Brief Information of the Compound and Protein
Compound Name
4-[[N-(5,6-dichloro-1-methylbenzimidazol-2-yl)-4-(trifluoromethoxy)anilino]methyl]-N-(2H-tetrazol-5-yl)benzamide
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PubChem ID
CID: 57403704
Canonical SMILES
Cn1c(nc2cc(Cl)c(Cl)cc12)N(Cc1ccc(cc1)C(=O)Nc1nnn[nH]1)c1ccc(OC(F)(F)F)cc1
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Compound Formula C24H17Cl2F3N8O2
Compound Structure
Protein Name
Glucagon receptor
Protein Classification
Membrane receptor
>
Family B G protein-coupled receptor
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Peptide receptor (family B GPCR)
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Glucagon-like receptor
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Glucagon receptor
Uniprot ID
P47871
Gene Name
GCGR
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  2
1
IC50 = 19 nM
   TI
   LI
   LO
   TS
2
IC50 = 670 nM
   TI
   LI
   LO
   TS