Brief Information of the Compound and Protein
Compound Name
N-[3-cyano-6-[(2,4-dichlorophenyl)methyl-propan-2-ylamino]-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-2-ethylbutanamide
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PubChem ID
CID: 10413333
SID: 15431030
Canonical SMILES
CCC(CC)C(=O)Nc1sc2CC(CCc2c1C#N)N(Cc1ccc(Cl)cc1Cl)C(C)C
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Compound Formula C25H31Cl2N3OS
Compound Structure
Protein Name
Glucagon receptor
Protein Classification
Membrane receptor
>
Family B G protein-coupled receptor
>
Peptide receptor (family B GPCR)
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Glucagon-like receptor
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Glucagon receptor
Uniprot ID
P47871
Gene Name
GCGR
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  2
1
IC50 = 59 nM
   TI
   LI
   LO
   TS
2
IC50 = 129 nM
   TI
   LI
   LO
   TS