Brief Information of the Compound and Protein
Compound Name
3-[[4-[2-[5-chloro-1-(2,3-dihydro-1,4-benzodioxin-6-yl)indole-2-carbonyl]pentyl]benzoyl]amino]propanoic acid
    Show/Hide
PubChem ID
CID: 16224781
SID: 24907288
Canonical SMILES
CCCC(Cc1ccc(cc1)C(=O)NCCC(O)=O)C(=O)c1cc2cc(Cl)ccc2n1-c1ccc2OCCOc2c1
    Show/Hide
Compound Formula C32H31ClN2O6
Compound Structure
Protein Name
Glucagon receptor
Protein Classification
Membrane receptor
>
Family B G protein-coupled receptor
>
Peptide receptor (family B GPCR)
>
Glucagon-like receptor
>
Glucagon receptor
Uniprot ID
P47871
Gene Name
GCGR
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  2
1
IC50 = 28 nM
   TI
   LI
   LO
   TS
2
IC50 = 49 nM
   TI
   LI
   LO
   TS