Brief Information of the Compound and Protein
Compound Name
 Compound Info 
10-(2-ethylpyridin-4-yl)-N-[3-(trifluoromethyl)phenyl]-5,6-dihydro-[1,2,4]triazolo[4,3-d][1,4]benzoxazepin-3-amine
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Canonical SMILES
CCc1cc(ccn1)-c1ccc2OCCn3c(Nc4cccc(c4)C(F)(F)F)nnc3-c2c1
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Compound Formula C24H20F3N5O
Compound Structure
Protein Name
 Protein Info 
Probable G-protein coupled receptor 142
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
Uniprot ID
Q7Z601
Gene Name
GPR142
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO
 Cell Line Info 
Cricetulus griseus (Chinese hamster)  1
1
IC50 = 74 nM
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