| Compound ID |
Compound Name |
Compound Formula |
|
CP0015176
|
3-[2-[(N-ethyl-4-fluoroanilino)methyl]-5-methyl-7-oxothieno[2,3-c]pyridin-6-yl]propanenitrile
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|
C20H20FN3OS
|
1
|
| 1 |
IC50 = 610 nM
|
|
|
|
CP0015330
|
3-[2-[(N-ethyl-4-fluoroanilino)methyl]-4-oxothieno[3,2-c]pyridin-5-yl]propanenitrile
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|
C19H18FN3OS
|
1
|
| 1 |
IC50 = 610 nM
|
|
|
|
CP0015363
|
3-[2-[(N-ethyl-4-fluoroanilino)methyl]-7-fluoro-4-oxopyrazolo[1,5-a]pyrazin-5-yl]propanenitrile
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|
C18H17F2N5O
|
1
|
| 1 |
IC50 = 2800 nM
|
|
|
|
CP0015152
|
3-[2-[[5-chloro-3-(trifluoromethyl)pyrazol-1-yl]methyl]-7-methyl-4-oxopyrazolo[1,5-a]pyrazin-5-yl]propanenitrile
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|
C15H12ClF3N6O
|
1
|
| 1 |
IC50 = 19000 nM
|
|
|
|
CP0014796
|
3-[2-[(N-ethyl-4-fluoroanilino)methyl]-4-oxopyrazolo[1,5-a]pyrazin-5-yl]propanenitrile
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|
C18H18FN5O
|
1
|
| 1 |
IC50 = 22000 nM
|
|
|
|
CP0015308
|
3-[2-[(N-ethyl-4-fluoroanilino)methyl]-7-methyl-4-oxopyrazolo[1,5-a]pyrazin-5-yl]propanenitrile
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|
C19H20FN5O
|
1
|
| 1 |
IC50 = 22000 nM
|
|
|
|
CP0013234
|
(3R)-3-[2-[[5-chloro-3-(difluoromethyl)pyrazol-1-yl]methyl]-7-methyl-4-oxopyrazolo[1,5-a]pyrazin-5-yl]butanenitrile
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|
C16H15ClF2N6O
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
|
CP0014797
|
3-[2-[(N-ethyl-4-fluoroanilino)methyl]-4-methyl-7-oxothieno[2,3-c]pyridin-6-yl]propanenitrile
Show/Hide
|
C20H20FN3OS
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
|
CP0015153
|
3-[2-[(3-bromo-5-chloropyrazol-1-yl)methyl]-7-methyl-4-oxopyrazolo[1,5-a]pyrazin-5-yl]propanenitrile
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|
C14H12BrClN6O
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
|
CP0015174
|
3-[2-[(N-ethyl-4-fluoroanilino)methyl]-7-oxothieno[2,3-c]pyridin-6-yl]propanenitrile
Show/Hide
|
C19H18FN3OS
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
|
CP0015175
|
3-[4-ethyl-2-[(N-ethyl-4-fluoroanilino)methyl]-7-oxothieno[2,3-c]pyridin-6-yl]propanenitrile
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|
C21H22FN3OS
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
|
CP0015177
|
3-[2-[(5-chloro-3-methylpyrazol-1-yl)methyl]-7-methyl-4-oxopyrazolo[1,5-a]pyrazin-5-yl]propanenitrile
Show/Hide
|
C15H15ClN6O
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
|
CP0015178
|
(3S)-3-[2-[[5-chloro-3-(difluoromethyl)pyrazol-1-yl]methyl]-7-methyl-4-oxopyrazolo[1,5-a]pyrazin-5-yl]butanenitrile
Show/Hide
|
C16H15ClF2N6O
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
|
CP0015179
|
2-[2-[(N-ethyl-4-fluoroanilino)methyl]-7-oxothieno[2,3-c]pyridin-6-yl]acetonitrile
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|
C18H16FN3OS
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
|
CP0015203
|
3-[2-[(3,5-dichloropyrazol-1-yl)methyl]-7-methyl-4-oxopyrazolo[1,5-a]pyrazin-5-yl]propanenitrile
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|
C14H12Cl2N6O
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
|
CP0015329
|
3-[2-[[5-chloro-3-(difluoromethyl)pyrazol-1-yl]methyl]-7-methyl-4-oxopyrazolo[1,5-a]pyrazin-5-yl]propanenitrile
Show/Hide
|
C15H13ClF2N6O
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
