Brief Information of the Compound and Protein
Compound Name
 Compound Info 
3-[2-[[5-chloro-3-(trifluoromethyl)pyrazol-1-yl]methyl]-7-methyl-4-oxopyrazolo[1,5-a]pyrazin-5-yl]propanenitrile
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 PubChem ID
CID: 168285906
Canonical SMILES
Cc1cn(CCC#N)c(=O)c2cc(Cn3nc(cc3Cl)C(F)(F)F)nn12
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Compound Formula C15H12ClF3N6O
Compound Structure
Protein Name
 Protein Info 
Glutamate receptor 2
Protein Classification
Ion channel
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Ligand-gated ion channel
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Ionotropic glutamate receptor
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AMPA receptor
Uniprot ID
P42262
Gene Name
GRIA2
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO
 Cell Line Info 
Cricetulus griseus (Chinese hamster)  1
1
IC50 = 19000 nM
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