Brief Information of the Compound and Protein
Compound Name
3-[[4-[(2S)-2-[5-chloro-1-[6-(trifluoromethyl)pyridin-2-yl]indole-2-carbonyl]pentyl]benzoyl]amino]propanoic acid
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PubChem ID
CID: 57399594
Canonical SMILES
CCC[C@@H](Cc1ccc(cc1)C(=O)NCCC(O)=O)C(=O)c1cc2cc(Cl)ccc2n1-c1cccc(n1)C(F)(F)F
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Compound Formula C30H27ClF3N3O4
Compound Structure
Protein Name
Glucagon receptor
Protein Classification
Membrane receptor
>
Family B G protein-coupled receptor
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Peptide receptor (family B GPCR)
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Glucagon-like receptor
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Glucagon receptor
Uniprot ID
P47871
Gene Name
GCGR
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  2
1
IC50 = 9.2 nM
   TI
   LI
   LO
   TS
2
IC50 = 34 nM
   TI
   LI
   LO
   TS