Brief Information of the Compound and Protein
Compound Name
3-[[4-[1-[3-(2-chloro-5-fluorophenyl)-6-[4-(trifluoromethoxy)phenyl]indazol-1-yl]ethyl]benzoyl]amino]propanoic acid
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PubChem ID
CID: 122189694
Canonical SMILES
CC(c1ccc(cc1)C(=O)NCCC(O)=O)n1nc(-c2cc(F)ccc2Cl)c2ccc(cc12)-c1ccc(OC(F)(F)F)cc1
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Compound Formula C32H24ClF4N3O4
Compound Structure
Protein Name
Glucagon receptor
Protein Classification
Membrane receptor
>
Family B G protein-coupled receptor
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Peptide receptor (family B GPCR)
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Glucagon-like receptor
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Glucagon receptor
Uniprot ID
P47871
Gene Name
GCGR
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  2
1
IC50 = 10 nM
   TI
   LI
   LO
   TS
2
IC50 = 140 nM
   TI
   LI
   LO
   TS