| Compound ID |
Compound Name |
Compound Formula |
|
CP0006743
|
4-methoxy-N-(2,4,6-trimethylphenyl)benzenesulfonamide
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|
C16H19NO3S
|
1
|
| 1 |
EC50 > 50118.72 nM
|
|
|
|
CP0186249
|
3-[[4-[1-[3-[2-methoxy-5-(trifluoromethyl)phenyl]-6-[4-(trifluoromethoxy)phenyl]indazol-1-yl]pentyl]benzoyl]amino]propanoic acid
Show/Hide
|
C37H33F6N3O5
|
2
|
| 1 |
IC50 = 0.8 nM
|
|
|
| 2 |
IC50 = 8 nM
|
|
|
|
CP0094595
|
4-[[(4-tert-butylcyclohexyl)-(1-methyl-5-phenylmethoxybenzimidazol-2-yl)amino]methyl]-N-(2H-tetrazol-5-yl)benzamide
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|
C34H40N8O2
|
2
|
| 1 |
IC50 = 1 nM
|
|
|
| 2 |
IC50 = 7 nM
|
|
|
|
CP0122551
|
4-[[(4-tert-butylcyclohexyl)-(1-methyl-6-propoxybenzimidazol-2-yl)amino]methyl]-N-(2H-tetrazol-5-yl)benzamide
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|
C30H40N8O2
|
2
|
| 1 |
IC50 = 1 nM
|
|
|
| 2 |
IC50 = 8 nM
|
|
|
|
CP0166401
|
4-[[(4-tert-butylcyclohexyl)-(5-cyclopentyloxy-1-methylbenzimidazol-2-yl)amino]methyl]-N-(2H-tetrazol-5-yl)benzamide
Show/Hide
|
C32H42N8O2
|
2
|
| 1 |
IC50 = 1 nM
|
|
|
| 2 |
IC50 = 9 nM
|
|
|
|
CP0235668
|
3-[[4-[1-[3-[2-methoxy-5-(trifluoromethyl)phenyl]-6-[4-(trifluoromethoxy)phenyl]indazol-1-yl]butyl]benzoyl]amino]propanoic acid
Show/Hide
|
C36H31F6N3O5
|
2
|
| 1 |
IC50 = 1 nM
|
|
|
| 2 |
IC50 = 5.6 nM
|
|
|
|
CP0738123
|
4-((3-methyl-4-propoxy-2-(4-(trifluoromethoxy)phenylimino)-6-(trifluoromethyl)-2,3-dihydro-1H-benzo[d]imidazol-1-yl)methyl)-N-(1H-tetrazol-5-yl)benzamide
Show/Hide
|
C28H24F6N8O3
|
2
|
| 1 |
IC50 = 1.3 nM
|
|
|
| 2 |
IC50 = 16.3 nM
|
|
|
|
CP0474757
|
3-[[4-[1-[3-[2-methoxy-5-(trifluoromethyl)phenyl]-6-(4-methylsulfanylphenyl)indazol-1-yl]pentyl]benzoyl]amino]propanoic acid
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|
C37H36F3N3O4S
|
2
|
| 1 |
IC50 = 1.5 nM
|
|
|
| 2 |
IC50 = 9 nM
|
|
|
|
CP0545453
|
3-[[4-[1-[6-(3-fluoro-4-methoxyphenyl)-3-[2-methoxy-5-(trifluoromethyl)phenyl]indazol-1-yl]pentyl]benzoyl]amino]propanoic acid
Show/Hide
|
C37H35F4N3O5
|
2
|
| 1 |
IC50 = 1.5 nM
|
|
|
| 2 |
IC50 = 18 nM
|
|
|
|
CP0415788
|
3-[[4-[1-[3-[2-methoxy-5-(trifluoromethyl)phenyl]-6-[4-(trifluoromethyl)phenyl]indazol-1-yl]pentyl]benzoyl]amino]propanoic acid
Show/Hide
|
C37H33F6N3O4
|
2
|
| 1 |
IC50 = 1.6 nM
|
|
|
| 2 |
IC50 = 14 nM
|
|
|
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CP0904767
|
4-((4-butyl-3-methyl-2-(4-(trifluoromethoxy)phenylimino)-6-(trifluoromethyl)-2,3-dihydro-1H-benzo[d]imidazol-1-yl)methyl)-N-(1H-tetrazol-5-yl)benzamide
Show/Hide
|
C29H26F6N8O2
|
2
|
| 1 |
IC50 = 1.7 nM
|
|
|
| 2 |
IC50 = 7.6 nM
|
|
|
|
CP0438941
|
3-(1-(N-((1r,4r)-4-tert-butylcyclohexyl)-2-(4-(trifluoromethoxy)phenyl)acetamido)-2,3-dihydro-1H-indene-5-carboxamido)propanoic acid
Show/Hide
|
C32H39F3N2O5
|
2
|
| 1 |
IC50 = 1.8 nM
|
|
|
| 2 |
IC50 = 500 nM
|
|
|
|
CP0445332
|
3-[[4-[(1S)-1-[3-[3-chloro-5-(trifluoromethyl)phenyl]-5-(6-methoxynaphthalen-2-yl)pyrazol-1-yl]ethyl]benzoyl]amino]propanoic acid
Show/Hide
|
C33H27ClF3N3O4
|
2
|
| 1 |
IC50 = 1.9 nM
|
|
|
| 2 |
IC50 = 5.7 nM
|
|
|
|
CP0411425
|
3-[[4-[1-[6-(4-methoxyphenyl)-3-[2-methoxy-5-(trifluoromethyl)phenyl]indazol-1-yl]pentyl]benzoyl]amino]propanoic acid
Show/Hide
|
C37H36F3N3O5
|
2
|
| 1 |
IC50 = 1.9 nM
|
|
|
| 2 |
IC50 = 14 nM
|
|
|
|
CP0043109
|
4-[[(4-tert-butylcyclohexyl)-(5-hydroxy-1-methylbenzimidazol-2-yl)amino]methyl]-N-(2H-tetrazol-5-yl)benzamide
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|
C27H34N8O2
|
2
|
| 1 |
IC50 = 2 nM
|
|
|
| 2 |
IC50 > 1000 nM
|
|
|
|
CP0043112
|
4-[[(4-tert-butylcyclohexyl)-(1-methyl-5-propoxybenzimidazol-2-yl)amino]methyl]-N-(2H-tetrazol-5-yl)benzamide
Show/Hide
|
C30H40N8O2
|
2
|
| 1 |
IC50 = 2 nM
|
|
|
| 2 |
IC50 = 4 nM
|
|
|
|
CP0156839
|
CHEMBL518939
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|
C29H38N8O2
|
2
|
| 1 |
IC50 = 2 nM
|
|
|
| 2 |
IC50 = 22 nM
|
|
|
|
CP0170481
|
4-[[(4-tert-butylcyclohexyl)-[5-(cyclopentylmethoxy)-1-methylbenzimidazol-2-yl]amino]methyl]-N-(2H-tetrazol-5-yl)benzamide
Show/Hide
|
C33H44N8O2
|
2
|
| 1 |
IC50 = 2 nM
|
|
|
| 2 |
IC50 = 19 nM
|
|
|
|
CP0380120
|
3-[[4-[1-[3-(2-carbamoyl-5-chlorophenyl)-6-[4-(trifluoromethoxy)phenyl]indazol-1-yl]ethyl]benzoyl]amino]propanoic acid
Show/Hide
|
C33H26ClF3N4O5
|
2
|
| 1 |
IC50 = 2 nM
|
|
|
| 2 |
IC50 = 220 nM
|
|
|
|
CP0545448
|
3-[[4-[1-[3-[2-methoxy-5-(trifluoromethyl)phenyl]-6-(4-methylphenyl)indazol-1-yl]butyl]benzoyl]amino]propanoic acid
Show/Hide
|
C36H34F3N3O4
|
2
|
| 1 |
IC50 = 2 nM
|
|
|
| 2 |
IC50 = 5 nM
|
|
|
|
CP0666275
|
4-((2-(4-tert-butylphenylimino)-3-methyl-4-propoxy-6-(trifluoromethyl)-2,3-dihydro-1H-benzo[d]imidazol-1-yl)methyl)-N-(1H-tetrazol-5-yl)benzamide
Show/Hide
|
C31H33F3N8O2
|
2
|
| 1 |
IC50 = 2.2 nM
|
|
|
| 2 |
IC50 = 13 nM
|
|
|
|
CP0513287
|
3-[[4-[(1S)-1-[3-(3,5-dichlorophenyl)-5-[6-(trifluoromethoxy)naphthalen-2-yl]pyrazol-1-yl]ethyl]benzoyl]amino]propanoic acid
Show/Hide
|
C32H24Cl2F3N3O4
|
2
|
| 1 |
IC50 = 2.5 nM
|
|
|
| 2 |
IC50 = 11.9 nM
|
|
|
|
CP0041074
|
3-[[4-[1-[3-[2-methoxy-5-(trifluoromethyl)phenyl]-6-(4-methylphenyl)indazol-1-yl]pentyl]benzoyl]amino]propanoic acid
Show/Hide
|
C37H36F3N3O4
|
2
|
| 1 |
IC50 = 2.6 nM
|
|
|
| 2 |
IC50 = 6.6 nM
|
|
|
|
CP0449415
|
3-[[4-[1-[3-[2-methoxy-5-(trifluoromethyl)phenyl]-6-(4-methylphenyl)indazol-1-yl]ethyl]benzoyl]amino]propanoic acid
Show/Hide
|
C34H30F3N3O4
|
2
|
| 1 |
IC50 = 2.6 nM
|
|
|
| 2 |
IC50 = 7.6 nM
|
|
|
|
CP0897011
|
4-((4-ethoxy-3-methyl-2-(4-(trifluoromethoxy)phenylimino)-6-(trifluoromethyl)-2,3-dihydro-1H-benzo[d]imidazol-1-yl)methyl)-N-(1H-tetrazol-5-yl)benzamide
Show/Hide
|
C27H22F6N8O3
|
2
|
| 1 |
IC50 = 2.8 nM
|
|
|
| 2 |
IC50 = 14.4 nM
|
|
|
|
CP0222546
|
4-[5-(4-Chloro-phenyl)-3-(2-isobutoxy-phenyl)-1H-pyrrol-2-yl]-pyridine
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|
C25H23ClN2O
|
2
|
| 1 |
IC50 = 3 nM
|
|
|
| 2 |
IC50 = 200 nM
|
|
|
|
CP0415829
|
3-[[4-[1-[3-[2-methoxy-5-(trifluoromethyl)phenyl]-6-phenylindazol-1-yl]pentyl]benzoyl]amino]propanoic acid
Show/Hide
|
C36H34F3N3O4
|
2
|
| 1 |
IC50 = 3 nM
|
|
|
| 2 |
IC50 = 18 nM
|
|
|
|
CP0445176
|
3-[[4-[1-[3-[3-chloro-5-(trifluoromethyl)phenyl]-6-[4-(trifluoromethoxy)phenyl]indazol-1-yl]ethyl]benzoyl]amino]propanoic acid
Show/Hide
|
C33H24ClF6N3O4
|
2
|
| 1 |
IC50 = 3 nM
|
|
|
| 2 |
IC50 = 56 nM
|
|
|
|
CP0570522
|
3-[[4-[1-[3-(5-chloro-2-methoxyphenyl)-6-[4-(trifluoromethoxy)phenyl]indazol-1-yl]ethyl]benzoyl]amino]propanoic acid
Show/Hide
|
C33H27ClF3N3O5
|
2
|
| 1 |
IC50 = 3 nM
|
|
|
| 2 |
IC50 = 36 nM
|
|
|
|
CP0851785
|
4-((4-butoxy-3-methyl-2-(4-(trifluoromethoxy)phenylimino)-6-(trifluoromethyl)-2,3-dihydro-1H-benzo[d]imidazol-1-yl)methyl)-N-(1H-tetrazol-5-yl)benzamide
Show/Hide
|
C29H26F6N8O3
|
2
|
| 1 |
IC50 = 3.1 nM
|
|
|
| 2 |
IC50 = 28 nM
|
|
|
|
CP0464681
|
4-[1-(4-tert-Butyl-cyclohexyl)-3-(4-trifluoromethoxy-phenyl)-ureidomethyl]-N-(1H-tetrazol-5-yl)-benzamide
Show/Hide
|
C27H32F3N7O3
|
2
|
| 1 |
IC50 = 3.2 nM
|
|
|
| 2 |
IC50 = 46 nM
|
|
|
|
CP0436930
|
4-[[(4-tert-butylcyclohexyl)-[[4-(trifluoromethoxy)phenyl]carbamoyl]amino]methyl]-N-(2H-tetrazol-5-yl)benzamide
Show/Hide
|
C27H32F3N7O3
|
2
|
| 1 |
IC50 = 3.2 nM
|
|
|
| 2 |
IC50 = 46 nM
|
|
|
|
CP0445218
|
3-[[4-[1-[6-(6-methoxypyridin-3-yl)-3-[2-methoxy-5-(trifluoromethyl)phenyl]indazol-1-yl]pentyl]benzoyl]amino]propanoic acid
Show/Hide
|
C36H35F3N4O5
|
2
|
| 1 |
IC50 = 3.4 nM
|
|
|
| 2 |
IC50 = 24 nM
|
|
|
|
CP0415790
|
3-[[4-[1-[3-[2-methoxy-5-(trifluoromethyl)phenyl]-6-(3,4,5-trifluorophenyl)indazol-1-yl]pentyl]benzoyl]amino]propanoic acid
Show/Hide
|
C36H31F6N3O4
|
2
|
| 1 |
IC50 = 3.5 nM
|
|
|
| 2 |
IC50 = 26 nM
|
|
|
|
CP0502906
|
4-[3-(4-Bromo-2-propoxy-phenyl)-5-(4-chloro-phenyl)-1H-pyrrol-2-yl]-pyridine
Show/Hide
|
C24H20BrClN2O
|
2
|
| 1 |
IC50 = 4 nM
|
|
|
| 2 |
IC50 = 130 nM
|
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|
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CP0265770
|
4-[[(4-tert-butylcyclohexyl)-(6-methoxy-1-methylbenzimidazol-2-yl)amino]methyl]-N-(2H-tetrazol-5-yl)benzamide
Show/Hide
|
C28H36N8O2
|
2
|
| 1 |
IC50 = 4 nM
|
|
|
| 2 |
IC50 = 213 nM
|
|
|
|
CP0333819
|
4-[[(4-tert-butylcyclohexyl)-(5-methoxy-1-methylbenzimidazol-2-yl)amino]methyl]-N-(2H-tetrazol-5-yl)benzamide
Show/Hide
|
C28H36N8O2
|
2
|
| 1 |
IC50 = 4 nM
|
|
|
| 2 |
IC50 = 38 nM
|
|
|
|
CP0401075
|
4-[[(4-tert-butylcyclohexyl)-(1-methylbenzimidazol-2-yl)amino]methyl]-N-(2H-tetrazol-5-yl)benzamide
Show/Hide
|
C27H34N8O
|
2
|
| 1 |
IC50 = 4 nM
|
|
|
| 2 |
IC50 = 55 nM
|
|
|
|
CP0892635
|
4-((5,6-dichloro-3-methyl-2-(4-(trifluoromethoxy)phenylimino)-2,3-dihydro-1H-benzo[d]imidazol-1-yl)methyl)-N-(1H-tetrazol-5-yl)benzamide
Show/Hide
|
C24H17Cl2F3N8O2
|
2
|
| 1 |
IC50 = 4 nM
|
|
|
| 2 |
IC50 = 23 nM
|
|
|
|
CP0442612
|
4-[(1R)-1-[8-tert-butyl-2-(3,5-dichlorophenyl)-3-oxo-1,4-diazaspiro[4.5]dec-1-en-4-yl]-4,4,4-trifluorobutyl]-N-(2H-tetrazol-5-ylmethyl)benzamide
Show/Hide
|
C31H34Cl2F3N7O2
|
2
|
| 1 |
IC50 = 4 nM
|
|
|
| 2 |
IC50 = 370 nM
|
|
|
|
CP0380118
|
3-[[4-[1-[3-(4,5-difluoro-2-methoxyphenyl)-6-[4-(trifluoromethoxy)phenyl]indazol-1-yl]ethyl]benzoyl]amino]propanoic acid
Show/Hide
|
C33H26F5N3O5
|
2
|
| 1 |
IC50 = 4 nM
|
|
|
| 2 |
IC50 = 37 nM
|
|
|
|
CP0406415
|
3-[[4-[1-[3-[2-methoxy-5-(trifluoromethyl)phenyl]-6-(4-methylphenyl)indazol-1-yl]-2-methylpropyl]benzoyl]amino]propanoic acid
Show/Hide
|
C36H34F3N3O4
|
2
|
| 1 |
IC50 = 4 nM
|
|
|
| 2 |
IC50 = 69 nM
|
|
|
|
CP0415828
|
3-[[4-[1-[3-[2-methoxy-5-(trifluoromethyl)phenyl]-6-(4-methylphenyl)indol-1-yl]butyl]benzoyl]amino]propanoic acid
Show/Hide
|
C37H35F3N2O4
|
2
|
| 1 |
IC50 = 4 nM
|
|
|
| 2 |
IC50 = 48 nM
|
|
|
|
CP0456653
|
3-[[4-[1-[3-[2-methoxy-5-(trifluoromethyl)phenyl]-6-(5-methylthiophen-2-yl)indazol-1-yl]pentyl]benzoyl]amino]propanoic acid
Show/Hide
|
C35H34F3N3O4S
|
2
|
| 1 |
IC50 = 4 nM
|
|
|
| 2 |
IC50 = 18 nM
|
|
|
|
CP0471990
|
3-[[4-[1-[6-(4-methoxyphenyl)-3-[2-methoxy-5-(trifluoromethyl)phenyl]indazol-1-yl]butyl]benzoyl]amino]propanoic acid
Show/Hide
|
C36H34F3N3O5
|
2
|
| 1 |
IC50 = 4 nM
|
|
|
| 2 |
IC50 = 11 nM
|
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|
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CP0539366
|
3-[[4-[1-[6-(2-chloro-4-methoxyphenyl)-3-[2-methoxy-5-(trifluoromethyl)phenyl]indazol-1-yl]pentyl]benzoyl]amino]propanoic acid
Show/Hide
|
C37H35ClF3N3O5
|
2
|
| 1 |
IC50 = 4 nM
|
|
|
| 2 |
IC50 = 18 nM
|
|
|
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CP0545455
|
3-[[4-[1-[3-(4-chloro-3-fluorophenyl)-6-[4-(trifluoromethoxy)phenyl]indazol-1-yl]ethyl]benzoyl]amino]propanoic acid
Show/Hide
|
C32H24ClF4N3O4
|
2
|
| 1 |
IC50 = 4 nM
|
|
|
| 2 |
IC50 = 44 nM
|
|
|
|
CP0545456
|
3-[[4-[1-[3-[2-methoxy-5-(trifluoromethyl)phenyl]-6-(4-methylphenyl)indazol-1-yl]propyl]benzoyl]amino]propanoic acid
Show/Hide
|
C35H32F3N3O4
|
2
|
| 1 |
IC50 = 4 nM
|
|
|
| 2 |
IC50 = 21 nM
|
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|
|
CP0446813
|
3-[[4-[(1S)-1-[3-[2-fluoro-5-(trifluoromethyl)phenyl]-5-(6-methoxynaphthalen-2-yl)pyrazol-1-yl]ethyl]benzoyl]amino]propanoic acid
Show/Hide
|
C33H27F4N3O4
|
2
|
| 1 |
IC50 = 4.1 nM
|
|
|
| 2 |
IC50 = 12.3 nM
|
|
|
|
CP0435866
|
3-[[4-[(1S)-1-[3-(3,5-dichlorophenyl)-5-(6-propan-2-ylnaphthalen-2-yl)pyrazol-1-yl]ethyl]benzoyl]amino]propanoic acid
Show/Hide
|
C34H31Cl2N3O3
|
2
|
| 1 |
IC50 = 4.3 nM
|
|
|
| 2 |
IC50 = 13.3 nM
|
|
|
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CP0932444
|
4-((2-(4-tert-butylphenylimino)-4-ethyl-3-methyl-6-(trifluoromethyl)-2,3-dihydro-1H-benzo[d]imidazol-1-yl)methyl)-N-(1H-tetrazol-5-yl)benzamide
Show/Hide
|
C30H31F3N8O
|
2
|
| 1 |
IC50 = 4.4 nM
|
|
|
| 2 |
IC50 = 17 nM
|
|
|
|
CP0359788
|
3-[[4-[(1S)-1-[3-(3,5-dichlorophenyl)-5-(6-methylnaphthalen-2-yl)pyrazol-1-yl]ethyl]benzoyl]amino]propanoic acid
Show/Hide
|
C32H27Cl2N3O3
|
2
|
| 1 |
IC50 = 4.6 nM
|
|
|
| 2 |
IC50 = 7.5 nM
|
|
|
|
CP0480311
|
1-(N-((1r,4r)-4-tert-butylcyclohexyl)-2-(4-(trifluoromethoxy)phenyl)acetamido)-N-(2H-tetrazol-5-yl)-2,3-dihydro-1H-indene-5-carboxamide
Show/Hide
|
C30H35F3N6O3
|
2
|
| 1 |
IC50 = 4.8 nM
|
|
|
| 2 |
IC50 = 67 nM
|
|
|
|
CP0480310
|
1-(5-((2H-tetrazol-5-yl)carbamoyl)-2,3-dihydro-1H-inden-1-yl)-1-((1r,4r)-4-tert-butylcyclohexyl)-3-(3,5-dichlorophenyl)urea
Show/Hide
|
C28H33Cl2N7O2
|
2
|
| 1 |
IC50 = 4.9 nM
|
|
|
| 2 |
IC50 = 5.9 nM
|
|
|
|
CP0486551
|
3-[[4-[1-[3-[2-fluoro-5-(trifluoromethyl)phenyl]-6-[4-(trifluoromethoxy)phenyl]indazol-1-yl]ethyl]benzoyl]amino]propanoic acid
Show/Hide
|
C33H24F7N3O4
|
2
|
| 1 |
IC50 = 5 nM
|
|
|
| 2 |
IC50 = 120 nM
|
|
|
|
CP0495580
|
3-[[4-[(1S)-1-[3-(3,4-dichlorophenyl)-5-(6-methoxynaphthalen-2-yl)pyrazol-1-yl]ethyl]benzoyl]amino]propanoic acid
Show/Hide
|
C32H27Cl2N3O4
|
2
|
| 1 |
IC50 = 5.2 nM
|
|
|
| 2 |
IC50 = 15.8 nM
|
|
|
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CP0452401
|
3-[[4-[(2S)-2-[5-(trifluoromethoxy)-1-[3-(trifluoromethyl)phenyl]indole-2-carbonyl]heptyl]benzoyl]amino]propanoic acid
Show/Hide
|
C34H32F6N2O5
|
2
|
| 1 |
IC50 = 5.7 nM
|
|
|
| 2 |
IC50 = 17 nM
|
|
|
|
CP0380783
|
4-[5-(4-Chloro-phenyl)-3-(5-chloro-2-propoxy-phenyl)-1H-pyrrol-2-yl]-pyridine
Show/Hide
|
C24H20Cl2N2O
|
2
|
| 1 |
IC50 = 6 nM
|
|
|
| 2 |
IC50 = 170 nM
|
|
|
|
CP0265769
|
4-[[(4-tert-butylcyclohexyl)-(5-fluoro-1-methylbenzimidazol-2-yl)amino]methyl]-N-(2H-tetrazol-5-yl)benzamide
Show/Hide
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C27H33FN8O
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2
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| 1 |
IC50 = 6 nM
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| 2 |
IC50 = 220 nM
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CP0333818
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4-[[(4-tert-butylcyclohexyl)-(1,5,6-trimethylbenzimidazol-2-yl)amino]methyl]-N-(2H-tetrazol-5-yl)benzamide
Show/Hide
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C29H38N8O
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2
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| 1 |
IC50 = 6 nM
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| 2 |
IC50 = 18 nM
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CP0669683
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4-((3-methyl-4-propoxy-6-(trifluoromethyl)-2-(4-(trifluoromethyl)phenylimino)-2,3-dihydro-1H-benzo[d]imidazol-1-yl)methyl)-N-(1H-tetrazol-5-yl)benzamide
Show/Hide
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C28H24F6N8O2
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2
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| 1 |
IC50 = 6 nM
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| 2 |
IC50 = 14 nM
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CP0488510
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CHEMBL3237900
Show/Hide
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C30H35ClFN3O4
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2
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| 1 |
IC50 = 6 nM
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| 2 |
IC50 = 110 nM
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CP0445217
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3-[[4-[1-[6-[4-(trifluoromethoxy)phenyl]-3-(3,4,5-trifluorophenyl)indazol-1-yl]ethyl]benzoyl]amino]propanoic acid
Show/Hide
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C32H23F6N3O4
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2
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| 1 |
IC50 = 6 nM
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| 2 |
IC50 = 20 nM
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CP0120350
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3-[[4-[(1S)-1-[3-(3,5-dichlorophenyl)-5-(6-methoxynaphthalen-2-yl)pyrazol-1-yl]ethyl]benzoyl]amino]propanoic acid
Show/Hide
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C32H27Cl2N3O4
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2
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| 1 |
IC50 = 6.6 nM
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| 2 |
IC50 = 15.7 nM
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CP0446805
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3-[[4-[(1S)-1-[3-(3-chloro-5-propoxyphenyl)-5-(6-methoxynaphthalen-2-yl)pyrazol-1-yl]ethyl]benzoyl]amino]propanoic acid
Show/Hide
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C35H34ClN3O5
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2
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| 1 |
IC50 = 6.9 nM
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| 2 |
IC50 = 47.2 nM
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CP0039137
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4-[3-(5-Bromo-2-propoxy-phenyl)-5-(4-chloro-phenyl)-1H-pyrrol-2-yl]-pyridine
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C24H20BrClN2O
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2
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| 1 |
IC50 = 7 nM
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| 2 |
IC50 = 170 nM
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CP0043111
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4-[[(5-bromo-1-methylbenzimidazol-2-yl)-(4-tert-butylcyclohexyl)amino]methyl]-N-(2H-tetrazol-5-yl)benzamide
Show/Hide
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C27H33BrN8O
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2
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| 1 |
IC50 = 7 nM
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| 2 |
IC50 = 62 nM
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CP0715176
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4-((3-methyl-4-propoxy-2-(3-(trifluoromethoxy)phenylimino)-6-(trifluoromethyl)-2,3-dihydro-1H-benzo[d]imidazol-1-yl)methyl)-N-(1H-tetrazol-5-yl)benzamide
Show/Hide
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C28H24F6N8O3
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2
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| 1 |
IC50 = 7 nM
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| 2 |
IC50 = 18 nM
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CP0894249
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4-((4-butoxy-6-chloro-3-methyl-2-(4-(trifluoromethoxy)phenylimino)-2,3-dihydro-1H-benzo[d]imidazol-1-yl)methyl)-N-(1H-tetrazol-5-yl)benzamide
Show/Hide
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C28H26ClF3N8O3
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2
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| 1 |
IC50 = 7 nM
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| 2 |
IC50 = 25 nM
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CP0904769
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4-((6-chloro-4-ethoxy-3-methyl-2-(4-(trifluoromethoxy)phenylimino)-2,3-dihydro-1H-benzo[d]imidazol-1-yl)methyl)-N-(1H-tetrazol-5-yl)benzamide
Show/Hide
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C26H22ClF3N8O3
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2
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| 1 |
IC50 = 7 nM
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| 2 |
IC50 = 19 nM
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CP0513181
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4-[(1R)-1-[8-tert-butyl-3-oxo-2-[4-(trifluoromethyl)phenyl]-1,4-diazaspiro[4.5]dec-1-en-4-yl]-4,4-dimethylpentyl]-N-(2H-tetrazol-5-ylmethyl)benzamide
Show/Hide
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C35H44F3N7O2
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2
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| 1 |
IC50 = 7 nM
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| 2 |
IC50 = 160 nM
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CP0374638
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3-[[4-[1-[6-(3-chloro-5-fluorophenyl)-3-[2-methoxy-5-(trifluoromethyl)phenyl]indazol-1-yl]pentyl]benzoyl]amino]propanoic acid
Show/Hide
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C36H32ClF4N3O4
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2
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| 1 |
IC50 = 7 nM
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| 2 |
IC50 = 46 nM
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CP0445175
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3-[[4-[1-[6-[4-(trifluoromethoxy)phenyl]-3-(2,3,5-trifluorophenyl)indazol-1-yl]ethyl]benzoyl]amino]propanoic acid
Show/Hide
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C32H23F6N3O4
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2
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| 1 |
IC50 = 7 nM
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| 2 |
IC50 = 52 nM
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CP0534733
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3-[[4-[1-[3-[2-methoxy-5-(trifluoromethoxy)phenyl]-6-[4-(trifluoromethoxy)phenyl]indazol-1-yl]ethyl]benzoyl]amino]propanoic acid
Show/Hide
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C34H27F6N3O6
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2
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| 1 |
IC50 = 7 nM
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| 2 |
IC50 = 11 nM
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CP0545454
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3-[[4-[1-[3-[2-methoxy-5-(trifluoromethyl)phenyl]-5-(4-methylphenyl)indazol-1-yl]butyl]benzoyl]amino]propanoic acid
Show/Hide
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C36H34F3N3O4
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2
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| 1 |
IC50 = 7 nM
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| 2 |
IC50 = 17 nM
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CP0352696
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3-[[4-[(1S)-1-[3-(2,5-dichlorophenyl)-5-(6-methoxynaphthalen-2-yl)pyrazol-1-yl]ethyl]benzoyl]amino]propanoic acid
Show/Hide
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C32H27Cl2N3O4
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2
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| 1 |
IC50 = 7.5 nM
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| 2 |
IC50 = 11.5 nM
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CP0426097
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3-[[4-[(1S)-1-[5-(6-chloronaphthalen-2-yl)-3-(3,5-dichlorophenyl)pyrazol-1-yl]ethyl]benzoyl]amino]propanoic acid
Show/Hide
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C31H24Cl3N3O3
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2
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| 1 |
IC50 = 7.5 nM
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| 2 |
IC50 = 12.5 nM
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CP0462756
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1-(5-((2H-tetrazol-5-yl)carbamoyl)-2,3-dihydro-1H-inden-1-yl)-3-(3,5-bis(trifluoromethyl)phenyl)-1-((1r,4r)-4-tert-butylcyclohexyl)urea
Show/Hide
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C30H33F6N7O2
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2
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| 1 |
IC50 = 7.6 nM
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| 2 |
IC50 = 61 nM
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CP0920306
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4-((2-(4-fluoro-3-(trifluoromethyl)phenylimino)-3-methyl-4-propoxy-6-(trifluoromethyl)-2,3-dihydro-1H-benzo[d]imidazol-1-yl)methyl)-N-(1H-tetrazol-5-yl)benzamide
Show/Hide
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C28H23F7N8O2
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2
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| 1 |
IC50 = 7.7 nM
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| 2 |
IC50 = 14 nM
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CP0222548
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4-[5-(4-Chloro-phenyl)-3-(2-propoxy-phenyl)-1H-pyrrol-2-yl]-pyridine
Show/Hide
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C24H21ClN2O
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2
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| 1 |
IC50 = 8 nM
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| 2 |
IC50 = 140 nM
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CP0449433
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3-[[4-[1-[3-(2,4-difluorophenyl)-6-[4-(trifluoromethoxy)phenyl]indazol-1-yl]ethyl]benzoyl]amino]propanoic acid
Show/Hide
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C32H24F5N3O4
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2
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| 1 |
IC50 = 8 nM
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| 2 |
IC50 = 41 nM
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CP0534732
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3-[[4-[1-[6-(4-methoxyphenyl)-3-[2-methoxy-5-(trifluoromethyl)phenyl]indol-1-yl]butyl]benzoyl]amino]propanoic acid
Show/Hide
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C37H35F3N2O5
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2
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| 1 |
IC50 = 8 nM
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| 2 |
IC50 = 130 nM
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CP0446171
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3-[[4-[[3-(3,5-dichlorophenyl)-5-[6-(trifluoromethoxy)naphthalen-2-yl]pyrazol-1-yl]methyl]benzoyl]amino]propanoic acid
Show/Hide
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C31H22Cl2F3N3O4
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2
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| 1 |
IC50 = 8.1 nM
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| 2 |
IC50 = 30.2 nM
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CP0492140
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3-[[4-[(1S)-1-[3-(3,5-dichlorophenyl)-5-(6-ethoxynaphthalen-2-yl)pyrazol-1-yl]ethyl]benzoyl]amino]propanoic acid
Show/Hide
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C33H29Cl2N3O4
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2
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| 1 |
IC50 = 8.1 nM
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| 2 |
IC50 = 23.6 nM
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CP0715177
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4-((6-chloro-3-methyl-4-propoxy-2-(4-(trifluoromethoxy)phenylimino)-2,3-dihydro-1H-benzo[d]imidazol-1-yl)methyl)-N-(1H-tetrazol-5-yl)benzamide
Show/Hide
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C27H24ClF3N8O3
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2
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| 1 |
IC50 = 8.3 nM
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| 2 |
IC50 = 19 nM
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CP0904768
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4-((4-methoxy-3-methyl-2-(4-(trifluoromethoxy)phenylimino)-6-(trifluoromethyl)-2,3-dihydro-1H-benzo[d]imidazol-1-yl)methyl)-N-(1H-tetrazol-5-yl)benzamide
Show/Hide
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C26H20F6N8O3
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2
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| 1 |
IC50 = 8.3 nM
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| 2 |
IC50 = 41 nM
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CP0170482
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4-[[(4-tert-butylcyclohexyl)-(5,6-dichloro-1-methylbenzimidazol-2-yl)amino]methyl]-N-(2H-tetrazol-5-yl)benzamide
Show/Hide
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C27H32Cl2N8O
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2
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| 1 |
IC50 = 9 nM
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| 2 |
IC50 = 23 nM
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CP0401073
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4-(((4-cyclohexylphenyl)(1-methyl-1H-benzo[d]imidazol-2-yl)amino)methyl)-N-(1H-tetrazol-5-yl)benzamide
Show/Hide
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C29H30N8O
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2
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| 1 |
IC50 = 9 nM
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| 2 |
IC50 = 28 nM
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CP0496123
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3-[[4-[(2S)-2-[5-chloro-1-[6-(trifluoromethyl)pyridin-2-yl]indole-2-carbonyl]pentyl]benzoyl]amino]propanoic acid
Show/Hide
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C30H27ClF3N3O4
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2
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| 1 |
IC50 = 9.2 nM
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| 2 |
IC50 = 34 nM
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CP0895597
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4-((6-chloro-4-isopropoxy-3-methyl-2-(4-(trifluoromethoxy)phenylimino)-2,3-dihydro-1H-benzo[d]imidazol-1-yl)methyl)-N-(1H-tetrazol-5-yl)benzamide
Show/Hide
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C27H24ClF3N8O3
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2
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| 1 |
IC50 = 9.3 nM
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| 2 |
IC50 = 29 nM
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CP0446169
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3-[[4-[(1S)-1-[5-(6-methoxynaphthalen-2-yl)-3-[2-methyl-5-(trifluoromethyl)phenyl]pyrazol-1-yl]ethyl]benzoyl]amino]propanoic acid
Show/Hide
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C34H30F3N3O4
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2
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| 1 |
IC50 = 9.3 nM
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| 2 |
IC50 = 27.4 nM
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CP0376681
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4-[3-(2-Butoxy-phenyl)-5-(4-chloro-phenyl)-1H-pyrrol-2-yl]-pyridine
Show/Hide
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C25H23ClN2O
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2
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| 1 |
IC50 = 10 nM
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| 2 |
IC50 = 180 nM
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CP0467127
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3-(1-(1-((1r,4r)-4-tert-butylcyclohexyl)-3-(3,5-dichlorophenyl)ureido)-2,3-dihydro-1H-indene-5-carboxamido)propanoic acid
Show/Hide
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C30H37Cl2N3O4
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2
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| 1 |
IC50 = 10 nM
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| 2 |
IC50 = 11 nM
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CP0432392
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4-[[(4-tert-butylcyclohexyl)-(6-methyl-1H-benzimidazol-2-yl)amino]methyl]-N-(2H-tetrazol-5-yl)benzamide
Show/Hide
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C27H34N8O
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2
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| 1 |
IC50 = 10 nM
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| 2 |
IC50 > 1000 nM
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CP0268151
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3-[[4-[(2S)-2-[5-chloro-1-[3-(trifluoromethyl)phenyl]indole-2-carbonyl]heptyl]benzoyl]amino]propanoic acid
Show/Hide
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C33H32ClF3N2O4
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2
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| 1 |
IC50 = 10 nM
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| 2 |
IC50 = 12 nM
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CP0452400
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3-[[4-[(2S)-2-[5-fluoro-1-[3-(trifluoromethyl)phenyl]indole-2-carbonyl]heptyl]benzoyl]amino]propanoic acid
Show/Hide
|
C33H32F4N2O4
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2
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| 1 |
IC50 = 10 nM
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| 2 |
IC50 = 20 nM
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CP0513140
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4-[(1R)-1-[8-tert-butyl-2-(3-chloro-5-fluorophenyl)-3-oxo-1,4-diazaspiro[4.5]dec-1-en-4-yl]-4,4-dimethylpentyl]-N-(2H-tetrazol-5-ylmethyl)benzamide
Show/Hide
|
C34H43ClFN7O2
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2
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| 1 |
IC50 = 10 nM
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| 2 |
IC50 = 42 nM
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CP0380119
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3-[[4-[1-[3-(2-chloro-5-fluorophenyl)-6-[4-(trifluoromethoxy)phenyl]indazol-1-yl]ethyl]benzoyl]amino]propanoic acid
Show/Hide
|
C32H24ClF4N3O4
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2
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| 1 |
IC50 = 10 nM
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| 2 |
IC50 = 140 nM
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CP0474753
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3-[[4-[1-[5-(4-methoxyphenyl)-3-[2-methoxy-5-(trifluoromethyl)phenyl]indazol-1-yl]butyl]benzoyl]amino]propanoic acid
Show/Hide
|
C36H34F3N3O5
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2
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| 1 |
IC50 = 10 nM
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| 2 |
IC50 = 26 nM
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CP0179650
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3-[[4-[(1S)-1-[3-(3,5-dichlorophenyl)-5-[6-(trifluoromethyl)naphthalen-2-yl]pyrazol-1-yl]ethyl]benzoyl]amino]propanoic acid
Show/Hide
|
C32H24Cl2F3N3O3
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2
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| 1 |
IC50 = 10.7 nM
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| 2 |
IC50 = 14.1 nM
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CP0140059
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4-[[(4-tert-butylcyclohexyl)-[1-methyl-5-(trifluoromethyl)benzimidazol-2-yl]amino]methyl]-N-(2H-tetrazol-5-yl)benzamide
Show/Hide
|
C28H33F3N8O
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2
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| 1 |
IC50 = 11 nM
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| 2 |
IC50 = 62 nM
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CP0894522
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4-((4-ethyl-3-methyl-2-(4-(trifluoromethoxy)phenylimino)-6-(trifluoromethyl)-2,3-dihydro-1H-benzo[d]imidazol-1-yl)methyl)-N-(1H-tetrazol-5-yl)benzamide
Show/Hide
|
C27H22F6N8O2
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2
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| 1 |
IC50 = 11 nM
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| 2 |
IC50 = 22 nM
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CP0452403
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3-[[4-[(2S)-2-[5-methyl-1-[3-(trifluoromethyl)phenyl]indole-2-carbonyl]heptyl]benzoyl]amino]propanoic acid
Show/Hide
|
C34H35F3N2O4
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2
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| 1 |
IC50 = 12 nM
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| 2 |
IC50 = 24 nM
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CP0492655
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3-[[4-[2-[5-chloro-1-[4-chloro-3-(trifluoromethyl)phenyl]indole-2-carbonyl]pentyl]benzoyl]amino]propanoic acid
Show/Hide
|
C31H27Cl2F3N2O4
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2
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| 1 |
IC50 = 12 nM
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| 2 |
IC50 = 17 nM
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CP0899733
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4-((6-chloro-4-methoxy-3-methyl-2-(4-(trifluoromethoxy)phenylimino)-2,3-dihydro-1H-benzo[d]imidazol-1-yl)methyl)-N-(1H-tetrazol-5-yl)benzamide
Show/Hide
|
C25H20ClF3N8O3
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2
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| 1 |
IC50 = 12 nM
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| 2 |
IC50 = 73 nM
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CP0445173
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3-[[4-[1-[3-[2-methoxy-5-(trifluoromethyl)phenyl]-6-[4-(trifluoromethoxy)phenyl]pyrrolo[2,3-b]pyridin-1-yl]butyl]benzoyl]amino]propanoic acid
Show/Hide
|
C36H31F6N3O5
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2
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| 1 |
IC50 = 12 nM
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| 2 |
IC50 = 360 nM
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CP0475035
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4-(((3-chloro-4-(4-chlorophenoxy)phenyl)(5-methyl-1H-benzo[d]imidazol-2-yl)amino)methyl)-N-(1H-tetrazol-5-yl)benzamide
Show/Hide
|
C29H22Cl2N8O2
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2
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| 1 |
IC50 = 13 nM
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| 2 |
IC50 > 1000 nM
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CP0853680
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4-((3-methyl-2-(4-(trifluoromethoxy)phenylimino)-6-(trifluoromethyl)-2,3-dihydro-1H-benzo[d]imidazol-1-yl)methyl)-N-(1H-tetrazol-5-yl)benzamide
Show/Hide
|
C25H18F6N8O2
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2
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| 1 |
IC50 = 13 nM
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| 2 |
IC50 = 49 nM
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CP0383830
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4-[(1R)-1-[8-tert-butyl-2-(3,4-difluorophenyl)-3-oxo-1,4-diazaspiro[4.5]dec-1-en-4-yl]-4,4-dimethylpentyl]-N-(2H-tetrazol-5-ylmethyl)benzamide
Show/Hide
|
C34H43F2N7O2
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2
|
| 1 |
IC50 = 13 nM
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| 2 |
IC50 = 180 nM
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CP0395568
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4-[(1R)-1-[8-tert-butyl-3-oxo-2-[3-(trifluoromethyl)phenyl]-1,4-diazaspiro[4.5]dec-1-en-4-yl]-4,4-dimethylpentyl]-N-(2H-tetrazol-5-ylmethyl)benzamide
Show/Hide
|
C35H44F3N7O2
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2
|
| 1 |
IC50 = 13 nM
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| 2 |
IC50 = 180 nM
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CP0411247
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4-[(1R)-1-[8-tert-butyl-2-(4-fluorophenyl)-3-oxo-1,4-diazaspiro[4.5]dec-1-en-4-yl]-4,4-dimethylpentyl]-N-(2H-tetrazol-5-ylmethyl)benzamide
Show/Hide
|
C34H44FN7O2
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2
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| 1 |
IC50 = 13 nM
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| 2 |
IC50 = 240 nM
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CP0461394
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(2R)-3-[[4-[[(4-tert-butylcyclohexyl)-(1-methylbenzimidazol-2-yl)amino]methyl]benzoyl]amino]-2-hydroxypropanoic acid
Show/Hide
|
C29H38N4O4
|
2
|
| 1 |
IC50 = 14 nM
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| 2 |
IC50 > 1000 nM
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CP0912382
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4-((3-methyl-2-(4-methyl-3-(trifluoromethyl)phenylimino)-4-propoxy-6-(trifluoromethyl)-2,3-dihydro-1H-benzo[d]imidazol-1-yl)methyl)-N-(1H-tetrazol-5-yl)benzamide
Show/Hide
|
C29H26F6N8O2
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2
|
| 1 |
IC50 = 14 nM
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| 2 |
IC50 = 19 nM
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CP0917424
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4-((5,6-dichloro-3-propyl-2-(4-(trifluoromethoxy)phenylimino)-2,3-dihydro-1H-benzo[d]imidazol-1-yl)methyl)-N-(1H-tetrazol-5-yl)benzamide
Show/Hide
|
C26H21Cl2F3N8O2
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2
|
| 1 |
IC50 = 14 nM
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| 2 |
IC50 = 61 nM
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CP0415753
|
CHEMBL3238218
Show/Hide
|
C34H44ClN7O2
|
2
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| 1 |
IC50 = 14 nM
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| 2 |
IC50 = 130 nM
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CP0446168
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3-[[4-[(1S)-1-[3-(3-chloro-5-methoxyphenyl)-5-(6-methoxynaphthalen-2-yl)pyrazol-1-yl]ethyl]benzoyl]amino]propanoic acid
Show/Hide
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C33H30ClN3O5
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2
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| 1 |
IC50 = 14.8 nM
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| 2 |
IC50 = 67.9 nM
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CP0475034
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4-[[(4-tert-butylcyclohexyl)-(1,5-dimethylbenzimidazol-2-yl)amino]methyl]-N-(2H-tetrazol-5-yl)benzamide
Show/Hide
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C28H36N8O
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2
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| 1 |
IC50 = 15 nM
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| 2 |
IC50 = 71 nM
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CP0395567
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4-[(1R)-1-[8-tert-butyl-2-(3,5-dichlorophenyl)-3-oxo-1,4-diazaspiro[4.5]dec-1-en-4-yl]-3-methylbutyl]-N-(2H-tetrazol-5-ylmethyl)benzamide
Show/Hide
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C32H39Cl2N7O2
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2
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| 1 |
IC50 = 15 nM
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| 2 |
IC50 = 760 nM
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CP0415754
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4-[(1R)-1-[8-tert-butyl-2-(3-methoxyphenyl)-3-oxo-1,4-diazaspiro[4.5]dec-1-en-4-yl]-4,4-dimethylpentyl]-N-(2H-tetrazol-5-ylmethyl)benzamide
Show/Hide
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C35H47N7O3
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2
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| 1 |
IC50 = 15 nM
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| 2 |
IC50 = 230 nM
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CP0474754
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3-[[4-[1-[3-(4-cyanophenyl)-6-[4-(trifluoromethoxy)phenyl]indazol-1-yl]ethyl]benzoyl]amino]propanoic acid
Show/Hide
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C33H25F3N4O4
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2
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| 1 |
IC50 = 15 nM
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| 2 |
IC50 = 43 nM
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CP0435868
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3-[[4-[(1S)-1-[5-(6-methoxynaphthalen-2-yl)-3-(trifluoromethyl)pyrazol-1-yl]ethyl]benzoyl]amino]propanoic acid
Show/Hide
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C27H24F3N3O4
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2
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| 1 |
IC50 = 15.3 nM
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| 2 |
IC50 = 63.1 nM
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CP0462844
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3-[[4-[[3-(3,5-dichlorophenyl)-5-(6-methoxynaphthalen-2-yl)pyrazol-1-yl]methyl]benzoyl]amino]propanoic acid
Show/Hide
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C31H25Cl2N3O4
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2
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| 1 |
IC50 = 15.6 nM
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| 2 |
IC50 = 90.9 nM
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CP0401074
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4-[[(4-tert-butylcyclohexyl)-(1-ethylbenzimidazol-2-yl)amino]methyl]-N-(2H-tetrazol-5-yl)benzamide
Show/Hide
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C28H36N8O
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1
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| 1 |
IC50 = 16 nM
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CP0475036
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4-[[(1-benzylbenzimidazol-2-yl)-(4-tert-butylcyclohexyl)amino]methyl]-N-(2H-tetrazol-5-yl)benzamide
Show/Hide
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C33H38N8O
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1
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| 1 |
IC50 = 16 nM
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CP0401179
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3-[[4-[(2S)-2-[5-(trifluoromethyl)-1-[3-(trifluoromethyl)phenyl]indole-2-carbonyl]heptyl]benzoyl]amino]propanoic acid
Show/Hide
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C34H32F6N2O4
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2
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| 1 |
IC50 = 16 nM
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| 2 |
IC50 = 44 nM
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CP0452399
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3-[[4-[(2S)-2-[5-chloro-1-[3-(trifluoromethyl)phenyl]indole-2-carbonyl]hexyl]benzoyl]amino]propanoic acid
Show/Hide
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C32H30ClF3N2O4
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2
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| 1 |
IC50 = 16 nM
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| 2 |
IC50 = 42 nM
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CP0522177
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3-[[4-[2-[1-[(4-tert-butylphenyl)methyl]-5-chloroindole-2-carbonyl]pentyl]benzoyl]amino]propanoic acid
Show/Hide
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C35H39ClN2O4
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1
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| 1 |
IC50 = 16 nM
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CP0484448
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3-[[4-[1-[5-(3-chloro-4-propoxyphenyl)-3-(3,5-dichlorophenyl)pyrazol-1-yl]ethyl]benzoyl]amino]propanoic acid
Show/Hide
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C30H28Cl3N3O4
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2
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| 1 |
IC50 = 16 nM
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| 2 |
IC50 = 64.8 nM
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CP0513184
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3-[[4-[(1R)-1-[8-tert-butyl-2-(3,5-dichlorophenyl)-3-oxo-1,4-diazaspiro[4.5]dec-1-en-4-yl]-4,4-dimethylpentyl]benzoyl]amino]propanoic acid
Show/Hide
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C35H45Cl2N3O4
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2
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| 1 |
IC50 = 16 nM
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| 2 |
IC50 = 48 nM
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CP0446077
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3-[[4-[(1R)-1-[3-(3,5-dichlorophenyl)-5-[6-(trifluoromethoxy)naphthalen-2-yl]pyrazol-1-yl]ethyl]benzoyl]amino]propanoic acid
Show/Hide
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C32H24Cl2F3N3O4
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2
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| 1 |
IC50 = 16.6 nM
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| 2 |
IC50 = 32.6 nM
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CP0222547
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4-[3-(2-Allyloxy-phenyl)-5-(4-chloro-phenyl)-1H-pyrrol-2-yl]-pyridine
Show/Hide
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C24H19ClN2O
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2
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| 1 |
IC50 = 17 nM
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| 2 |
IC50 = 260 nM
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CP0431146
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3-[[4-[(2S)-2-[5-chloro-1-[3-(trifluoromethyl)phenyl]indole-2-carbonyl]-5-methylhexyl]benzoyl]amino]propanoic acid
Show/Hide
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C33H32ClF3N2O4
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2
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| 1 |
IC50 = 17 nM
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| 2 |
IC50 = 36 nM
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CP0496125
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3-[[4-[(2S)-2-[5-chloro-1-[3-(trifluoromethyl)phenyl]indole-2-carbonyl]pentyl]benzoyl]amino]propanoic acid
Show/Hide
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C31H28ClF3N2O4
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2
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| 1 |
IC50 = 17 nM
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| 2 |
IC50 = 55 nM
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CP0465688
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CHEMBL3238215
Show/Hide
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C34H41Cl2N7O2
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2
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| 1 |
IC50 = 17 nM
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| 2 |
IC50 = 100 nM
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CP0394196
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(4S)-5-[(2S)-1-[(2S)-1-[(2S)-6-amino-1-[(2S)-1-[(2S)-1-[(2S)-1-[(2S)-1-[(2S)-5-carbamimidamido-1-[(2S)-5-carbamimidamido-1-[(2S)-1-[(2S)-1-[(2S)-3-carboxy-1-[(2S)-1-[(2S)-1-[(2S)-1-[(2S)-1-[(2S)-1-[(2S)-1-[(2S)-1-[(2S,3R)-1,3-dihydroxy-1-iminobutan-2-yl]imino-1,4-dihydroxy-4-iminobutan-2-yl]imino-1-hydroxy-4-methylsulfanylbutan-2-yl]imino-1-hydroxy-4-methylpentan-2-yl]imino-1-hydroxy-3-(1H-indol-3-yl)propan-2-yl]imino-1,5-dihydroxy-5-iminopentan-2-yl]imino-1-hydroxy-3-methylbutan-2-yl]imino-1-hydroxy-3-phenylpropan-2-yl]imino-1-hydroxypropan-2-yl]imino-1,5-dihydroxy-5-iminopentan-2-yl]imino-1-hydroxypropan-2-yl]imino-1-hydroxypentan-2-yl]imino-1-hydroxypentan-2-yl]imino-1,3-dihydroxypropan-2-yl]imino-3-carboxy-1-hydroxypropan-2-yl]imino-1-hydroxy-4-methylpentan-2-yl]imino-1-hydroxy-3-(4-hydroxyphenyl)propan-2-yl]imino-1-hydroxyhexan-2-yl]imino-1,3-dihydroxypropan-2-yl]imino-1-hydroxy-3-(4-hydroxyphenyl)propan-2-yl]imino-4-[[(2S)-2-[[(2S,3R)-2-[[(2S)-2-[[(2S,3R)-2-[[2-[[(2S)-2-[[(2S)-1,3-dihydroxy-2-[[(2S)-1-hydroxy-3-(1H-imidazol-5-yl)-2-(methylamino)propylidene]amino]propylidene]amino]-1,5-dihydroxy-5-iminopentylidene]amino]-1-hydroxyethylidene]amino]-1,3-dihydroxybutylidene]amino]-1-hydroxy-3-phenylpropylidene]amino]-1,3-dihydroxybutylidene]amino]-1,3-dihydroxypropylidene]amino]-5-hydroxypentanoic acid
Show/Hide
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C155H230N44O48S
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1
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| 1 |
IC50 = 18 nM
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CP0888570
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4-((5,6-dichloro-3-ethyl-2-(4-(trifluoromethoxy)phenylimino)-2,3-dihydro-1H-benzo[d]imidazol-1-yl)methyl)-N-(1H-tetrazol-5-yl)benzamide
Show/Hide
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C25H19Cl2F3N8O2
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2
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| 1 |
IC50 = 18 nM
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| 2 |
IC50 = 73 nM
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CP0904759
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4-((6-chloro-3-methyl-2-(4-(trifluoromethoxy)phenylimino)-2,3-dihydro-1H-benzo[d]imidazol-1-yl)methyl)-N-(1H-tetrazol-5-yl)benzamide
Show/Hide
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C24H18ClF3N8O2
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2
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| 1 |
IC50 = 18 nM
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| 2 |
IC50 = 96 nM
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CP0459951
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4-[[N-(5,6-dichloro-1-methylbenzimidazol-2-yl)-4-(trifluoromethoxy)anilino]methyl]-N-(2H-tetrazol-5-yl)benzamide
Show/Hide
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C24H17Cl2F3N8O2
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2
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| 1 |
IC50 = 19 nM
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| 2 |
IC50 = 670 nM
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CP0384133
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2-[5-(4-chlorophenyl)-2-pyridin-4-yl-1H-pyrrol-3-yl]-N-propylaniline
Show/Hide
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C24H22ClN3
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2
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| 1 |
IC50 = 20 nM
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| 2 |
IC50 = 270 nM
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CP0286734
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4-[2-(4-Chloro-phenyl)-5-(4-fluoro-phenyl)-3H-imidazol-4-yl]-3-methyl-pyridine
Show/Hide
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C21H15ClFN3
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1
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| 1 |
IC50 = 20.04 nM
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CP0435017
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3-(4-((1-(4-tert-butylcyclohexyl)-3-(4-(trifluoromethoxy)phenyl)ureido)methyl)benzamido)propanoic acid
Show/Hide
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C29H36F3N3O5
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2
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| 1 |
IC50 = 21 nM
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| 2 |
IC50 = 144 nM
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CP0047783
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3-{4-[1-(4-tert-Butyl-cyclohexyl)-3-(4-trifluoromethoxy-phenyl)-ureidomethyl]-benzoylamino}-propionic acid
Show/Hide
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C29H36F3N3O5
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2
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| 1 |
IC50 = 21 nM
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| 2 |
IC50 = 140 nM
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CP0395564
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4-[(1R)-1-[8-tert-butyl-2-(3-fluorophenyl)-3-oxo-1,4-diazaspiro[4.5]dec-1-en-4-yl]-4,4-dimethylpentyl]-N-(2H-tetrazol-5-ylmethyl)benzamide
Show/Hide
|
C34H44FN7O2
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2
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| 1 |
IC50 = 21 nM
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| 2 |
IC50 = 140 nM
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CP0484377
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1-(5-((2H-tetrazol-5-yl)carbamoyl)-2,3-dihydro-1H-inden-1-yl)-1-(4-cyclohexylphenyl)-3-(4-(trifluoromethoxy)phenyl)urea
Show/Hide
|
C31H30F3N7O3
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2
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| 1 |
IC50 = 22 nM
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| 2 |
IC50 = 85 nM
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CP0666274
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4-((3-methyl-4-propoxy-6-(trifluoromethyl)-2-(3-(trifluoromethyl)phenylimino)-2,3-dihydro-1H-benzo[d]imidazol-1-yl)methyl)-N-(1H-tetrazol-5-yl)benzamide
Show/Hide
|
C28H24F6N8O2
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2
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| 1 |
IC50 = 22 nM
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| 2 |
IC50 = 31 nM
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CP0411598
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4-[(1R)-1-[8-tert-butyl-2-(3,5-dichlorophenyl)-3-oxo-1,4-diazaspiro[4.5]dec-1-en-4-yl]-4-methylpentyl]-N-(2H-tetrazol-5-ylmethyl)benzamide
Show/Hide
|
C33H41Cl2N7O2
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2
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| 1 |
IC50 = 22 nM
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| 2 |
IC50 = 150 nM
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CP0540262
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4-[(1R)-1-[8-tert-butyl-3-oxo-2-[4-(trifluoromethyl)pyridin-3-yl]-1,4-diazaspiro[4.5]dec-1-en-4-yl]-4,4-dimethylpentyl]-N-(2H-tetrazol-5-ylmethyl)benzamide
Show/Hide
|
C34H43F3N8O2
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2
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| 1 |
IC50 = 22 nM
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| 2 |
IC50 = 1200 nM
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CP0401177
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3-[[4-[2-[5-chloro-1-[4-methoxy-3-(trifluoromethyl)phenyl]indole-2-carbonyl]pentyl]benzoyl]amino]propanoic acid
Show/Hide
|
C32H30ClF3N2O5
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2
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| 1 |
IC50 = 23 nM
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| 2 |
IC50 = 39 nM
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CP0411597
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4-[(1R)-1-[8-tert-butyl-2-(3,5-dichlorophenyl)-3-oxo-1,4-diazaspiro[4.5]dec-1-en-4-yl]pentyl]-N-(2H-tetrazol-5-ylmethyl)benzamide
Show/Hide
|
C32H39Cl2N7O2
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2
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| 1 |
IC50 = 23 nM
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| 2 |
IC50 = 380 nM
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CP0414508
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4-[(1R)-1-[8-tert-butyl-2-(3,5-difluorophenyl)-3-oxo-1,4-diazaspiro[4.5]dec-1-en-4-yl]-4,4-dimethylpentyl]-N-(2H-tetrazol-5-ylmethyl)benzamide
Show/Hide
|
C34H43F2N7O2
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2
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| 1 |
IC50 = 23 nM
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| 2 |
IC50 = 110 nM
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CP0139955
|
4-[2,5-Bis-(4-chloro-phenyl)-3H-imidazol-4-yl]-pyridine
Show/Hide
|
C20H13Cl2N3
|
1
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| 1 |
IC50 = 23.01 nM
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CP0468491
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4-[[(4-tert-butylcyclohexyl)-(1-propylbenzimidazol-2-yl)amino]methyl]-N-(2H-tetrazol-5-yl)benzamide
Show/Hide
|
C29H38N8O
|
1
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| 1 |
IC50 = 24 nM
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CP0476580
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3-[[4-[2-[5-chloro-1-[3-(trifluoromethoxy)phenyl]indole-2-carbonyl]pentyl]benzoyl]amino]propanoic acid
Show/Hide
|
C31H28ClF3N2O5
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2
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| 1 |
IC50 = 24 nM
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| 2 |
IC50 = 35 nM
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CP0914640
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4-((3-methyl-6-(trifluoromethoxy)-2-(4-(trifluoromethoxy)phenylimino)-2,3-dihydro-1H-benzo[d]imidazol-1-yl)methyl)-N-(1H-tetrazol-5-yl)benzamide
Show/Hide
|
C25H18F6N8O3
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2
|
| 1 |
IC50 = 24 nM
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| 2 |
IC50 = 180 nM
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CP0124750
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4-[(1R)-1-[8-tert-butyl-2-(3,5-dichlorophenyl)-3-oxo-1,4-diazaspiro[4.5]dec-1-en-4-yl]-4,4-dimethylpentyl]-N-(2H-tetrazol-5-ylmethyl)benzamide
Show/Hide
|
C34H43Cl2N7O2
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2
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| 1 |
IC50 = 24 nM
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| 2 |
IC50 = 46 nM
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CP0435171
|
CHEMBL3237925
Show/Hide
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C33H41Cl2N7O2
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2
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| 1 |
IC50 = 24 nM
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| 2 |
IC50 = 130 nM
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CP0287590
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4-[3-(2-Bromo-phenyl)-5-(4-chloro-phenyl)-1H-pyrrol-2-yl]-pyridine
Show/Hide
|
C21H14BrClN2
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2
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| 1 |
IC50 = 26 nM
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| 2 |
IC50 = 2300 nM
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CP0452402
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3-[[4-[(2S)-2-[5-methoxy-1-[3-(trifluoromethyl)phenyl]indole-2-carbonyl]heptyl]benzoyl]amino]propanoic acid
Show/Hide
|
C34H35F3N2O5
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2
|
| 1 |
IC50 = 26 nM
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| 2 |
IC50 = 35 nM
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CP0411599
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4-[(1R)-1-[8-tert-butyl-2-(4-methoxyphenyl)-3-oxo-1,4-diazaspiro[4.5]dec-1-en-4-yl]-4,4-dimethylpentyl]-N-(2H-tetrazol-5-ylmethyl)benzamide
Show/Hide
|
C35H47N7O3
|
2
|
| 1 |
IC50 = 26 nM
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| 2 |
IC50 = 360 nM
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CP0474755
|
3-[[4-[1-[3-(6-methoxypyridin-3-yl)-6-[4-(trifluoromethoxy)phenyl]indazol-1-yl]ethyl]benzoyl]amino]propanoic acid
Show/Hide
|
C32H27F3N4O5
|
2
|
| 1 |
IC50 = 26 nM
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| 2 |
IC50 = 65 nM
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CP0393098
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3-(1-(3-(3,5-bis(trifluoromethyl)phenyl)-1-((1r,4r)-4-tert-butylcyclohexyl)ureido)-2,3-dihydro-1H-indene-5-carboxamido)propanoic acid
Show/Hide
|
C32H37F6N3O4
|
2
|
| 1 |
IC50 = 28 nM
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| 2 |
IC50 = 46 nM
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CP0465995
|
(R)-3-(4-((3-(3,5-dichlorophenyl)-5-(4-(trifluoromethoxy)phenyl)-1H-pyrazol-1-yl)methyl)benzamido)-2-hydroxypropanoic acid
Show/Hide
|
C27H20Cl2F3N3O5
|
1
|
| 1 |
IC50 = 28 nM
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CP0492656
|
3-[[4-[2-[5-chloro-1-(2,3-dihydro-1,4-benzodioxin-6-yl)indole-2-carbonyl]pentyl]benzoyl]amino]propanoic acid
Show/Hide
|
C32H31ClN2O6
|
2
|
| 1 |
IC50 = 28 nM
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| 2 |
IC50 = 49 nM
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CP0522178
|
3-[[4-[2-[5-chloro-1-[4-(trifluoromethoxy)phenyl]indole-2-carbonyl]pentyl]benzoyl]amino]propanoic acid
Show/Hide
|
C31H28ClF3N2O5
|
2
|
| 1 |
IC50 = 28 nM
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| 2 |
IC50 = 45 nM
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CP0306397
|
4-[5-(4-Chloro-phenyl)-3-(2-isopropoxy-phenyl)-1H-pyrrol-2-yl]-pyridine
Show/Hide
|
C24H21ClN2O
|
2
|
| 1 |
IC50 = 30 nM
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|
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| 2 |
IC50 = 910 nM
|
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CP0464688
|
4-{3-[1-(4-Bromo-phenyl)-ethyl]-8-tert-butyl-2-oxo-1,3-diaza-spiro[4.5]dec-1-ylmethyl}-N-(2H-tetrazol-5-yl)-benzamide
Show/Hide
|
C29H36BrN7O2
|
2
|
| 1 |
IC50 = 30 nM
|
|
|
| 2 |
IC50 = 164 nM
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CP0452395
|
3-[[4-[2-[5-chloro-1-[4-(trifluoromethyl)phenyl]indole-2-carbonyl]pentyl]benzoyl]amino]propanoic acid
Show/Hide
|
C31H28ClF3N2O4
|
2
|
| 1 |
IC50 = 30 nM
|
|
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| 2 |
IC50 = 31 nM
|
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CP0904766
|
4-((3,4-dimethyl-2-(4-(trifluoromethoxy)phenylimino)-6-(trifluoromethyl)-2,3-dihydro-1H-benzo[d]imidazol-1-yl)methyl)-N-(1H-tetrazol-5-yl)benzamide
Show/Hide
|
C26H20F6N8O2
|
2
|
| 1 |
IC50 = 30 nM
|
|
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| 2 |
IC50 = 130 nM
|
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CP0439152
|
4-(((4-tert-butylphenyl)(1-methyl-1H-benzo[d]imidazol-2-yl)amino)methyl)-N-(1H-tetrazol-5-yl)benzamide
Show/Hide
|
C27H28N8O
|
2
|
| 1 |
IC50 = 31 nM
|
|
|
| 2 |
IC50 = 810 nM
|
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|
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CP0465689
|
4-[(1R)-1-[2-(3,5-dichlorophenyl)-3-oxo-8-propan-2-yl-1,4-diazaspiro[4.5]dec-1-en-4-yl]-4,4-dimethylpentyl]-N-(2H-tetrazol-5-ylmethyl)benzamide
Show/Hide
|
C33H41Cl2N7O2
|
2
|
| 1 |
IC50 = 31 nM
|
|
|
| 2 |
IC50 = 52 nM
|
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CP0461393
|
4-[[9-tert-butyl-2-oxo-3-[4-(trifluoromethoxy)phenyl]-1,3-diazaspiro[5.5]undecan-1-yl]methyl]-N-(2H-tetrazol-5-yl)benzamide
Show/Hide
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C29H34F3N7O3
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1
|
| 1 |
IC50 = 32 nM
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CP0401176
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3-[[4-[2-[5-chloro-1-(4-chlorophenyl)indole-2-carbonyl]pentyl]benzoyl]amino]propanoic acid
Show/Hide
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C30H28Cl2N2O4
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2
|
| 1 |
IC50 = 32 nM
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| 2 |
IC50 = 100 nM
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CP0464689
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4-[8-tert-Butyl-2-oxo-3-(3-trifluoromethoxy-phenyl)-1,3-diaza-spiro[4.5]dec-1-ylmethyl]-N-(2H-tetrazol-5-yl)-benzamide
Show/Hide
|
C28H32F3N7O3
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2
|
| 1 |
IC50 = 33 nM
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| 2 |
IC50 = 234 nM
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CP0394847
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N-[3-cyano-5-[3-[(2,4-dichlorophenyl)methyl]-1,2,4-oxadiazol-5-yl]-4-methylthiophen-2-yl]-2-ethylbutanamide
Show/Hide
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C21H20Cl2N4O2S
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2
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| 1 |
IC50 = 34 nM
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| 2 |
IC50 = 89 nM
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CP0134870
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4-[9-tert-Butyl-2-oxo-3-(4-trifluoromethoxy-phenyl)-1,3-diaza-spiro[5.5]undec-1-ylmethyl]-N-(1H-tetrazol-5-yl)-benzamide
Show/Hide
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C29H34F3N7O3
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2
|
| 1 |
IC50 = 34 nM
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| 2 |
IC50 = 92 nM
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CP0503082
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3-[[4-[2-[5-chloro-1-(6-methoxynaphthalen-2-yl)indole-2-carbonyl]pentyl]benzoyl]amino]propanoic acid
Show/Hide
|
C35H33ClN2O5
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2
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| 1 |
IC50 = 34 nM
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| 2 |
IC50 = 95 nM
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CP0465994
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4-((5-(3,5-dichlorophenyl)-3-(4-(trifluoromethoxy)phenyl)-1H-pyrazol-1-yl)methyl)-N-(2H-tetrazol-5-yl)benzamide
Show/Hide
|
C25H16Cl2F3N7O2
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2
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| 1 |
IC50 = 35 nM
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| 2 |
IC50 = 36 nM
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CP0456654
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3-[[4-[1-[3-(2-methoxypyrimidin-4-yl)-6-[4-(trifluoromethoxy)phenyl]indazol-1-yl]ethyl]benzoyl]amino]propanoic acid
Show/Hide
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C31H26F3N5O5
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2
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| 1 |
IC50 = 35 nM
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| 2 |
IC50 = 84 nM
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CP0508233
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4-[8-tert-Butyl-3-(3,5-dichloro-phenyl)-2-oxo-1,3-diaza-spiro[4.5]dec-1-ylmethyl]-N-(2H-tetrazol-5-yl)-benzamide
Show/Hide
|
C27H31Cl2N7O2
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2
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| 1 |
IC50 = 36 nM
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| 2 |
IC50 = 116 nM
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CP0415755
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CHEMBL3238231
Show/Hide
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C31H37Cl2N7O2
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2
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| 1 |
IC50 = 36 nM
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| 2 |
IC50 = 260 nM
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CP0492500
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3-[[4-[(2S)-3-[5-chloro-1-[3-(trifluoromethyl)phenyl]indol-2-yl]-2-(cyclopropylmethyl)-3-oxopropyl]benzoyl]amino]propanoic acid
Show/Hide
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C32H28ClF3N2O4
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2
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| 1 |
IC50 = 37 nM
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| 2 |
IC50 = 55 nM
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CP0462961
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3-[[4-[[5-(3-chloro-4-propoxyphenyl)-3-(3,5-dichlorophenyl)pyrazol-1-yl]methyl]benzoyl]amino]propanoic acid
Show/Hide
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C29H26Cl3N3O4
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2
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| 1 |
IC50 = 37.9 nM
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| 2 |
IC50 = 100.7 nM
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CP0894248
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4-((5-chloro-3-methyl-2-(4-(trifluoromethoxy)phenylimino)-2,3-dihydro-1H-benzo[d]imidazol-1-yl)methyl)-N-(1H-tetrazol-5-yl)benzamide
Show/Hide
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C24H18ClF3N8O2
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2
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| 1 |
IC50 = 38 nM
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| 2 |
IC50 = 440 nM
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CP0435174
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4-[(1R)-1-[8-tert-butyl-2-(5-chloropyridin-3-yl)-3-oxo-1,4-diazaspiro[4.5]dec-1-en-4-yl]-4,4-dimethylpentyl]-N-(2H-tetrazol-5-ylmethyl)benzamide
Show/Hide
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C33H43ClN8O2
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2
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| 1 |
IC50 = 38 nM
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| 2 |
IC50 = 480 nM
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CP0478584
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4-((3-(3,5-dichlorophenyl)-5-(4-(trifluoromethoxy)phenyl)-1H-pyrazol-1-yl)methyl)-N-(2H-tetrazol-5-yl)benzamide
Show/Hide
|
C25H16Cl2F3N7O2
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2
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| 1 |
IC50 = 39 nM
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| 2 |
IC50 = 330 nM
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CP0534728
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3-[[4-[[3-[2-methoxy-5-(trifluoromethyl)phenyl]-6-(4-methylphenyl)indazol-1-yl]methyl]benzoyl]amino]propanoic acid
Show/Hide
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C33H28F3N3O4
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2
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| 1 |
IC50 = 39 nM
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| 2 |
IC50 = 140 nM
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CP0063255
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4-[5-(2,4-Dichloro-phenyl)-3-(4-fluoro-phenyl)-1H-pyrrol-2-yl]-pyridine
Show/Hide
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C21H13Cl2FN2
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2
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| 1 |
IC50 = 40 nM
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| 2 |
IC50 = 950 nM
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CP0147411
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4-[5-(4-Chloro-phenyl)-3-(2-hexyloxy-phenyl)-1H-pyrrol-2-yl]-pyridine
Show/Hide
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C27H27ClN2O
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2
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| 1 |
IC50 = 40 nM
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| 2 |
IC50 = 500 nM
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CP0280722
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4-[5-(4-Chloro-phenyl)-3-(2-ethoxy-phenyl)-1H-pyrrol-2-yl]-pyridine
Show/Hide
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C23H19ClN2O
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2
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| 1 |
IC50 = 40 nM
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| 2 |
IC50 = 500 nM
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CP0313977
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4-[5-(3-Chloro-phenyl)-3-(4-fluoro-phenyl)-1H-pyrrol-2-yl]-pyridine
Show/Hide
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C21H14ClFN2
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2
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| 1 |
IC50 = 40 nM
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| 2 |
IC50 = 990 nM
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CP0375132
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4-[5-(4-Chloro-phenyl)-3-(2,6-dipropoxy-phenyl)-1H-pyrrol-2-yl]-pyridine
Show/Hide
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C27H27ClN2O2
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2
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| 1 |
IC50 = 40 nM
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| 2 |
IC50 = 290 nM
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CP0545452
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3-[[4-[1-[3-[4-(dimethylamino)benzoyl]-6-[4-(trifluoromethoxy)phenyl]indazol-1-yl]ethyl]benzoyl]amino]propanoic acid
Show/Hide
|
C35H31F3N4O5
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2
|
| 1 |
IC50 = 40 nM
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| 2 |
IC50 = 210 nM
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CP0329193
|
4-[2-(4-Bromo-phenyl)-5-phenyl-3H-imidazol-4-yl]-pyridine
Show/Hide
|
C20H14BrN3
|
1
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| 1 |
IC50 = 40.09 nM
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CP0396444
|
3-[[4-[[3-(3,5-dichlorophenyl)-5-[5-(trifluoromethoxy)naphthalen-2-yl]pyrazol-1-yl]methyl]benzoyl]amino]propanoic acid
Show/Hide
|
C31H22Cl2F3N3O4
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2
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| 1 |
IC50 = 40.5 nM
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| 2 |
IC50 = 114.2 nM
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CP0394835
|
4-Cyano-5-(2-ethyl-butyrylamino)-3-methyl-thiophene-2-carboxylic acid (2,4-dichloro-benzyl)-isopropyl-amide
Show/Hide
|
C23H27Cl2N3O2S
|
2
|
| 1 |
IC50 = 41 nM
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| 2 |
IC50 = 153 nM
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CP0914638
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4-((3-methyl-4-propoxy-2-(4-(trifluoromethoxy)phenylimino)-2,3-dihydro-1H-benzo[d]imidazol-1-yl)methyl)-N-(1H-tetrazol-5-yl)benzamide
Show/Hide
|
C27H25F3N8O3
|
2
|
| 1 |
IC50 = 42 nM
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| 2 |
IC50 = 250 nM
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CP0509348
|
3-{4-[8-tert-Butyl-3-(3,5-dichloro-phenyl)-2-oxo-1,3-diaza-spiro[4.5]dec-1-ylmethyl]-benzoylamino}-propionic acid
Show/Hide
|
C29H35Cl2N3O4
|
2
|
| 1 |
IC50 = 43 nM
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| 2 |
IC50 = 423 nM
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CP0404398
|
4-((3,5-bis(4-(trifluoromethoxy)phenyl)-1H-pyrazol-1-yl)methyl)-N-(2H-tetrazol-5-yl)benzamide
Show/Hide
|
C26H17F6N7O3
|
2
|
| 1 |
IC50 = 43 nM
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|
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| 2 |
IC50 = 47 nM
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CP0297243
|
3-(4-((3-(3,5-dichlorophenyl)-5-(4-(trifluoromethoxy)phenyl)-1H-pyrazol-1-yl)methyl)benzamido)propanoic acid
Show/Hide
|
C27H20Cl2F3N3O4
|
4
|
| 1 |
IC50 = 44 nM
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|
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| 2 |
IC50 = 84 nM
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| 3 |
IC50 = 86.2 nM
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| 4 |
IC50 = 113.8 nM
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CP0465712
|
CHEMBL3238230
Show/Hide
|
C32H39Cl2N7O2
|
2
|
| 1 |
IC50 = 44 nM
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| 2 |
IC50 = 66 nM
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CP0488515
|
3-[[4-[(1R)-1-[8-tert-butyl-2-(3-chloro-4-fluorophenyl)-3-oxo-1,4-diazaspiro[4.5]dec-1-en-4-yl]ethyl]benzoyl]amino]propanoic acid
Show/Hide
|
C30H35ClFN3O4
|
2
|
| 1 |
IC50 = 44 nM
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| 2 |
IC50 = 440 nM
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CP0442473
|
3-(1-(1-(cis-4-tert-butylcyclohexyl)-3-(4-(trifluoromethoxy)phenyl)ureido)-2,3-dihydro-1H-indene-5-carboxamido)propanoic acid
Show/Hide
|
C31H38F3N3O5
|
1
|
| 1 |
IC50 = 46 nM
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CP0488404
|
3-[[4-[2-[5-chloro-1-(3-fluorophenyl)indole-2-carbonyl]pentyl]benzoyl]amino]propanoic acid
Show/Hide
|
C30H28ClFN2O4
|
2
|
| 1 |
IC50 = 47 nM
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| 2 |
IC50 = 150 nM
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CP0437829
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1-(N-((1r,4r)-4-tert-butylcyclohexyl)-4-(trifluoromethoxy)benzamido)-N-(2H-tetrazol-5-yl)-2,3-dihydro-1H-indene-5-carboxamide
Show/Hide
|
C29H33F3N6O3
|
2
|
| 1 |
IC50 = 49 nM
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| 2 |
IC50 = 1467 nM
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CP0445495
|
4-[2-(4-chlorophenyl)-5-(4-fluorophenyl)-1H-imidazol-4-yl]-2-methylpyridine
Show/Hide
|
C21H15ClFN3
|
1
|
| 1 |
IC50 = 50 nM
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CP0486552
|
3-[[4-[1-[3-(5-methoxypyridin-3-yl)-6-[4-(trifluoromethoxy)phenyl]indazol-1-yl]ethyl]benzoyl]amino]propanoic acid
Show/Hide
|
C32H27F3N4O5
|
2
|
| 1 |
IC50 = 50 nM
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| 2 |
IC50 = 100 nM
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CP0496122
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N-(2H-tetrazol-5-yl)-4-[[2-[4-(trifluoromethoxy)benzoyl]-6-(trifluoromethyl)indol-1-yl]methyl]benzamide
Show/Hide
|
C26H16F6N6O3
|
1
|
| 1 |
IC50 = 51 nM
|
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CP0496124
|
3-[[4-[2-[1-(4-tert-butylphenyl)-5-chloroindole-2-carbonyl]pentyl]benzoyl]amino]propanoic acid
Show/Hide
|
C34H37ClN2O4
|
1
|
| 1 |
IC50 = 52 nM
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CP0888569
|
4-((3-methyl-6-propoxy-2-(4-(trifluoromethoxy)phenylimino)-2,3-dihydro-1H-benzo[d]imidazol-1-yl)methyl)-N-(1H-tetrazol-5-yl)benzamide
Show/Hide
|
C27H25F3N8O3
|
2
|
| 1 |
IC50 = 55 nM
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| 2 |
IC50 = 1200 nM
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CP0415752
|
CHEMBL3237923
Show/Hide
|
C31H37Cl2N7O2
|
2
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| 1 |
IC50 = 55 nM
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| 2 |
IC50 = 220 nM
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CP0434513
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3-[[4-[(1R)-1-[8-tert-butyl-2-(3-cyclopropylphenyl)-3-oxo-1,4-diazaspiro[4.5]dec-1-en-4-yl]ethyl]benzoyl]amino]propanoic acid
Show/Hide
|
C33H41N3O4
|
2
|
| 1 |
IC50 = 56 nM
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| 2 |
IC50 = 340 nM
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CP0452397
|
3-[[4-[2-(5-chloro-1-quinolin-3-ylindole-2-carbonyl)pentyl]benzoyl]amino]propanoic acid
Show/Hide
|
C33H30ClN3O4
|
2
|
| 1 |
IC50 = 58 nM
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| 2 |
IC50 = 718 nM
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CP0499372
|
3-[[4-[[3-(3,5-dichlorophenyl)-5-naphthalen-2-ylpyrazol-1-yl]methyl]benzoyl]amino]propanoic acid
Show/Hide
|
C30H23Cl2N3O3
|
2
|
| 1 |
IC50 = 58.5 nM
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| 2 |
IC50 = 60.6 nM
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CP0497047
|
N-[3-cyano-6-[(2,4-dichlorophenyl)methyl-propan-2-ylamino]-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-2-ethylbutanamide
Show/Hide
|
C25H31Cl2N3OS
|
2
|
| 1 |
IC50 = 59 nM
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| 2 |
IC50 = 129 nM
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CP0051820
|
4-[5-(4-Chloro-phenyl)-3-phenyl-1H-pyrrol-2-yl]-pyridine
Show/Hide
|
C21H15ClN2
|
2
|
| 1 |
IC50 = 60 nM
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| 2 |
IC50 = 380 nM
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CP0357281
|
4-[5-(4-Chloro-phenyl)-3-(3-methoxy-phenyl)-1H-pyrrol-2-yl]-pyridine
Show/Hide
|
C22H17ClN2O
|
2
|
| 1 |
IC50 = 60 nM
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| 2 |
IC50 = 450 nM
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CP0509122
|
5-(4-Chloro-phenyl)-2-pyridin-4-yl-1H-pyrrole-3-carboxylic acid benzyl ester
Show/Hide
|
C23H17ClN2O2
|
2
|
| 1 |
IC50 = 60 nM
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| 2 |
IC50 = 1300 nM
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CP0492072
|
3-{4-[8-tert-Butyl-2-oxo-3-(3-trifluoromethoxy-phenyl)-1,3-diaza-spiro[4.5]dec-1-ylmethyl]-benzoylamino}-propionic acid
Show/Hide
|
C30H36F3N3O5
|
2
|
| 1 |
IC50 = 60 nM
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| 2 |
IC50 = 515 nM
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CP0484379
|
1-(5-((2H-tetrazol-5-yl)carbamoyl)-2,3-dihydro-1H-inden-1-yl)-1,3-bis(4-(trifluoromethoxy)phenyl)urea
Show/Hide
|
C26H19F6N7O4
|
2
|
| 1 |
IC50 = 62 nM
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| 2 |
IC50 = 3434 nM
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CP0430193
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N-[3-cyano-6-[(2,4-dichlorophenyl)methyl-methylamino]-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-2-ethylbutanamide
Show/Hide
|
C23H27Cl2N3OS
|
2
|
| 1 |
IC50 = 63 nM
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| 2 |
IC50 = 92 nM
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CP0372626
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4-[[5-(4-tert-butylcyclohexyl)-3-[4-(trifluoromethoxy)phenyl]pyrazol-1-yl]methyl]-N-(2H-tetrazol-5-yl)benzamide
Show/Hide
|
C29H32F3N7O2
|
2
|
| 1 |
IC50 = 63 nM
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| 2 |
IC50 = 170 nM
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CP0899731
|
4-((5,6-dichloro-3-isopropyl-2-(4-(trifluoromethoxy)phenylimino)-2,3-dihydro-1H-benzo[d]imidazol-1-yl)methyl)-N-(1H-tetrazol-5-yl)benzamide
Show/Hide
|
C26H21Cl2F3N8O2
|
2
|
| 1 |
IC50 = 64 nM
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| 2 |
IC50 = 210 nM
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CP0405060
|
3-[[4-[[3-(3,5-dichlorophenyl)-5-[7-(trifluoromethoxy)naphthalen-2-yl]pyrazol-1-yl]methyl]benzoyl]amino]propanoic acid
Show/Hide
|
C31H22Cl2F3N3O4
|
2
|
| 1 |
IC50 = 64.2 nM
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| 2 |
IC50 = 189 nM
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CP0223176
|
(R)-1-[4-(4-Fluoro-phenyl)-2,6-diisopropyl-5-propyl-pyridin-3-yl]-ethanol
Show/Hide
|
C22H30FNO
|
2
|
| 1 |
IC50 = 65 nM
|
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| 2 |
IC50 = 110 nM
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CP0492073
|
4-[8-tert-Butyl-3-(3,4-difluoro-phenyl)-2-oxo-1,3-diaza-spiro[4.5]dec-1-ylmethyl]-N-(2H-tetrazol-5-yl)-benzamide
Show/Hide
|
C27H31F2N7O2
|
2
|
| 1 |
IC50 = 65 nM
|
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| 2 |
IC50 = 227 nM
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CP0411624
|
4-[(1R)-1-[8-tert-butyl-2-(3,5-dichlorophenyl)-3-oxo-1,4-diazaspiro[4.5]dec-1-en-4-yl]-4,4-dimethylpentyl]-N-[2-(2,3-dihydro-1H-tetrazol-5-yl)ethyl]benzamide
Show/Hide
|
C35H47Cl2N7O2
|
2
|
| 1 |
IC50 = 65 nM
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| 2 |
IC50 = 890 nM
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|
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CP0435172
|
CHEMBL3237915
Show/Hide
|
C31H36F3N3O5
|
2
|
| 1 |
IC50 = 67 nM
|
|
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| 2 |
IC50 = 1100 nM
|
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CP0484378
|
3-(1-(1-(4-cyclohexylphenyl)-3-(4-(trifluoromethoxy)phenyl)ureido)-2,3-dihydro-1H-indene-5-carboxamido)propanoic acid
Show/Hide
|
C33H34F3N3O5
|
2
|
| 1 |
IC50 = 68 nM
|
|
|
| 2 |
IC50 = 189 nM
|
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CP0115930
|
4-[5-(4-Chloro-phenyl)-3-(2-methoxy-phenyl)-1H-pyrrol-2-yl]-pyridine
Show/Hide
|
C22H17ClN2O
|
2
|
| 1 |
IC50 = 70 nM
|
|
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| 2 |
IC50 = 500 nM
|
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|
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CP0170867
|
4-[4-(4-Fluoro-phenyl)-5-pyridin-4-yl-1H-imidazol-2-yl]-phenylamine
Show/Hide
|
C20H15FN4
|
1
|
| 1 |
IC50 = 70.15 nM
|
|
|
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CP0411280
|
4-[(R)-[8-tert-butyl-2-(3,5-dichlorophenyl)-3-oxo-1,4-diazaspiro[4.5]dec-1-en-4-yl]-cyclopropylmethyl]-N-(2H-tetrazol-5-ylmethyl)benzamide
Show/Hide
|
C31H35Cl2N7O2
|
2
|
| 1 |
IC50 = 72 nM
|
|
|
| 2 |
IC50 = 540 nM
|
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CP0380122
|
3-[[4-[1-[3-(2-methoxypyridin-3-yl)-6-[4-(trifluoromethoxy)phenyl]indazol-1-yl]ethyl]benzoyl]amino]propanoic acid
Show/Hide
|
C32H27F3N4O5
|
2
|
| 1 |
IC50 = 72 nM
|
|
|
| 2 |
IC50 = 77 nM
|
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CP0484435
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3-[[4-[1-[3-(3,5-dichlorophenyl)-5-[4-(trifluoromethoxy)phenyl]pyrazol-1-yl]ethyl]benzoyl]amino]propanoic acid
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C28H22Cl2F3N3O4
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2
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| 1 |
IC50 = 77.5 nM
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| 2 |
IC50 = 100.3 nM
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CP0096778
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4-[5-(4-Chloro-phenyl)-3-(4-fluoro-phenyl)-1H-pyrrol-2-yl]-pyridine
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C21H14ClFN2
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2
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| 1 |
IC50 = 80 nM
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| 2 |
IC50 = 800 nM
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CP0904604
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4-((4-ethyl-3-methyl-2-(p-tolylimino)-6-(trifluoromethyl)-2,3-dihydro-1H-benzo[d]imidazol-1-yl)methyl)-N-(1H-tetrazol-5-yl)benzamide
Show/Hide
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C27H25F3N8O
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2
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| 1 |
IC50 = 80 nM
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| 2 |
IC50 = 230 nM
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CP0016202
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4-(4-Fluorophenyl)-2-(4-hydroxyphenyl)-5-(4-pyridyl)-1H-imidazole
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C20H14FN3O
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1
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| 1 |
IC50 = 80.17 nM
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CP0057065
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4-[2-(4-Chloro-phenyl)-5-(4-fluoro-phenyl)-3H-imidazol-4-yl]-pyridine
Show/Hide
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C20H13ClFN3
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1
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| 1 |
IC50 = 80.17 nM
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CP0495578
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3-[[4-[(1S)-1-[3-tert-butyl-5-(6-methoxynaphthalen-2-yl)pyrazol-1-yl]ethyl]benzoyl]amino]propanoic acid
Show/Hide
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C30H33N3O4
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2
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| 1 |
IC50 = 81.8 nM
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| 2 |
IC50 = 108 nM
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CP0383829
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4-[(1R)-1-[8-tert-butyl-2-(3,5-dichlorophenyl)-3-oxo-1,4-diazaspiro[4.5]dec-1-en-4-yl]propyl]-N-(2H-tetrazol-5-ylmethyl)benzamide
Show/Hide
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C30H35Cl2N7O2
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2
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| 1 |
IC50 = 82 nM
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| 2 |
IC50 = 270 nM
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CP0424380
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4-(((3-chloro-4-(4-chlorophenoxy)phenyl)(4-phenylthiazol-2-yl)amino)methyl)-N-(1H-tetrazol-5-yl)benzamide
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C30H21Cl2N7O2S
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1
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| 1 |
IC50 = 85 nM
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CP0414517
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3-[[4-[(1R)-1-[8-tert-butyl-2-(4-fluorophenyl)-3-oxo-1,4-diazaspiro[4.5]dec-1-en-4-yl]ethyl]benzoyl]amino]propanoic acid
Show/Hide
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C30H36FN3O4
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2
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| 1 |
IC50 = 85 nM
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| 2 |
IC50 = 430 nM
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CP0488522
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(2S)-3-[[4-[(1R)-1-[8-tert-butyl-2-(3,5-dichlorophenyl)-3-oxo-1,4-diazaspiro[4.5]dec-1-en-4-yl]-4,4-dimethylpentyl]benzoyl]amino]-2-hydroxypropanoic acid
Show/Hide
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C35H45Cl2N3O5
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2
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| 1 |
IC50 = 86 nM
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| 2 |
IC50 = 370 nM
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CP0091849
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5-(4-Chloro-phenyl)-2-pyridin-4-yl-1H-pyrrole-3-carboxylic acid ethyl ester
Show/Hide
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C18H15ClN2O2
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2
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| 1 |
IC50 = 90 nM
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| 2 |
IC50 = 400 nM
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CP0182277
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4-[5-Cyclohexyl-3-(4-fluoro-phenyl)-1H-pyrrol-2-yl]-pyridine
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C21H21FN2
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2
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| 1 |
IC50 = 90 nM
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| 2 |
IC50 = 490 nM
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CP0222552
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4-[3,5-Bis-(4-fluoro-phenyl)-1H-pyrrol-2-yl]-pyridine
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C21H14F2N2
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2
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| 1 |
IC50 = 90 nM
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| 2 |
IC50 = 350 nM
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CP0468492
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4-(((1-methyl-1H-benzo[d]imidazol-2-yl)(4-(trifluoromethoxy)phenyl)amino)methyl)-N-(1H-tetrazol-5-yl)benzamide
Show/Hide
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C24H19F3N8O2
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2
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| 1 |
IC50 = 90 nM
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| 2 |
IC50 > 1000 nM
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CP0324127
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4-[5-(4-Fluoro-phenyl)-2-p-tolyl-3H-imidazol-4-yl]-pyridine
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C21H16FN3
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1
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| 1 |
IC50 = 90.16 nM
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CP0395748
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4-[2-(2-Bromo-phenyl)-5-(4-fluoro-phenyl)-3H-imidazol-4-yl]-pyridine
Show/Hide
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C20H13BrFN3
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1
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| 1 |
IC50 = 90.16 nM
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CP0494656
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4-[9-tert-Butyl-2-oxo-3-(4-trifluoromethoxy-phenyl)-1,3-diaza-spiro[5.5]undec-1-ylmethyl]-N-(1H-tetrazol-5-ylmethyl)-benzamide
Show/Hide
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C30H36F3N7O3
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2
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| 1 |
IC50 = 92 nM
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| 2 |
IC50 = 1975 nM
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CP0436677
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4-[8-tert-Butyl-3-(3-chloro-phenyl)-2-oxo-1,3-diaza-spiro[4.5]dec-1-ylmethyl]-N-(2H-tetrazol-5-yl)-benzamide
Show/Hide
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C27H32ClN7O2
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2
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| 1 |
IC50 = 94 nM
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| 2 |
IC50 = 353 nM
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CP0505160
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3-(4-((5-(3,5-dichlorophenyl)-3-(4-(trifluoromethoxy)phenyl)-1H-pyrazol-1-yl)methyl)benzamido)propanoic acid
Show/Hide
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C27H20Cl2F3N3O4
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2
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| 1 |
IC50 = 95 nM
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| 2 |
IC50 = 230 nM
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CP0488511
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3-[[4-[(1R)-1-[8-tert-butyl-2-(3,4-dichlorophenyl)-3-oxo-1,4-diazaspiro[4.5]dec-1-en-4-yl]ethyl]benzoyl]amino]propanoic acid
Show/Hide
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C30H35Cl2N3O4
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2
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| 1 |
IC50 = 95 nM
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| 2 |
IC50 = 550 nM
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CP0540674
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3-[[4-[(1R)-1-[8-tert-butyl-2-(3,5-dichlorophenyl)-3-oxo-1,4-diazaspiro[4.5]dec-1-en-4-yl]ethyl]benzoyl]amino]propanoic acid
Show/Hide
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C30H35Cl2N3O4
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2
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| 1 |
IC50 = 96 nM
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| 2 |
IC50 = 140 nM
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CP0245884
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4-[5-(4-Chloro-phenyl)-3-cyclohexyl-1H-pyrrol-2-yl]-pyridine
Show/Hide
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C21H21ClN2
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2
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| 1 |
IC50 = 100 nM
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| 2 |
IC50 > 3000 nM
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CP0310029
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4-[5-(4-Chloro-phenyl)-3-(4-methoxy-phenyl)-1H-pyrrol-2-yl]-pyridine
Show/Hide
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C22H17ClN2O
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2
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| 1 |
IC50 = 100 nM
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| 2 |
IC50 = 1600 nM
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CP0082326
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4-[2,5-Bis-(4-fluoro-phenyl)-3H-imidazol-4-yl]-pyridine
Show/Hide
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C20H13F2N3
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1
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| 1 |
IC50 = 100 nM
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CP0139965
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4-[5-(4-Fluoro-phenyl)-2-(4-methoxy-phenyl)-3H-imidazol-4-yl]-pyridine
Show/Hide
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C21H16FN3O
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1
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| 1 |
IC50 = 100 nM
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CP0276117
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4-[5-(4-Fluoro-phenyl)-2-(4-iodo-phenyl)-3H-imidazol-4-yl]-pyridine
Show/Hide
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C20H13FIN3
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1
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| 1 |
IC50 = 100 nM
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CP0363451
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4-[2-(4-Bromo-phenyl)-5-phenyl-3H-imidazol-4-yl]-phenol
Show/Hide
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C21H15BrN2O
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1
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| 1 |
IC50 = 100 nM
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CP0428256
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4-[8-tert-Butyl-2-oxo-3-(4-trifluoromethoxy-phenyl)-1,3-diaza-spiro[4.5]dec-1-ylmethyl]-N-(1H-tetrazol-5-yl)-benzamide
Show/Hide
|
C28H32F3N7O3
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2
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| 1 |
IC50 = 105 nM
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| 2 |
IC50 = 193 nM
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CP0063780
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4-[5-(4-Chloro-phenyl)-3-isopropyl-1H-pyrrol-2-yl]-pyridine
Show/Hide
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C18H17ClN2
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2
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| 1 |
IC50 = 110 nM
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| 2 |
IC50 = 3032 nM
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CP0522179
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3-[[4-[2-[5-chloro-1-(3,5-dichlorophenyl)indole-2-carbonyl]pentyl]benzoyl]amino]propanoic acid
Show/Hide
|
C30H27Cl3N2O4
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1
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| 1 |
IC50 = 110 nM
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CP0916009
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4-((4-ethyl-2-(4-fluorophenylimino)-3-methyl-6-(trifluoromethyl)-2,3-dihydro-1H-benzo[d]imidazol-1-yl)methyl)-N-(1H-tetrazol-5-yl)benzamide
Show/Hide
|
C26H22F4N8O
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2
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| 1 |
IC50 = 110 nM
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| 2 |
IC50 = 1200 nM
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CP0380121
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3-[[4-[1-[3-(4-methoxypyridin-3-yl)-6-[4-(trifluoromethoxy)phenyl]indazol-1-yl]ethyl]benzoyl]amino]propanoic acid
Show/Hide
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C32H27F3N4O5
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2
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| 1 |
IC50 = 110 nM
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| 2 |
IC50 = 760 nM
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CP0095585
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4-[2-(5-Bromo-thiophen-2-yl)-5-(4-fluoro-phenyl)-3H-imidazol-4-yl]-pyridine
Show/Hide
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C18H11BrFN3S
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1
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| 1 |
IC50 = 110.15 nM
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CP0464524
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4-[8-tert-Butyl-2-oxo-3-(4-trifluoromethyl-phenyl)-1,3-diaza-spiro[4.5]dec-1-ylmethyl]-N-(2H-tetrazol-5-yl)-benzamide
Show/Hide
|
C28H32F3N7O2
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2
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| 1 |
IC50 = 113 nM
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| 2 |
IC50 = 135 nM
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CP0496028
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4-[8-tert-Butyl-3-(4-chloro-phenyl)-2-oxo-1,3-diaza-spiro[4.5]dec-1-ylmethyl]-N-(2H-tetrazol-5-yl)-benzamide
Show/Hide
|
C27H32ClN7O2
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2
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| 1 |
IC50 = 116 nM
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| 2 |
IC50 = 446 nM
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CP0155748
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5-Fluoro-2-(3-hydroxymethyl-2,6-diisopropyl-5-pentyl-pyridin-4-yl)-phenol
Show/Hide
|
C23H32FNO2
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2
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| 1 |
IC50 = 120 nM
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| 2 |
IC50 = 190 nM
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CP0463750
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4-(((4-tert-butylcyclohexyl)(1-cyclopentyl-1H-benzo[d]imidazol-2-yl)amino)methyl)-N-(1H-tetrazol-5-yl)benzamide
Show/Hide
|
C31H40N8O
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1
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| 1 |
IC50 = 120 nM
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CP0436967
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4-[[3-(3,5-dichlorophenyl)-5-[4-(trifluoromethoxy)phenyl]pyrazol-1-yl]methyl]-N-(2H-tetrazol-5-ylmethyl)benzamide
Show/Hide
|
C26H18Cl2F3N7O2
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2
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| 1 |
IC50 = 120 nM
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| 2 |
IC50 = 650 nM
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CP0522121
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4-((5-cyclohexyl-3-(4-(trifluoromethoxy)phenyl)-1H-pyrazol-1-yl)methyl)-N-(2H-tetrazol-5-yl)benzamide
Show/Hide
|
C25H24F3N7O2
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2
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| 1 |
IC50 = 120 nM
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| 2 |
IC50 = 160 nM
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CP0488405
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3-[[4-[2-[5-chloro-1-(3,5-dimethylphenyl)indole-2-carbonyl]pentyl]benzoyl]amino]propanoic acid
Show/Hide
|
C32H33ClN2O4
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1
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| 1 |
IC50 = 120 nM
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CP0395565
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(3R)-3-[[4-[(1R)-1-[8-tert-butyl-2-(3,5-dichlorophenyl)-3-oxo-1,4-diazaspiro[4.5]dec-1-en-4-yl]-4,4-dimethylpentyl]benzoyl]amino]butanoic acid
Show/Hide
|
C36H47Cl2N3O4
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2
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| 1 |
IC50 = 120 nM
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| 2 |
IC50 = 530 nM
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CP0036291
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4-[5-(4-Fluoro-phenyl)-2-phenethyl-3H-imidazol-4-yl]-pyridine
Show/Hide
|
C22H18FN3
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1
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| 1 |
IC50 = 120.23 nM
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CP0446167
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3-[[4-[[3-(3,5-dichlorophenyl)-5-[8-(trifluoromethoxy)naphthalen-2-yl]pyrazol-1-yl]methyl]benzoyl]amino]propanoic acid
Show/Hide
|
C31H22Cl2F3N3O4
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2
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| 1 |
IC50 = 121.5 nM
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| 2 |
IC50 = 239.8 nM
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CP0409276
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N-[3-cyano-6-(2-methylbutan-2-yl)-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-2-ethylbutanamide
Show/Hide
|
C20H30N2OS
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2
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| 1 |
IC50 = 129 nM
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| 2 |
IC50 = 181 nM
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CP0438940
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3-(1-(N-((1r,4r)-4-tert-butylcyclohexyl)-4-(trifluoromethoxy)benzamido)-2,3-dihydro-1H-indene-5-carboxamido)propanoic acid
Show/Hide
|
C31H37F3N2O5
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2
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| 1 |
IC50 = 130 nM
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| 2 |
IC50 = 2778 nM
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CP0505708
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4-(1-(3,5-bis(4-(trifluoromethoxy)phenyl)-1H-pyrazol-1-yl)ethyl)-N-(2H-tetrazol-5-yl)benzamide
Show/Hide
|
C27H19F6N7O3
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2
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| 1 |
IC50 = 130 nM
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| 2 |
IC50 = 1300 nM
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CP0419923
|
CHEMBL3237906
Show/Hide
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C30H36ClN3O4
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2
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| 1 |
IC50 = 130 nM
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| 2 |
IC50 = 480 nM
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CP0488512
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4-[(1R)-1-[8-tert-butyl-2-(3,5-dichlorophenyl)-3-oxo-1,4-diazaspiro[4.5]dec-1-en-4-yl]ethyl]-N-(2H-tetrazol-5-ylmethyl)benzamide
Show/Hide
|
C29H33Cl2N7O2
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2
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| 1 |
IC50 = 130 nM
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| 2 |
IC50 = 180 nM
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CP0057386
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4-[5-(4-Fluoro-phenyl)-2-phenyl-3H-imidazol-4-yl]-pyridine
Show/Hide
|
C20H14FN3
|
1
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| 1 |
IC50 = 130.02 nM
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CP0038573
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4-[3-(4-Bromo-phenyl)-5-(4-chloro-phenyl)-1H-pyrrol-2-yl]-pyridine
Show/Hide
|
C21H14BrClN2
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2
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| 1 |
IC50 = 140 nM
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| 2 |
IC50 = 2300 nM
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CP0101836
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4-[5-(4-Chloro-phenyl)-1H-pyrrol-2-yl]-pyridine
Show/Hide
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C15H11ClN2
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2
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| 1 |
IC50 = 140 nM
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| 2 |
IC50 > 3000 nM
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CP0112393
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4-[4-(4-Fluoro-phenyl)-5-pyridin-4-yl-1H-pyrrol-2-yl]-benzonitrile
Show/Hide
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C22H14FN3
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2
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| 1 |
IC50 = 140 nM
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| 2 |
IC50 = 4900 nM
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CP0415751
|
CHEMBL3237899
Show/Hide
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C31H37Cl2N3O4
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2
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| 1 |
IC50 = 140 nM
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| 2 |
IC50 = 190 nM
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CP0056450
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4-[2-(4-Chloro-phenyl)-5-(4-iodo-phenyl)-3H-imidazol-4-yl]-pyridine
Show/Hide
|
C20H13ClIN3
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1
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| 1 |
IC50 = 140.28 nM
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CP0411623
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(2R)-3-[[4-[(1R)-1-[8-tert-butyl-2-(3,5-dichlorophenyl)-3-oxo-1,4-diazaspiro[4.5]dec-1-en-4-yl]-4,4-dimethylpentyl]benzoyl]amino]-2-hydroxypropanoic acid
Show/Hide
|
C35H45Cl2N3O5
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2
|
| 1 |
IC50 = 149 nM
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| 2 |
IC50 = 400 nM
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CP0222549
|
4-[3-(3-Bromo-phenyl)-5-(4-chloro-phenyl)-1H-pyrrol-2-yl]-pyridine
Show/Hide
|
C21H14BrClN2
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2
|
| 1 |
IC50 = 150 nM
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| 2 |
IC50 = 1700 nM
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CP0411243
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3-[[4-[(1R)-1-[8-tert-butyl-2-(3-methylphenyl)-3-oxo-1,4-diazaspiro[4.5]dec-1-en-4-yl]ethyl]benzoyl]amino]propanoic acid
Show/Hide
|
C31H39N3O4
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2
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| 1 |
IC50 = 150 nM
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| 2 |
IC50 = 490 nM
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CP0036234
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4-[2-(4-Chloro-phenyl)-5-(2-phenoxy-phenyl)-3H-imidazol-4-yl]-pyridine
Show/Hide
|
C26H18ClN3O
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1
|
| 1 |
IC50 = 150.31 nM
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CP0303465
|
4-[2-(3-Bromo-phenyl)-5-(4-fluoro-phenyl)-3H-imidazol-4-yl]-pyridine
Show/Hide
|
C20H13BrFN3
|
1
|
| 1 |
IC50 = 150.31 nM
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CP0496029
|
4-[3-(4-Bromo-phenyl)-8-tert-butyl-2-oxo-1,3-diaza-spiro[4.5]dec-1-ylmethyl]-N-(2H-tetrazol-5-yl)-benzamide
Show/Hide
|
C27H32BrN7O2
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2
|
| 1 |
IC50 = 156 nM
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| 2 |
IC50 = 655 nM
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CP0375406
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4-[[(4-tert-butylcyclohexyl)-(1-methylbenzimidazol-2-yl)amino]methyl]-N-(2H-tetrazol-5-ylmethyl)benzamide
Show/Hide
|
C28H36N8O
|
1
|
| 1 |
IC50 = 160 nM
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CP0894250
|
4-((5,6-dichloro-3-(2-methoxyethyl)-2-(4-(trifluoromethoxy)phenylimino)-2,3-dihydro-1H-benzo[d]imidazol-1-yl)methyl)-N-(1H-tetrazol-5-yl)benzamide
Show/Hide
|
C26H21Cl2F3N8O3
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2
|
| 1 |
IC50 = 160 nM
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| 2 |
IC50 = 640 nM
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CP0399811
|
(2S)-3-[[4-[(1R)-1-[8-tert-butyl-2-(3,5-dichlorophenyl)-3-oxo-1,4-diazaspiro[4.5]dec-1-en-4-yl]ethyl]benzoyl]amino]-2-hydroxypropanoic acid
Show/Hide
|
C30H35Cl2N3O5
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2
|
| 1 |
IC50 = 160 nM
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| 2 |
IC50 > 10000 nM
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CP0166177
|
4-[2-(4-Bromo-phenyl)-5-(4-fluoro-phenyl)-3H-imidazol-4-yl]-pyridine
Show/Hide
|
C20H13BrFN3
|
1
|
| 1 |
IC50 = 160.03 nM
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CP0432393
|
4-[[(4-tert-butylcyclohexyl)-(1-methylbenzimidazol-2-yl)amino]methyl]-N-(2H-tetrazol-5-yl)benzamide
Show/Hide
|
C27H34N8O
|
2
|
| 1 |
IC50 = 170 nM
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| 2 |
IC50 = 430 nM
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CP0488514
|
3-[[4-[2-[8-tert-butyl-2-(3,5-dichlorophenyl)-3-oxo-1,4-diazaspiro[4.5]dec-1-en-4-yl]ethyl]benzoyl]amino]propanoic acid
Show/Hide
|
C30H35Cl2N3O4
|
1
|
| 1 |
IC50 = 170 nM
|
|
|
|
CP0416122
|
CHEMBL3237914
Show/Hide
|
C31H36F3N3O4
|
2
|
| 1 |
IC50 = 170 nM
|
|
|
| 2 |
IC50 = 910 nM
|
|
|
|
CP0516003
|
4-[8-tert-Butyl-3-(4-fluoro-phenyl)-2-oxo-1,3-diaza-spiro[4.5]dec-1-ylmethyl]-N-(2H-tetrazol-5-yl)-benzamide
Show/Hide
|
C27H32FN7O2
|
2
|
| 1 |
IC50 = 178 nM
|
|
|
| 2 |
IC50 = 611 nM
|
|
|
|
CP0464684
|
3-{4-[9-tert-Butyl-2-oxo-3-(4-trifluoromethoxy-phenyl)-1,3-diaza-spiro[5.5]undec-1-ylmethyl]-benzoylamino}-propionic acid
Show/Hide
|
C31H38F3N3O5
|
2
|
| 1 |
IC50 = 182 nM
|
|
|
| 2 |
IC50 = 282 nM
|
|
|
|
CP0495078
|
N-[3-cyano-4-methyl-5-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]thiophen-2-yl]-2-ethylbutanamide
Show/Hide
|
C18H24N4O2S
|
2
|
| 1 |
IC50 = 185 nM
|
|
|
| 2 |
IC50 = 368 nM
|
|
|
|
CP0202930
|
4-[3,5-Bis-(4-chloro-phenyl)-1H-pyrrol-2-yl]-pyridine
Show/Hide
|
C21H14Cl2N2
|
2
|
| 1 |
IC50 = 190 nM
|
|
|
| 2 |
IC50 = 810 nM
|
|
|
|
CP0411600
|
(2R)-3-[[4-[(1R)-1-[8-tert-butyl-2-(3,5-dichlorophenyl)-3-oxo-1,4-diazaspiro[4.5]dec-1-en-4-yl]ethyl]benzoyl]amino]-2-hydroxypropanoic acid
Show/Hide
|
C30H35Cl2N3O5
|
2
|
| 1 |
IC50 = 190 nM
|
|
|
| 2 |
IC50 > 10000 nM
|
|
|
|
CP0097184
|
4-[2-(5-Bromo-furan-2-yl)-5-(4-fluoro-phenyl)-3H-imidazol-4-yl]-pyridine
Show/Hide
|
C18H11BrFN3O
|
1
|
| 1 |
IC50 = 190.11 nM
|
|
|
|
CP0541406
|
4-[(1R)-1-[2-(3,5-dichlorophenyl)-3-oxo-1,4-diazaspiro[4.5]dec-1-en-4-yl]-4,4-dimethylpentyl]-N-(2H-tetrazol-5-ylmethyl)benzamide
Show/Hide
|
C30H35Cl2N7O2
|
2
|
| 1 |
IC50 = 195 nM
|
|
|
| 2 |
IC50 = 510 nM
|
|
|
|
CP0328303
|
4-[4-(4-Fluoro-phenyl)-5-pyridin-4-yl-1H-imidazol-2-yl]-benzonitrile
Show/Hide
|
C21H13FN4
|
1
|
| 1 |
IC50 = 210.38 nM
|
|
|
|
CP0410069
|
4-((5-(4-(methylsulfonyl)phenyl)-3-(4-(trifluoromethoxy)phenyl)-1H-pyrazol-1-yl)methyl)-N-(2H-tetrazol-5-yl)benzamide
Show/Hide
|
C26H20F3N7O4S
|
1
|
| 1 |
IC50 = 220 nM
|
|
|
|
CP0036294
|
4-[2-(4-Chloro-phenyl)-5-(3-phenoxy-phenyl)-3H-imidazol-4-yl]-pyridine
Show/Hide
|
C26H18ClN3O
|
1
|
| 1 |
IC50 = 220.29 nM
|
|
|
|
CP0424381
|
3-[[4-[[(4-tert-butylcyclohexyl)-(1-methylbenzimidazol-2-yl)amino]methyl]benzoyl]amino]propanoic acid
Show/Hide
|
C29H38N4O3
|
1
|
| 1 |
IC50 = 230 nM
|
|
|
|
CP0446166
|
3-[[4-[[3-(3,5-dichlorophenyl)-5-[3-(trifluoromethoxy)phenyl]pyrazol-1-yl]methyl]benzoyl]amino]propanoic acid
Show/Hide
|
C27H20Cl2F3N3O4
|
2
|
| 1 |
IC50 = 233.6 nM
|
|
|
| 2 |
IC50 = 238 nM
|
|
|
|
CP0222551
|
4-[3-(4-Fluoro-phenyl)-5-p-tolyl-1H-pyrrol-2-yl]-pyridine
Show/Hide
|
C22H17FN2
|
2
|
| 1 |
IC50 = 250 nM
|
|
|
| 2 |
IC50 = 2200 nM
|
|
|
|
CP0478586
|
3-(4-(1-(3,5-bis(4-(trifluoromethoxy)phenyl)-1H-pyrazol-1-yl)ethyl)benzamido)propanoic acid
Show/Hide
|
C29H23F6N3O5
|
1
|
| 1 |
IC50 = 250 nM
|
|
|
|
CP0245745
|
4-[2-(4-Chloro-phenyl)-5-(4-phenoxy-phenyl)-3H-imidazol-4-yl]-pyridine
Show/Hide
|
C26H18ClN3O
|
1
|
| 1 |
IC50 = 250.03 nM
|
|
|
|
CP0411278
|
3-[[4-[1-[8-tert-butyl-2-(3,5-dichlorophenyl)-3-oxo-1,4-diazaspiro[4.5]dec-1-en-4-yl]propan-2-yl]benzoyl]amino]propanoic acid
Show/Hide
|
C31H37Cl2N3O4
|
2
|
| 1 |
IC50 = 260 nM
|
|
|
| 2 |
IC50 = 890 nM
|
|
|
|
CP0465713
|
4-[[4-[(1R)-1-[8-tert-butyl-2-(3,5-dichlorophenyl)-3-oxo-1,4-diazaspiro[4.5]dec-1-en-4-yl]-4,4-dimethylpentyl]benzoyl]amino]butanoic acid
Show/Hide
|
C36H47Cl2N3O4
|
2
|
| 1 |
IC50 = 270 nM
|
|
|
| 2 |
IC50 = 350 nM
|
|
|
|
CP0411279
|
3-[[4-[(1R)-1-[8-tert-butyl-3-oxo-2-[3-(trifluoromethyl)phenyl]-1,4-diazaspiro[4.5]dec-1-en-4-yl]ethyl]benzoyl]amino]propanoic acid
Show/Hide
|
C31H36F3N3O4
|
2
|
| 1 |
IC50 = 280 nM
|
|
|
| 2 |
IC50 = 720 nM
|
|
|
|
CP0088613
|
4-[5-(4-Fluoro-phenyl)-2-(4-isopropyl-phenyl)-3H-imidazol-4-yl]-pyridine
Show/Hide
|
C23H20FN3
|
1
|
| 1 |
IC50 = 280.54 nM
|
|
|
|
CP0508243
|
4-[8-tert-Butyl-3-(2,4-dichloro-phenyl)-2-oxo-1,3-diaza-spiro[4.5]dec-1-ylmethyl]-N-(2H-tetrazol-5-yl)-benzamide
Show/Hide
|
C27H31Cl2N7O2
|
2
|
| 1 |
IC50 = 286 nM
|
|
|
| 2 |
IC50 = 1416 nM
|
|
|
|
CP0182300
|
4-[3-(4-Fluoro-phenyl)-5-(4-methylsulfanyl-phenyl)-1H-pyrrol-2-yl]-pyridine
Show/Hide
|
C22H17FN2S
|
1
|
| 1 |
IC50 = 290 nM
|
|
|
|
CP0411239
|
3-[[4-[[8-tert-butyl-2-(3,5-dichlorophenyl)-3-oxo-1,4-diazaspiro[4.5]dec-1-en-4-yl]methyl]benzoyl]amino]propanoic acid
Show/Hide
|
C29H33Cl2N3O4
|
2
|
| 1 |
IC50 = 290 nM
|
|
|
| 2 |
IC50 = 520 nM
|
|
|
|
CP0507189
|
3-[[4-[(1R)-1-[3-(3,5-dichlorophenyl)-5-(6-methoxynaphthalen-2-yl)pyrazol-1-yl]ethyl]benzoyl]amino]propanoic acid
Show/Hide
|
C32H27Cl2N3O4
|
2
|
| 1 |
IC50 = 298 nM
|
|
|
| 2 |
IC50 = 728.3 nM
|
|
|
|
CP0217515
|
4-[2-Biphenyl-4-yl-5-(4-fluoro-phenyl)-3H-imidazol-4-yl]-pyridine
Show/Hide
|
C26H18FN3
|
1
|
| 1 |
IC50 = 300.61 nM
|
|
|
|
CP0345817
|
4-[4-(4-Fluoro-phenyl)-5-pyridin-4-yl-1H-imidazol-2-yl]-benzoic acid methyl ester
Show/Hide
|
C22H16FN3O2
|
1
|
| 1 |
IC50 = 300.61 nM
|
|
|
|
CP0496734
|
(2R)-3-[[4-[[9-tert-butyl-2-oxo-3-[4-(trifluoromethoxy)phenyl]-1,3-diazaspiro[5.5]undecan-1-yl]methyl]benzoyl]amino]-2-hydroxypropanoic acid
Show/Hide
|
C31H38F3N3O6
|
1
|
| 1 |
IC50 = 303 nM
|
|
|
|
CP0479238
|
3-(3-((3,5-bis(4-(trifluoromethoxy)phenyl)-1H-pyrazol-1-yl)methyl)benzamido)propanoic acid
Show/Hide
|
C28H21F6N3O5
|
1
|
| 1 |
IC50 = 330 nM
|
|
|
|
CP0382054
|
3-[[4-[(1R)-1-[8-tert-butyl-3-oxo-2-[3-(trifluoromethoxy)phenyl]-1,4-diazaspiro[4.5]dec-1-en-4-yl]ethyl]benzoyl]amino]propanoic acid
Show/Hide
|
C31H36F3N3O5
|
2
|
| 1 |
IC50 = 330 nM
|
|
|
| 2 |
IC50 = 840 nM
|
|
|
|
CP0464682
|
3-{4-[8-tert-Butyl-2-oxo-3-(4-trifluoromethoxy-phenyl)-1,3-diaza-spiro[4.5]dec-1-ylmethyl]-benzoylamino}-propionic acid
Show/Hide
|
C30H36F3N3O5
|
2
|
| 1 |
IC50 = 336 nM
|
|
|
| 2 |
IC50 = 459 nM
|
|
|
|
CP0449556
|
3-[[4-[1-[5-(2-cyclohexylphenyl)-3-(3,5-dichlorophenyl)pyrazol-1-yl]ethyl]benzoyl]amino]propanoic acid
Show/Hide
|
C33H33Cl2N3O3
|
2
|
| 1 |
IC50 = 337.4 nM
|
|
|
| 2 |
IC50 = 362 nM
|
|
|
|
CP0414505
|
3-[[4-[(1R)-1-[8-tert-butyl-2-(5-chloro-2-fluorophenyl)-3-oxo-1,4-diazaspiro[4.5]dec-1-en-4-yl]ethyl]benzoyl]amino]propanoic acid
Show/Hide
|
C30H35ClFN3O4
|
2
|
| 1 |
IC50 = 340 nM
|
|
|
| 2 |
IC50 = 750 nM
|
|
|
|
CP0078098
|
4-[5-(4-Fluoro-phenyl)-2-naphthalen-1-yl-3H-imidazol-4-yl]-pyridine
Show/Hide
|
C24H16FN3
|
1
|
| 1 |
IC50 = 340.41 nM
|
|
|
|
CP0401231
|
3-[[4-[(1R)-1-[8-tert-butyl-2-(2-fluorophenyl)-3-oxo-1,4-diazaspiro[4.5]dec-1-en-4-yl]ethyl]benzoyl]amino]propanoic acid
Show/Hide
|
C30H36FN3O4
|
2
|
| 1 |
IC50 = 350 nM
|
|
|
| 2 |
IC50 = 1100 nM
|
|
|
|
CP0464687
|
3-{4-[8-tert-Butyl-3-(3-chloro-phenyl)-2-oxo-1,3-diaza-spiro[4.5]dec-1-ylmethyl]-benzoylamino}-propionic acid
Show/Hide
|
C29H36ClN3O4
|
2
|
| 1 |
IC50 = 351 nM
|
|
|
| 2 |
IC50 = 601 nM
|
|
|
|
CP0144083
|
4-[3-(4-Fluoro-phenyl)-5-(4-nitro-phenyl)-1H-pyrrol-2-yl]-pyridine
Show/Hide
|
C21H14FN3O2
|
1
|
| 1 |
IC50 = 360 nM
|
|
|
|
CP0383827
|
3-[[4-[(1R)-1-(8-tert-butyl-3-oxo-2-phenyl-1,4-diazaspiro[4.5]dec-1-en-4-yl)ethyl]benzoyl]amino]propanoic acid
Show/Hide
|
C30H37N3O4
|
2
|
| 1 |
IC50 = 360 nM
|
|
|
| 2 |
IC50 = 630 nM
|
|
|
|
CP0101935
|
4-[5-(4-Ethyl-phenyl)-3-(4-fluoro-phenyl)-1H-pyrrol-2-yl]-pyridine
Show/Hide
|
C23H19FN2
|
1
|
| 1 |
IC50 = 370 nM
|
|
|
|
CP0373345
|
3-(4-((3,5-bis(4-(trifluoromethoxy)phenyl)-1H-pyrazol-1-yl)methyl)benzamido)propanoic acid
Show/Hide
|
C28H21F6N3O5
|
2
|
| 1 |
IC50 = 370 nM
|
|
|
| 2 |
IC50 = 490 nM
|
|
|
|
CP0337062
|
4-[3-(4-Fluoro-phenyl)-5-phenyl-1H-pyrrol-2-yl]-pyridine
Show/Hide
|
C21H15FN2
|
1
|
| 1 |
IC50 = 390 nM
|
|
|
|
CP0213431
|
[4-(4-fluorophenyl)-5-pentyl-2,6-di(propan-2-yl)pyridin-3-yl]methanol
Show/Hide
|
C23H32FNO
|
1
|
| 1 |
IC50 = 400 nM
|
|
|
|
CP0496736
|
4-[8-tert-Butyl-3-(4-methanesulfonyl-phenyl)-2-oxo-1,3-diaza-spiro[4.5]dec-1-ylmethyl]-N-(2H-tetrazol-5-yl)-benzamide
Show/Hide
|
C28H35N7O4S
|
1
|
| 1 |
IC50 = 407 nM
|
|
|
|
CP0428239
|
4-(8-tert-Butyl-2-oxo-3-p-tolyl-1,3-diaza-spiro[4.5]dec-1-ylmethyl)-N-(2H-tetrazol-5-yl)-benzamide
Show/Hide
|
C28H35N7O2
|
1
|
| 1 |
IC50 = 427 nM
|
|
|
|
CP0436929
|
4-((3-(1-(4-chlorophenyl)ethyl)-5-(4-(trifluoromethoxy)phenyl)-1H-pyrazol-1-yl)methyl)-N-(2H-tetrazol-5-yl)benzamide
Show/Hide
|
C27H21ClF3N7O2
|
1
|
| 1 |
IC50 = 430 nM
|
|
|
|
CP0496126
|
3-[[4-[(2R)-2-[5-chloro-1-[6-(trifluoromethyl)pyridin-2-yl]indole-2-carbonyl]pentyl]benzoyl]amino]propanoic acid
Show/Hide
|
C30H27ClF3N3O4
|
1
|
| 1 |
IC50 = 450 nM
|
|
|
|
CP0419924
|
4-[(1R)-1-[8-tert-butyl-2-(3,5-dichlorophenyl)-3-oxo-1,4-diazaspiro[4.5]dec-1-en-4-yl]ethyl]-N-(2H-tetrazol-5-yl)benzamide
Show/Hide
|
C28H31Cl2N7O2
|
2
|
| 1 |
IC50 = 470 nM
|
|
|
| 2 |
IC50 = 750 nM
|
|
|
|
CP0372624
|
3-[[4-[[5-(4-tert-butylcyclohexyl)-3-[4-(trifluoromethoxy)phenyl]pyrazol-1-yl]methyl]benzoyl]amino]propanoic acid
Show/Hide
|
C31H36F3N3O4
|
1
|
| 1 |
IC50 = 480 nM
|
|
|
|
CP0533323
|
1-(3-chloro-4-(4-chlorophenoxy)phenyl)-3-(2-chlorobenzoyl)urea
Show/Hide
|
C20H13Cl3N2O3
|
1
|
| 1 |
IC50 = 482 nM
|
|
|
|
CP0259487
|
4-[5-(4-Fluoro-phenyl)-2-(4-methylsulfanyl-phenyl)-1H-imidazol-4-yl]-pyridine
Show/Hide
|
C21H16FN3S
|
1
|
| 1 |
IC50 = 490 nM
|
|
|
|
CP0415758
|
CHEMBL3237909
Show/Hide
|
C30H36FN3O4
|
2
|
| 1 |
IC50 = 490 nM
|
|
|
| 2 |
IC50 = 560 nM
|
|
|
|
CP0467989
|
2-(3-Hydroxymethyl-2,6-diisopropyl-5-pentyl-pyridin-4-yl)-phenol
Show/Hide
|
C23H33NO2
|
1
|
| 1 |
IC50 = 500 nM
|
|
|
|
CP0465716
|
3-[[4-[[8-tert-butyl-3-oxo-2-[3-(trifluoromethyl)phenyl]-1,4-diazaspiro[4.5]dec-1-en-4-yl]methyl]benzoyl]amino]propanoic acid
Show/Hide
|
C30H34F3N3O4
|
1
|
| 1 |
IC50 = 510 nM
|
|
|
|
CP0410070
|
4-((5-(4-(1-(4-chlorophenyl)ethyl)phenyl)-3-(4-(trifluoromethoxy)phenyl)-1H-pyrazol-1-yl)methyl)-N-(2H-tetrazol-5-yl)benzamide
Show/Hide
|
C33H25ClF3N7O2
|
1
|
| 1 |
IC50 = 520 nM
|
|
|
|
CP0510474
|
3-[[4-[(1R)-1-[8-tert-butyl-2-(2-chlorophenyl)-3-oxo-1,4-diazaspiro[4.5]dec-1-en-4-yl]ethyl]benzoyl]amino]propanoic acid
Show/Hide
|
C30H36ClN3O4
|
2
|
| 1 |
IC50 = 520 nM
|
|
|
| 2 |
IC50 = 2900 nM
|
|
|
|
CP0203388
|
4-[5-(4-Fluoro-phenyl)-3-methyl-2-(4-methylsulfanyl-phenyl)-3H-imidazol-4-yl]-pyridine
Show/Hide
|
C22H18FN3S
|
1
|
| 1 |
IC50 = 521.19 nM
|
|
|
|
CP0540827
|
3-[[4-[[3-(3,5-dichlorophenyl)-5-[2-(trifluoromethoxy)phenyl]pyrazol-1-yl]methyl]benzoyl]amino]propanoic acid
Show/Hide
|
C27H20Cl2F3N3O4
|
1
|
| 1 |
IC50 = 527.5 nM
|
|
|
|
CP0405297
|
2-(4-((3,5-bis(4-(trifluoromethoxy)phenyl)-1H-pyrazol-1-yl)methyl)benzamido)acetic acid
Show/Hide
|
C27H19F6N3O5
|
2
|
| 1 |
IC50 = 560 nM
|
|
|
| 2 |
IC50 = 3000 nM
|
|
|
|
CP0372630
|
4-((3-(4-(methylsulfonyl)phenyl)-5-(4-(trifluoromethoxy)phenyl)-1H-pyrazol-1-yl)methyl)-N-(2H-tetrazol-5-yl)benzamide
Show/Hide
|
C26H20F3N7O4S
|
1
|
| 1 |
IC50 = 570 nM
|
|
|
|
CP0295139
|
4-[3-(4-Fluoro-phenyl)-5-(4-methoxy-phenyl)-1H-pyrrol-2-yl]-pyridine
Show/Hide
|
C22H17FN2O
|
1
|
| 1 |
IC50 = 590 nM
|
|
|
|
CP0324497
|
4-[5-Biphenyl-3-yl-2-(4-chloro-phenyl)-3H-imidazol-4-yl]-pyridine
Show/Hide
|
C26H18ClN3
|
1
|
| 1 |
IC50 = 590.2 nM
|
|
|
|
CP0401232
|
4-[(1R)-1-[8-tert-butyl-2-(3,5-dichlorophenyl)-3-oxo-1,4-diazaspiro[4.5]dec-1-en-4-yl]-4,4-dimethylpentyl]-N-(2H-tetrazol-5-yl)benzamide
Show/Hide
|
C33H41Cl2N7O2
|
2
|
| 1 |
IC50 = 600 nM
|
|
|
| 2 |
IC50 = 850 nM
|
|
|
|
CP0442624
|
CHEMBL3237911
Show/Hide
|
C30H35ClFN3O4
|
2
|
| 1 |
IC50 = 620 nM
|
|
|
| 2 |
IC50 = 630 nM
|
|
|
|
CP0464683
|
4-[8-tert-Butyl-2,4-dioxo-3-(4-trifluoromethoxy-phenyl)-1,3-diaza-spiro[4.5]dec-1-ylmethyl]-N-(1H-tetrazol-5-yl)-benzamide
Show/Hide
|
C28H30F3N7O4
|
1
|
| 1 |
IC50 = 631 nM
|
|
|
|
CP0508242
|
4-(8-tert-Butyl-3-cyclohexyl-2-oxo-1,3-diaza-spiro[4.5]dec-1-ylmethyl)-N-(2H-tetrazol-5-yl)-benzamide
Show/Hide
|
C27H39N7O2
|
1
|
| 1 |
IC50 = 700 nM
|
|
|
|
CP0436934
|
3-(4-((5-(4-(1-(4-chlorophenyl)ethyl)phenyl)-3-(4-(trifluoromethoxy)phenyl)-1H-pyrazol-1-yl)methyl)benzamido)propanoic acid
Show/Hide
|
C35H29ClF3N3O4
|
1
|
| 1 |
IC50 = 730 nM
|
|
|
|
CP0435176
|
3-[[4-[[8-tert-butyl-2-(2-fluorophenyl)-3-oxo-1,4-diazaspiro[4.5]dec-1-en-4-yl]methyl]benzoyl]amino]propanoic acid
Show/Hide
|
C29H34FN3O4
|
2
|
| 1 |
IC50 = 730 nM
|
|
|
| 2 |
IC50 > 10000 nM
|
|
|
|
CP0436676
|
4-[8-tert-Butyl-3-(2-chloro-phenyl)-2-oxo-1,3-diaza-spiro[4.5]dec-1-ylmethyl]-N-(2H-tetrazol-5-yl)-benzamide
Show/Hide
|
C27H32ClN7O2
|
1
|
| 1 |
IC50 = 739 nM
|
|
|
|
CP0488513
|
3-[[4-[[8-tert-butyl-2-(3-chlorophenyl)-3-oxo-1,4-diazaspiro[4.5]dec-1-en-4-yl]methyl]benzoyl]amino]propanoic acid
Show/Hide
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C29H34ClN3O4
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1
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| 1 |
IC50 = 770 nM
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CP0534730
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3-[[4-[1-[3-[2-methoxy-5-(trifluoromethyl)phenyl]-7-(4-methylphenyl)indazol-1-yl]butyl]benzoyl]amino]propanoic acid
Show/Hide
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C36H34F3N3O4
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2
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| 1 |
IC50 = 780 nM
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| 2 |
IC50 = 3800 nM
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CP0438237
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[4-(4-chlorophenyl)-5-pentyl-2,6-di(propan-2-yl)pyridin-3-yl]methanol
Show/Hide
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C23H32ClNO
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1
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| 1 |
IC50 = 800 nM
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CP0548968
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3-[[4-[[8-tert-butyl-3-oxo-2-[4-(trifluoromethyl)phenyl]-1,4-diazaspiro[4.5]dec-1-en-4-yl]methyl]benzoyl]amino]propanoic acid
Show/Hide
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C30H34F3N3O4
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1
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| 1 |
IC50 = 800 nM
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CP0505163
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4-((3-cyclohexyl-5-(4-(trifluoromethoxy)phenyl)-1H-pyrazol-1-yl)methyl)-N-(2H-tetrazol-5-yl)benzamide
Show/Hide
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C25H24F3N7O2
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1
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| 1 |
IC50 = 810 nM
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CP0480312
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3-(1-(1,3-bis(4-(trifluoromethoxy)phenyl)ureido)-2,3-dihydro-1H-indene-5-carboxamido)propanoic acid
Show/Hide
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C28H23F6N3O6
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1
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| 1 |
IC50 = 820 nM
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CP0222550
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4-[4-(4-Fluoro-phenyl)-5-pyridin-4-yl-1H-pyrrol-2-yl]-benzoic acid ethyl ester
Show/Hide
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C24H19FN2O2
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1
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| 1 |
IC50 = 850 nM
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CP0343507
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4-[5-(4-tert-Butyl-phenyl)-3-(4-fluoro-phenyl)-1H-pyrrol-2-yl]-pyridine
Show/Hide
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C25H23FN2
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1
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| 1 |
IC50 = 850 nM
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CP0449482
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3-{4-[8-tert-Butyl-2,4-dioxo-3-(4-trifluoromethoxy-phenyl)-1,3-diaza-spiro[4.5]dec-1-ylmethyl]-benzoylamino}-propionic acid
Show/Hide
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C30H34F3N3O6
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1
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| 1 |
IC50 = 856 nM
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CP0184827
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4-[5-(4-Fluoro-phenyl)-1-methyl-2-(4-methylsulfanyl-phenyl)-1H-imidazol-4-yl]-pyridine
Show/Hide
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C22H18FN3S
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1
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| 1 |
IC50 = 860.99 nM
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CP0436479
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6-(1,1-Dimethyl-propyl)-2-(2-ethyl-butyrylamino)-4,5,6,7-tetrahydro-benzo[b]thiophene-3-carboxylic acid amide
Show/Hide
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C20H32N2O2S
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1
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| 1 |
IC50 = 870 nM
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CP0428284
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4-(8-tert-Butyl-2-oxo-3-phenyl-1,3-diaza-spiro[4.5]dec-1-ylmethyl)-N-(2H-tetrazol-5-yl)-benzamide
Show/Hide
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C27H33N7O2
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1
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| 1 |
IC50 = 894 nM
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CP0359167
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4-[4-(4-Fluoro-phenyl)-2-(4-methylsulfanyl-phenyl)-oxazol-5-yl]-pyridine
Show/Hide
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C21H15FN2OS
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1
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| 1 |
IC50 = 931.11 nM
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CP0434523
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3-[[4-[[8-tert-butyl-2-(4-chlorophenyl)-3-oxo-1,4-diazaspiro[4.5]dec-1-en-4-yl]methyl]benzoyl]amino]propanoic acid
Show/Hide
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C29H34ClN3O4
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2
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| 1 |
IC50 = 940 nM
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| 2 |
IC50 = 1400 nM
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CP0525960
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4-[[(4-tert-butylcyclohexyl)-(1-phenylbenzimidazol-2-yl)amino]methyl]-N-(2H-tetrazol-5-yl)benzamide
Show/Hide
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C32H36N8O
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1
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| 1 |
IC50 = 950 nM
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CP0458852
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(2,6-Diisopropyl-5-pentyl-4-p-tolyl-pyridin-3-yl)-methanol
Show/Hide
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C24H35NO
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1
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| 1 |
IC50 = 1000 nM
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CP0278708
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4-(3-(4-fluorophenyl)-5-(4-(methylsulfinyl)phenyl)-1H-pyrrol-2-yl)pyridine
Show/Hide
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C22H17FN2OS
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1
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| 1 |
IC50 = 1100 nM
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CP0383242
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[4-(3,4-difluorophenyl)-5-pentyl-2,6-di(propan-2-yl)pyridin-3-yl]methanol
Show/Hide
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C23H31F2NO
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1
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| 1 |
IC50 = 1100 nM
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CP0374015
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3-((3,5-bis(4-(trifluoromethoxy)phenyl)-1H-pyrazol-1-yl)methyl)-N-(2H-tetrazol-5-yl)benzamide
Show/Hide
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C26H17F6N7O3
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1
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| 1 |
IC50 = 1100 nM
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CP0378511
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4-(3-((3,5-bis(4-(trifluoromethoxy)phenyl)-1H-pyrazol-1-yl)methyl)benzamido)butanoic acid
Show/Hide
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C29H23F6N3O5
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1
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| 1 |
IC50 = 1100 nM
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CP0479281
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4-(4-((3,5-bis(4-(trifluoromethoxy)phenyl)-1H-pyrazol-1-yl)methyl)benzamido)butanoic acid
Show/Hide
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C29H23F6N3O5
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1
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| 1 |
IC50 = 1100 nM
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CP0378515
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3-(4-((3-cyclohexyl-1-(4-(trifluoromethoxy)phenyl)-1H-pyrazol-4-yl)methyl)benzamido)propanoic acid
Show/Hide
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C27H28F3N3O4
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1
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| 1 |
IC50 = 1200 nM
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CP0472467
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3-(4-((5-(4-(methylsulfonyl)phenyl)-3-(4-(trifluoromethoxy)phenyl)-1H-pyrazol-1-yl)methyl)benzamido)propanoic acid
Show/Hide
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C28H24F3N3O6S
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1
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| 1 |
IC50 = 1200 nM
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CP0202931
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4-[4-(4-Fluoro-phenyl)-5-pyridin-4-yl-1H-pyrrol-2-yl]-phenylamine
Show/Hide
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C21H16FN3
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1
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| 1 |
IC50 = 1400 nM
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CP0050873
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(2,6-Diisopropyl-5-pentyl-4-phenyl-pyridin-3-yl)-methanol
Show/Hide
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C23H33NO
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1
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| 1 |
IC50 = 1400 nM
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CP0411603
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3-[[4-[[8-tert-butyl-2-(3,4-dichlorophenyl)-3-oxo-1,4-diazaspiro[4.5]dec-1-en-4-yl]methyl]benzoyl]amino]propanoic acid
Show/Hide
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C29H33Cl2N3O4
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1
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| 1 |
IC50 = 1600 nM
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CP0435175
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CHEMBL3238227
Show/Hide
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C34H43F3N8O2
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1
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| 1 |
IC50 = 1600 nM
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CP0464686
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4-(3,8-Di-tert-butyl-2-oxo-1,3-diaza-spiro[4.5]dec-1-ylmethyl)-N-(2H-tetrazol-5-yl)-benzamide
Show/Hide
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C25H37N7O2
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1
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| 1 |
IC50 = 1663 nM
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CP0436672
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3-{4-[9-tert-Butyl-2,4-dioxo-3-(4-trifluoromethoxy-phenyl)-1,3-diaza-spiro[5.5]undec-1-ylmethyl]-benzoylamino}-propionic acid
Show/Hide
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C31H36F3N3O6
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1
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| 1 |
IC50 = 1691 nM
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CP0479282
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3-(4-((1-cyclohexyl-5-(4-(trifluoromethoxy)phenyl)-1H-pyrazol-3-yl)methyl)benzamido)propanoic acid
Show/Hide
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C27H28F3N3O4
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1
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| 1 |
IC50 = 1700 nM
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CP0445174
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3-[[4-[1-[7-(4-methoxyphenyl)-3-[2-methoxy-5-(trifluoromethyl)phenyl]indazol-1-yl]butyl]benzoyl]amino]propanoic acid
Show/Hide
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C36H34F3N3O5
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2
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| 1 |
IC50 = 1700 nM
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| 2 |
IC50 = 2700 nM
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CP0411240
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3-[[4-[[8-tert-butyl-3-oxo-2-[4-(trifluoromethoxy)phenyl]-1,4-diazaspiro[4.5]dec-1-en-4-yl]methyl]benzoyl]amino]propanoic acid
Show/Hide
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C30H34F3N3O5
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1
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| 1 |
IC50 = 1900 nM
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CP0435177
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3-[[4-[[8-tert-butyl-2-(4-fluorophenyl)-3-oxo-1,4-diazaspiro[4.5]dec-1-en-4-yl]methyl]benzoyl]amino]propanoic acid
Show/Hide
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C29H34FN3O4
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1
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| 1 |
IC50 = 1900 nM
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CP0464685
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4-[9-tert-Butyl-2,4-dioxo-3-(4-trifluoromethoxy-phenyl)-1,3-diaza-spiro[5.5]undec-1-ylmethyl]-N-(1H-tetrazol-5-yl)-benzamide
Show/Hide
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C29H32F3N7O4
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1
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| 1 |
IC50 = 1965 nM
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CP0373348
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4-((3-cyclohexyl-5-(4-(trifluoromethoxy)phenyl)-1H-pyrazol-1-yl)methyl)benzoic acid
Show/Hide
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C24H23F3N2O3
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1
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| 1 |
IC50 = 2000 nM
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CP0170868
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2-(4-Bromo-phenyl)-4,5-diphenyl-1H-imidazole
Show/Hide
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C21H15BrN2
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1
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| 1 |
IC50 = 2200 nM
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CP0565369
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4-[(1R)-1-[8-tert-butyl-2-(3,5-dichlorophenyl)-3-oxo-1,4-diazaspiro[4.5]dec-1-en-4-yl]-2-methylpropyl]-N-(2H-tetrazol-5-ylmethyl)benzamide
Show/Hide
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C31H37Cl2N7O2
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1
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| 1 |
IC50 = 2200 nM
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CP0457107
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[4-(2-aminophenyl)-5-pentyl-2,6-di(propan-2-yl)pyridin-3-yl]methanol
Show/Hide
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C23H34N2O
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1
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| 1 |
IC50 = 2300 nM
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CP0473502
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3-(4-((3-(1-(4-chlorophenyl)ethyl)-5-(4-(trifluoromethoxy)phenyl)-1H-pyrazol-1-yl)methyl)benzamido)propanoic acid
Show/Hide
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C29H25ClF3N3O4
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1
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| 1 |
IC50 = 2400 nM
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CP0215714
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4-[2-(4-Chloro-phenyl)-5-(2,4-dipropoxy-phenyl)-3H-imidazol-4-yl]-pyridine
Show/Hide
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C26H26ClN3O2
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1
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| 1 |
IC50 = 2404.36 nM
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CP0436675
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4-(8-tert-Butyl-3-isopropyl-2-oxo-1,3-diaza-spiro[4.5]dec-1-ylmethyl)-N-(2H-tetrazol-5-yl)-benzamide
Show/Hide
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C24H35N7O2
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1
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| 1 |
IC50 = 2556 nM
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CP0436968
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3-(4-((3-(4-(methylsulfonyl)phenyl)-5-(4-(trifluoromethoxy)phenyl)-1H-pyrazol-1-yl)methyl)benzamido)propanoic acid
Show/Hide
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C28H24F3N3O6S
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1
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| 1 |
IC50 = 2700 nM
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CP0382057
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2-[[4-[(1R)-1-[8-tert-butyl-2-(3,5-dichlorophenyl)-3-oxo-1,4-diazaspiro[4.5]dec-1-en-4-yl]-4,4-dimethylpentyl]benzoyl]amino]acetic acid
Show/Hide
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C34H43Cl2N3O4
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1
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| 1 |
IC50 = 2700 nM
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CP0371944
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4-((1-cyclohexyl-5-(4-(trifluoromethoxy)phenyl)-1H-pyrazol-3-yl)methyl)-N-(2H-tetrazol-5-yl)benzamide
Show/Hide
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C25H24F3N7O2
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1
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| 1 |
IC50 = 2900 nM
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CP0410071
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2-(3-((3,5-bis(4-(trifluoromethoxy)phenyl)-1H-pyrazol-1-yl)methyl)benzamido)acetic acid
Show/Hide
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C27H19F6N3O5
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1
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| 1 |
IC50 = 2900 nM
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CP0522120
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3-(4-((1-cyclohexyl-3-(4-(trifluoromethoxy)phenyl)-1H-pyrazol-5-yl)methyl)benzamido)propanoic acid
Show/Hide
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C27H28F3N3O4
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1
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| 1 |
IC50 = 2900 nM
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CP0539583
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[4-(3-fluorophenyl)-5-pentyl-2,6-di(propan-2-yl)pyridin-3-yl]methanol
Show/Hide
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C23H32FNO
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1
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| 1 |
IC50 = 3000 nM
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CP0382053
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3-[[4-[(8-tert-butyl-3-oxo-2-phenyl-1,4-diazaspiro[4.5]dec-1-en-4-yl)methyl]benzoyl]amino]propanoic acid
Show/Hide
|
C29H35N3O4
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1
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| 1 |
IC50 = 3200 nM
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CP0394836
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N-[3-cyano-4-methyl-5-[5-(2-methylpropyl)-1,3,4-oxadiazol-2-yl]thiophen-2-yl]-2-ethylbutanamide
Show/Hide
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C18H24N4O2S
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1
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| 1 |
IC50 = 3210 nM
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CP0297388
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4-[5-Biphenyl-4-yl-2-(4-chloro-phenyl)-3H-imidazol-4-yl]-pyridine
Show/Hide
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C26H18ClN3
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1
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| 1 |
IC50 = 3303.7 nM
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CP0540263
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US8633231, 2
Show/Hide
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C27H31Cl2N7O2
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1
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| 1 |
IC50 = 3700 nM
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CP0412066
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3-(4-((5-cyclohexyl-3-(4-(trifluoromethoxy)phenyl)-1H-pyrazol-1-yl)methyl)benzamido)propanoic acid
Show/Hide
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C27H28F3N3O4
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1
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| 1 |
IC50 = 3800 nM
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CP0436480
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N-[6-[benzyl(methyl)amino]-3-cyano-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-2-ethylbutanamide
Show/Hide
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C23H29N3OS
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1
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| 1 |
IC50 = 3820 nM
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CP0475998
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4-((1-cyclohexyl-3-(4-(trifluoromethoxy)phenyl)-1H-pyrazol-5-yl)methyl)-N-(2H-tetrazol-5-yl)benzamide
Show/Hide
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C25H24F3N7O2
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1
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| 1 |
IC50 = 4200 nM
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CP0382058
|
CHEMBL3238245
Show/Hide
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C35H45Cl2N7O2
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1
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| 1 |
IC50 = 4500 nM
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CP0414503
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3-[[4-[(1S)-1-[8-tert-butyl-2-(3,5-dichlorophenyl)-3-oxo-1,4-diazaspiro[4.5]dec-1-en-4-yl]ethyl]benzoyl]amino]propanoic acid
Show/Hide
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C30H35Cl2N3O4
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1
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| 1 |
IC50 = 5100 nM
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CP0478581
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4-((3-cyclohexyl-1-(4-(trifluoromethoxy)phenyl)-1H-pyrazol-4-yl)methyl)-N-(2H-tetrazol-5-yl)benzamide
Show/Hide
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C25H24F3N7O2
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1
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| 1 |
IC50 = 5300 nM
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CP0455346
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3-(3-Hydroxymethyl-2,6-diisopropyl-5-pentyl-pyridin-4-yl)-phenol
Show/Hide
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C23H33NO2
|
1
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| 1 |
IC50 = 6000 nM
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CP0411625
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3-[[4-[[8-tert-butyl-2-(2-chlorophenyl)-3-oxo-1,4-diazaspiro[4.5]dec-1-en-4-yl]methyl]benzoyl]amino]propanoic acid
Show/Hide
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C29H34ClN3O4
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1
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| 1 |
IC50 = 6800 nM
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CP0463633
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4-(4-Fluoro-phenyl)-2,6-diisopropyl-5-(2-methyl-propenyl)-pyridin-3-ol
Show/Hide
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C21H26FNO
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1
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| 1 |
IC50 = 7000 nM
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CP0465996
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3-(4-((3,5-bis(4-(trifluoromethoxy)phenyl)-1H-pyrazol-1-yl)methyl)-N-methylbenzamido)propanoic acid
Show/Hide
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C29H23F6N3O5
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1
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| 1 |
IC50 = 7200 nM
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CP0478585
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3-(4-((5-cyclohexyl-1-(4-(trifluoromethoxy)phenyl)-1H-pyrazol-4-yl)methyl)benzamido)propanoic acid
Show/Hide
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C27H28F3N3O4
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1
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| 1 |
IC50 = 7200 nM
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CP0469502
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2-[[4-[(1R)-1-[8-tert-butyl-2-(3,5-dichlorophenyl)-3-oxo-1,4-diazaspiro[4.5]dec-1-en-4-yl]-4,4-dimethylpentyl]benzoyl]amino]ethanesulfonic acid
Show/Hide
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C34H45Cl2N3O5S
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1
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| 1 |
IC50 = 8500 nM
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CP0541984
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[4-(2-fluorophenyl)-5-pentyl-2,6-di(propan-2-yl)pyridin-3-yl]methanol
Show/Hide
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C23H32FNO
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1
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| 1 |
IC50 = 9000 nM
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CP0395570
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4-[(1R)-1-[8-tert-butyl-2-(3,5-dichlorophenyl)-3-oxo-1,4-diazaspiro[4.5]dec-1-en-4-yl]-4,4-dimethylpentyl]-N-[(1S)-1-(2H-tetrazol-5-yl)ethyl]benzamide
Show/Hide
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C35H45Cl2N7O2
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1
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| 1 |
IC50 > 10000 nM
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CP0411601
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(3S)-3-[[4-[(1R)-1-[8-tert-butyl-2-(3,5-dichlorophenyl)-3-oxo-1,4-diazaspiro[4.5]dec-1-en-4-yl]-4,4-dimethylpentyl]benzoyl]amino]butanoic acid
Show/Hide
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C36H47Cl2N3O4
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1
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| 1 |
IC50 > 10000 nM
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CP0511104
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[4-(2,4-difluorophenyl)-5-pentyl-2,6-di(propan-2-yl)pyridin-3-yl]methanol
Show/Hide
|
C23H31F2NO
|
1
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| 1 |
IC50 = 11000 nM
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CP0378510
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4-((5-cyclohexyl-1-(4-(trifluoromethoxy)phenyl)-1H-pyrazol-4-yl)methyl)-N-(2H-tetrazol-5-yl)benzamide
Show/Hide
|
C25H24F3N7O2
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1
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| 1 |
IC50 = 16000 nM
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CP0488974
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[2-fluoro-5-[3-(hydroxymethyl)-5-pentyl-2,6-di(propan-2-yl)pyridin-4-yl]phenyl]methanol
Show/Hide
|
C24H34FNO2
|
1
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| 1 |
IC50 = 19000 nM
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CP0390915
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4-Bromo-N-[3-cyano-6-(1,1-dimethyl-propyl)-4,5,6,7-tetrahydro-benzo[b]thiophen-2-yl]-benzamide
Show/Hide
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C21H23BrN2OS
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1
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| 1 |
IC50 > 20000 nM
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CP0466514
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[4-(3-methoxyphenyl)-5-pentyl-2,6-di(propan-2-yl)pyridin-3-yl]methanol
Show/Hide
|
C24H35NO2
|
1
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| 1 |
IC50 = 48000 nM
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CP0440531
|
4-((methyl(1-methyl-1H-benzo[d]imidazol-2-yl)amino)methyl)-N-(1H-tetrazol-5-yl)benzamide
Show/Hide
|
C18H18N8O
|
1
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| 1 |
IC50 > 1000 nM
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CP0522763
|
N-[3-chloro-4-(4-chlorophenoxy)phenyl]-4-phenyl-1,3-thiazol-2-amine
Show/Hide
|
C21H14Cl2N2OS
|
1
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| 1 |
IC50 > 1000 nM
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CP0050171
|
4-[4-(4-Fluoro-phenyl)-5-pyridin-4-yl-1H-pyrrol-2-yl]-benzoic acid
Show/Hide
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C22H15FN2O2
|
1
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| 1 |
IC50 > 3000 nM
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CP0085243
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4-[3-(4-Fluoro-phenyl)-5-methyl-1H-pyrrol-2-yl]-pyridine
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C16H13FN2
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1
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| 1 |
IC50 > 3000 nM
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CP0251081
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5-(4-Chloro-phenyl)-2-pyridin-4-yl-1H-pyrrole-3-carboxylic acid
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C16H11ClN2O2
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1
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| 1 |
IC50 > 3000 nM
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CP0436200
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5-(4-Chloro-phenyl)-2-pyridin-4-yl-1H-pyrrole-3-carboxylic acid benzylamide
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C23H18ClN3O
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1
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| 1 |
IC50 > 3000 nM
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CP0271630
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4-[3-(4-Fluoro-phenyl)-1H-pyrrol-2-yl]-pyridine
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C15H11FN2
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1
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| 1 |
IC50 > 3000 nM
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