General Information of the Compound
Compound ID
CP0410568
Compound Name
(2R)-3-Chloro-4-(4-(4-fluoro-2-(trifluoromethyl)phenyl)-2-methylpiperazin-1-ylsulfonyl)phenol
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Structure
Formula
C18H17ClF4N2O3S
Molecular Weight
452.857
Canonical SMILES
C[C@@H]1CN(CCN1S(=O)(=O)c1ccc(O)cc1Cl)c1ccc(F)cc1C(F)(F)F
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InChI
InChI=1S/C18H17ClF4N2O3S/c1-11-10-24(16-4-2-12(20)8-14(16)18(21,22)23)6-7-25(11)29(27,28)17-5-3-13(26)9-15(17)19/h2-5,8-9,11,26H,6-7,10H2,1H3/t11-/m1/s1
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InChIKey
HCVJPQNTGDAVPA-LLVKDONJSA-N
Physicochemical Property
logP
4.1029
Rotatable Bonds
3
Heavy Atom Count
29
Polar Areas
60.85
Hydrogen Bond Donor Count
1
Hydrogen Bond Acceptor Count
4
Complexity
29

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 44248454
SID: 85282167
ChEMBL ID
CHEMBL563036
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01109, 11-beta-hydroxysteroid dehydrogenase 1
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  2
1
IC50 = 12 nM
   TI
   LI
   LO
   TS
2
IC50 = 38 nM
   TI
   LI
   LO
   TS
Protein ID: PT01107, 11-beta-hydroxysteroid dehydrogenase 1
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
IC50 = 50 nM
   TI
   LI
   LO
   TS