General Information of the Protein
Protein ID
PT02988
Protein Name
Prostaglandin E2 receptor EP1 subtype
Secondarily
Protein Name
Prostanoid EP1 receptor
Gene Name
PTGER1
Secondarily
Gene Name
Ptgerep1
Sequence
MSPCGLNLSLADEAATCATPRLPNTSVVLPTGDNGTSPALPIFSMTLGAVSNVLALALLAQVAGRMRRRRSAATFLLFVASLLAIDLAGHVIPGALVLRLYTAGRAPAGGACHFLGGCMVFFGLCPLLLGCGMAVERCVGVTQPLIHAARVSVARARLALAVLAAMALAVALLPLVHVGRYELQYPGTWCFISLGPRGGWRQALLAGLFAGLGLAALLAALVCNTLSGLALLRARWRRRRSRRFRKTAGPDDRRRWGSRGPRLASASSASSITSATATLRSSRGGGSARRVHAHDVEMVGQLVGIMVVSCICWSPLLVLVVLAIGGWNSNSLQRPLFLAVRLASWNQILDPWVYILLRQAMLRQLLRLLPLRVSAKGGPTELGLTKSAWEASSLRSSRHSGFSHL
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Organism
Mus musculus, Mouse
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
>
Small molecule receptor (family A GPCR)
>
Lipid-like ligand receptor (family A GPCR)
>
Prostanoid receptor
Function
Receptor for prostaglandin E2 (PGE2). The activity of this receptor is mediated by G(q) proteins which activate a phosphatidylinositol-calcium second messenger system. May play a role as an important modulator of renal function. Implicated the smooth muscle contractile response to PGE2 in various tissues.
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Uniprot ID
P35375
Subcellular Location
Cell membrane
Map of Molecular Bioactivity Related to the Protein
Map of Molecular Bioactivity Related to the Protein

Protein
Cell Line
Compound

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Protein
Cell Line ID: CL000011 , CHO
 Cell Line Info 
Compound ID Compound Name Compound Formula
CP0055947
 Compound Info 
(15S)-prostaglandin E2
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C20H32O5
  1
1
Ki = 6 nM
 Bioactivity Info 
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CP0377772
 Compound Info 
6-[(1R,2S,3R)-3-Hydroxy-2-((E)-(3S,5S)-3-hydroxy-5-methyl-non-1-enyl)-5-oxo-cyclopentylsulfanyl]-hexanoic acid
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C21H36O5S
  1
1
Ki = 11 nM
 Bioactivity Info 
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CP0403791
 Compound Info 
(Z)-7-[(1R,2R,3R)-3-Hydroxy-2-((E)-(R)-3-hydroxy-oct-1-enyl)-5-oxo-cyclopentyl]-hept-5-enoic acid
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C20H32O5
  1
1
Ki = 18 nM
 Bioactivity Info 
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CP0062070
 Compound Info 
(11alpha,13E,15S)-11,15-dihydroxy-9-oxoprost-13-en-1-oic acid
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C20H34O5
  2
1
Ki = 22 nM
 Bioactivity Info 
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2
Ki = 100 nM
 Bioactivity Info 
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CP0406251
 Compound Info 
3-{(S)-3-[(R)-3-Hydroxy-2-((1R,2R)-3-hydroxy-oct-1-enyl)-5-oxo-cyclopentyl]-propylsulfanyl}-propionic acid
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C19H32O5S
  1
1
Ki = 27 nM
 Bioactivity Info 
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CP0381675
 Compound Info 
2-[2-[[(1R,2R,3R)-3-hydroxy-2-[(E,3S)-3-hydroxyoct-1-enyl]-5-oxocyclopentyl]methylsulfanyl]ethylsulfanyl]acetic acid
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C18H30O5S2
  1
1
Ki = 50 nM
 Bioactivity Info 
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CP0383420
 Compound Info 
4-{(S)-2-[(R)-3-Hydroxy-2-((1R,2R)-3-hydroxy-oct-1-enyl)-5-oxo-cyclopentyl]-ethylsulfanyl}-butyric acid
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C19H32O5S
  1
1
Ki = 52 nM
 Bioactivity Info 
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CP0404505
 Compound Info 
5-[(S)-(R)-3-Hydroxy-2-((1R,2R)-3-hydroxy-oct-1-enyl)-5-oxo-cyclopentylmethylsulfanyl]-pentanoic acid
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C19H32O5S
  1
1
Ki = 95 nM
 Bioactivity Info 
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CP0397271
 Compound Info 
6-[(S)-(R)-3-Hydroxy-2-((1S,2R)-3-hydroxy-oct-1-enyl)-5-oxo-cyclopentylsulfanyl]-hexanoic acid
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C19H32O5S
  1
1
Ki = 120 nM
 Bioactivity Info 
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CP0406253
 Compound Info 
2-[4-[(1R,2R,3R)-3-hydroxy-2-[(E,3S)-3-hydroxyoct-1-enyl]-5-oxocyclopentyl]butylsulfanyl]acetic acid
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C19H32O5S
  1
1
Ki = 200 nM
 Bioactivity Info 
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CP0378129
 Compound Info 
2-[2-[(2R)-2-[(E,3S)-3-hydroxy-4-[3-(6-methyl-1,3-benzoxazol-2-yl)phenyl]but-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]-1,3-thiazole-4-carboxylic acid
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C28H27N3O5S2
  1
1
Ki = 200 nM
 Bioactivity Info 
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CP0400279
 Compound Info 
3-(4-((1H-pyrazol-1-yl)methyl)-2-(2-(methyl(phenyl)amino)ethoxy)phenyl)-N-(3,4-difluorophenylsulfonyl)propanamide
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C28H28F2N4O4S
  1
1
Ki = 260 nM
 Bioactivity Info 
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CP0486399
 Compound Info 
2-[2-methyl-1-[4-(2-phenylethoxy)benzoyl]indol-4-yl]acetic acid
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C26H23NO4
  1
1
Ki = 400 nM
 Bioactivity Info 
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CP0430729
 Compound Info 
3-(4-((1H-pyrazol-1-yl)methyl)-2-(3-morpholinophenethoxy)phenyl)-N-(3,4-difluorophenylsulfonyl)propanamide
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C31H32F2N4O5S
  1
1
Ki = 560 nM
 Bioactivity Info 
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CP0403755
 Compound Info 
2-[3-[(1R,2S,3R)-3-hydroxy-2-[(E,3S)-3-hydroxyoct-1-enyl]-5-oxocyclopentyl]sulfanylpropylsulfanyl]acetic acid
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C18H30O5S2
  1
1
Ki = 610 nM
 Bioactivity Info 
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CP0458692
 Compound Info 
3-{2-[(S)-(R)-3-Hydroxy-2-((1S,2R)-3-hydroxy-oct-1-enyl)-5-oxo-cyclopentylsulfanyl]-ethylsulfanyl}-propionic acid
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C18H30O5S2
  1
1
Ki = 610 nM
 Bioactivity Info 
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CP0410311
 Compound Info 
2-[2-[(2R)-2-[(E,3S)-4-[3-(5-chloro-1,3-benzoxazol-2-yl)phenyl]-3-hydroxybut-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]-1,3-thiazole-4-carboxylic acid
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C27H24ClN3O5S2
  1
1
Ki = 650 nM
 Bioactivity Info 
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CP0410235
 Compound Info 
2-[2-[(2R)-2-[(E,3S)-4-[3-(5-chloro-1,3-benzothiazol-2-yl)phenyl]-3-hydroxybut-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]-1,3-thiazole-4-carboxylic acid
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C27H24ClN3O4S3
  1
1
Ki = 680 nM
 Bioactivity Info 
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CP0383212
 Compound Info 
(Z)-7-{(1R,2R,3R)-2-[(E)-(S)-4-(1-Butyl-cyclobutyl)-4-hydroxy-but-1-enyl]-3-hydroxy-5-oxo-cyclopentyl}-hept-5-enoic acid
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C24H38O5
  1
1
Ki = 780 nM
 Bioactivity Info 
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CP0486387
 Compound Info 
2-[1-[4-(1,3-benzodioxol-2-ylmethoxy)benzoyl]-2-methylindol-4-yl]acetic acid
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C26H21NO6
  1
1
Ki = 780 nM
 Bioactivity Info 
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CP0402069
 Compound Info 
(E)-7-{(1R,2R,3R,5R)-5-Chloro-3-hydroxy-2-[(E)-(S)-3-hydroxy-4-(3-methoxymethyl-phenyl)-but-1-enyl]-cyclopentyl}-hept-5-enoic acid
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C24H33ClO5
  1
1
Ki = 980 nM
 Bioactivity Info 
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CP0418822
 Compound Info 
2-[3-[(1R,2S,3R)-3-hydroxy-2-[(E,3S)-3-hydroxyoct-1-enyl]-5-oxocyclopentyl]sulfanylpropoxy]acetic acid
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C18H30O6S
  1
1
Ki = 1200 nM
 Bioactivity Info 
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CP0442227
 Compound Info 
2-[2-methyl-1-(4-phenylmethoxybenzoyl)indol-4-yl]acetic acid
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C25H21NO4
  1
1
Ki = 1200 nM
 Bioactivity Info 
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CP0401105
 Compound Info 
4-[2-[(4S)-4-[(E,3S)-4-(3-fluorophenyl)-3-hydroxybut-1-enyl]-2-oxo-1,3-oxazolidin-3-yl]ethylsulfanyl]butanoic acid
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C19H24FNO5S
  1
1
Ki = 1200 nM
 Bioactivity Info 
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CP0504299
 Compound Info 
3-(4-((1H-pyrazol-1-yl)methyl)-2-phenethoxyphenyl)-N-(3,4-difluorophenylsulfonyl)propanamide
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C27H25F2N3O4S
  1
1
Ki = 1300 nM
 Bioactivity Info 
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CP0375591
 Compound Info 
2-[3-[ethyl-[4-[[(2S)-4-methyl-2,3-dihydro-1,4-benzoxazin-2-yl]methoxy]benzoyl]amino]phenyl]acetic acid
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C27H28N2O5
  1
1
Ki = 1300 nM
 Bioactivity Info 
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CP0410240
 Compound Info 
2-[2-[(2R)-2-[(E,3S)-3-hydroxy-4-[3-(5-methyl-1,3-benzoxazol-2-yl)phenyl]but-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]-1,3-thiazole-4-carboxylic acid
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C28H27N3O5S2
  1
1
Ki = 1300 nM
 Bioactivity Info 
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CP0398224
 Compound Info 
(Z)-7-{(1R,2R,3R)-3-Hydroxy-2-[(E)-(S)-4-hydroxy-4-(1-pentyl-cyclobutyl)-but-1-enyl]-5-oxo-cyclopentyl}-hept-5-enoic acid
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C25H40O5
  1
1
Ki = 1600 nM
 Bioactivity Info 
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CP0415386
 Compound Info 
(E)-7-{(1R,2R,3R,5R)-5-Fluoro-3-hydroxy-2-[(E)-(S)-3-hydroxy-4-(3-methoxymethyl-phenyl)-but-1-enyl]-cyclopentyl}-hept-5-enoic acid
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C24H33FO5
  1
1
Ki = 1700 nM
 Bioactivity Info 
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CP0459036
 Compound Info 
N-(3,4-difluorophenyl)sulfonyl-3-[2-(2-naphthalen-2-ylethoxy)-4-(pyridin-3-yloxymethyl)phenyl]propanamide
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C33H28F2N2O5S
  1
1
Ki = 1700 nM
 Bioactivity Info 
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CP0474029
 Compound Info 
2-[2-[(2R)-2-[(E,3S)-3-hydroxy-4-[3-(2,2,2-trifluoroethoxymethyl)phenyl]but-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]-1,3-thiazole-4-carboxylic acid
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C23H25F3N2O5S2
  1
1
Ki = 1900 nM
 Bioactivity Info 
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CP0439527
 Compound Info 
2-[1-[4-[[(3R)-2,3-dihydro-1,4-benzodioxin-3-yl]methoxy]benzoyl]-2-methylindol-4-yl]acetic acid
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C27H23NO6
  1
1
Ki = 2000 nM
 Bioactivity Info 
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CP0447742
 Compound Info 
3-(4-((1H-pyrazol-1-yl)methyl)-2-(2-(naphthalen-2-yl)ethoxy)phenyl)-N-(3,4-difluorophenylsulfonyl)propanamide
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C31H27F2N3O4S
  1
1
Ki = 2100 nM
 Bioactivity Info 
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CP0424870
 Compound Info 
2-[3-[[4-[[(2S)-4-methyl-2,3-dihydro-1,4-benzoxazin-2-yl]methoxy]benzoyl]amino]phenyl]acetic acid
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C25H24N2O5
  1
1
Ki = 2100 nM
 Bioactivity Info 
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CP0442380
 Compound Info 
2-[1-[4-[[(3S)-2,3-dihydro-1,4-benzodioxin-3-yl]methoxy]benzoyl]-2-methylindol-4-yl]acetic acid
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C27H23NO6
  1
1
Ki = 2300 nM
 Bioactivity Info 
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CP0400837
 Compound Info 
4-[2-[(4S)-4-[(E,3S)-4-(3-ethylphenyl)-3-hydroxybut-1-enyl]-2-oxo-1,3-oxazolidin-3-yl]ethylsulfanyl]butanoic acid
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C21H29NO5S
  1
1
Ki = 2400 nM
 Bioactivity Info 
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CP0410313
 Compound Info 
2-[2-[(2R)-2-[(E,3S)-4-[3-(2,4-dimethylphenyl)phenyl]-3-hydroxybut-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]-1,3-thiazole-4-carboxylic acid
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C28H30N2O4S2
  1
1
Ki = 2400 nM
 Bioactivity Info 
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CP0410239
 Compound Info 
2-[2-[(2R)-2-[(E,3S)-4-[3-(3,4-dimethylphenyl)phenyl]-3-hydroxybut-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]-1,3-thiazole-4-carboxylic acid
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C28H30N2O4S2
  1
1
Ki = 2500 nM
 Bioactivity Info 
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CP0381808
 Compound Info 
2-[3-[(1R,2S,3R)-3-hydroxy-2-[(E,3S)-3-hydroxy-4-phenylbut-1-enyl]-5-oxocyclopentyl]sulfanylpropylsulfanyl]acetic acid
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C20H26O5S2
  1
1
Ki = 2600 nM
 Bioactivity Info 
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CP0482040
 Compound Info 
2-[3-[[4-[[(2S)-4-methyl-2,3-dihydro-1,4-benzoxazin-2-yl]methoxy]phenyl]sulfonylamino]phenyl]acetic acid
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C24H24N2O6S
  1
1
Ki = 2700 nM
 Bioactivity Info 
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CP0423877
 Compound Info 
2-[2-[(2R)-2-[(E,3S)-4-[3-(1-benzofuran-2-yl)phenyl]-3-hydroxybut-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]-1,3-thiazole-4-carboxylic acid
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C28H26N2O5S2
  1
1
Ki = 2700 nM
 Bioactivity Info 
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CP0430637
 Compound Info 
3-(4-((1H-pyrazol-1-yl)methyl)-2-(2-phenoxyethoxy)phenyl)-N-(3,4-difluorophenylsulfonyl)propanamide
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C27H25F2N3O5S
  1
1
Ki = 2800 nM
 Bioactivity Info 
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CP0391384
 Compound Info 
4-[2-[(2R)-2-[(E,3S)-3-hydroxy-4-(3-methylphenyl)but-1-enyl]-5-sulfanylidenepyrrolidin-1-yl]ethylsulfanyl]butanoic acid
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C21H29NO3S2
  1
1
Ki = 2800 nM
 Bioactivity Info 
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CP0239876
 Compound Info 
acrylic acid derivative, 4
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C25H22N2O3
  1
1
Ki = 2900 nM
 Bioactivity Info 
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CP0425413
 Compound Info 
2-[2-methyl-1-[2-methyl-4-[[(2S)-4-methyl-2,3-dihydro-1,4-benzoxazin-2-yl]methoxy]benzoyl]indol-3-yl]acetic acid
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C29H28N2O5
  1
1
Ki = 2900 nM
 Bioactivity Info 
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CP0397228
 Compound Info 
(3-{(1R,2S,3R)-3-Hydroxy-2-[(E)-(S)-3-hydroxy-4-(4-methoxy-phenyl)-but-1-enyl]-5-oxo-cyclopentylsulfanyl}-propylsulfanyl)-acetic acid
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C21H28O6S2
  1
1
Ki = 3100 nM
 Bioactivity Info 
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CP0402233
 Compound Info 
(E)-7-{(1R,2R,3R,5R)-5-Chloro-3-hydroxy-2-[(E)-(S)-3-hydroxy-4-(4-hydroxy-3-methyl-phenyl)-but-1-enyl]-cyclopentyl}-hept-5-enoic acid
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C23H31ClO5
  1
1
Ki = 3100 nM
 Bioactivity Info 
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CP0410241
 Compound Info 
2-[2-[(2R)-2-[(E,3S)-4-[3-(5,7-dimethyl-1,3-benzoxazol-2-yl)phenyl]-3-hydroxybut-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]-1,3-thiazole-4-carboxylic acid
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C29H29N3O5S2
  1
1
Ki = 3200 nM
 Bioactivity Info 
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CP0059258
 Compound Info 
(Z)-7-{(1R,2R,3R,5R)-5-Chloro-2-[(E)-(S)-4-(1-ethyl-cyclobutyl)-4-hydroxy-but-1-enyl]-3-hydroxy-cyclopentyl}-hept-5-enoic acid
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C22H35ClO4
  1
1
Ki = 3400 nM
 Bioactivity Info 
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CP0431608
 Compound Info 
2-[2-[(2R)-2-[(E,3S)-3-hydroxyoct-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]-1,3-thiazole-4-carboxylic acid
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C18H26N2O4S2
  1
1
Ki = 3400 nM
 Bioactivity Info 
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CP0486394
 Compound Info 
2-[1-[4-(3,4-dihydro-2H-chromen-2-ylmethoxy)benzoyl]-2-methylindol-4-yl]acetic acid
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C28H25NO5
  1
1
Ki = 3800 nM
 Bioactivity Info 
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CP0463776
 Compound Info 
phenylbutanoic acid analogue, 20
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C26H26N2O3
  1
1
Ki = 4000 nM
 Bioactivity Info 
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CP0510260
 Compound Info 
3-{2-({[(1R)-1-(3,5-Dimethylphenyl)-3-methylbutyl]-amino}carbonyl)-4-[(2-methoxyphenoxy)methyl]phenyl}-propanoic acid
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C31H37NO5
  1
1
Ki = 4100 nM
 Bioactivity Info 
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CP0410233
 Compound Info 
2-[2-[(2R)-2-[(E,3S)-3-hydroxy-4-(3-phenylphenyl)but-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]-1,3-thiazole-4-carboxylic acid
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C26H26N2O4S2
  1
1
Ki = 4200 nM
 Bioactivity Info 
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CP0401812
 Compound Info 
3-[4-[(3-Chlorophenoxy)methyl]-2-({[(1R)-1-(3,5-dimethylphenyl)-3-methylbutyl]amino}carbonyl)phenyl]propanoicacid
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C30H34ClNO4
  1
1
Ki = 4400 nM
 Bioactivity Info 
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CP0407028
 Compound Info 
3-[4-[(2-Chlorophenoxy)methyl]-2-({[(1R)-1-(3,5-dimethylphenyl)-3-methylbutyl]amino}carbonyl)phenyl]propanoicacid
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C30H34ClNO4
  1
1
Ki = 4400 nM
 Bioactivity Info 
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CP0427503
 Compound Info 
4-[2-[(4S)-4-[(E,3S)-3-hydroxy-4-(3-methylphenyl)but-1-enyl]-2-oxo-1,3-oxazolidin-3-yl]ethylsulfanyl]butanoic acid
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C20H27NO5S
  1
1
Ki = 4400 nM
 Bioactivity Info 
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CP0401107
 Compound Info 
4-[2-[(4S)-4-[(E,3S)-4-(3-ethylphenyl)-3-hydroxybut-1-enyl]-2-oxo-1,3-thiazolidin-3-yl]ethylsulfanyl]butanoic acid
   Show/Hide
C21H29NO4S2
  1
1
Ki = 4600 nM
 Bioactivity Info 
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CP0390113
 Compound Info 
N-(3,4-difluorophenyl)sulfonyl-3-[4-(morpholin-4-ylmethyl)-2-(2-naphthalen-2-ylethoxy)phenyl]propanamide
   Show/Hide
C32H32F2N2O5S
  1
1
Ki = 5000 nM
 Bioactivity Info 
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CP0328974
 Compound Info 
3-[2-{[(1-Naphthylmethyl)amino]carbonyl}-4-(phenoxymethyl)phenyl]propanoic acid
   Show/Hide
C28H25NO4
  1
1
Ki = 5000 nM
 Bioactivity Info 
   TI
   LI
   LO
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CP0432929
 Compound Info 
4-[2-[(2R)-2-[(E,3S)-4-[3-(1,3-benzoxazol-2-yl)phenyl]-3-hydroxybut-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]butanoic acid
   Show/Hide
C27H30N2O5S
  1
1
Ki = 5000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0448394
 Compound Info 
(Z)-7-{(1R,2S,3R)-2-[(E)-(S)-4-(1-Ethyl-cyclobutyl)-4-hydroxy-but-1-enyl]-3-hydroxy-cyclopentyl}-hept-5-enoic acid
   Show/Hide
C22H36O4
  1
1
Ki = 5100 nM
 Bioactivity Info 
   TI
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   LO
   TS
CP0419026
 Compound Info 
2-[3-[2-[(2R)-2-[(E,3S)-4-(3-chlorophenyl)-3-hydroxybut-1-enyl]-5-oxopyrrolidin-1-yl]ethyl]phenyl]acetic acid
   Show/Hide
C24H26ClNO4
  1
1
Ki = 5100 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0376006
 Compound Info 
2-[2,5-dimethyl-1-[4-[[(2S)-4-methyl-2,3-dihydro-1,4-benzoxazin-2-yl]methoxy]benzoyl]indol-3-yl]acetic acid
   Show/Hide
C29H28N2O5
  1
1
Ki = 5200 nM
 Bioactivity Info 
   TI
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   LO
   TS
CP0376532
 Compound Info 
3-(4-((1H-pyrazol-1-yl)methyl)-2-(naphthalen-1-ylmethylaminooxy)phenyl)-N-(3,4-difluorophenylsulfonyl)propanamide
   Show/Hide
C30H26F2N4O4S
  1
1
Ki = 5300 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0492173
 Compound Info 
7-{(1R,2R,3R,5R)-5-Chloro-3-hydroxy-2-[(E)-(S)-3-hydroxy-4-(3-methoxymethyl-phenyl)-but-1-enyl]-cyclopentyl}-heptanoic acid
   Show/Hide
C24H35ClO5
  1
1
Ki = 5400 nM
 Bioactivity Info 
   TI
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   LO
   TS
CP0410234
 Compound Info 
2-[2-[(2R)-2-[(E,3S)-3-hydroxy-4-[3-(4-methoxyphenyl)phenyl]but-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]-1,3-thiazole-4-carboxylic acid
   Show/Hide
C27H28N2O5S2
  1
1
Ki = 5400 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0374553
 Compound Info 
2-[2-methyl-1-[4-(2-phenoxyethoxy)benzoyl]indol-4-yl]acetic acid
   Show/Hide
C26H23NO5
  1
1
Ki = 5600 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0378130
 Compound Info 
2-[2-[(2R)-2-[(E,3S)-3-hydroxy-4-[3-(4-methylphenyl)phenyl]but-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]-1,3-thiazole-4-carboxylic acid
   Show/Hide
C27H28N2O4S2
  1
1
Ki = 6100 nM
 Bioactivity Info 
   TI
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   LO
   TS
CP0400679
 Compound Info 
2-[2-methyl-1-[4-[[(2S)-4-methyl-2,3-dihydro-1,4-benzoxazin-2-yl]methoxy]benzoyl]indol-4-yl]acetic acid
   Show/Hide
C28H26N2O5
  1
1
Ki = 6200 nM
 Bioactivity Info 
   TI
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   LO
   TS
CP0410236
 Compound Info 
2-[2-[(2R)-2-[(E,3S)-4-[3-(4-chlorophenyl)phenyl]-3-hydroxybut-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]-1,3-thiazole-4-carboxylic acid
   Show/Hide
C26H25ClN2O4S2
  1
1
Ki = 6300 nM
 Bioactivity Info 
   TI
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   LO
   TS
CP0430839
 Compound Info 
acrylic acid derivative, 13
   Show/Hide
C26H25NO4
  1
1
Ki = 6400 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0380709
 Compound Info 
2-[4-chloro-3-[[2-chloro-4-[[(2S)-4-methyl-2,3-dihydro-1,4-benzoxazin-2-yl]methoxy]benzoyl]amino]phenyl]acetic acid
   Show/Hide
C25H22Cl2N2O5
  1
1
Ki = 6600 nM
 Bioactivity Info 
   TI
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   LO
   TS
CP0239946
 Compound Info 
phenylpropanoic acid analogue, 5
   Show/Hide
C25H24N2O3
  1
1
Ki = 7100 nM
 Bioactivity Info 
   TI
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   LO
   TS
CP0410238
 Compound Info 
4-[2-[(2R)-2-[(E,3S)-4-[3-(1,3-dihydroisoindol-2-yl)phenyl]-3-hydroxybut-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]butanoic acid
   Show/Hide
C28H34N2O4S
  1
1
Ki = 7100 nM
 Bioactivity Info 
   TI
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   LO
   TS
CP0445848
 Compound Info 
2-[2-methyl-1-[4-(3-phenylpropoxy)benzoyl]indol-4-yl]acetic acid
   Show/Hide
C27H25NO4
  1
1
Ki = 7700 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0410310
 Compound Info 
2-[2-[(2R)-2-[(E,3S)-3-hydroxy-4-[3-(4-methyl-1,3-benzoxazol-2-yl)phenyl]but-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]-1,3-thiazole-4-carboxylic acid
   Show/Hide
C28H27N3O5S2
  1
1
Ki = 7700 nM
 Bioactivity Info 
   TI
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   LO
   TS
CP0451828
 Compound Info 
2-[1-[4-(2,3-dihydro-1-benzofuran-2-ylmethoxy)benzoyl]-2-methylindol-4-yl]acetic acid
   Show/Hide
C27H23NO5
  1
1
Ki = 7800 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0410237
 Compound Info 
2-[2-[(2R)-2-[(E,3S)-4-[3-(1,3-benzothiazol-2-yl)phenyl]-3-hydroxybut-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]-1,3-thiazole-4-carboxylic acid
   Show/Hide
C27H25N3O4S3
  1
1
Ki = 8000 nM
 Bioactivity Info 
   TI
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   LO
   TS
CP0390811
 Compound Info 
3-[4-[(3-Cyanophenyl)amino]-2-({[(1R)-1-(3,5-dimethylphenyl)-3-methylbutyl]amino}carbonyl)phenyl]propanoic acid
   Show/Hide
C30H33N3O3
  1
1
Ki = 8700 nM
 Bioactivity Info 
   TI
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   LO
   TS
CP0374669
 Compound Info 
4-(2-{(1R,3R)-3-Hydroxy-2-[(E)-(S)-4-hydroxy-4-(1-propyl-cyclobutyl)-but-1-enyl]-5-oxo-cyclopentyl}-ethyl)-benzoic acid
   Show/Hide
C25H34O5
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0383213
 Compound Info 
(Z)-7-{(1R,2R,3R)-3-Hydroxy-2-[(E)-(S)-4-hydroxy-4-(1-isobutyl-cyclobutyl)-but-1-enyl]-5-oxo-cyclopentyl}-hept-5-enoic acid
   Show/Hide
C24H38O5
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0395500
 Compound Info 
(Z)-7-{(1R,2R,3R)-3-Hydroxy-2-[(E)-(S)-4-hydroxy-4-(1-propyl-cyclopentyl)-but-1-enyl]-5-oxo-cyclopentyl}-hept-5-enoic acid
   Show/Hide
C24H38O5
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0397704
 Compound Info 
7-{(1R,3R)-3-Hydroxy-2-[(E)-(S)-4-hydroxy-4-(1-propyl-cyclobutyl)-but-1-enyl]-5-oxo-cyclopentyl}-heptanoic acid methyl ester
   Show/Hide
C24H40O5
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0397705
 Compound Info 
(Z)-7-{(1R,2R,3R)-2-[(E)-(S)-4-(1-Ethyl-cyclobutyl)-4-hydroxy-but-1-enyl]-3-hydroxy-5-oxo-cyclopentyl}-hept-5-enoic acid
   Show/Hide
C22H34O5
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
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   LO
   TS
CP0403034
 Compound Info 
(E)-7-{(1R,3R)-3-Hydroxy-2-[(E)-(S)-4-hydroxy-4-(1-propyl-cyclobutyl)-but-1-enyl]-5-oxo-cyclopentyl}-hept-5-enoic acid
   Show/Hide
C23H36O5
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0403813
 Compound Info 
7-{(1R,3R)-3-Hydroxy-2-[(E)-(S)-4-hydroxy-4-(1-propyl-cyclobutyl)-but-1-enyl]-5-oxo-cyclopentyl}-heptanoic acid
   Show/Hide
C23H38O5
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0406799
 Compound Info 
(Z)-7-{(1R,2R,3R)-3-Hydroxy-2-[(E)-(S)-4-hydroxy-4-(1-propyl-cyclobutyl)-but-1-enyl]-5-oxo-cyclopentyl}-hept-5-enoic acid
   Show/Hide
C23H36O5
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0429334
 Compound Info 
(Z)-7-{(1R,2R,3R,5S)-5-Chloro-2-[(E)-(S)-4-(1-ethyl-cyclobutyl)-4-hydroxy-but-1-enyl]-3-hydroxy-cyclopentyl}-hept-5-enoic acid
   Show/Hide
C22H35ClO4
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0448597
 Compound Info 
7-{(1R,3R)-3-Hydroxy-2-[(E)-(S)-4-hydroxy-4-(1-propyl-cyclobutyl)-but-1-enyl]-5-oxo-cyclopentyl}-hept-5-ynoic acid
   Show/Hide
C23H34O5
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0449050
 Compound Info 
(Z)-7-{(1R,2R,3R)-3-Hydroxy-2-[(E)-(S)-4-hydroxy-4-(1-propyl-cyclohexyl)-but-1-enyl]-5-oxo-cyclopentyl}-hept-5-enoic acid
   Show/Hide
C25H40O5
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0380810
 Compound Info 
(3-{(1R,2S,3R)-3-Hydroxy-2-[(E)-(S)-3-hydroxy-4-(2-methoxy-phenyl)-but-1-enyl]-5-oxo-cyclopentylsulfanyl}-propylsulfanyl)-acetic acid
   Show/Hide
C21H28O6S2
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0381692
 Compound Info 
(3-{(1R,2S,3R)-3-Hydroxy-2-[(E)-(S)-3-hydroxy-4-(3-methoxy-phenyl)-but-1-enyl]-5-oxo-cyclopentylsulfanyl}-propylsulfanyl)-acetic acid
   Show/Hide
C21H28O6S2
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0381766
 Compound Info 
2-[3-[(1R,2S,3R)-3-hydroxy-2-[(E,3S)-3-hydroxy-4-(4-methylphenyl)but-1-enyl]-5-oxocyclopentyl]sulfanylpropylsulfanyl]acetic acid
   Show/Hide
C21H28O5S2
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0403665
 Compound Info 
(3-{(1R,2S,3R)-3-Hydroxy-2-[(E)-(S)-3-hydroxy-4-(3-propoxymethyl-phenyl)-but-1-enyl]-5-oxo-cyclopentylsulfanyl}-propylsulfanyl)-acetic acid
   Show/Hide
C24H34O6S2
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0403849
 Compound Info 
(3-{(1R,2S,3R)-2-[(E)-(S)-4-(3-Ethoxymethyl-phenyl)-3-hydroxy-but-1-enyl]-3-hydroxy-5-oxo-cyclopentylsulfanyl}-propylsulfanyl)-acetic acid
   Show/Hide
C23H32O6S2
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0403886
 Compound Info 
2-[3-[(1R,2S,3R)-3-hydroxy-2-[(E,3S)-3-hydroxy-4-(2-methylphenyl)but-1-enyl]-5-oxocyclopentyl]sulfanylpropylsulfanyl]acetic acid
   Show/Hide
C21H28O5S2
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0419283
 Compound Info 
(3-{(1R,2S,3R)-3-Hydroxy-2-[(E)-(S)-3-hydroxy-4-(3-methoxymethyl-phenyl)-but-1-enyl]-5-oxo-cyclopentylsulfanyl}-propylsulfanyl)-acetic acid
   Show/Hide
C22H30O6S2
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0432233
 Compound Info 
2-[3-[(1R,2S,3R)-3-hydroxy-2-[(E,3S)-3-hydroxy-4-(3-methylphenyl)but-1-enyl]-5-oxocyclopentyl]sulfanylpropylsulfanyl]acetic acid
   Show/Hide
C21H28O5S2
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0437604
 Compound Info 
(3-{(1R,2S,3R)-3-Hydroxy-2-[(E)-(S)-3-hydroxy-4-(3-methylsulfanylmethyl-phenyl)-but-1-enyl]-5-oxo-cyclopentylsulfanyl}-propylsulfanyl)-acetic acid
   Show/Hide
C22H30O5S3
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0438957
 Compound Info 
2-[3-[(1R,2S,3R)-3-hydroxy-2-[(E,3S)-3-hydroxy-4-[3-(3-methoxypropyl)phenyl]but-1-enyl]-5-oxocyclopentyl]sulfanylpropylsulfanyl]acetic acid
   Show/Hide
C24H34O6S2
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0458667
 Compound Info 
2-[3-[(1R,2S,3R)-3-hydroxy-2-[(E,3S)-3-hydroxy-4-[3-(2-methoxyethyl)phenyl]but-1-enyl]-5-oxocyclopentyl]sulfanylpropylsulfanyl]acetic acid
   Show/Hide
C23H32O6S2
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0224474
 Compound Info 
4-(2-((1R,2R,3R)-3-hydroxy-2-((S,E)-3-hydroxy-4-(3-(methoxymethyl)phenyl)but-1-enyl)-5-oxocyclopentyl)ethylthio)butanoic acid
   Show/Hide
C23H32O6S
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0415385
 Compound Info 
4-(2-{(1R,2R,3R)-3-Hydroxy-2-[(E)-(S)-3-hydroxy-4-(4-hydroxy-3-methyl-phenyl)-but-1-enyl]-5-oxo-cyclopentyl}-ethylsulfanyl)-butyric acid
   Show/Hide
C22H30O6S
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0448302
 Compound Info 
4-(2-{(1R,2R,3R,5R)-5-Fluoro-3-hydroxy-2-[(E)-(S)-3-hydroxy-4-(3-methoxymethyl-phenyl)-but-1-enyl]-cyclopentyl}-ethylsulfanyl)-butyric acid
   Show/Hide
C23H33FO5S
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0437055
 Compound Info 
2-[1-[4-[[(2S)-7-fluoro-4-methyl-2,3-dihydro-1,4-benzoxazin-2-yl]methoxy]benzoyl]-2-methylindol-4-yl]acetic acid
   Show/Hide
C28H25FN2O5
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0445860
 Compound Info 
2-[1-[4-(3,4-dihydro-2H-chromen-3-ylmethoxy)benzoyl]-2-methylindol-4-yl]acetic acid
   Show/Hide
C28H25NO5
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0485456
 Compound Info 
2-[1-(4-butoxybenzoyl)-2-methylindol-4-yl]acetic acid
   Show/Hide
C22H23NO4
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0485482
 Compound Info 
2-[2-methyl-1-[4-[[(2R)-4-methyl-2,3-dihydro-1,4-benzoxazin-2-yl]methoxy]benzoyl]indol-4-yl]acetic acid
   Show/Hide
C28H26N2O5
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0239945
 Compound Info 
acrylic acid derivative, 12
   Show/Hide
C25H22N2O3
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0405515
 Compound Info 
acrylic acid derivative, 17
   Show/Hide
C28H24O4
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0421513
 Compound Info 
acrylic acid derivative, 7
   Show/Hide
C25H30O5
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0421542
 Compound Info 
acrylic acid derivative, 8
   Show/Hide
C25H30O6
  1
1
Ki > 10000 nM
 Bioactivity Info 
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   LI
   LO
   TS
CP0428946
 Compound Info 
acrylic acid derivative, 11
   Show/Hide
C23H20N2O4
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0428955
 Compound Info 
phenoxyacetic acid analogue, 19
   Show/Hide
C24H22N2O4
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0430840
 Compound Info 
acrylic acid derivative, 10
   Show/Hide
C23H24N2O4
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0430841
 Compound Info 
benzyloxyacetic acid analogue, 21
   Show/Hide
C25H24N2O4
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0430842
 Compound Info 
acrylic acid derivative, 3
   Show/Hide
C28H32N2O5
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0438911
 Compound Info 
acrylic acid derivative, 9
   Show/Hide
C22H22N2O4
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0463775
 Compound Info 
acrylic acid derivative, 15
   Show/Hide
C26H22O3S
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0463777
 Compound Info 
phenylpropynoic acid analogue, 18
   Show/Hide
C25H20N2O3
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0477288
 Compound Info 
acrylic acid derivative, 14
   Show/Hide
C28H24O3
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0494377
 Compound Info 
acrylic acid derivative, 16
   Show/Hide
C28H24O4
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0497108
 Compound Info 
acrylic acid derivative, 6
   Show/Hide
C24H28O5
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0390115
 Compound Info 
N-(3,4-difluorophenyl)sulfonyl-3-[4-[(dimethylamino)methyl]-2-(2-naphthalen-2-ylethoxy)phenyl]propanamide
   Show/Hide
C30H30F2N2O4S
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0430730
 Compound Info 
3-(4-((3-cyanophenoxy)methyl)-2-(2-(naphthalen-2-yl)ethoxy)phenyl)-N-(3,4-difluorophenylsulfonyl)propanamide
   Show/Hide
C35H28F2N2O5S
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0373665
 Compound Info 
3-[2-({[1-(4-Fluoro-3-methylphenyl)-3-methylbutyl]-amino}carbonyl)-4-(phenoxymethyl)phenyl]propanoic acid
   Show/Hide
C29H32FNO4
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0373666
 Compound Info 
3-[2-({[1-(3,5-Dimethylphenyl)-3-methylbutyl]amino}-carbonyl)-4-(phenoxymethyl)phenyl]propanoic acid
   Show/Hide
C30H35NO4
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0373674
 Compound Info 
3-[4-[(3-Cyanophenoxy)methyl]-2-({[1-(3,5-dimethylphenyl)-3-methylbutyl]amino}carbonyl)phenyl]propanoic acid
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C31H34N2O4
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
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   LO
   TS
CP0373705
 Compound Info 
3-{2-({[1-(3,5-Dimethylphenyl)-3-methylbutyl]amino}-carbonyl)-4-[(3-fluorophenoxy)methyl]phenyl}propanoic acid
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C30H34FNO4
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0373980
 Compound Info 
3-[4-[(2,5-Difluorophenoxy)methyl]-2-({[1-(3,5-dimethylphenyl)-3-methylbutyl]amino}carbonyl)phenyl]propanoic acid
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C30H33F2NO4
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0390421
 Compound Info 
3-{2-({[1-(3,5-Dimethylphenyl)-3-methylbutyl]amino}-carbonyl)-4-[(2-methylphenoxy)methyl]phenyl}propanoic acid
   Show/Hide
C31H37NO4
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
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   LO
   TS
CP0181716
 Compound Info 
3-[2-({[3-Methyl-1-(1-naphthyl)butyl]amino}carbonyl)-4-(phenoxymethyl)phenyl]propanoic acid
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C32H33NO4
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0375769
 Compound Info 
3-[2-{[(1-Benzyl-3-methylbutyl)amino]carbonyl}-4-(phenoxymethyl)phenyl]propanoic acid
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C29H33NO4
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
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   LO
   TS
CP0390196
 Compound Info 
3-(4-(Phenoxymethyl)-2-{[(2-phenylethyl)amino]carbonyl}phenyl)propanoic acid
   Show/Hide
C25H25NO4
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0401370
 Compound Info 
3-(2-(3-methyl-1-phenylbutylcarbamoyl)-4-(phenoxymethyl)phenyl)propanoic acid
   Show/Hide
C28H31NO4
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
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   LO
   TS
CP0440188
 Compound Info 
3-[2-({[(1S)-1-(1-Naphthyl)ethyl]amino}carbonyl)-4-(phenoxymethyl)phenyl]propanoic acid
   Show/Hide
C29H27NO4
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0440189
 Compound Info 
3-[2-({[(1R)-1-(1-Naphthyl)ethyl]amino}carbonyl)-4-(phenoxymethyl)phenyl]propanoic acid
   Show/Hide
C29H27NO4
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0373058
 Compound Info 
3-[2-({[(1R)-1-(3,5-Dimethylphenyl)-3-methylbutyl]-amino}carbonyl)-4-phenoxyphenyl]propanoic acid
   Show/Hide
C29H33NO4
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0373059
 Compound Info 
3-[4-(3,5-Dimethylphenoxy)-2-({[(1R)-1-(3,5-dimethylphenyl)-3-methylbutyl]amino}carbonyl)phenyl]propanoic acid
   Show/Hide
C31H37NO4
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0383546
 Compound Info 
3-[2-({[(1R)-1-(3,5-Dimethylphenyl)-3-methylbutyl]amino}-carbonyl)-4-(phenoxymethyl)phenyl]propanoic acid
   Show/Hide
C30H35NO4
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0383547
 Compound Info 
3-{2-({[(1R)-1-(3,5-Dimethylphenyl)-3-methylbutyl]amino}-carbonyl)-4-[(3-fluorophenoxy)methyl]phenyl}propanoic acid
   Show/Hide
C30H34FNO4
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0390806
 Compound Info 
3-[4-(3,5-Difluorophenoxy)-2-({[(1R)-1-(3,5-dimethylphenyl)-3-methylbutyl]amino}carbonyl)phenyl]propanoic acid
   Show/Hide
C29H31F2NO4
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0390809
 Compound Info 
3-[4-[(3,5-Difluorophenyl)amino]-2-({[(1R)-1-(3,5-dimethylphenyl)-3-methylbutyl]amino}carbonyl)phenyl]-propanoic acid
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C29H32F2N2O3
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0390810
 Compound Info 
3-(4-[(3,5-Dimethylphenyl)amino]-2-{[(1R)-1-(3,5-dimethylphenyl)-3-methylbutyl]carbamoyl}phenyl)propanoic acid
   Show/Hide
C31H38N2O3
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0390821
 Compound Info 
3-[4-[(2,4-Difluorophenoxy)methyl]-2-({[(1R)-1-(3,5-dimethylphenyl)-3-methylbutyl]amino}carbonyl)phenyl]-propanoic acid
   Show/Hide
C30H33F2NO4
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0390824
 Compound Info 
3-[4-[(2,4-Dimethylphenoxy)methyl]-2-({[(1R)-1-(3,5-dimethylphenyl)-3-methylbutyl]amino}carbonyl)phenyl]-propanoic acid
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C32H39NO4
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0390971
 Compound Info 
3-{2-({[(1R)-1-(3,5-Dimethylphenyl)-3-methylbutyl]-amino}carbonyl)-4-[(pyridin-3-yloxy)methyl]phenyl}propanoicacid
   Show/Hide
C29H34N2O4
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0390972
 Compound Info 
3-(2-({[(1R)-1-(3,5-Dimethylphenyl)-3-methylbutyl]-amino}carbonyl)-4-{[(2-methylpyridin-3-yl)oxy]methyl}-phenyl)propanoic acid
   Show/Hide
C30H36N2O4
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0391021
 Compound Info 
3-[4-[(2,5-Difluorophenoxy)methyl]-2-({[(1R)-1-(3,5-dimethylphenyl)-3-methylbutyl]amino}carbonyl)phenyl]-propanoic acid
   Show/Hide
C30H33F2NO4
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0401854
 Compound Info 
3-[4-(3-Cyanophenoxy)-2-({[(1R)-1-(3,5-dimethylphenyl)-3-methylbutyl]amino}carbonyl)phenyl]propanoic acid
   Show/Hide
C30H32N2O4
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0402252
 Compound Info 
3-{2-({[(1R)-1-(3,5-Dimethylphenyl)-3-methylbutyl]-amino}carbonyl)-4-[(2-methylphenoxy)methyl]phenyl}-propanoic acid
   Show/Hide
C31H37NO4
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0414920
 Compound Info 
3-{2-({[(1R)-1-(3,5-Dimethylphenyl)-3-methylbutyl]-amino}carbonyl)-4-[(3-methylphenyl)amino]phenyl}propanoic acid
   Show/Hide
C30H36N2O3
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0417692
 Compound Info 
3-[4-[(3-Cyanophenoxy)methyl]-2-({[(1R)-1-(3,5-dimethylphenyl)-3-methylbutyl]amino}carbonyl)phenyl]propanoicacid
   Show/Hide
C31H34N2O4
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0435130
 Compound Info 
3-[4-[(2,5-Difluorophenoxy)methyl]-2-({[(1S)-1-(3,5-dimethylphenyl)-3-methylbutyl]amino}carbonyl)phenyl]-propanoic acid
   Show/Hide
C30H33F2NO4
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0435134
 Compound Info 
3-[4-[(2,5-Dimethylphenoxy)methyl]-2-({[(1R)-1-(3,5-dimethylphenyl)-3-methylbutyl]amino}carbonyl)phenyl]-propanoic acid
   Show/Hide
C32H39NO4
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0469066
 Compound Info 
3-(2-({[(1R)-1-(3,5-Dimethylphenyl)-3-methylbutyl]-amino}carbonyl)-4-{[(6-methylpyridin-3-yl)oxy]methyl}-phenyl)propanoic acid
   Show/Hide
C30H36N2O4
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0010057
 Compound Info 
2-{1-[(4-chlorophenyl)carbonyl]-5-methoxy-2-methyl-1H-indol-3-yl}acetic acid
   Show/Hide
C19H16ClNO4
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0378355
 Compound Info 
2-[5-fluoro-2-methyl-1-[4-[[(2S)-4-methyl-2,3-dihydro-1,4-benzoxazin-2-yl]methoxy]benzoyl]indol-3-yl]acetic acid
   Show/Hide
C28H25FN2O5
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0378356
 Compound Info 
2-[5-methoxy-2-methyl-1-[4-[[(2S)-4-methyl-2,3-dihydro-1,4-benzoxazin-2-yl]methoxy]benzoyl]indol-3-yl]acetic acid
   Show/Hide
C29H28N2O6
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0388261
 Compound Info 
2-[2-methyl-1-[4-[[(2S)-4-methyl-2,3-dihydro-1,4-benzoxazin-2-yl]methoxy]benzoyl]indol-3-yl]acetic acid
   Show/Hide
C28H26N2O5
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0388266
 Compound Info 
2-[1-[2-chloro-4-[[(2S)-4-methyl-2,3-dihydro-1,4-benzoxazin-2-yl]methoxy]benzoyl]-2-methylindol-3-yl]acetic acid
   Show/Hide
C28H25ClN2O5
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
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   LO
   TS
CP0388465
 Compound Info 
2-[1-[4-[[(2R)-1-ethyl-2,3-dihydroindol-2-yl]methoxy]-2-methylbenzoyl]-2-methylindol-3-yl]acetic acid
   Show/Hide
C30H30N2O4
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0428289
 Compound Info 
2-[5-chloro-2-methyl-1-[4-[[(2S)-4-methyl-2,3-dihydro-1,4-benzoxazin-2-yl]methoxy]benzoyl]indol-3-yl]acetic acid
   Show/Hide
C28H25ClN2O5
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0431698
 Compound Info 
2-[1-[2-chloro-4-[[(2S)-4-methyl-2,3-dihydro-1,4-benzoxazin-2-yl]methoxy]benzoyl]-5-fluoro-2-methylindol-3-yl]acetic acid
   Show/Hide
C28H24ClFN2O5
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0377711
 Compound Info 
2-[4-methyl-3-[[2-methyl-4-[[(2S)-4-methyl-2,3-dihydro-1,4-benzoxazin-2-yl]methoxy]benzoyl]amino]phenyl]acetic acid
   Show/Hide
C27H28N2O5
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0387733
 Compound Info 
2-[3-methyl-5-[[2-methyl-4-[[(2S)-4-methyl-2,3-dihydro-1,4-benzoxazin-2-yl]methoxy]benzoyl]amino]phenyl]acetic acid
   Show/Hide
C27H28N2O5
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0390164
 Compound Info 
2-[3-[[2-chloro-4-[[(2S)-4-methyl-2,3-dihydro-1,4-benzoxazin-2-yl]methoxy]benzoyl]amino]-4-fluorophenyl]acetic acid
   Show/Hide
C25H22ClFN2O5
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0426154
 Compound Info 
2-[3-[methyl-[4-[[(2S)-4-methyl-2,3-dihydro-1,4-benzoxazin-2-yl]methoxy]benzoyl]amino]phenyl]acetic acid
   Show/Hide
C26H26N2O5
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0431260
 Compound Info 
2-[3-[[4-[[(2S)-4-methyl-2,3-dihydro-1,4-benzoxazin-2-yl]methoxy]phenyl]carbamoyl]phenyl]acetic acid
   Show/Hide
C25H24N2O5
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0494477
 Compound Info 
2-[3-[[2-methyl-4-[[(2S)-4-methyl-2,3-dihydro-1,4-benzoxazin-2-yl]methoxy]benzoyl]amino]phenyl]acetic acid
   Show/Hide
C26H26N2O5
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0388029
 Compound Info 
4-[2-[(4S)-4-[(E,3S)-3-hydroxy-4-(3-propylphenyl)but-1-enyl]-2-oxo-1,3-oxazolidin-3-yl]ethylsulfanyl]butanoic acid
   Show/Hide
C22H31NO5S
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0388030
 Compound Info 
4-[2-[(4S)-4-[(E,3S)-4-(3-chlorophenyl)-3-hydroxybut-1-enyl]-2-oxo-1,3-oxazolidin-3-yl]ethylsulfanyl]butanoic acid
   Show/Hide
C19H24ClNO5S
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0388031
 Compound Info 
7-[(2R)-2-[(E,3S)-4-(3-fluorophenyl)-3-hydroxybut-1-enyl]-5-sulfanylidenepyrrolidin-1-yl]heptanoic acid
   Show/Hide
C21H28FNO3S
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0388032
 Compound Info 
4-[2-[(4S)-4-[(E,3S)-3-hydroxy-4-phenylbut-1-enyl]-2-oxo-1,3-thiazolidin-3-yl]ethylsulfanyl]butanoic acid
   Show/Hide
C19H25NO4S2
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0388033
 Compound Info 
4-[2-[(4S)-4-[(E,3S)-3-hydroxy-4-[3-(trifluoromethyl)phenyl]but-1-enyl]-2-oxo-1,3-thiazolidin-3-yl]ethylsulfanyl]butanoic acid
   Show/Hide
C20H24F3NO4S2
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0388034
 Compound Info 
7-[(2R)-2-[(E,3S)-3-hydroxy-4-phenylbut-1-enyl]-5-sulfanylidenepyrrolidin-1-yl]heptanoic acid
   Show/Hide
C21H29NO3S
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0391383
 Compound Info 
7-[(2R)-2-[(E,3S)-4-(3-ethylphenyl)-3-hydroxybut-1-enyl]-5-sulfanylidenepyrrolidin-1-yl]heptanoic acid
   Show/Hide
C23H33NO3S
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0392256
 Compound Info 
7-[(2R)-2-[(E,3S)-3-hydroxy-4-(3-propylphenyl)but-1-enyl]-5-sulfanylidenepyrrolidin-1-yl]heptanoic acid
   Show/Hide
C24H35NO3S
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0395226
 Compound Info 
4-[2-[(2R)-2-[(E,3S)-3-hydroxy-4-[3-(methoxymethyl)phenyl]but-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]butanoic acid
   Show/Hide
C22H31NO5S
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0395230
 Compound Info 
4-[2-[(1R,2R)-2-[(E,3S)-3-hydroxy-4-[3-(methoxymethyl)phenyl]but-1-enyl]-5-oxocyclopentyl]ethylsulfanyl]butanoic acid
   Show/Hide
C23H32O5S
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0395231
 Compound Info 
4-[2-[(4S)-4-[(E,3S)-3-hydroxy-4-[3-(trifluoromethyl)phenyl]but-1-enyl]-2-oxo-1,3-oxazolidin-3-yl]ethylsulfanyl]butanoic acid
   Show/Hide
C20H24F3NO5S
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0400838
 Compound Info 
7-[(2R)-2-[(E,3S)-3-hydroxy-4-[3-(trifluoromethyl)phenyl]but-1-enyl]-5-sulfanylidenepyrrolidin-1-yl]heptanoic acid
   Show/Hide
C22H28F3NO3S
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0400839
 Compound Info 
7-[(2R)-2-[(E,3S)-3-hydroxy-4-[3-(methoxymethyl)phenyl]but-1-enyl]-5-sulfanylidenepyrrolidin-1-yl]heptanoic acid
   Show/Hide
C23H33NO4S
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0400840
 Compound Info 
4-[2-[(4S)-4-[(E,3S)-3-hydroxy-4-[3-(trifluoromethoxy)phenyl]but-1-enyl]-2-oxo-1,3-oxazolidin-3-yl]ethylsulfanyl]butanoic acid
   Show/Hide
C20H24F3NO6S
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0401106
 Compound Info 
4-[2-[(4S)-4-[(E,3S)-3-hydroxy-4-[3-(methoxymethyl)phenyl]but-1-enyl]-2-oxo-1,3-oxazolidin-3-yl]ethylsulfanyl]butanoic acid
   Show/Hide
C21H29NO6S
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0403544
 Compound Info 
7-[(2R)-2-[(E,3S)-3-hydroxy-4-[3-(methoxymethyl)phenyl]but-1-enyl]-5-oxopyrrolidin-1-yl]heptanoic acid
   Show/Hide
C23H33NO5
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0403545
 Compound Info 
4-[2-[(4S)-4-[(E,3S)-3-hydroxy-4-phenylbut-1-enyl]-2-oxo-1,3-oxazolidin-3-yl]ethylsulfanyl]butanoic acid
   Show/Hide
C19H25NO5S
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0427837
 Compound Info 
4-[2-[(4S)-4-[(E,3S)-4-(3-fluorophenyl)-3-hydroxybut-1-enyl]-2-oxo-1,3-thiazolidin-3-yl]ethylsulfanyl]butanoic acid
   Show/Hide
C19H24FNO4S2
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0431080
 Compound Info 
4-[2-[(4S)-4-[(E,3S)-3-hydroxy-4-[3-(methoxymethyl)phenyl]but-1-enyl]-2-oxo-1,3-thiazolidin-3-yl]ethylsulfanyl]butanoic acid
   Show/Hide
C21H29NO5S2
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0431204
 Compound Info 
4-[2-[(4S)-4-[(E,3S)-3-hydroxy-4-(3-propylphenyl)but-1-enyl]-2-oxo-1,3-thiazolidin-3-yl]ethylsulfanyl]butanoic acid
   Show/Hide
C22H31NO4S2
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0463502
 Compound Info 
4-[2-[(4S)-4-[(E,3S)-3-hydroxy-4-(3-phenylphenyl)but-1-enyl]-2-oxo-1,3-oxazolidin-3-yl]ethylsulfanyl]butanoic acid
   Show/Hide
C25H29NO5S
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0038951
 Compound Info 
4-(2-((R)-2-((S,E)-3-hydroxyoct-1-enyl)-5-oxopyrrolidin-1-yl)ethylthio)butanoic acid
   Show/Hide
C18H31NO4S
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0050749
 Compound Info 
4-(2-((R)-2-((S)-3-hydroxyoct-1-enyl)-5-oxopyrrolidin-1-yl)ethyl)benzoate
   Show/Hide
C21H29NO4
  1
1
Ki > 10000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0144553
 Compound Info 
7-[(R)-2-((E)-(S)-3-Hydroxy-oct-1-enyl)-5-oxo-pyrrolidin-1-yl]-heptanoic acid
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C19H33NO4
  1
1
Ki > 10000 nM
 Bioactivity Info 
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CP0378128
 Compound Info 
4-[2-[(2R)-2-[(E,3S)-3-hydroxy-4-(3-methylphenyl)but-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]butanoic acid
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C21H29NO4S
  1
1
Ki > 10000 nM
 Bioactivity Info 
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CP0387595
 Compound Info 
2-[2-[(2R)-2-[(E,3S)-3-hydroxy-4-(3-methylphenyl)but-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]-1,3-thiazole-4-carboxylic acid
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C21H24N2O4S2
  1
1
Ki > 10000 nM
 Bioactivity Info 
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CP0387596
 Compound Info 
2-[2-[(2R)-2-[(E,3S)-3-hydroxy-4-(3-methylphenyl)but-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]-1,3-thiazole-5-carboxylic acid
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C21H24N2O4S2
  1
1
Ki > 10000 nM
 Bioactivity Info 
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CP0387602
 Compound Info 
4-[2-[(2R)-2-[(E,3S)-3-hydroxy-4-(3-methylphenyl)but-1-enyl]-5-oxopyrrolidin-1-yl]ethyl]benzoic acid
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C24H27NO4
  1
1
Ki > 10000 nM
 Bioactivity Info 
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CP0387603
 Compound Info 
2-[2-[(2R)-2-[(E,3S)-3-hydroxy-4-phenylbut-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]-1,3-thiazole-4-carboxylic acid
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C20H22N2O4S2
  1
1
Ki > 10000 nM
 Bioactivity Info 
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CP0387618
 Compound Info 
5-[3-[(2R)-2-[(E,3S)-3-hydroxy-4-(3-methylphenyl)but-1-enyl]-5-oxopyrrolidin-1-yl]propyl]thiophene-2-carboxylic acid
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C23H27NO4S
  1
1
Ki > 10000 nM
 Bioactivity Info 
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CP0392891
 Compound Info 
2-[2-[(2R)-2-[(E,3S)-3-hydroxy-4-(5-methylfuran-2-yl)but-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]-1,3-thiazole-4-carboxylic acid
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C19H22N2O5S2
  1
1
Ki > 10000 nM
 Bioactivity Info 
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CP0431607
 Compound Info 
2-[3-[(2R)-2-[(E,3S)-3-hydroxy-4-(3-methylphenyl)but-1-enyl]-5-oxopyrrolidin-1-yl]propyl]-1,3-oxazole-4-carboxylic acid
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C22H26N2O5
  1
1
Ki > 10000 nM
 Bioactivity Info 
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CP0438240
 Compound Info 
2-[3-[(2R)-2-[(E,3S)-3-hydroxy-4-(3-methylphenyl)but-1-enyl]-5-oxopyrrolidin-1-yl]propyl]-1,3-thiazole-4-carboxylic acid
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C22H26N2O4S
  1
1
Ki > 10000 nM
 Bioactivity Info 
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CP0475478
 Compound Info 
2-[2-[(2R)-2-[(E,3S)-4-cyclopentyl-3-hydroxybut-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]-1,3-thiazole-4-carboxylic acid
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C19H26N2O4S2
  1
1
Ki > 10000 nM
 Bioactivity Info 
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CP0387597
 Compound Info 
2-[2-[(2R)-2-[(E,3S)-3-hydroxy-4-(3-naphthalen-2-ylphenyl)but-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]-1,3-thiazole-4-carboxylic acid
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C30H28N2O4S2
  1
1
Ki > 10000 nM
 Bioactivity Info 
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CP0387598
 Compound Info 
5-[3-[(2R)-2-[(E,3S)-4-(3-chlorophenyl)-3-hydroxybut-1-enyl]-5-oxopyrrolidin-1-yl]propyl]thiophene-2-carboxylic acid
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C22H24ClNO4S
  1
1
Ki > 10000 nM
 Bioactivity Info 
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CP0387600
 Compound Info 
3-[3-[(2R)-2-[(E,3S)-4-(3-chlorophenyl)-3-hydroxybut-1-enyl]-5-oxopyrrolidin-1-yl]phenyl]propanoic acid
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C23H24ClNO4
  1
1
Ki > 10000 nM
 Bioactivity Info 
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CP0387601
 Compound Info 
2-[3-[[(2R)-2-[(E,3S)-3-hydroxy-4-(3-methylphenyl)but-1-enyl]-5-oxopyrrolidin-1-yl]methyl]phenyl]acetic acid
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C24H27NO4
  1
1
Ki > 10000 nM
 Bioactivity Info 
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CP0438238
 Compound Info 
4-[2-[(2R)-2-[(E,3S)-4-(3-chlorophenyl)-3-hydroxybut-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]butanoic acid
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C20H26ClNO4S
  1
1
Ki > 10000 nM
 Bioactivity Info 
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CP0438239
 Compound Info 
5-[2-[(2R)-2-[(E,3S)-3-hydroxy-4-(3-methylphenyl)but-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]thiophene-2-carboxylic acid
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C22H25NO4S2
  1
1
Ki > 10000 nM
 Bioactivity Info 
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CP0378146
 Compound Info 
4-[2-[(2R)-2-[(E,3S)-3-hydroxy-4-(3-pyridin-2-ylphenyl)but-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]butanoic acid
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C25H30N2O4S
  1
1
Ki > 10000 nM
 Bioactivity Info 
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CP0378148
 Compound Info 
2-[2-[(2R)-2-[(E,3S)-4-[3-(1,3-benzoxazol-2-yl)phenyl]-3-hydroxybut-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]-1,3-thiazole-4-carboxylic acid
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C27H25N3O5S2
  1
1
Ki > 10000 nM
 Bioactivity Info 
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CP0410231
 Compound Info 
4-[2-[(2R)-2-[(E,3S)-4-[3-(1,3-benzothiazol-2-yl)phenyl]-3-hydroxybut-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]butanoic acid
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C27H30N2O4S2
  1
1
Ki > 10000 nM
 Bioactivity Info 
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CP0410232
 Compound Info 
4-[2-[(2R)-2-[(E,3S)-3-hydroxy-4-[3-(pyridin-4-ylmethoxy)phenyl]but-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]butanoic acid
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C26H32N2O5S
  1
1
Ki > 10000 nM
 Bioactivity Info 
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CP0410312
 Compound Info 
4-[2-[(2R)-2-[(E,3S)-3-hydroxy-4-[3-(pyridin-2-ylmethoxy)phenyl]but-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]butanoic acid
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C26H32N2O5S
  1
1
Ki > 10000 nM
 Bioactivity Info 
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CP0416072
 Compound Info 
4-[2-[(2R)-2-[(E,3S)-3-hydroxy-4-[3-(1H-indol-5-yl)phenyl]but-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]butanoic acid
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C28H32N2O4S
  1
1
Ki > 10000 nM
 Bioactivity Info 
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CP0423859
 Compound Info 
4-[2-[(2R)-2-[(E,3S)-3-hydroxy-4-(3-naphthalen-2-ylphenyl)but-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]butanoic acid
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C30H33NO4S
  1
1
Ki > 10000 nM
 Bioactivity Info 
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CP0423860
 Compound Info 
4-[2-[(2R)-2-[(E,3S)-3-hydroxy-4-[3-(pyridin-3-ylmethoxy)phenyl]but-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]butanoic acid
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C26H32N2O5S
  1
1
Ki > 10000 nM
 Bioactivity Info 
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CP0423862
 Compound Info 
4-[2-[(2R)-2-[(E,3S)-3-hydroxy-4-(3-phenylphenyl)but-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]butanoic acid
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C26H31NO4S
  1
1
Ki > 10000 nM
 Bioactivity Info 
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CP0480109
 Compound Info 
4-[2-[(2R)-2-[(E,3S)-4-[3-(1-benzofuran-2-yl)phenyl]-3-hydroxybut-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]butanoic acid
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C28H31NO5S
  1
1
Ki > 10000 nM
 Bioactivity Info 
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Biochemical Assays
Compound ID Compound Name Compound Formula
CP0010057
 Compound Info 
2-{1-[(4-chlorophenyl)carbonyl]-5-methoxy-2-methyl-1H-indol-3-yl}acetic acid
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C19H16ClNO4
  1
1 Ki > 10000 nM
Similar Protein(s) and Bioactivity Statistics
90% Identity
Protein ID Protein Name Protein Organism
PT05403 Prostaglandin E2 receptor EP1 subtype Rattus norvegicus, Rat
 Protein Info