| Compound ID |
Compound Name |
Compound Formula |
|
CP0011042
|
4-(4-(4-chlorophenyl)-4-hydroxypiperidin-1-yl)-N,N-dimethyl-2,2-diphenylbutanamide
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|
C29H33ClN2O2
|
1
|
| 1 |
EC50 = 58 nM
|
|
|
|
CP0424922
|
(S)-2-amino-3-(4-hydroxyphenyl)-1-((S)-2-(5-methyl-4-phenyl-1H-imidazol-2-yl)piperidin-1-yl)propan-1-one
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|
C24H28N4O2
|
1
|
| 1 |
EC50 = 153 nM
|
|
|
|
CP0497069
|
2-Amino-3-(4-hydroxy-phenyl)-1-[2-(5-methyl-4-phenyl-1H-imidazol-2-yl)-pyrrolidin-1-yl]-propan-1-one
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|
C23H26N4O2
|
1
|
| 1 |
EC50 = 1300 nM
|
|
|
|
CP0467149
|
2-[2-Amino-3-(4-hydroxy-phenyl)-propionyl]-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid phenethyl-amide
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|
C27H29N3O3
|
1
|
| 1 |
EC50 = 2120 nM
|
|
|
|
CP0247738
|
(S)-2-amino-3-(4-hydroxyphenyl)-1-((S)-3-(4-phenyl-1H-imidazol-2-yl)-3,4-dihydroisoquinolin-2(1H)-yl)propan-1-one
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|
C27H26N4O2
|
1
|
| 1 |
EC50 = 2400 nM
|
|
|
|
CP0446690
|
(S)-2-amino-3-(4-hydroxyphenyl)-1-((S)-3-(5-methyl-4-phenyl-1H-imidazol-2-yl)-3,4-dihydroisoquinolin-2(1H)-yl)propan-1-one
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|
C28H28N4O2
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0462009
|
2-Amino-1-[3-(5-bromo-4-phenyl-1H-imidazol-2-yl)-3,4-dihydro-1H-isoquinolin-2-yl]-3-(4-hydroxy-phenyl)-propan-1-one
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|
C27H25BrN4O2
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0505485
|
2-Amino-1-[3-(1H-benzoimidazol-2-yl)-3,4-dihydro-1H-isoquinolin-2-yl]-3-(4-hydroxy-phenyl)-propan-1-one
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|
C25H24N4O2
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0091844
|
BDBM50241435
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|
C75H126N24O15
|
1
|
| 1 |
Ki = 0.92 nM
|
|
|
|
CP0042625
|
Analog of Dynorphin A
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|
C73H119N21O17
|
1
|
| 1 |
Ki = 1.2 nM
|
|
|
|
CP0267602
|
Analog of Dynorphin A
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|
C70H113N19O17
|
1
|
| 1 |
Ki = 1.5 nM
|
|
|
|
CP0056102
|
Analog of Dynorphin A
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|
C72H115N19O16
|
1
|
| 1 |
Ki = 3.2 nM
|
|
|
|
CP0151231
|
Analog of Dynorphin A
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|
C70H111N19O16
|
1
|
| 1 |
Ki = 4.4 nM
|
|
|
|
CP0123441
|
Analog of Dynorphin A
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|
C71H113N19O16
|
1
|
| 1 |
Ki = 4.8 nM
|
|
|
|
CP0303774
|
Analog of Dynorphin A
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|
C73H120N24O17
|
1
|
| 1 |
Ki = 6.1 nM
|
|
|
|
CP0274780
|
Analog of Dynorphin A
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|
C70H115N25O17
|
1
|
| 1 |
Ki = 8.3 nM
|
|
|
|
CP0091810
|
Analog of Dynorphin A
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|
C71H115N25O16
|
1
|
| 1 |
Ki = 40 nM
|
|
|
|
CP0183020
|
Analog of Dynorphin A
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|
C72H117N25O16
|
1
|
| 1 |
Ki = 62 nM
|
|
|
|
CP0267780
|
Analog of Dynorphin A
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|
C70H113N25O16
|
1
|
| 1 |
Ki = 75 nM
|
|
|
|
CP0267761
|
Analog of Dynorphin A
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|
C77H128N24O17
|
1
|
| 1 |
Ki = 180 nM
|
|
|
