| Compound ID |
Compound Name |
Compound Formula |
|
CP0943875
|
[2-fluoro-3-(2-morpholinopyrimidin-5-yl)phenyl]methyl-N-carbamimidoylcarbamate hydrochloride
Show/Hide
|
C17H20ClFN6O3
|
1
|
| 1 |
IC50 = 9.2 nM
|
|
|
|
CP0956592
|
3-[4-(Pyridin-4-yl)piperazin-1-yl]benzyl-N-carbamimidoylcarbamate trihydrochloride
Show/Hide
|
C18H25Cl3N6O2
|
1
|
| 1 |
IC50 = 13 nM
|
|
|
|
CP0904633
|
2-Fluoro-3-[4-(pyridin-3-yl)piperazin-1-yl]benzyl-N-carbamimidoylcarbamate (2R,3R)-tartrate
Show/Hide
|
C22H27FN6O8
|
1
|
| 1 |
IC50 = 17 nM
|
|
|
|
CP0658461
|
N-[4-(2-{4-[(2-Amino-1H-imidazol-4-yl)methyl]phenyl}ethyl)thiazol-2-yl]acetamide hydrochloride
Show/Hide
|
C17H20ClN5OS
|
1
|
| 1 |
IC50 = 19 nM
|
|
|
|
CP0049270
|
2-phenylethylhydrazine
Show/Hide
|
C8H12N2
|
1
|
| 1 |
IC50 = 19.95 nM
|
|
|
|
CP0456931
|
N-[4-[2-[4-(diaminomethylideneamino)phenyl]ethyl]-5-[(4-methylsulfonylphenyl)methyl]-1,3-thiazol-2-yl]acetamide
Show/Hide
|
C22H25N5O3S2
|
1
|
| 1 |
IC50 = 20 nM
|
|
|
|
CP0860492
|
2-Fluoro-3-[3-(pyridin-3-yloxy)azetidin-1-yl]benzyl-N-carbamimidoylcarbamate hemi(2R,3R)-tartrate
Show/Hide
|
C38H42F2N10O12
|
1
|
| 1 |
IC50 = 24 nM
|
|
|
|
CP0954479
|
4-{4-[5-(3-{[Glycyl(methyl)amino]methyl}phenyl)pyrimidin-2-yl]piperazin-1-yl}benzoic acid dihydrochloride
Show/Hide
|
C25H30Cl2N6O3
|
1
|
| 1 |
IC50 = 24 nM
|
|
|
|
CP0905705
|
2-Fluoro-3-{3-[(6-methylpyridin-3-yl)oxy]azetidin-1-yl}benzyl-N-carbamimidoylcarbamate (2R,3R)-tartrate
Show/Hide
|
C22H26FN5O9
|
1
|
| 1 |
IC50 = 25 nM
|
|
|
|
CP0904605
|
3-Chloro-4-{4-[5-(3-{[glycyl(methyl)amino]methyl}phenyl)pyrimidin-2-yl]piperazin-1-yl}benzoic acid dihydrochloride
Show/Hide
|
C25H29Cl3N6O3
|
1
|
| 1 |
IC50 = 25 nM
|
|
|
|
CP0473477
|
2-hydrazinyl-1-(4-methoxyphenyl)ethanol
Show/Hide
|
C9H14N2O2
|
1
|
| 1 |
IC50 = 28.84 nM
|
|
|
|
CP0948428
|
2-amino-N-methyl-N-(3-(2-morpholinopyrimidin-5-yl)benzyl)acetamide (2R,3R)-tartrate
Show/Hide
|
C22H29N5O8
|
1
|
| 1 |
IC50 = 31 nM
|
|
|
|
CP0965396
|
3-[4-(Pyridin-3-yl)piperazin-1-yl]benzyl-N-carbamimidoylcarbamate trihydrochloride
Show/Hide
|
C18H25Cl3N6O2
|
1
|
| 1 |
IC50 = 31 nM
|
|
|
|
CP0915844
|
N-Methyl-N-{3-[2-(morpholin-4-yl)pyrimidin-5-yl]benzyl}glycinamide (2R,3R)-tartrate
Show/Hide
|
C22H29N5O8
|
1
|
| 1 |
IC50 = 31 nM
|
|
|
|
CP0901202
|
N-{4-[2-(4-{[Amino(imino)methyl]amino}phenyl)ethyl]-5-[4-(methylsulfonyl)phenyl]-1,3-thiazol-2-yl}acetamidehydrochloride
Show/Hide
|
C21H24ClN5O3S2
|
1
|
| 1 |
IC50 = 34 nM
|
|
|
|
CP0465625
|
N-[4-[2-[4-(diaminomethylideneamino)phenyl]ethyl]-5-[(3-methylsulfonylphenyl)methyl]-1,3-thiazol-2-yl]acetamide
Show/Hide
|
C22H25N5O3S2
|
1
|
| 1 |
IC50 = 36 nM
|
|
|
|
CP0466202
|
(R)-2-Hydrazino-1-phenylethanol
Show/Hide
|
C8H12N2O
|
1
|
| 1 |
IC50 = 40 nM
|
|
|
|
CP0960957
|
2-Fluoro-3-{3-[(2-methylpyridin-3-yl)oxy]azetidin-1-yl}benzyl-N-carbamimidoylcarbamate (2R,3R)-tartrate
Show/Hide
|
C22H26FN5O9
|
1
|
| 1 |
IC50 = 40 nM
|
|
|
|
CP0965533
|
2-Fluoro-3-[4-(pyridin-3-yloxy)piperidin-1-yl]benzyl-N-carbamimidoylcarbamate (2R,3R)-tartrate
Show/Hide
|
C23H28FN5O9
|
1
|
| 1 |
IC50 = 45 nM
|
|
|
|
CP0857302
|
N-(3-{2-[4-(2-Hydroxyethyl)piperidin-1-yl]pyrimidin-5-yl}benzyl)-N-methylglycinamide (2R,3R)-tartrate
Show/Hide
|
C25H35N5O8
|
1
|
| 1 |
IC50 = 45 nM
|
|
|
|
CP0947025
|
[3-(2-morpholinopyrimidin-5-yl)phenyl]methyl N-carbamimidoylcarbamate (2R,3R)-tartrate
Show/Hide
|
C21H26N6O9
|
1
|
| 1 |
IC50 = 47 nM
|
|
|
|
CP0492979
|
2-hydrazinyl-1-(3-methoxyphenyl)ethanol
Show/Hide
|
C9H14N2O2
|
1
|
| 1 |
IC50 = 52.48 nM
|
|
|
|
CP0900912
|
N-{4-[2-(4-{[Amino(imino)methyl]amino}phenyl)ethyl]-5-[4-(aminosulfonyl)benzyl]-1,3-thiazol-2-yl}acetamidehydrochloride
Show/Hide
|
C21H25ClN6O3S2
|
1
|
| 1 |
IC50 = 53 nM
|
|
|
|
CP0956589
|
N-Carbamimidoyl-2-(3-{2-[2-(morpholin-4-yl)pyrimidin-5-yl]ethyl}phenyl)acetamide hemi(2R,3R)-tartrate
Show/Hide
|
C42H54N12O10
|
1
|
| 1 |
IC50 = 54 nM
|
|
|
|
CP0946801
|
N-Methyl-N-{3-[6-(morpholin-4-yl)pyridin-3-yl]benzyl}glycinamide (2R,3R)-tartrate
Show/Hide
|
C23H30N4O8
|
1
|
| 1 |
IC50 = 55 nM
|
|
|
|
CP0862694
|
N-Carbamimidoyl-2-{3-[2-(morpholin-4-yl)pyrimidin-5-yl]phenyl}acetamide (2R,3R)-tartrate
Show/Hide
|
C21H26N6O8
|
1
|
| 1 |
IC50 = 56 nM
|
|
|
|
CP0522093
|
2-phenylpropylhydrazine
Show/Hide
|
C9H14N2
|
1
|
| 1 |
IC50 = 58.88 nM
|
|
|
|
CP0533344
|
1-[2-(4-methoxyphenyl)ethyl]-1-methylhydrazine
Show/Hide
|
C10H16N2O
|
1
|
| 1 |
IC50 = 60.26 nM
|
|
|
|
CP0912480
|
2-Hydrazino-1-phenylethanol
Show/Hide
|
C8H12N2O
|
1
|
| 1 |
IC50 = 64.57 nM
|
|
|
|
CP0488637
|
1-[2-(4-chlorophenyl)ethyl]-1-methylhydrazine
Show/Hide
|
C9H13ClN2
|
1
|
| 1 |
IC50 = 70.79 nM
|
|
|
|
CP0956590
|
2,4-Difluoro-3-[2-(morpholin-4-yl)pyrimidin-5-yl]benzylcarbamimidoylcarbamate hemi(2R,3R)-tartrate
Show/Hide
|
C38H42F4N12O12
|
1
|
| 1 |
IC50 = 77 nM
|
|
|
|
CP0473478
|
1-ethyl-1-[2-(4-methoxyphenyl)ethyl]hydrazine
Show/Hide
|
C11H18N2O
|
1
|
| 1 |
IC50 = 79.43 nM
|
|
|
|
CP0967423
|
N-(3'-{[Glycyl(methyl)amino]methyl}biphenyl-4-yl)morpholine-4-carboxamide ethanedioate
Show/Hide
|
C23H28N4O7
|
1
|
| 1 |
IC50 = 83 nM
|
|
|
|
CP0488636
|
1-[2-(3-methoxyphenyl)ethyl]-1-methylhydrazine
Show/Hide
|
C10H16N2O
|
1
|
| 1 |
IC50 = 89.13 nM
|
|
|
|
CP0513558
|
1-[2-(2-fluorophenyl)ethyl]-1-methylhydrazine
Show/Hide
|
C9H13FN2
|
1
|
| 1 |
IC50 = 91.2 nM
|
|
|
|
CP0915494
|
[4-fluoro-3-(2-morpholinopyrimidin-5-yl)phenyl]methyl-N-carbamimidoylcarbamate dihydrochloride
Show/Hide
|
C17H21Cl2FN6O3
|
1
|
| 1 |
IC50 = 99 nM
|
|
|
|
CP0492983
|
1-[2-(4-fluorophenyl)ethyl]-1-methylhydrazine
Show/Hide
|
C9H13FN2
|
1
|
| 1 |
IC50 = 109.65 nM
|
|
|
|
CP0492984
|
1-methyl-1-(2-phenylethyl)hydrazine
Show/Hide
|
C9H14N2
|
1
|
| 1 |
IC50 = 109.65 nM
|
|
|
|
CP0904632
|
3-[4-(Tetrahydro-2H-pyran-4-yl)piperazin-1-yl]benzyl-N-carbamimidoylcarbamate (2R,3R)-tartrate
Show/Hide
|
C22H33N5O9
|
1
|
| 1 |
IC50 = 110 nM
|
|
|
|
CP0406047
|
1-[2-(3-chlorophenyl)ethyl]-1-methylhydrazine
Show/Hide
|
C9H13ClN2
|
1
|
| 1 |
IC50 = 120.23 nM
|
|
|
|
CP0954478
|
N-{3-[2-(4-Hydroxypiperidin-1-yl)pyrimidin-5-yl]benzyl}-N-methylglycinamide (2R,3R)-tartrate
Show/Hide
|
C23H31N5O8
|
1
|
| 1 |
IC50 = 130 nM
|
|
|
|
CP0860491
|
3-[4-(Pyridin-2-yl)piperazin-1-yl]benzyl-N-carbamimidoylcarbamate trihydrochloride
Show/Hide
|
C18H25Cl3N6O2
|
1
|
| 1 |
IC50 = 140 nM
|
|
|
|
CP0964602
|
3-{1-[5-(3-{[Glycyl(methyl)amino]methyl}phenyl)pyrimidin-2-yl]piperidin-4-yl}propanoic acid dihydrochloride
Show/Hide
|
C22H31Cl2N5O3
|
1
|
| 1 |
IC50 = 140 nM
|
|
|
|
CP0460357
|
(S)-2-Hydrazino-1-phenylethanol
Show/Hide
|
C8H12N2O
|
1
|
| 1 |
IC50 = 150 nM
|
|
|
|
CP0900911
|
N-(4-[2-(4-{[Amino(imino)methyl]amino}phenyl)ethyl]-5-{4-[(dimethylamino)sulfonyl]benzyl}-1,3-thiazol-2-yl)acetamide hydrochloride
Show/Hide
|
C23H29ClN6O3S2
|
1
|
| 1 |
IC50 = 150 nM
|
|
|
|
CP0940284
|
N-(4-[2-(4-{[Amino(imino)methyl]amino}phenyl)ethyl]-5-{2-[4-(methylsulfonyl)phenyl]ethyl}-1,3-thiazol-2-yl)acetamide hydrochloride
Show/Hide
|
C23H28ClN5O3S2
|
1
|
| 1 |
IC50 = 160 nM
|
|
|
|
CP0956591
|
3-[4-(Morpholin-4-yl)piperidin-1-yl]benzyl-N-carbamimidoylcarbamate trihydrochloride
Show/Hide
|
C18H30Cl3N5O3
|
1
|
| 1 |
IC50 = 160 nM
|
|
|
|
CP0509285
|
1-[2-(2-chlorophenyl)ethyl]-1-methylhydrazine
Show/Hide
|
C9H13ClN2
|
1
|
| 1 |
IC50 = 169.82 nM
|
|
|
|
CP0887128
|
N-(Biphenyl-3-ylmethyl)glycinamide hydrochloride
Show/Hide
|
C15H17ClN2O
|
1
|
| 1 |
IC50 = 180 nM
|
|
|
|
CP0492981
|
1-ethyl-1-(2-phenylethyl)hydrazine
Show/Hide
|
C10H16N2
|
1
|
| 1 |
IC50 = 181.97 nM
|
|
|
|
CP0501967
|
2-[amino(methyl)amino]-1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethanol
Show/Hide
|
C11H16N2O3
|
1
|
| 1 |
IC50 = 199.53 nM
|
|
|
|
CP0406044
|
2-[amino(methyl)amino]-1-phenylethanol
Show/Hide
|
C9H14N2O
|
1
|
| 1 |
IC50 = 208.93 nM
|
|
|
|
CP0900922
|
N-{4-[2-(4-{[Amino(imino)methyl]amino}phenyl)ethyl]-5-benzyl-1,3-thiazol-2-yl}acetamide hydrochloride
Show/Hide
|
C21H24ClN5OS
|
1
|
| 1 |
IC50 = 210 nM
|
|
|
|
CP0492973
|
2-[amino(methyl)amino]-1-(2,3,4-trimethoxyphenyl)ethanol
Show/Hide
|
C12H20N2O4
|
1
|
| 1 |
IC50 = 218.78 nM
|
|
|
|
CP0533335
|
1-(2-methoxy-2-naphthalen-2-ylethyl)-1-methylhydrazine
Show/Hide
|
C14H18N2O
|
1
|
| 1 |
IC50 = 229.09 nM
|
|
|
|
CP0200164
|
N-[4-[2-[4-(diaminomethylideneamino)phenyl]ethyl]-1,3-thiazol-2-yl]acetamide
Show/Hide
|
C14H17N5OS
|
1
|
| 1 |
IC50 = 230 nM
|
|
|
|
CP0493610
|
1-methyl-1-(3-phenylpropyl)hydrazine
Show/Hide
|
C10H16N2
|
1
|
| 1 |
IC50 = 239.88 nM
|
|
|
|
CP0900663
|
N-[(4'-Chlorobiphenyl-3-yl)methyl]-N-methylglycinamide hydrochloride
Show/Hide
|
C16H18Cl2N2O
|
1
|
| 1 |
IC50 = 240 nM
|
|
|
|
CP0541504
|
2-[[3-[2-[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]pyrimidin-5-yl]phenyl]methyl-methylamino]acetamide;dihydrochloride
Show/Hide
|
C19H27Cl2N5O2
|
1
|
| 1 |
IC50 = 240 nM
|
|
|
|
CP0911121
|
N-Methyl-N-{3-[2-(piperidin-1-yl)pyrimidin-5-yl]benzyl}glycinamide dihydrochloride
Show/Hide
|
C19H27Cl2N5O
|
1
|
| 1 |
IC50 = 250 nM
|
|
|
|
CP0406045
|
1-[2-(4-methoxyphenyl)ethyl]-1-(2-methylpropyl)hydrazine
Show/Hide
|
C13H22N2O
|
1
|
| 1 |
IC50 = 257.04 nM
|
|
|
|
CP0492969
|
(1R,2S)-2-[amino(methyl)amino]-1-phenylbutan-1-ol
Show/Hide
|
C11H18N2O
|
1
|
| 1 |
IC50 = 257.04 nM
|
|
|
|
CP0522092
|
(1R,2S)-2-[amino(methyl)amino]-1-phenylpentan-1-ol
Show/Hide
|
C12H20N2O
|
1
|
| 1 |
IC50 = 257.04 nM
|
|
|
|
CP0406043
|
2-[amino(methyl)amino]-1-(2-chlorophenyl)ethanol
Show/Hide
|
C9H13ClN2O
|
1
|
| 1 |
IC50 = 269.15 nM
|
|
|
|
CP0492968
|
1-benzyl-1-methylhydrazine
Show/Hide
|
C8H12N2
|
1
|
| 1 |
IC50 = 269.15 nM
|
|
|
|
CP0486828
|
(1R,2S)-2-(1-Methylhydrazino)-1,2-diphenylethanol
Show/Hide
|
C15H18N2O
|
1
|
| 1 |
IC50 = 280 nM
|
|
|
|
CP0930280
|
N-({4'-[(Dimethylcarbamoyl)amino]biphenyl-3-yl}methyl)-N-methylglycinamide ethanedioate
Show/Hide
|
C21H26N4O6
|
1
|
| 1 |
IC50 = 280 nM
|
|
|
|
CP0406042
|
2-[amino(methyl)amino]-1-(3-methoxyphenyl)ethanol
Show/Hide
|
C10H16N2O2
|
1
|
| 1 |
IC50 = 281.84 nM
|
|
|
|
CP0541499
|
2-[[3-[2-[(2R)-2-(hydroxymethyl)pyrrolidin-1-yl]pyrimidin-5-yl]phenyl]methyl-methylamino]acetamide;dihydrochloride
Show/Hide
|
C19H27Cl2N5O2
|
1
|
| 1 |
IC50 = 300 nM
|
|
|
|
CP0492976
|
2-[amino(methyl)amino]-1-(4-methoxyphenyl)ethanol
Show/Hide
|
C10H16N2O2
|
1
|
| 1 |
IC50 = 309.03 nM
|
|
|
|
CP0509283
|
2-[amino(methyl)amino]-1-(4-chlorophenyl)ethanol
Show/Hide
|
C9H13ClN2O
|
1
|
| 1 |
IC50 = 309.03 nM
|
|
|
|
CP0940898
|
Methyl 4-({2-(acetylamino)-4-[2-(4-{[amino(imino)methyl]amino}phenyl)ethyl]-1,3-thiazol-5-yl}methyl)benzoatehydrochloride
Show/Hide
|
C23H26ClN5O3S
|
1
|
| 1 |
IC50 = 320 nM
|
|
|
|
CP0493609
|
2-[amino(methyl)amino]-1-(4-fluorophenyl)ethanol
Show/Hide
|
C9H13FN2O
|
1
|
| 1 |
IC50 = 323.59 nM
|
|
|
|
CP0509284
|
1-methyl-1-[2-(3,4,5-trimethoxyphenyl)ethyl]hydrazine
Show/Hide
|
C12H20N2O3
|
1
|
| 1 |
IC50 = 323.59 nM
|
|
|
|
CP0522091
|
1-[2-methoxy-2-(3-methylphenyl)ethyl]-1-methylhydrazine
Show/Hide
|
C11H18N2O
|
1
|
| 1 |
IC50 = 323.59 nM
|
|
|
|
CP0520902
|
(1S,2R)-2-(1-Methylhydrazino)-1,2-diphenylethanol
Show/Hide
|
C15H18N2O
|
1
|
| 1 |
IC50 = 330 nM
|
|
|
|
CP0908166
|
N-{4-[4-(2-{[Amino(imino)methyl]amino}ethyl)phenyl]-1,3-thiazol-2-yl}acetamide hydrochloride
Show/Hide
|
C14H18ClN5OS
|
1
|
| 1 |
IC50 = 330 nM
|
|
|
|
CP0897696
|
N-Methyl-N-{[4'-(4-methylpiperazin-1-yl)biphenyl-3-yl]methyl}glycinamide (2R,3R)-tartrate
Show/Hide
|
C25H34N4O7
|
1
|
| 1 |
IC50 = 330 nM
|
|
|
|
CP0531259
|
1-methyl-1-[2-(2,3,4-trimethoxyphenyl)ethyl]hydrazine
Show/Hide
|
C12H20N2O3
|
1
|
| 1 |
IC50 = 331.13 nM
|
|
|
|
CP0906413
|
N-Methyl-N-{[4'-(morpholin-4-yl)biphenyl-3-yl]methyl}glycinamide ethanedioate
Show/Hide
|
C22H27N3O6
|
1
|
| 1 |
IC50 = 340 nM
|
|
|
|
CP0406093
|
1-[amino(methyl)amino]-2-(4-methoxyphenyl)propan-2-ol
Show/Hide
|
C11H18N2O2
|
1
|
| 1 |
IC50 = 346.74 nM
|
|
|
|
CP0479553
|
(1R,2S)-2-[amino(methyl)amino]-1-phenylpropan-1-ol
Show/Hide
|
C10H16N2O
|
1
|
| 1 |
IC50 = 346.74 nM
|
|
|
|
CP0492971
|
2-[amino(2-methylpropyl)amino]-1-phenylethanol
Show/Hide
|
C12H20N2O
|
1
|
| 1 |
IC50 = 346.74 nM
|
|
|
|
CP0493611
|
1-[2-(2-methoxyphenyl)ethyl]-1-methylhydrazine
Show/Hide
|
C10H16N2O
|
1
|
| 1 |
IC50 = 346.74 nM
|
|
|
|
CP0508013
|
1-[2-(3,4-dimethoxyphenyl)ethyl]-1-methylhydrazine
Show/Hide
|
C11H18N2O2
|
1
|
| 1 |
IC50 = 346.74 nM
|
|
|
|
CP0492982
|
1-[2-(2,5-dimethoxyphenyl)ethyl]-1-methylhydrazine
Show/Hide
|
C11H18N2O2
|
1
|
| 1 |
IC50 = 371.54 nM
|
|
|
|
CP0492874
|
1-[2-(4-methoxyphenyl)-2-phenylmethoxyethyl]-1-methylhydrazine
Show/Hide
|
C17H22N2O2
|
1
|
| 1 |
IC50 = 389.05 nM
|
|
|
|
CP0857184
|
N-{1-[2-(4-Carbamimidamidophenyl)ethyl]-5-[4-(methylsulfonyl)phenyl]-1H-pyrazol-3-yl}acetamidehydrochloride
Show/Hide
|
C21H25ClN6O3S
|
1
|
| 1 |
IC50 = 390 nM
|
|
|
|
CP0509282
|
1-(2-methoxy-2-naphthalen-1-ylethyl)-1-methylhydrazine
Show/Hide
|
C14H18N2O
|
1
|
| 1 |
IC50 = 398.11 nM
|
|
|
|
CP0860490
|
[2-fluoro-3-(4-methyl-2-morpholino-pyrimidin-5-yl)phenyl]methyl N-carbamimidoylcarbamate (2R,3R)-tartrate
Show/Hide
|
C22H27FN6O9
|
1
|
| 1 |
IC50 = 400 nM
|
|
|
|
CP0513555
|
1-[2-methoxy-2-(3-methoxyphenyl)ethyl]-1-methylhydrazine
Show/Hide
|
C11H18N2O2
|
1
|
| 1 |
IC50 = 407.38 nM
|
|
|
|
CP0513557
|
1-[2-(3-chlorophenyl)-2-methoxyethyl]-1-methylhydrazine
Show/Hide
|
C10H15ClN2O
|
1
|
| 1 |
IC50 = 407.38 nM
|
|
|
|
CP0903574
|
[2-methyl-3-(2-morpholinopyrimidin-5-yl)phenyl]methyl-N-carbamimidoylcarbamate (2R,3R)-tartrate
Show/Hide
|
C22H28N6O9
|
1
|
| 1 |
IC50 = 410 nM
|
|
|
|
CP0520877
|
1-[2-methoxy-2-(4-methoxyphenyl)ethyl]-1-methylhydrazine
Show/Hide
|
C11H18N2O2
|
1
|
| 1 |
IC50 = 416.87 nM
|
|
|
|
CP0917664
|
N-Methyl-N-{[4'-(morpholin-4-ylcarbonyl)biphenyl-3-yl]methyl}glycinamide (2R,3R)-tartrate
Show/Hide
|
C25H31N3O9
|
1
|
| 1 |
IC50 = 420 nM
|
|
|
|
CP0406041
|
2-[amino(methyl)amino]-1-naphthalen-2-ylethanol
Show/Hide
|
C13H16N2O
|
1
|
| 1 |
IC50 = 426.58 nM
|
|
|
|
CP0513556
|
1-[2-(4-chlorophenyl)-2-methoxyethyl]-1-methylhydrazine
Show/Hide
|
C10H15ClN2O
|
1
|
| 1 |
IC50 = 426.58 nM
|
|
|
|
CP0406046
|
1-(2-methylpropyl)-1-(2-phenylethyl)hydrazine
Show/Hide
|
C12H20N2
|
1
|
| 1 |
IC50 = 436.52 nM
|
|
|
|
CP0520879
|
1-[2-(3-fluorophenyl)-2-methoxyethyl]-1-methylhydrazine
Show/Hide
|
C10H15FN2O
|
1
|
| 1 |
IC50 = 436.52 nM
|
|
|
|
CP0958224
|
N-[(4'-Acetamidobiphenyl-3-yl)methyl]-N-methylglycinamide hydrochloride
Show/Hide
|
C18H22ClN3O2
|
1
|
| 1 |
IC50 = 460 nM
|
|
|
|
CP0502138
|
1-methyl-1-(2-phenylpropyl)hydrazine
Show/Hide
|
C10H16N2
|
1
|
| 1 |
IC50 = 467.74 nM
|
|
|
|
CP0899707
|
N-({4'-[(Diethylamino)methyl]biphenyl-3-yl}methyl)-Nmethylglycinamide dihydrochloride
Show/Hide
|
C21H31Cl2N3O
|
1
|
| 1 |
IC50 = 480 nM
|
|
|
|
CP0431910
|
N-[4-[2-[4-(diaminomethylideneamino)phenyl]ethyl]-1,3-thiazol-2-yl]-2-methylpropanamide
Show/Hide
|
C16H21N5OS
|
1
|
| 1 |
IC50 = 520 nM
|
|
|
|
CP0878529
|
3-Carbamimidoyl-1-methyl-1-{3-[2-(morpholin-4-yl)pyrimidin-5-yl]benzyl}urea (2R,3R)-tartrate
Show/Hide
|
C22H29N7O8
|
1
|
| 1 |
IC50 = 530 nM
|
|
|
|
CP0962609
|
N,N-Diethyl-3'-{[glycyl(methyl)amino]methyl}biphenyl-4-carboxamide ethanedioate
Show/Hide
|
C23H29N3O6
|
1
|
| 1 |
IC50 = 560 nM
|
|
|
|
CP0473476
|
2-[amino(methyl)amino]-2-methyl-1-phenylpropan-1-ol
Show/Hide
|
C11H18N2O
|
1
|
| 1 |
IC50 = 562.34 nM
|
|
|
|
CP0520878
|
1-[2-(4-fluorophenyl)-2-methoxyethyl]-1-methylhydrazine
Show/Hide
|
C10H15FN2O
|
1
|
| 1 |
IC50 = 575.44 nM
|
|
|
|
CP0860489
|
[2-chloro-3-(2-morpholinopyrimidin-5-yl)phenyl]methyl N-carbamimidoylcarbamate dihydrochloride
Show/Hide
|
C17H21Cl3N6O3
|
1
|
| 1 |
IC50 = 600 nM
|
|
|
|
CP0952405
|
N-Ethyl-3'-{[glycyl(methyl)amino]methyl}biphenyl-4-carboxamide hydrochloride
Show/Hide
|
C19H24ClN3O2
|
1
|
| 1 |
IC50 = 610 nM
|
|
|
|
CP0473475
|
1-[2-methoxy-2-(2,3,4-trimethoxyphenyl)ethyl]-1-methylhydrazine
Show/Hide
|
C13H22N2O4
|
1
|
| 1 |
IC50 = 630.96 nM
|
|
|
|
CP0462379
|
N-[4-[2-[4-[(N'-ethylcarbamimidoyl)amino]phenyl]ethyl]-1,3-thiazol-2-yl]acetamide
Show/Hide
|
C16H21N5OS
|
1
|
| 1 |
IC50 = 680 nM
|
|
|
|
CP0522738
|
N-[4-[2-[4-(aminomethylideneamino)phenyl]ethyl]-1,3-thiazol-2-yl]acetamide
Show/Hide
|
C14H16N4OS
|
1
|
| 1 |
IC50 = 730 nM
|
|
|
|
CP0573219
|
2-amino-N-methyl-N-[(3-phenylphenyl)methyl]acetamide
Show/Hide
|
C16H18N2O
|
1
|
| 1 |
IC50 = 800 nM
|
|
|
|
CP0494328
|
(1R,2R)-2-(1-Methylhydrazino)-1,2-diphenylethanol
Show/Hide
|
C15H18N2O
|
1
|
| 1 |
IC50 = 1060 nM
|
|
|
|
CP0505475
|
N-[4-[2-[4-[(N'-propan-2-ylcarbamimidoyl)amino]phenyl]ethyl]-1,3-thiazol-2-yl]acetamide
Show/Hide
|
C17H23N5OS
|
1
|
| 1 |
IC50 = 1100 nM
|
|
|
|
CP0908167
|
Methyl N-{4-[2-(2-acetamido-1,3-thiazol-4-yl)ethyl]phenyl}carbamimidothioate hydroiodide
Show/Hide
|
C15H19IN4OS2
|
1
|
| 1 |
IC50 = 1100 nM
|
|
|
|
CP0386177
|
N-[4-[2-[4-(diaminomethylideneamino)phenyl]ethyl]-5-[(4-methylsulfanylphenyl)methyl]-1,3-thiazol-2-yl]acetamide
Show/Hide
|
C22H25N5OS2
|
1
|
| 1 |
IC50 = 1100 nM
|
|
|
|
CP0513246
|
(1S,2S)-2-(1-Methylhydrazino)-1,2-diphenylethanol
Show/Hide
|
C15H18N2O
|
1
|
| 1 |
IC50 = 1180 nM
|
|
|
|
CP0478597
|
2-Hydrazino-1-phenylpentanol
Show/Hide
|
C11H18N2O
|
1
|
| 1 |
IC50 = 1200 nM
|
|
|
|
CP0528271
|
[5-(3-methylsulfonyl-5-phenylphenyl)sulfonyl-1,3-thiazol-2-yl]methanamine
Show/Hide
|
C17H16N2O4S3
|
1
|
| 1 |
IC50 = 1200 nM
|
|
|
|
CP0967422
|
N-[(3'-Chlorobiphenyl-3-yl)methyl]-N-methylglycinamide ethanedioate
Show/Hide
|
C18H19ClN2O5
|
1
|
| 1 |
IC50 = 1300 nM
|
|
|
|
CP0439960
|
[5-[3-(4-methylphenyl)-5-methylsulfonylphenyl]sulfonyl-1,3-thiazol-2-yl]methanamine
Show/Hide
|
C18H18N2O4S3
|
1
|
| 1 |
IC50 = 1300 nM
|
|
|
|
CP0867965
|
N-Methyl-N-({5-[4-(morpholin-4-yl)phenyl]pyridin-3-yl}methyl)glycinamide (2R,3R)-tartrate
Show/Hide
|
C23H30N4O8
|
1
|
| 1 |
IC50 = 1500 nM
|
|
|
|
CP0930370
|
3'-{[Glycyl(methyl)amino]methyl}biphenyl-4-carboxamide hydrochloride
Show/Hide
|
C17H20ClN3O2
|
1
|
| 1 |
IC50 = 1600 nM
|
|
|
|
CP0904616
|
1-[5-(3-{[Glycyl(methyl)amino]methyl}phenyl)pyrimidin-2-yl]piperidine-4-carboxylic acid dihydrochloride
Show/Hide
|
C20H27Cl2N5O3
|
1
|
| 1 |
IC50 = 1700 nM
|
|
|
|
CP0901840
|
N-Methyl-N-{[4'-(morpholin-4-yl)biphenyl-3-yl]methyl}ethane-1,2-diamine (2R,3R)-tartrate
Show/Hide
|
C24H33N3O7
|
1
|
| 1 |
IC50 = 1800 nM
|
|
|
|
CP0962610
|
2-Amino-1-{5-[4-(morpholin-4-yl)phenyl]-1,3-dihydro-2H-isoindol-2-yl}ethanone hydrochloride
Show/Hide
|
C20H24ClN3O2
|
1
|
| 1 |
IC50 = 2000 nM
|
|
|
|
CP0852596
|
N-Methyl-N-({6-[4-(morpholin-4-yl)phenyl]pyridin-2-yl}methyl)glycinamide dihydrochloride
Show/Hide
|
C19H26Cl2N4O2
|
1
|
| 1 |
IC50 = 2000 nM
|
|
|
|
CP0456932
|
N-[1-(4-fluorophenyl)-5-(4-methylsulfonylphenyl)pyrazol-3-yl]acetamide
Show/Hide
|
C18H16FN3O3S
|
1
|
| 1 |
IC50 = 2100 nM
|
|
|
|
CP0949294
|
N-[4-(2-{4-[(2-Amino-1H-imidazol-4-yl)ethyl]phenyl}ethyl)thiazol-2-yl]acetamide hydrochloride
Show/Hide
|
C18H22ClN5OS
|
1
|
| 1 |
IC50 = 2200 nM
|
|
|
|
CP0492980
|
1-ethyl-1-[2-(3,4,5-trimethoxyphenyl)ethyl]hydrazine
Show/Hide
|
C13H22N2O3
|
1
|
| 1 |
IC50 = 2238.72 nM
|
|
|
|
CP0433342
|
N-[4-[2-[4-(4,5-dihydro-1H-imidazol-2-ylamino)phenyl]ethyl]-1,3-thiazol-2-yl]acetamide
Show/Hide
|
C16H19N5OS
|
1
|
| 1 |
IC50 = 3000 nM
|
|
|
|
CP0967412
|
N-{[4'-(Dimethylamino)biphenyl-3-yl]methyl}-N-methylglycinamide ethanedioate
Show/Hide
|
C20H25N3O5
|
1
|
| 1 |
IC50 = 3000 nM
|
|
|
|
CP0431913
|
N-[4-[2-[4-(4,5-dihydro-1,3-thiazol-2-ylamino)phenyl]ethyl]-1,3-thiazol-2-yl]acetamide
Show/Hide
|
C16H18N4OS2
|
1
|
| 1 |
IC50 = 3500 nM
|
|
|
|
CP0349042
|
[5-(3-ethyl-5-phenylphenyl)sulfonyl-1,3-thiazol-2-yl]methanamine
Show/Hide
|
C18H18N2O2S2
|
1
|
| 1 |
IC50 = 3600 nM
|
|
|
|
CP0930281
|
N-Methyl-N-{[4'-(morpholin-4-yl)biphenyl-3-yl]methyl}-beta-alaninamide (2R,3R)-tartrate
Show/Hide
|
C25H33N3O8
|
1
|
| 1 |
IC50 = 4000 nM
|
|
|
|
CP0014376
|
1H-1,3-benzodiazol-2-amine
Show/Hide
|
C7H7N3
|
1
|
| 1 |
IC50 = 4100 nM
|
|
|
|
CP0923138
|
N-[(2'-Chlorobiphenyl-3-yl)methyl]-N-methylglycinamide hydrochloride
Show/Hide
|
C16H18Cl2N2O
|
1
|
| 1 |
IC50 = 4100 nM
|
|
|
|
CP0431911
|
N-[4-[2-[4-(2-aminoethyl)phenyl]ethyl]-1,3-thiazol-2-yl]acetamide
Show/Hide
|
C15H19N3OS
|
1
|
| 1 |
IC50 = 5000 nM
|
|
|
|
CP0860488
|
N-(4-{2-[2-(Morpholin-4-yl)pyrimidin-5-yl]ethyl}phenyl)guanidine dihydrochloride
Show/Hide
|
C17H24Cl2N6O
|
1
|
| 1 |
IC50 = 5100 nM
|
|
|
|
CP0920792
|
N-{4-[3-(4-{[Amino(imino)methyl]amino}phenyl)propyl]-1,3-thiazol-2-yl}acetamide hydrochloride
Show/Hide
|
C15H20ClN5OS
|
1
|
| 1 |
IC50 = 8800 nM
|
|
|
|
CP0932776
|
N-{5-[2-(4-{[Amino(imino)methyl]amino}phenyl)ethyl]-1,3-thiazol-2-yl}acetamide hydrochloride
Show/Hide
|
C14H18ClN5OS
|
1
|
| 1 |
IC50 = 9600 nM
|
|
|
|
CP0431912
|
N-[4-[2-[4-(carbamothioylamino)phenyl]ethyl]-1,3-thiazol-2-yl]acetamide
Show/Hide
|
C14H16N4OS2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0943874
|
N-[2-(3-{2-[2-(Morpholin-4-yl)pyrimidin-5-yl]ethyl}phenyl)ethyl]guanidine dihydrochloride
Show/Hide
|
C19H28Cl2N6O
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0943880
|
N-(3-{2-[2-(Morpholin-4-yl)pyrimidin-5-yl]ethyl}phenyl)guanidine dihydrochloride
Show/Hide
|
C17H24Cl2N6O
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0851035
|
N-{4-[2-(4-{[Amino(imino)methyl]amino}phenyl)ethyl]-1,3-thiazol-2-yl}benzamide hydrochloride
Show/Hide
|
C19H20ClN5OS
|
1
|
| 1 |
IC50 = 11000 nM
|
|
|
|
CP0857664
|
N-(4-{2-[4-(2-Amino-1H-imidazol-4-yl)phenyl]ethyl}thiazol-2-yl)acetamide hydrochloride
Show/Hide
|
C16H18ClN5OS
|
1
|
| 1 |
IC50 = 13000 nM
|
|
|
|
CP0384458
|
[5-[3-(1-methylpyrazol-4-yl)-5-methylsulfonylphenyl]sulfonyl-1,3-thiazol-2-yl]methanamine
Show/Hide
|
C15H16N4O4S3
|
1
|
| 1 |
IC50 = 13300 nM
|
|
|
|
CP0957621
|
3'-{[Glycyl(methyl)amino]methyl}biphenyl-4-carboxylicacid hydrochloride
Show/Hide
|
C17H19ClN2O3
|
1
|
| 1 |
IC50 = 14000 nM
|
|
|
|
CP0871650
|
N-{3-[2-(4-Carbamimidamidophenyl)ethyl]phenyl}acetamide hydrochloride
Show/Hide
|
C17H21ClN4O
|
1
|
| 1 |
IC50 = 15000 nM
|
|
|
|
CP0893965
|
N-{4-[2-(4-Carbamimidamidophenyl)ethyl]phenyl}acetamide hydrochloride
Show/Hide
|
C17H21ClN4O
|
1
|
| 1 |
IC50 = 18000 nM
|
|
|
|
CP0384459
|
[5-[3-ethyl-5-(1-methylpyrazol-4-yl)phenyl]sulfonyl-1,3-thiazol-2-yl]methanamine
Show/Hide
|
C16H18N4O2S2
|
1
|
| 1 |
IC50 = 19600 nM
|
|
|
|
CP0904144
|
1-{4-[2-(2-Amino-1,3-thiazol-4-yl)ethyl]phenyl}guanidine dihydrochloride
Show/Hide
|
C12H17Cl2N5S
|
1
|
| 1 |
IC50 = 22000 nM
|
|
|
|
CP0413873
|
5-benzyl-1H-imidazol-2-amine
Show/Hide
|
C10H11N3
|
1
|
| 1 |
IC50 = 32000 nM
|
|
|
|
CP0559457
|
[5-[3-fluoro-5-(1-methylpyrazol-4-yl)phenyl]sulfonyl-1,3-thiazol-2-yl]methanamine
Show/Hide
|
C14H13FN4O2S2
|
1
|
| 1 |
IC50 = 36300 nM
|
|
|
|
CP0920136
|
N-[4-(4-Carbamimidamidobenzyl)-1,3-thiazol-2-yl]acetamide hydrochloride
Show/Hide
|
C13H16ClN5OS
|
1
|
| 1 |
IC50 = 42000 nM
|
|
|
|
CP0528276
|
(5-naphthalen-2-ylsulfonyl-1,3-thiazol-2-yl)methanamine
Show/Hide
|
C14H12N2O2S2
|
1
|
| 1 |
IC50 = 47100 nM
|
|
|
|
CP0478596
|
(1R*,2S*)-2-Hydrazino-1,2-diphenylethanol
Show/Hide
|
C14H16N2O
|
1
|
| 1 |
IC50 = 50000 nM
|
|
|
|
CP0946353
|
1H-indol-2-amine hydrochloride
Show/Hide
|
C8H9ClN2
|
1
|
| 1 |
IC50 = 74000 nM
|
|
|
|
CP0426810
|
[4-[3-ethyl-5-(1-methylpyrazol-4-yl)phenyl]sulfonyl-1,3-thiazol-2-yl]methanamine
Show/Hide
|
C16H18N4O2S2
|
1
|
| 1 |
IC50 = 74300 nM
|
|
|
|
CP0522739
|
N-[4-[2-[4-[[amino(dimethylamino)methylidene]amino]phenyl]ethyl]-1,3-thiazol-2-yl]acetamide
Show/Hide
|
C16H21N5OS
|
1
|
| 1 |
IC50 > 100000 nM
|
|
|
|
CP0522740
|
N-[4-[2-(4-aminophenyl)ethyl]-1,3-thiazol-2-yl]acetamide
Show/Hide
|
C13H15N3OS
|
1
|
| 1 |
IC50 > 100000 nM
|
|
|
|
CP0057720
|
1,3-benzothiazol-2-amine
Show/Hide
|
C7H6N2S
|
1
|
| 1 |
IC50 > 100000 nM
|
|
|
|
CP0142371
|
1H-1,3-benzodiazole
Show/Hide
|
C7H6N2
|
1
|
| 1 |
IC50 > 100000 nM
|
|
|
|
CP0222047
|
1-phenylguanidine
Show/Hide
|
C7H9N3
|
1
|
| 1 |
IC50 > 100000 nM
|
|
|
|
CP0245992
|
quinazolin-2-amine
Show/Hide
|
C8H7N3
|
1
|
| 1 |
IC50 > 100000 nM
|
|
|
|
CP0389020
|
5-(2-phenylethyl)-1H-imidazol-2-amine
Show/Hide
|
C11H13N3
|
1
|
| 1 |
IC50 > 100000 nM
|
|
|
|
CP0418891
|
6-methyl-1H-benzimidazol-2-amine
Show/Hide
|
C8H9N3
|
1
|
| 1 |
IC50 > 100000 nM
|
|
|
|
CP0418892
|
4-methyl-1H-benzimidazol-2-amine
Show/Hide
|
C8H9N3
|
1
|
| 1 |
IC50 > 100000 nM
|
|
|
|
CP0509177
|
5-phenyl-1H-imidazol-2-amine
Show/Hide
|
C9H9N3
|
1
|
| 1 |
IC50 > 100000 nM
|
|
|
|
CP0545959
|
1-methyl-1H-1,3-benzodiazol-2-amine
Show/Hide
|
C8H9N3
|
1
|
| 1 |
IC50 > 100000 nM
|
|
|
|
CP0755319
|
(1H-benzo[d]imidazol-2-yl)methanamine dihydrochloride
Show/Hide
|
C8H11Cl2N3
|
1
|
| 1 |
IC50 > 100000 nM
|
|
|
|
CP0857663
|
1-Phenyl-imidazolidin-2-ylideneamine hydrobromide
Show/Hide
|
C9H12BrN3
|
1
|
| 1 |
IC50 > 100000 nM
|
|
|
|
CP0906015
|
N-phenyl-4,5-dihydro-1H-imidazol-2-amine hydrochloride
Show/Hide
|
C9H12ClN3
|
1
|
| 1 |
IC50 > 100000 nM
|
|
|
|
CP0946352
|
1H-imidazol-2-amine hemisulfate
Show/Hide
|
C3H7N3O4S
|
1
|
| 1 |
IC50 > 100000 nM
|
|
|
|
CP0887127
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N,N2,N2-Trimethyl-N-{[4'-(morpholin-4-yl)biphenyl-3-yl]methyl}glycinamide (2R,3R)-tartrate
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C26H35N3O8
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1
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| 1 |
IC50 > 100000 nM
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CP0901839
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N,N2-Dimethyl-N-{[4'-(morpholin-4-yl)biphenyl-3-yl]methyl}glycinamide (2R,3R)-tartrate
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C25H33N3O8
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1
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| 1 |
IC50 > 100000 nM
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CP0902848
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N,2-Dimethyl-N-{[4'-(morpholin-4-yl)biphenyl-3-yl]methyl}alaninamide (2R,3R)-tartrate
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C26H35N3O8
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1
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| 1 |
IC50 > 100000 nM
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CP0919349
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N-Isopropyl-N-{[4'-(morpholin-4-yl)biphenyl-3-yl]methyl}glycinamide (2R,3R)-tartrate
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C26H35N3O8
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1
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| 1 |
IC50 > 100000 nM
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CP0952406
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N-(2-Aminoethyl)-N-methyl-4'-(morpholin-4-yl)biphenyl-3-carboxamide (2R,3R)-tartrate
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C24H31N3O8
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1
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| 1 |
IC50 > 100000 nM
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CP0421556
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[4-(3-methylsulfonyl-5-phenylphenyl)sulfonyl-1,3-thiazol-2-yl]methanamine
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C17H16N2O4S3
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1
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| 1 |
IC50 > 100000 nM
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CP0426167
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[4-[3-(1-methylpyrazol-4-yl)-5-methylsulfonylphenyl]sulfonyl-1,3-thiazol-2-yl]methanamine
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C15H16N4O4S3
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1
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| 1 |
IC50 > 100000 nM
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