Brief Information of the Compound and Protein
Compound Name
5-Fluoro-2-(3-hydroxymethyl-2,6-diisopropyl-5-pentyl-pyridin-4-yl)-phenol
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PubChem ID
CID: 135819137
Canonical SMILES
CCCCCc1c(nc(C(C)C)c(CO)c1-c1ccc(F)cc1O)C(C)C
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Compound Formula C23H32FNO2
Compound Structure
Protein Name
Glucagon receptor
Protein Classification
Membrane receptor
>
Family B G protein-coupled receptor
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Peptide receptor (family B GPCR)
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Glucagon-like receptor
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Glucagon receptor
Uniprot ID
P47871
Gene Name
GCGR
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  2
1
IC50 = 120 nM
   TI
   LI
   LO
   TS
2
IC50 = 190 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 IC50 = 190 nM