Brief Information of the Cell Line and Protein
Cell Line ID: CL000011 , CHO
Synonyms
Chinese Hamster Ovary
CHO-ori
Category Spontaneously immortalized cell line
Organism
Cricetulus griseus (Chinese hamster)
Cellosaurus ID
CVCL_0213
Protein ID: PT03559 , Orexin/Hypocretin receptor type 1
Gene Name HCRTR1
Organism Rattus norvegicus, Rat
Protein Classification Membrane receptor
Uniprot ID P56718
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000011  Protein ID: PT03559
 
Compound ID Compound Name Compound Formula
CP0087270
SB-649868
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C26H24FN3O3S
 1
1
Ki = 0.1175 nM
   TI
   LI
   LO
   TS
CP0385441
US8623863, 3-8
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C24H27FN4O3
 1
1
Ki = 5.1 nM
   TI
   LI
   LO
   TS
CP0471684
US8623863, 2-8
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C25H29FN4O2
 1
1
Ki = 8.7 nM
   TI
   LI
   LO
   TS
CP0468161
US8623863, 1-8
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C24H27FN4O2
 1
1
Ki = 15 nM
   TI
   LI
   LO
   TS
CP0519859
US8623863, 3-2
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C26H29FN2O2S
 1
1
Ki = 29 nM
   TI
   LI
   LO
   TS
CP0463175
US8623863, 4-9
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C23H25FN4O3
 1
1
Ki = 39 nM
   TI
   LI
   LO
   TS
CP0403002
US8623863, 3-3
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C27H30FN3O2
 1
1
Ki = 42 nM
   TI
   LI
   LO
   TS
CP0441542
US8623863, 2-9
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C24H27FN4O2
 1
1
Ki = 50 nM
   TI
   LI
   LO
   TS
CP0544447
US8623863, 3-5
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C24H26FN3O2S
 1
1
Ki = 73 nM
   TI
   LI
   LO
   TS
CP0472606
US8623863, 3-4
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C24H26FN3O3
 1
1
Ki = 110 nM
   TI
   LI
   LO
   TS
CP0438206
US8623863, 2-10
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C23H26FN5O2
 1
1
Ki = 150 nM
   TI
   LI
   LO
   TS
CP0542117
US8623863, 2-11
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C22H24FN5O2
 1
1
Ki = 190 nM
   TI
   LI
   LO
   TS
CP0474805
US8623863, 3-6
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C25H27FN4O2
 1
1
Ki = 310 nM
   TI
   LI
   LO
   TS