Brief Information of the Cell Line and Protein
Cell Line ID: CL000011 , CHO
Synonyms
Chinese Hamster Ovary
CHO-ori
Category Spontaneously immortalized cell line
Organism
Cricetulus griseus (Chinese hamster)
Cellosaurus ID
CVCL_0213
Protein ID: PT01102 , Voltage-dependent L-type calcium channel subunit alpha-1C
Gene Name CACNA1C
Organism Homo sapiens, Human
Protein Classification Ion channel
Uniprot ID Q13936
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000011  Protein ID: PT01102
 
Compound ID Compound Name Compound Formula
CP0072914
US20230414632, Compound I-e
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C20H24N2O6
 1
1
IC50 = 3 nM
   TI
   LI
   LO
   TS
CP0046619
Adalat
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C17H18N2O6
 1
1
IC50 = 50 nM
   TI
   LI
   LO
   TS
CP0454037
10-[4-(2,1,3-benzoxadiazol-4-yl)-2,6-dimethyl-5-propan-2-yloxycarbonyl-1,4-dihydropyridine-3-carbonyl]oxydecyl-trimethylazanium
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C31H47N4O5+
 1
1
IC50 = 70 nM
   TI
   LI
   LO
   TS
CP0406371
Pinaverium
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C26H41BrNO4+
 1
1
IC50 = 1750 nM
   TI
   LI
   LO
   TS
CP0002225
Doribax
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C15H24N4O6S2
 1
1
IC50 = 1995.26 nM
   TI
   LI
   LO
   TS
CP0013111
ADL 8-2698
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C25H32N2O4
 1
1
IC50 = 5011.87 nM
   TI
   LI
   LO
   TS
CP0002227
SOLIFENACIN
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C23H26N2O2
 1
1
IC50 = 6309.57 nM
   TI
   LI
   LO
   TS
CP0002231
2-{2-ethoxy-5-[(4-ethylpiperazine-1-)sulfonyl]phenyl}-5-methyl-7-propyl-3H,4H-imidazo[1,5-a][1,2,4]triazin-4-one
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C23H32N6O4S
 1
1
IC50 = 15848.93 nM
   TI
   LI
   LO
   TS
CP0036382
CAS_52-53-9
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C27H38N2O4
 1
1
IC50 = 23500 nM
   TI
   LI
   LO
   TS
CP0271660
(R)-1-(Methylsulfonylamino)-3-[2-(4-methoxyphenyl)ethyl]-4-(4-methoxy-phenyl)-2-imidazolidinone
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C20H25N3O5S
 1
1
IC50 > 30000 nM
   TI
   LI
   LO
   TS
CP0010753
N-[[1-[2-(tert-butylcarbamoylamino)ethyl]-4-(hydroxymethyl)piperidin-4-yl]methyl]-3,5-dichlorobenzamide
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C21H32Cl2N4O3
 1
1
IC50 > 31600 nM
   TI
   LI
   LO
   TS
CP0014435
(2R)-2-acetylamino-N-benzyl-3-methoxypropanamide
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C13H18N2O3
 1
1
IC50 = 50118.72 nM
   TI
   LI
   LO
   TS
CP0002211
N-[2-(diethylamino)ethyl]-5-[(Z)-(5-fluoro-2-oxo-1H-indol-3-ylidene)methyl]-2,4-dimethyl-1H-pyrrole-3-carboxamide
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C22H27FN4O2
 1
1
IC50 = 79432.82 nM
   TI
   LI
   LO
   TS
CP0008168
CAS_136434-34-9
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C18H19NOS
 1
1
IC50 = 100000 nM
   TI
   LI
   LO
   TS
CP0010658
5-[2-ethoxy-5-(4-methyl-1-piperazinylsulfonyl)phenyl]-1-methyl-3-n-propyl-1,6-dihydro-7H-pyrazolo[4,3-d]pyrimidin-7-one
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C22H30N6O4S
 1
1
IC50 = 100000 nM
   TI
   LI
   LO
   TS