| Compound ID |
Compound Name |
Compound Formula |
|
CP0155420
|
N-(2,3-dichlorophenyl)-2-[4-[4-(2-methylimidazol-1-yl)phenyl]triazol-1-yl]acetamide
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|
C20H16Cl2N6O
|
2
|
| 1 |
EC50 = 12 nM
|
|
|
| 2 |
EC50 = 25 nM
|
|
|
|
CP0432996
|
N-(2,3-dichlorophenyl)-2-[4-[4-(4-methylimidazol-1-yl)phenyl]triazol-1-yl]acetamide
Show/Hide
|
C20H16Cl2N6O
|
2
|
| 1 |
EC50 = 14 nM
|
|
|
| 2 |
EC50 = 34 nM
|
|
|
|
CP0475865
|
N-(2,3-dichlorophenyl)-2-[4-(4-imidazol-1-ylphenyl)triazol-1-yl]acetamide
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|
C19H14Cl2N6O
|
2
|
| 1 |
EC50 = 16 nM
|
|
|
| 2 |
EC50 = 26 nM
|
|
|
|
CP0155419
|
N-(2,3-dichlorophenyl)-2-[4-[6-(2-methylimidazol-1-yl)pyridin-3-yl]triazol-1-yl]acetamide
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|
C19H15Cl2N7O
|
1
|
| 1 |
EC50 = 24 nM
|
|
|
|
CP0094466
|
N-(2,3-dichlorophenyl)-2-[4-[3-fluoro-4-(4-methylimidazol-1-yl)phenyl]triazol-1-yl]acetamide
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|
C20H15Cl2FN6O
|
2
|
| 1 |
EC50 = 32 nM
|
|
|
| 2 |
EC50 = 38 nM
|
|
|
|
CP0419292
|
N-(2,3-dichlorophenyl)-2-[4-[3-methoxy-4-(4-methylimidazol-1-yl)phenyl]triazol-1-yl]acetamide
Show/Hide
|
C21H18Cl2N6O2
|
2
|
| 1 |
EC50 = 40 nM
|
|
|
| 2 |
EC50 = 77 nM
|
|
|
|
CP0433029
|
N-(2,3-dimethylphenyl)-2-[4-[3-methoxy-4-(4-methylimidazol-1-yl)phenyl]triazol-1-yl]acetamide
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|
C23H24N6O2
|
2
|
| 1 |
EC50 = 70 nM
|
|
|
| 2 |
EC50 = 115 nM
|
|
|
|
CP0419296
|
N-(2,3-dichlorophenyl)-2-[4-[2-fluoro-4-(4-methylimidazol-1-yl)phenyl]triazol-1-yl]acetamide
Show/Hide
|
C20H15Cl2FN6O
|
2
|
| 1 |
EC50 = 77 nM
|
|
|
| 2 |
EC50 = 79 nM
|
|
|
|
CP0008174
|
2-[4-[3-methoxy-4-(4-methylimidazol-1-yl)phenyl]triazol-1-yl]-N-naphthalen-1-ylacetamide
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|
C25H22N6O2
|
2
|
| 1 |
EC50 = 115 nM
|
|
|
| 2 |
EC50 = 252 nM
|
|
|
|
CP0432995
|
N-(2,3-dichlorophenyl)-2-[4-[4-[(2-methylimidazol-1-yl)methyl]phenyl]triazol-1-yl]acetamide
Show/Hide
|
C21H18Cl2N6O
|
2
|
| 1 |
EC50 = 589 nM
|
|
|
| 2 |
EC50 = 716 nM
|
|
|
|
CP0432994
|
N-(2,3-difluorophenyl)-2-[4-[3-methoxy-4-(4-methylimidazol-1-yl)phenyl]triazol-1-yl]acetamide
Show/Hide
|
C21H18F2N6O2
|
2
|
| 1 |
EC50 = 634 nM
|
|
|
| 2 |
EC50 > 20000 nM
|
|
|
|
CP0432997
|
N-(2,3-dichlorophenyl)-N-methyl-2-[4-[4-(2-methylimidazol-1-yl)phenyl]triazol-1-yl]acetamide
Show/Hide
|
C21H18Cl2N6O
|
1
|
| 1 |
EC50 = 4995 nM
|
|
|
|
CP0419293
|
N-(2,3-dichlorophenyl)-2-methyl-2-[4-[4-(2-methylimidazol-1-yl)phenyl]triazol-1-yl]propanamide
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|
C22H20Cl2N6O
|
1
|
| 1 |
EC50 > 20000 nM
|
|
|
|
CP0445954
|
2-[4-[3-methoxy-4-(4-methylimidazol-1-yl)phenyl]triazol-1-yl]-N-(1,2,3,4-tetrahydronaphthalen-1-yl)acetamide
Show/Hide
|
C25H26N6O2
|
1
|
| 1 |
EC50 > 20000 nM
|
|
|
|
CP0400990
|
N-[[4-[3-methoxy-4-(4-methylimidazol-1-yl)phenyl]triazol-1-yl]methyl]naphthalen-1-amine
Show/Hide
|
C24H22N6O
|
1
|
| 1 |
EC50 > 20000 nM
|
|
|
|
CP0431887
|
N-[[4-[3-methoxy-4-(4-methylimidazol-1-yl)phenyl]triazol-1-yl]methyl]naphthalene-1-carboxamide
Show/Hide
|
C25H22N6O2
|
1
|
| 1 |
EC50 > 20000 nM
|
|
|
|
CP0432998
|
1-[[4-[3-methoxy-4-(4-methylimidazol-1-yl)phenyl]triazol-1-yl]methyl]-3-naphthalen-1-ylurea
Show/Hide
|
C25H23N7O2
|
1
|
| 1 |
EC50 > 20000 nM
|
|
|
|
CP0466144
|
N-(3-chlorophenyl)-10-(2-methylpyridin-4-yl)-5,6-dihydro-[1,2,4]triazolo[4,3-d][1,4]benzoxazepin-3-amine
Show/Hide
|
C22H18ClN5O
|
1
|
| 1 |
IC50 = 37 nM
|
|
|
|
CP0466143
|
10-(2-methylpyridin-4-yl)-N-[3-(trifluoromethoxy)phenyl]-5,6-dihydro-[1,2,4]triazolo[4,3-d][1,4]benzoxazepin-3-amine
Show/Hide
|
C23H18F3N5O2
|
1
|
| 1 |
IC50 = 45 nM
|
|
|
|
CP0421592
|
10-pyridin-4-yl-N-[3-(trifluoromethyl)phenyl]-5,6-dihydro-[1,2,4]triazolo[4,3-d][1,4]benzoxazepin-3-amine
Show/Hide
|
C22H16F3N5O
|
1
|
| 1 |
IC50 = 48 nM
|
|
|
|
CP0568480
|
3-(3-chloro-2-fluorophenoxy)-10-(2-methylpyridin-4-yl)-5,6-dihydro-[1,2,4]triazolo[4,3-d][1,4]benzoxazepine
Show/Hide
|
C22H16ClFN4O2
|
1
|
| 1 |
IC50 = 56 nM
|
|
|
|
CP0558265
|
3-(3-chlorophenoxy)-10-(2-methylpyridin-4-yl)-5,6-dihydro-[1,2,4]triazolo[4,3-d][1,4]benzoxazepine
Show/Hide
|
C22H17ClN4O2
|
1
|
| 1 |
IC50 = 58 nM
|
|
|
|
CP0566008
|
10-pyridin-4-yl-N-[3-(trifluoromethoxy)phenyl]-5,6-dihydro-[1,2,4]triazolo[4,3-d][1,4]benzoxazepin-3-amine
Show/Hide
|
C22H16F3N5O2
|
1
|
| 1 |
IC50 = 63 nM
|
|
|
|
CP0568481
|
10-(2-methylpyridin-4-yl)-N-[3-(trifluoromethyl)phenyl]-5,6-dihydro-[1,2,4]triazolo[4,3-d][1,4]benzoxazepin-3-amine
Show/Hide
|
C23H18F3N5O
|
1
|
| 1 |
IC50 = 63 nM
|
|
|
|
CP0546099
|
10-(2-ethylpyridin-4-yl)-N-[3-(trifluoromethyl)phenyl]-5,6-dihydro-[1,2,4]triazolo[4,3-d][1,4]benzoxazepin-3-amine
Show/Hide
|
C24H20F3N5O
|
1
|
| 1 |
IC50 = 74 nM
|
|
|
|
CP0421591
|
10-(2-methylpyridin-4-yl)-3-[3-(trifluoromethoxy)phenoxy]-5,6-dihydro-[1,2,4]triazolo[4,3-d][1,4]benzoxazepine
Show/Hide
|
C23H17F3N4O3
|
1
|
| 1 |
IC50 = 78 nM
|
|
|
|
CP0421603
|
N-(3-cyanophenyl)-7-pyridin-4-yl-3,5-dihydro-2H-1,4-benzoxazepine-4-carboxamide
Show/Hide
|
C22H18N4O2
|
1
|
| 1 |
IC50 = 80 nM
|
|
|
|
CP0421590
|
10-(2-methylpyridin-4-yl)-3-[2-(trifluoromethoxy)phenoxy]-5,6-dihydro-[1,2,4]triazolo[4,3-d][1,4]benzoxazepine
Show/Hide
|
C23H17F3N4O3
|
1
|
| 1 |
IC50 = 89 nM
|
|
|
|
CP0546098
|
3-(2-chlorophenoxy)-10-(2-methylpyridin-4-yl)-5,6-dihydro-[1,2,4]triazolo[4,3-d][1,4]benzoxazepine
Show/Hide
|
C22H17ClN4O2
|
1
|
| 1 |
IC50 = 102 nM
|
|
|
|
CP0466150
|
N-(3-chlorophenyl)-7-pyridin-4-yl-3,5-dihydro-2H-1,4-benzoxazepine-4-carboxamide
Show/Hide
|
C21H18ClN3O2
|
1
|
| 1 |
IC50 = 108 nM
|
|
|
|
CP0421594
|
N-(3-cyanophenyl)-7-imidazol-1-yl-3,5-dihydro-2H-1,4-benzoxazepine-4-carboxamide
Show/Hide
|
C20H17N5O2
|
1
|
| 1 |
IC50 = 110 nM
|
|
|
|
CP0497286
|
N-(3-chloro-4-fluorophenyl)-7-pyridin-4-yl-3,5-dihydro-2H-1,4-benzoxazepine-4-carboxamide
Show/Hide
|
C21H17ClFN3O2
|
1
|
| 1 |
IC50 = 132 nM
|
|
|
|
CP0421600
|
N-(3,4-dichlorophenyl)-7-pyridin-4-yl-3,5-dihydro-2H-1,4-benzoxazepine-4-carboxamide
Show/Hide
|
C21H17Cl2N3O2
|
1
|
| 1 |
IC50 = 140 nM
|
|
|
|
CP0421597
|
N-(3,4-dichlorophenyl)-7-pyridin-4-yl-1,2,3,5-tetrahydro-1,4-benzodiazepine-4-carboxamide
Show/Hide
|
C21H18Cl2N4O
|
1
|
| 1 |
IC50 = 146 nM
|
|
|
|
CP0560535
|
7-pyridin-4-yl-N-[3-(trifluoromethyl)phenyl]-3,5-dihydro-2H-1,4-benzoxazepine-4-carboxamide
Show/Hide
|
C22H18F3N3O2
|
1
|
| 1 |
IC50 = 158 nM
|
|
|
|
CP0558267
|
N-(3-chloro-2-fluorophenyl)-7-pyridin-4-yl-3,5-dihydro-2H-1,4-benzoxazepine-4-carboxamide
Show/Hide
|
C21H17ClFN3O2
|
1
|
| 1 |
IC50 = 163 nM
|
|
|
|
CP0546100
|
N-(3-methoxyphenyl)-7-(3-methoxypyridin-4-yl)-3,5-dihydro-2H-1,4-benzoxazepine-4-carboxamide
Show/Hide
|
C23H23N3O4
|
1
|
| 1 |
IC50 = 187 nM
|
|
|
|
CP0560536
|
N-(3-fluorophenyl)-7-pyridin-4-yl-3,5-dihydro-2H-1,4-benzoxazepine-4-carboxamide
Show/Hide
|
C21H18FN3O2
|
1
|
| 1 |
IC50 = 224 nM
|
|
|
|
CP0560537
|
N-(3-methoxyphenyl)-7-pyridin-4-yl-3,5-dihydro-2H-1,4-benzoxazepine-4-carboxamide
Show/Hide
|
C22H21N3O3
|
1
|
| 1 |
IC50 = 249 nM
|
|
|
|
CP0490372
|
N-(3-phenylphenyl)-7-pyridin-4-yl-3,5-dihydro-2H-1,4-benzoxazepine-4-carboxamide
Show/Hide
|
C27H23N3O2
|
1
|
| 1 |
IC50 = 343 nM
|
|
|
|
CP0572990
|
N-(3-methoxyphenyl)-7-(2-methylpyridin-4-yl)-3,5-dihydro-2H-1,4-benzoxazepine-4-carboxamide
Show/Hide
|
C23H23N3O3
|
1
|
| 1 |
IC50 = 374 nM
|
|
|
|
CP0485432
|
N-(3-methoxyphenyl)-7-(3-methylpyridin-4-yl)-3,5-dihydro-2H-1,4-benzoxazepine-4-carboxamide
Show/Hide
|
C23H23N3O3
|
1
|
| 1 |
IC50 = 394 nM
|
|
|
|
CP0500791
|
N-(2-methoxyphenyl)-7-pyridin-4-yl-3,5-dihydro-2H-1,4-benzoxazepine-4-carboxamide
Show/Hide
|
C22H21N3O3
|
1
|
| 1 |
IC50 = 517 nM
|
|
|
|
CP0500788
|
3-[(3-chlorophenyl)methyl]-10-(2-methylpyridin-4-yl)-5,6-dihydro-[1,2,4]triazolo[4,3-d][1,4]benzoxazepine
Show/Hide
|
C23H19ClN4O
|
1
|
| 1 |
IC50 = 593 nM
|
|
|
|
CP0568468
|
N-(2,3-dichlorophenyl)-7-pyridin-4-yl-3,5-dihydro-2H-1,4-benzoxazepine-4-carboxamide
Show/Hide
|
C21H17Cl2N3O2
|
1
|
| 1 |
IC50 = 708 nM
|
|
|
|
CP0421604
|
N-phenyl-7-pyridin-4-yl-3,5-dihydro-2H-1,4-benzoxazepine-4-carboxamide
Show/Hide
|
C21H19N3O2
|
1
|
| 1 |
IC50 = 793 nM
|
|
|
|
CP0500790
|
7-(2-aminopyridin-4-yl)-N-(3-cyanophenyl)-3,5-dihydro-2H-1,4-benzoxazepine-4-carboxamide
Show/Hide
|
C22H19N5O2
|
1
|
| 1 |
IC50 = 810 nM
|
|
|
|
CP0421595
|
N-(3,4-dichlorophenyl)-8-pyridin-4-yl-1,3,4,5-tetrahydro-2-benzazepine-2-carboxamide
Show/Hide
|
C22H19Cl2N3O
|
1
|
| 1 |
IC50 = 839 nM
|
|
|
|
CP0466145
|
N-(3-methoxyphenyl)-7-quinolin-4-yl-3,5-dihydro-2H-1,4-benzoxazepine-4-carboxamide
Show/Hide
|
C26H23N3O3
|
1
|
| 1 |
IC50 = 962 nM
|
|
|
|
CP0466148
|
N-(4-fluorophenyl)-7-pyridin-4-yl-3,5-dihydro-2H-1,4-benzoxazepine-4-carboxamide
Show/Hide
|
C21H18FN3O2
|
1
|
| 1 |
IC50 = 1220 nM
|
|
|
|
CP0574306
|
N-(3-methoxyphenyl)-7-pyrimidin-4-yl-3,5-dihydro-2H-1,4-benzoxazepine-4-carboxamide
Show/Hide
|
C21H20N4O3
|
1
|
| 1 |
IC50 = 1600 nM
|
|
|
|
CP0466149
|
1-(7-pyridin-4-yl-3,5-dihydro-2H-1,4-benzoxazepin-4-yl)-2-[3-(trifluoromethyl)phenyl]ethanone
Show/Hide
|
C23H19F3N2O2
|
1
|
| 1 |
IC50 = 1640 nM
|
|
|
|
CP0421602
|
N-(3-phenoxyphenyl)-7-pyridin-4-yl-3,5-dihydro-2H-1,4-benzoxazepine-4-carboxamide
Show/Hide
|
C27H23N3O3
|
1
|
| 1 |
IC50 = 1720 nM
|
|
|
|
CP0558266
|
N-(3,4-dichlorophenyl)-7-pyridin-4-yl-3,4-dihydro-1H-isoquinoline-2-carboxamide
Show/Hide
|
C21H17Cl2N3O
|
1
|
| 1 |
IC50 = 1850 nM
|
|
|
|
CP0466147
|
7-pyridin-4-yl-4-[[3-(trifluoromethyl)phenyl]methylsulfonyl]-3,5-dihydro-2H-1,4-benzoxazepine
Show/Hide
|
C22H19F3N2O3S
|
1
|
| 1 |
IC50 = 2290 nM
|
|
|
|
CP0549438
|
N-(3-methoxyphenyl)-7-(2-methoxypyridin-4-yl)-3,5-dihydro-2H-1,4-benzoxazepine-4-carboxamide
Show/Hide
|
C23H23N3O4
|
1
|
| 1 |
IC50 = 2800 nM
|
|
|
|
CP0564323
|
N-(2-fluorophenyl)-7-pyridin-4-yl-3,5-dihydro-2H-1,4-benzoxazepine-4-carboxamide
Show/Hide
|
C21H18FN3O2
|
1
|
| 1 |
IC50 = 13100 nM
|
|
|
|
CP0421598
|
N-(3,4-dichlorophenyl)-5-pyridin-4-yl-1,3-dihydroisoindole-2-carboxamide
Show/Hide
|
C20H15Cl2N3O
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0421599
|
N-(3,4-dichlorophenyl)-1-methyl-7-pyridin-4-yl-3,5-dihydro-2H-1,4-benzodiazepine-4-carboxamide
Show/Hide
|
C22H20Cl2N4O
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0421601
|
N-(3-methoxyphenyl)-N-methyl-7-pyridin-4-yl-3,5-dihydro-2H-1,4-benzoxazepine-4-carboxamide
Show/Hide
|
C23H23N3O3
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0466146
|
N-(3,4-dichlorophenyl)-7-pyridin-4-yl-3,4-dihydro-2H-quinoline-1-carboxamide
Show/Hide
|
C21H17Cl2N3O
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0466151
|
N-(4-methoxyphenyl)-7-pyridin-4-yl-3,5-dihydro-2H-1,4-benzoxazepine-4-carboxamide
Show/Hide
|
C22H21N3O3
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0497287
|
1-butyl-N-(3,4-dichlorophenyl)-7-pyridin-4-yl-3,5-dihydro-2H-1,4-benzodiazepine-4-carboxamide
Show/Hide
|
C25H26Cl2N4O
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0546101
|
N-(3,4-dichlorophenyl)-6-pyridin-4-yl-2,3-dihydroindole-1-carboxamide
Show/Hide
|
C20H15Cl2N3O
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
