| Compound ID |
Compound Name |
Compound Formula |
|
CP0052587
|
(2R,3R)-1-[4-(2-Chloro-4-fluoro-benzyloxy)-benzenesulfonyl]-3-hydroxy-3-methyl-piperidine-2-carboxylic acid hydroxyamide
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|
C20H22ClFN2O6S
|
1
|
| 1 |
IC50 = 6.3 nM
|
|
|
|
CP0191349
|
N-[[(2R)-1-[4-(but-3-enylamino)-6-[(2-thiophen-2-yl-1,3-thiazol-4-yl)methylamino]-1,3,5-triazin-2-yl]pyrrolidin-2-yl]methyl]-4-propylbenzenesulfonamide
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|
C29H36N8O2S3
|
1
|
| 1 |
IC50 = 30 nM
|
|
|
|
CP0191351
|
N-[[(2R)-1-[4-[(1-methylimidazol-4-yl)methylamino]-6-(propylamino)-1,3,5-triazin-2-yl]pyrrolidin-2-yl]methyl]-4-propylbenzenesulfonamide
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|
C25H37N9O2S
|
1
|
| 1 |
IC50 = 30 nM
|
|
|
|
CP0191353
|
N-[[(2R)-1-[4-(but-3-enylamino)-6-[(2-thiophen-2-yl-1,3-thiazol-4-yl)methylamino]-1,3,5-triazin-2-yl]pyrrolidin-2-yl]methyl]naphthalene-2-sulfonamide
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|
C30H32N8O2S3
|
1
|
| 1 |
IC50 = 40 nM
|
|
|
|
CP0191350
|
N-[[(2R)-1-[4-(but-3-enylamino)-6-[(2-thiophen-2-yl-1,3-thiazol-4-yl)methylamino]-1,3,5-triazin-2-yl]pyrrolidin-2-yl]methyl]-4-(trifluoromethyl)benzenesulfonamide
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|
C27H29F3N8O2S3
|
1
|
| 1 |
IC50 = 50 nM
|
|
|
|
CP0446326
|
N-[[(2R)-1-[4-[(2-phenyl-1,3-thiazol-4-yl)methylamino]-6-(propylamino)-1,3,5-triazin-2-yl]pyrrolidin-2-yl]methyl]-4-propylbenzenesulfonamide
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|
C30H38N8O2S2
|
1
|
| 1 |
IC50 = 50 nM
|
|
|
|
CP0534190
|
N-[[(2R)-1-[4-(but-3-enylamino)-6-[(2-phenyl-1,3-thiazol-4-yl)methylamino]-1,3,5-triazin-2-yl]pyrrolidin-2-yl]methyl]-4-methoxybenzenesulfonamide
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|
C29H34N8O3S2
|
1
|
| 1 |
IC50 = 50 nM
|
|
|
|
CP0413961
|
N-[[(2R)-1-[4-(but-3-enylamino)-6-[(2-phenyl-1,3-thiazol-4-yl)methylamino]-1,3,5-triazin-2-yl]pyrrolidin-2-yl]methyl]-4-(trifluoromethyl)benzenesulfonamide
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|
C29H31F3N8O2S2
|
1
|
| 1 |
IC50 = 60 nM
|
|
|
|
CP0120704
|
N-[[(2R)-1-[4-(cyclopropylamino)-6-[(2-phenyl-1,3-thiazol-4-yl)methylamino]-1,3,5-triazin-2-yl]pyrrolidin-2-yl]methyl]-4-propylbenzenesulfonamide
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|
C30H36N8O2S2
|
1
|
| 1 |
IC50 = 70 nM
|
|
|
|
CP0110474
|
N-[[(2R)-1-[4-(2-cyanoethylamino)-6-[(2-phenyl-1,3-thiazol-4-yl)methylamino]-1,3,5-triazin-2-yl]pyrrolidin-2-yl]methyl]-4-propylbenzenesulfonamide
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|
C30H35N9O2S2
|
1
|
| 1 |
IC50 = 90 nM
|
|
|
|
CP0449949
|
N-[[(2R)-1-[4-(cyclopropylmethylamino)-6-[(2-thiophen-2-yl-1,3-thiazol-4-yl)methylamino]-1,3,5-triazin-2-yl]pyrrolidin-2-yl]methyl]-4-(trifluoromethyl)benzenesulfonamide
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|
C27H29F3N8O2S3
|
1
|
| 1 |
IC50 = 110 nM
|
|
|
|
CP0408592
|
N-[[(2R)-1-[4-(2-methylpropylamino)-6-[(2-phenyl-1,3-thiazol-4-yl)methylamino]-1,3,5-triazin-2-yl]pyrrolidin-2-yl]methyl]-4-propylbenzenesulfonamide
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|
C31H40N8O2S2
|
1
|
| 1 |
IC50 = 120 nM
|
|
|
|
CP0413962
|
N-[[(2R)-1-[4-(2-methoxyethylamino)-6-[(2-phenyl-1,3-thiazol-4-yl)methylamino]-1,3,5-triazin-2-yl]pyrrolidin-2-yl]methyl]-4-propylbenzenesulfonamide
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|
C30H38N8O3S2
|
1
|
| 1 |
IC50 = 210 nM
|
|
|
|
CP0523351
|
N-[[(2R)-1-[4-(but-3-enylamino)-6-[(2-phenyl-1,3-thiazol-4-yl)methylamino]-1,3,5-triazin-2-yl]pyrrolidin-2-yl]methyl]benzenesulfonamide
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|
C28H32N8O2S2
|
1
|
| 1 |
IC50 = 230 nM
|
|
|
|
CP0534192
|
N-[[(2R)-1-[4-(butylamino)-6-[(2-thiophen-2-yl-1,3-thiazol-4-yl)methylamino]-1,3,5-triazin-2-yl]pyrrolidin-2-yl]methyl]-4-(trifluoromethyl)benzenesulfonamide
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|
C27H31F3N8O2S3
|
1
|
| 1 |
IC50 = 240 nM
|
|
|
|
CP0553415
|
N-[[(2R)-1-[4-(2-hydroxyethylamino)-6-[(2-phenyl-1,3-thiazol-4-yl)methylamino]-1,3,5-triazin-2-yl]pyrrolidin-2-yl]methyl]-4-propylbenzenesulfonamide
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|
C29H36N8O3S2
|
1
|
| 1 |
IC50 = 260 nM
|
|
|
|
CP0413963
|
N-[[(2R)-1-[4-(methylamino)-6-[(2-thiophen-2-yl-1,3-thiazol-4-yl)methylamino]-1,3,5-triazin-2-yl]pyrrolidin-2-yl]methyl]-4-(trifluoromethyl)benzenesulfonamide
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|
C24H25F3N8O2S3
|
1
|
| 1 |
IC50 = 390 nM
|
|
|
|
CP0534191
|
N-[[(2R)-1-[4-(butylamino)-6-[(6-methylpyridin-2-yl)methylamino]-1,3,5-triazin-2-yl]pyrrolidin-2-yl]methyl]-4-propylbenzenesulfonamide
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|
C28H40N8O2S
|
1
|
| 1 |
IC50 = 410 nM
|
|
|
|
CP0553414
|
N-[[(2R)-1-[4-(but-3-enylamino)-6-[(2-methyl-1,3-thiazol-4-yl)methylamino]-1,3,5-triazin-2-yl]pyrrolidin-2-yl]methyl]-4-(trifluoromethyl)benzenesulfonamide
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|
C24H29F3N8O2S2
|
1
|
| 1 |
IC50 = 430 nM
|
|
|
|
CP0523350
|
N-[[(2R)-1-[4-(butylamino)-6-[(2-thiophen-2-yl-1,3-thiazol-4-yl)methylamino]-1,3,5-triazin-2-yl]pyrrolidin-2-yl]methyl]-4-chlorobenzenesulfonamide
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|
C26H31ClN8O2S3
|
1
|
| 1 |
IC50 = 460 nM
|
|
|
|
CP0513291
|
N-[[(2R)-1-[4-(butylamino)-6-[(2-thiophen-2-yl-1,3-thiazol-4-yl)methylamino]-1,3,5-triazin-2-yl]pyrrolidin-2-yl]methyl]-3-chlorobenzenesulfonamide
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|
C26H31ClN8O2S3
|
1
|
| 1 |
IC50 = 700 nM
|
|
|
|
CP0553411
|
N-[[(2R)-1-[4-(butylamino)-6-[(2-thiophen-2-yl-1,3-thiazol-4-yl)methylamino]-1,3,5-triazin-2-yl]pyrrolidin-2-yl]methyl]-3,4-dimethylbenzenesulfonamide
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|
C28H36N8O2S3
|
1
|
| 1 |
IC50 = 720 nM
|
|
|
|
CP0553413
|
N-[[(2R)-1-[4-(benzylamino)-6-(but-3-enylamino)-1,3,5-triazin-2-yl]pyrrolidin-2-yl]methyl]-4-(trifluoromethyl)benzenesulfonamide
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|
C26H30F3N7O2S
|
1
|
| 1 |
IC50 = 870 nM
|
|
|
|
CP0396384
|
N-[[(2R)-1-[4-(butylamino)-6-(thiophen-3-ylmethylamino)-1,3,5-triazin-2-yl]pyrrolidin-2-yl]methyl]-4-propylbenzenesulfonamide
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|
C26H37N7O2S2
|
1
|
| 1 |
IC50 = 1170 nM
|
|
|
|
CP0413955
|
N-[[(2R)-1-[4-(butylamino)-6-[(2-thiophen-2-yl-1,3-thiazol-4-yl)methylamino]-1,3,5-triazin-2-yl]pyrrolidin-2-yl]methyl]-4-phenylbenzenesulfonamide
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|
C32H36N8O2S3
|
1
|
| 1 |
IC50 = 1250 nM
|
|
|
|
CP0446323
|
N-[[(2R)-1-[4-(butylamino)-6-[(2-thiophen-2-yl-1,3-thiazol-4-yl)methylamino]-1,3,5-triazin-2-yl]pyrrolidin-2-yl]methyl]-4-fluorobenzenesulfonamide
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|
C26H31FN8O2S3
|
1
|
| 1 |
IC50 = 1500 nM
|
|
|
|
CP0553412
|
N-[[(2S)-1-[4-(but-3-enylamino)-6-[(2-phenyl-1,3-thiazol-4-yl)methylamino]-1,3,5-triazin-2-yl]pyrrolidin-2-yl]methyl]-4-(trifluoromethyl)benzenesulfonamide
Show/Hide
|
C29H31F3N8O2S2
|
1
|
| 1 |
IC50 = 1560 nM
|
|
|
|
CP0413954
|
N-[[(2R)-1-[4-(butylamino)-6-[(2-thiophen-2-yl-1,3-thiazol-4-yl)methylamino]-1,3,5-triazin-2-yl]pyrrolidin-2-yl]methyl]-3-hydroxybenzenesulfonamide
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|
C26H32N8O3S3
|
1
|
| 1 |
IC50 = 1600 nM
|
|
|
|
CP0446325
|
N-[[(2R)-1-[4-(cyclopentylamino)-6-[(2-phenyl-1,3-thiazol-4-yl)methylamino]-1,3,5-triazin-2-yl]pyrrolidin-2-yl]methyl]-4-propylbenzenesulfonamide
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|
C32H40N8O2S2
|
1
|
| 1 |
IC50 = 1600 nM
|
|
|
|
CP0513290
|
N-[[(2R)-1-[4-(butylamino)-6-[(2-thiophen-2-yl-1,3-thiazol-4-yl)methylamino]-1,3,5-triazin-2-yl]pyrrolidin-2-yl]methyl]-4-cyanobenzenesulfonamide
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|
C27H31N9O2S3
|
1
|
| 1 |
IC50 = 1800 nM
|
|
|
|
CP0523355
|
N-[[(2R)-1-[4-(oxan-4-ylmethylamino)-6-[(2-phenyl-1,3-thiazol-4-yl)methylamino]-1,3,5-triazin-2-yl]pyrrolidin-2-yl]methyl]-4-propylbenzenesulfonamide
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|
C33H42N8O3S2
|
1
|
| 1 |
IC50 = 2140 nM
|
|
|
|
CP0408577
|
N-[[(2R)-1-[4-(butylamino)-6-[(2-thiophen-2-yl-1,3-thiazol-4-yl)methylamino]-1,3,5-triazin-2-yl]pyrrolidin-2-yl]methyl]-4-hydroxybenzenesulfonamide
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|
C26H32N8O3S3
|
1
|
| 1 |
IC50 = 2600 nM
|
|
|
|
CP0515629
|
N-[[(2R)-1-[4-[(2-thiophen-2-yl-1,3-thiazol-4-yl)methylamino]-1,3,5-triazin-2-yl]pyrrolidin-2-yl]methyl]-4-(trifluoromethyl)benzenesulfonamide
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|
C23H22F3N7O2S3
|
1
|
| 1 |
IC50 = 3500 nM
|
|
|
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CP0523356
|
N-[[(2R)-1-[4-(2-cyclopropylethylamino)-6-[(2-phenyl-1,3-thiazol-4-yl)methylamino]-1,3,5-triazin-2-yl]pyrrolidin-2-yl]methyl]-4-propylbenzenesulfonamide
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|
C32H40N8O2S2
|
1
|
| 1 |
IC50 = 3800 nM
|
|
|
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CP0396382
|
N-[[(2R)-1-[4-(butylamino)-6-[(2-thiophen-2-yl-1,3-thiazol-4-yl)methylamino]-1,3,5-triazin-2-yl]pyrrolidin-2-yl]methyl]-3-cyanobenzenesulfonamide
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|
C27H31N9O2S3
|
1
|
| 1 |
IC50 = 4100 nM
|
|
|
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CP0413957
|
N-[[(2R)-1-[4-(butylamino)-6-[(4-cyanothiophen-2-yl)methylamino]-1,3,5-triazin-2-yl]pyrrolidin-2-yl]methyl]-4-propylbenzenesulfonamide
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|
C27H36N8O2S2
|
1
|
| 1 |
IC50 = 4100 nM
|
|
|
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CP0513898
|
N-[[(2R)-1-[4-(butylamino)-6-[(2-thiophen-2-yl-1,3-thiazol-4-yl)methylamino]-1,3,5-triazin-2-yl]pyrrolidin-2-yl]methyl]-4-methylsulfonylbenzenesulfonamide
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|
C27H34N8O4S4
|
1
|
| 1 |
IC50 = 5300 nM
|
|
|
|
CP0523357
|
N-[[(2R)-1-[2-oxo-6-[(2-thiophen-2-yl-1,3-thiazol-4-yl)methylamino]-1H-1,3,5-triazin-4-yl]pyrrolidin-2-yl]methyl]-4-(trifluoromethyl)benzenesulfonamide
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|
C23H22F3N7O3S3
|
1
|
| 1 |
IC50 = 5300 nM
|
|
|
|
CP0452222
|
N-[[(2R)-1-[4-(butylamino)-6-(propan-2-ylamino)-1,3,5-triazin-2-yl]pyrrolidin-2-yl]methyl]-4-propylbenzenesulfonamide
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|
C24H39N7O2S
|
1
|
| 1 |
IC50 = 5800 nM
|
|
|
|
CP0446324
|
N-[[(2R)-1-[4-(butylamino)-6-(cyclopropylmethylamino)-1,3,5-triazin-2-yl]pyrrolidin-2-yl]methyl]-4-propylbenzenesulfonamide
Show/Hide
|
C25H39N7O2S
|
1
|
| 1 |
IC50 = 6500 nM
|
|
|
|
CP0413956
|
N-[[(2R)-1-[4-(butylamino)-6-(cyclopentylamino)-1,3,5-triazin-2-yl]pyrrolidin-2-yl]methyl]-4-propylbenzenesulfonamide
Show/Hide
|
C26H41N7O2S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0413959
|
N-[[(2R)-1-[4-(but-3-enylamino)-6-[(3-phenylphenyl)methylamino]-1,3,5-triazin-2-yl]pyrrolidin-2-yl]methyl]-4-(trifluoromethyl)benzenesulfonamide
Show/Hide
|
C32H34F3N7O2S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0449935
|
N-[[(2R)-1-[4-(but-3-enylamino)-6-[(2-phenyl-1,3-thiazol-4-yl)methylamino]-1,3,5-triazin-2-yl]pyrrolidin-2-yl]methyl]-3-(trifluoromethyl)benzenesulfonamide
Show/Hide
|
C29H31F3N8O2S2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0449936
|
N-[[(2R)-1-[4-(butylamino)-6-[(4-butylphenyl)methylamino]-1,3,5-triazin-2-yl]pyrrolidin-2-yl]methyl]-4-propylbenzenesulfonamide
Show/Hide
|
C32H47N7O2S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
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CP0452223
|
N-[[(2R)-1-[4-(butylamino)-6-[(4-methylthiophen-2-yl)methylamino]-1,3,5-triazin-2-yl]pyrrolidin-2-yl]methyl]-4-propylbenzenesulfonamide
Show/Hide
|
C27H39N7O2S2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0513292
|
N-[[(2R)-1-[4-(but-3-enylamino)-6-[(2-phenyl-1,3-thiazol-4-yl)methylamino]-1,3,5-triazin-2-yl]pyrrolidin-2-yl]methyl]-2-(trifluoromethyl)benzenesulfonamide
Show/Hide
|
C29H31F3N8O2S2
|
1
|
| 1 |
IC50 > 10000 nM
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|
|
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CP0513293
|
3-fluoro-4-methyl-N-[(3R)-1-[4-(2-naphthalen-1-ylethylamino)-6-[[(3S)-2-oxoazepan-3-yl]amino]-1,3,5-triazin-2-yl]pyrrolidin-3-yl]benzenesulfonamide
Show/Hide
|
C32H37FN8O3S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0513846
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N-[[(2R)-1-[4-[methyl(propyl)amino]-6-[(2-phenyl-1,3-thiazol-4-yl)methylamino]-1,3,5-triazin-2-yl]pyrrolidin-2-yl]methyl]-4-propylbenzenesulfonamide
Show/Hide
|
C31H40N8O2S2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
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CP0513901
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N-[(3R)-1-[4-(benzylamino)-6-[[(3S)-2-oxoazepan-3-yl]amino]-1,3,5-triazin-2-yl]pyrrolidin-3-yl]-3-fluoro-4-methylbenzenesulfonamide
Show/Hide
|
C27H33FN8O3S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
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CP0523352
|
N-[[(3R)-1-[4-(but-3-enylamino)-6-[(2-phenyl-1,3-thiazol-4-yl)methylamino]-1,3,5-triazin-2-yl]pyrrolidin-3-yl]methyl]-4-(trifluoromethyl)benzenesulfonamide
Show/Hide
|
C29H31F3N8O2S2
|
1
|
| 1 |
IC50 > 10000 nM
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|
|
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CP0523353
|
N-[[(2R)-1-[4-(butylamino)-6-[(3-methylphenyl)methylamino]-1,3,5-triazin-2-yl]pyrrolidin-2-yl]methyl]-4-propylbenzenesulfonamide
Show/Hide
|
C29H41N7O2S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
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CP0523354
|
N-[[(2R)-1-[4-(but-3-enylamino)-6-[(4-phenylphenyl)methylamino]-1,3,5-triazin-2-yl]pyrrolidin-2-yl]methyl]-4-(trifluoromethyl)benzenesulfonamide
Show/Hide
|
C32H34F3N7O2S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
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CP0545199
|
N-[[(2R)-1-[4-(but-3-enylamino)-6-[(2-phenyl-1,3-thiazol-4-yl)methylamino]-1,3,5-triazin-2-yl]pyrrolidin-2-yl]methyl]cyclopropanesulfonamide
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C25H32N8O2S2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
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CP0545200
|
N-[[(3S)-1-[4-(but-3-enylamino)-6-[(2-phenyl-1,3-thiazol-4-yl)methylamino]-1,3,5-triazin-2-yl]pyrrolidin-3-yl]methyl]-4-(trifluoromethyl)benzenesulfonamide
Show/Hide
|
C29H31F3N8O2S2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
