Brief Information of the Compound and Protein
Compound Name
N-[3-cyano-4-methyl-5-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]thiophen-2-yl]-2-ethylbutanamide
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PubChem ID
CID: 10383925
SID: 15399234
Canonical SMILES
CCC(CC)C(=O)Nc1sc(c(C)c1C#N)-c1nc(CC(C)C)no1
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Compound Formula C18H24N4O2S
Compound Structure
Protein Name
Glucagon receptor
Protein Classification
Membrane receptor
>
Family B G protein-coupled receptor
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Peptide receptor (family B GPCR)
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Glucagon-like receptor
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Glucagon receptor
Uniprot ID
P47871
Gene Name
GCGR
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  2
1
IC50 = 185 nM
   TI
   LI
   LO
   TS
2
IC50 = 368 nM
   TI
   LI
   LO
   TS