1-one    Show/Hide	C22H23F2N5O	1
1	TC50 > 12000 nM	TI    LI    LO    TS
CP0377875  Compound Info	[(2R,5R)-5-(6-aminopurin-9-yl)-4-fluoro-2,5-dihydrofuran-2-yl]oxymethylphosphonic acid    Show/Hide	C10H11FN5O5P	1
1	CC50 >= 95000 nM	TI    LI    LO    TS
CP0398356  Compound Info	2-(2-chloro-6-fluorophenyl)-5-(6-methoxy-4-methylpyridin-3-yl)-1H-pyrrolo[2,3-b]pyridine    Show/Hide	C20H15ClFN3O	1
1	IC50 > 100000 nM	TI    LI    LO    TS
CP0426396  Compound Info	BDBM50246180    Show/Hide	C20H23N5O2	1
1	IC50 > 2000000 nM	TI    LI    LO    TS
CP0440597  Compound Info	7,8-dichloro-1-[(3-fluorophenyl)methylamino]-3-(trifluoromethyl)pyrido[1,2-a]benzimidazole-4-carbonitrile    Show/Hide	C20H10Cl2F4N4	1
1	IC50 = 7030 nM	TI    LI    LO    TS
CP0523655  Compound Info	2-(2-chloro-6-fluorophenyl)-5-(4,6-dimethoxypyridin-3-yl)-1H-pyrrolo[2,3-b]pyridine    Show/Hide	C20H15ClFN3O2	1
1	IC50 > 100000 nM	TI    LI    LO    TS
CP0569231  Compound Info	N-benzyl-3-[(8-pyridin-4-yl-1,5-naphthyridin-2-yl)amino]benzenesulfonamide    Show/Hide	C26H21N5O2S	1
1	IC50 > 50000 nM	TI    LI    LO    TS
CP0575677  Compound Info	N-(2-hydroxyethyl)-3-[(8-pyridin-4-yl-1,5-naphthyridin-2-yl)amino]benzenesulfonamide    Show/Hide	C21H19N5O3S	1
1	IC50 = 4000 nM	TI    LI    LO    TS
CP0857303  Compound Info	(R)-1-(3-(4-Amino-3-(3-chloro-4-(pyridin-2-ylmethoxy)phenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl)piperidin-1-yl)propan-1-one    Show/Hide	C25H26ClN7O2	1
1	GI50 > 10000 nM	TI    LI    LO    TS
CP0909620  Compound Info	3-(4-(methylsulfinyl)phenyl)-N-(3-(methylsulfonyl)phenyl)imidazo[1,2-b]pyridazin-6-amine    Show/Hide	C20H18N4O3S2	1
1	IC50 = 123000 nM	TI    LI    LO    TS
CP0946923  Compound Info	4-((3-(4-(Methylsulfinyl)phenyl)imidazo[1,2-b]pyridazin-6-yl)amino)tetrahydro-2Hthiopyran-1,1-dioxide    Show/Hide	C18H20N4O3S2	1
1	IC50 > 247000 nM	TI    LI    LO    TS
CP0949178  Compound Info	3-(4-(methylsulfinyl)phenyl)-N-(pyrazin-2-yl)imidazo[1,2-b]pyridazin-6-amine    Show/Hide	C17H14N6OS	1
1	IC50 = 277000 nM	TI    LI    LO    TS