General Information of the Protein
Protein ID
PT00676
Protein Name
Glucagon receptor
Gene Name
GCGR
Sequence
MPPCQPRRPLLLLLLLLACQPQAPSAQVMDFLFEKWKLYGDQCHHNLSLLPPPTELVCNRTFDKYSCWPDTPANTTANISCPWYLPWHHKVQHRFVFKRCGPDGQWVRGPRGQPWRDASQCQMDGEELEVQKEVAKMYSSFQVMYTVGYSLSLGALLLALAVLGGISKLHCTRNAIHSNLFVSFVLKASSVLVIDGLLRTRYSQKIGDDLSVSIWLSDGAVAGCRVAAVFMQYGVVANYCWLLVEGLYLHNLLGLATLPERSFFSLYLGIGWGAPMLFIIPWVVVRCLFENIQCWTSNDNMGFWWILRFPVFLAILINFFIFIRIVHLLVAKLRAREMHHTDYKFRLAKSTLTLIPLLGVHEVVFAFVTDEHAQGTLRFAKLFFDLFLSSFQGLLVAVLYCFLNKEVQSELRRHWHRWRLGKVLQEERGTSNHKAPSAPGQGLSGKKLQSGRDGGSQDSSAEIPLAGGLPRLAESPFSTLLGPQLGLDSGT
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Organism
Macaca mulatta, Rhesus macaque
Protein Classification
Unclassified protein
Uniprot ID
A0A1D5QZY8
Subcellular Location
Cell membrane
Membrane
Map of Molecular Bioactivity Related to the Protein
Map of Molecular Bioactivity Related to the Protein

Protein
Cell Line
Compound

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Protein
Cell Line ID: CL000011 , CHO
Compound ID Compound Name Compound Formula
CP0120350
3-[[4-[(1S)-1-[3-(3,5-dichlorophenyl)-5-(6-methoxynaphthalen-2-yl)pyrazol-1-yl]ethyl]benzoyl]amino]propanoic acid
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C32H27Cl2N3O4
 1
1
IC50 = 55.5 nM
   TI
   LI
   LO
   TS
Similar Protein(s) and Bioactivity Statistics
50% Identity
Protein ID Protein Name Protein Organism
PT01473 Glucagon receptor Homo sapiens, Human