Brief Information of the Compound and Protein
Compound Name
 Compound Info 
4-[[(5-bromo-1-methylbenzimidazol-2-yl)-(4-tert-butylcyclohexyl)amino]methyl]-N-(2H-tetrazol-5-yl)benzamide
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Canonical SMILES
Cn1c(nc2cc(Br)ccc12)N(Cc1ccc(cc1)C(=O)Nc1nnn[nH]1)[C@H]1CC[C@@H](CC1)C(C)(C)C
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Compound Formula C27H33BrN8O
Compound Structure
Protein Name
 Protein Info 
Glucagon receptor
Protein Classification
Membrane receptor
>
Family B G protein-coupled receptor
>
Peptide receptor (family B GPCR)
>
Glucagon-like receptor
>
Glucagon receptor
Uniprot ID
P47871
Gene Name
GCGR
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO
 Cell Line Info 
Cricetulus griseus (Chinese hamster)  2
1
IC50 = 7 nM
   TI
   LI
   LO
   TS
2
IC50 = 62 nM
   TI
   LI
   LO
   TS