Brief Information of the Compound and Protein
Compound Name
(3S)-3-[2-[[5-chloro-3-(difluoromethyl)pyrazol-1-yl]methyl]-7-methyl-4-oxopyrazolo[1,5-a]pyrazin-5-yl]butanenitrile
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PubChem ID
CID: 166625943
Canonical SMILES
C[C@@H](CC#N)n1cc(C)n2nc(Cn3nc(cc3Cl)C(F)F)cc2c1=O
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Compound Formula C16H15ClF2N6O
Compound Structure
Protein Name
Glutamate receptor 2
Protein Classification
Ion channel
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Ligand-gated ion channel
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Ionotropic glutamate receptor
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AMPA receptor
Uniprot ID
P42262
Gene Name
GRIA2
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
IC50 > 30000 nM
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   LI
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