Brief Information of the Compound and Protein
Compound Name
7-pyridin-4-yl-4-[[3-(trifluoromethyl)phenyl]methylsulfonyl]-3,5-dihydro-2H-1,4-benzoxazepine
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Canonical SMILES
FC(F)(F)c1cccc(CS(=O)(=O)N2CCOc3ccc(cc3C2)-c2ccncc2)c1
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Compound Formula C22H19F3N2O3S
Compound Structure
Protein Name
Probable G-protein coupled receptor 142
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
Uniprot ID
Q7Z601
Gene Name
GPR142
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
IC50 = 2290 nM
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