Brief Information of the Compound and Protein
Compound Name
 Compound Info 
4-[[(4-tert-butylcyclohexyl)-(1,5,6-trimethylbenzimidazol-2-yl)amino]methyl]-N-(2H-tetrazol-5-yl)benzamide
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Canonical SMILES
Cc1cc2nc(N(Cc3ccc(cc3)C(=O)Nc3nnn[nH]3)[C@H]3CC[C@@H](CC3)C(C)(C)C)n(C)c2cc1C
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Compound Formula C29H38N8O
Compound Structure
Protein Name
 Protein Info 
Glucagon receptor
Protein Classification
Membrane receptor
>
Family B G protein-coupled receptor
>
Peptide receptor (family B GPCR)
>
Glucagon-like receptor
>
Glucagon receptor
Uniprot ID
P47871
Gene Name
GCGR
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO
 Cell Line Info 
Cricetulus griseus (Chinese hamster)  2
1
IC50 = 6 nM
   TI
   LI
   LO
   TS
2
IC50 = 18 nM
   TI
   LI
   LO
   TS