Brief Information of the Compound and Protein
Compound Name
4-((5-cyclohexyl-3-(4-(trifluoromethoxy)phenyl)-1H-pyrazol-1-yl)methyl)-N-(2H-tetrazol-5-yl)benzamide
    Show/Hide
PubChem ID
CID: 10324097
SID: 15333613
Canonical SMILES
FC(F)(F)Oc1ccc(cc1)-c1cc(C2CCCCC2)n(Cc2ccc(cc2)C(=O)Nc2nnn[nH]2)n1
    Show/Hide
Compound Formula C25H24F3N7O2
Compound Structure
Protein Name
Glucagon receptor
Protein Classification
Membrane receptor
>
Family B G protein-coupled receptor
>
Peptide receptor (family B GPCR)
>
Glucagon-like receptor
>
Glucagon receptor
Uniprot ID
P47871
Gene Name
GCGR
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  2
1
IC50 = 120 nM
   TI
   LI
   LO
   TS
2
IC50 = 160 nM
   TI
   LI
   LO
   TS