Compound ID |
Compound Name |
Compound Formula |
CP0545822
|
N-[[1-(oxan-4-ylmethyl)piperidin-4-yl]methyl]-2-propan-2-ylpyrazolo[1,5-a]pyridine-7-carboxamide
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|
C23H34N4O2
|
1
|
1 |
EC50 = 0.1 nM
|
|
|
CP0409231
|
N-[[1-(3-methoxypropyl)piperidin-4-yl]methyl]-2-propan-2-ylpyrazolo[1,5-a]pyridine-7-carboxamide
Show/Hide
|
C21H32N4O2
|
1
|
1 |
EC50 = 0.3 nM
|
|
|
CP0538685
|
N-[[1-[(1-hydroxycyclohexyl)methyl]piperidin-4-yl]methyl]-2-propan-2-ylimidazo[1,2-a]pyridine-8-carboxamide
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|
C24H36N4O2
|
1
|
1 |
EC50 = 0.3 nM
|
|
|
CP0549075
|
N-[[1-[(4-hydroxyoxan-4-yl)methyl]piperidin-4-yl]methyl]-2-propan-2-ylimidazo[1,2-a]pyridine-8-carboxamide
Show/Hide
|
C23H34N4O3
|
1
|
1 |
EC50 = 0.4 nM
|
|
|
CP0204174
|
N-[[1-[(4-hydroxyoxan-4-yl)methyl]piperidin-4-yl]methyl]-2-oxo-3-propan-2-ylbenzimidazole-1-carboxamide
Show/Hide
|
C23H34N4O4
|
1
|
1 |
EC50 = 0.5 nM
|
|
|
CP0414039
|
N-[[1-(oxan-4-ylmethyl)piperidin-4-yl]methyl]-2-propan-2-ylimidazo[1,2-a]pyridine-8-carboxamide
Show/Hide
|
C23H34N4O2
|
1
|
1 |
EC50 = 0.6 nM
|
|
|
CP0462167
|
methyl 4-[[4-[[(2-propan-2-ylimidazo[1,2-a]pyridine-8-carbonyl)amino]methyl]piperidin-1-yl]methyl]piperidine-1-carboxylate
Show/Hide
|
C25H37N5O3
|
1
|
1 |
EC50 = 0.6 nM
|
|
|
CP0538686
|
N-[[1-(2-hydroxy-2-methylpropyl)piperidin-4-yl]methyl]-2-propan-2-ylimidazo[1,2-a]pyridine-8-carboxamide
Show/Hide
|
C21H32N4O2
|
1
|
1 |
EC50 = 0.7 nM
|
|
|
CP0148502
|
4-[[4-[[4-[(3R)-oxolan-3-yl]oxy-1,2-benzoxazol-3-yl]oxymethyl]piperidin-1-yl]methyl]oxan-4-ol
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|
C23H32N2O6
|
3
|
1 |
EC50 = 1.3 nM
|
|
|
2 |
EC50 = 1.5 nM
|
|
|
3 |
Ki = 0.32 nM
|
|
|
CP0043344
|
methyl 4-[[4-[[(2-propan-2-yl-1H-benzimidazole-4-carbonyl)amino]methyl]piperidin-1-yl]methyl]piperidine-1-carboxylate
Show/Hide
|
C25H37N5O3
|
1
|
1 |
EC50 = 1.5 nM
|
|
|
CP0409229
|
N-[[1-(3-methoxypropyl)piperidin-4-yl]methyl]-2-propan-2-ylimidazo[1,2-a]pyridine-8-carboxamide
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|
C21H32N4O2
|
1
|
1 |
EC50 = 1.5 nM
|
|
|
CP0097781
|
CAS_183782
Show/Hide
|
C19H29ClN2O2
|
1
|
1 |
EC50 = 2 nM
|
|
|
CP0290551
|
2-Piperidinoethyl 4-amino-5-chloro-2-methoxybenzoate
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|
C15H21ClN2O3
|
3
|
1 |
EC50 = 2.5 nM
|
|
|
2 |
Ki = 3.5 nM
|
|
|
3 |
Ki = 5.7 nM
|
|
|
CP0540782
|
3-propan-2-yl-N-(1-propan-2-ylpiperidin-4-yl)imidazo[1,5-a]pyridine-1-carboxamide
Show/Hide
|
C19H28N4O
|
1
|
1 |
EC50 = 3.4 nM
|
|
|
CP0429690
|
N-[1-(2-fluoroethyl)piperidin-4-yl]-3-propan-2-ylimidazo[1,5-a]pyridine-1-carboxamide
Show/Hide
|
C18H25FN4O
|
1
|
1 |
EC50 = 3.9 nM
|
|
|
CP0429686
|
N-[[1-(3-methoxypropyl)piperidin-4-yl]methyl]-3-propan-2-ylimidazo[1,5-a]pyridine-1-carboxamide
Show/Hide
|
C21H32N4O2
|
1
|
1 |
EC50 = 4.8 nM
|
|
|
CP0409232
|
methyl 4-[[4-[[(1-propan-2-ylimidazo[1,5-a]pyridine-3-carbonyl)amino]methyl]piperidin-1-yl]methyl]piperidine-1-carboxylate
Show/Hide
|
C25H37N5O3
|
1
|
1 |
EC50 = 4.9 nM
|
|
|
CP0106868
|
4-Amino-5-chloro-2,3-dihydro-benzofuran-7-carboxylic acid [1-(3-methoxy-propyl)-piperidin-4-yl]-amide
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|
C18H26ClN3O3
|
1
|
1 |
EC50 = 5.2 nM
|
|
|
CP0388931
|
N-[[(1R,5S)-3-(3-hydroxy-2,2-dimethylpropyl)-3-azabicyclo[3.1.0]hexan-6-yl]methyl]-3-propan-2-ylimidazo[1,5-a]pyridine-1-carboxamide
Show/Hide
|
C22H32N4O2
|
1
|
1 |
EC50 = 5.7 nM
|
|
|
CP0462169
|
2-[1-(3-methoxypropyl)piperidin-4-yl]-5-(2-propan-2-ylpyrazolo[1,5-a]pyridin-7-yl)-1,3,4-oxadiazole
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|
C21H29N5O2
|
2
|
1 |
EC50 = 6 nM
|
|
|
2 |
EC50 = 62 nM
|
|
|
CP0532800
|
2-[1-(oxan-4-ylmethyl)piperidin-4-yl]-5-(2-propan-2-ylpyrazolo[1,5-a]pyridin-7-yl)-1,3,4-oxadiazole
Show/Hide
|
C23H31N5O2
|
2
|
1 |
EC50 = 6 nM
|
|
|
2 |
EC50 = 21 nM
|
|
|
CP0390034
|
N-[[3-(3-methoxypropyl)-3-azabicyclo[3.1.0]hexan-6-yl]methyl]-2-propan-2-ylpyrazolo[1,5-a]pyridine-7-carboxamide
Show/Hide
|
C21H30N4O2
|
1
|
1 |
EC50 = 7.3 nM
|
|
|
CP0409234
|
methyl 4-[[6-[[(2-propan-2-ylpyrazolo[1,5-a]pyridine-7-carbonyl)amino]methyl]-3-azabicyclo[3.1.0]hexan-3-yl]methyl]piperidine-1-carboxylate
Show/Hide
|
C25H35N5O3
|
1
|
1 |
EC50 = 8.4 nM
|
|
|
CP0540512
|
methyl 4-[4-[[(2-propan-2-ylimidazo[1,2-a]pyridine-8-carbonyl)amino]methyl]piperidin-1-yl]piperidine-1-carboxylate
Show/Hide
|
C24H35N5O3
|
1
|
1 |
EC50 = 8.4 nM
|
|
|
CP0435278
|
methyl 4-[[(1S,5R)-6-[[(3-propan-2-ylimidazo[1,5-a]pyridine-1-carbonyl)amino]methyl]-3-azabicyclo[3.1.0]hexan-3-yl]methyl]piperidine-1-carboxylate
Show/Hide
|
C25H35N5O3
|
1
|
1 |
EC50 = 8.7 nM
|
|
|
CP0564792
|
N-[[3-(oxan-4-ylmethyl)-3-azabicyclo[3.1.0]hexan-6-yl]methyl]-2-propan-2-ylpyrazolo[1,5-a]pyridine-7-carboxamide
Show/Hide
|
C23H32N4O2
|
1
|
1 |
EC50 = 8.7 nM
|
|
|
CP0390001
|
N-[[1-(oxan-4-ylmethyl)piperidin-4-yl]methyl]-1-propan-2-ylimidazo[1,5-a]pyridine-3-carboxamide
Show/Hide
|
C23H34N4O2
|
1
|
1 |
EC50 = 8.8 nM
|
|
|
CP0415573
|
2-propan-2-yl-N-[(1-propan-2-ylpiperidin-4-yl)methyl]imidazo[1,2-a]pyridine-8-carboxamide
Show/Hide
|
C20H30N4O
|
1
|
1 |
EC50 = 9 nM
|
|
|
CP0380218
|
methyl 4-[(1R,5S)-6-[[(3-propan-2-ylimidazo[1,5-a]pyridine-1-carbonyl)amino]methyl]-3-azabicyclo[3.1.0]hexan-3-yl]piperidine-1-carboxylate
Show/Hide
|
C24H33N5O3
|
1
|
1 |
EC50 = 9.7 nM
|
|
|
CP0380209
|
N-[(1-cyclobutylpiperidin-4-yl)methyl]-3-propan-2-ylimidazo[1,5-a]pyridine-1-carboxamide
Show/Hide
|
C21H30N4O
|
1
|
1 |
EC50 = 9.8 nM
|
|
|
CP0380210
|
N-[[1-(oxan-4-ylmethyl)piperidin-4-yl]methyl]-3-propan-2-ylimidazo[1,5-a]pyridine-1-carboxamide
Show/Hide
|
C23H34N4O2
|
1
|
1 |
EC50 = 10 nM
|
|
|
CP0462168
|
N-[[3-(oxan-4-yl)-3-azabicyclo[3.1.0]hexan-6-yl]methyl]-1-propan-2-ylimidazo[1,5-a]pyridine-3-carboxamide
Show/Hide
|
C22H30N4O2
|
1
|
1 |
EC50 = 10.4 nM
|
|
|
CP0429634
|
N-[[1-(oxan-4-yl)piperidin-4-yl]methyl]-3-propan-2-ylimidazo[1,5-a]pyridine-1-carboxamide
Show/Hide
|
C22H32N4O2
|
1
|
1 |
EC50 = 11 nM
|
|
|
CP0395412
|
N-[[(1S,5R)-3-(cyclobutylmethyl)-3-azabicyclo[3.1.0]hexan-6-yl]methyl]-3-propan-2-ylimidazo[1,5-a]pyridine-1-carboxamide
Show/Hide
|
C22H30N4O
|
1
|
1 |
EC50 = 13.2 nM
|
|
|
CP0546973
|
N-[[3-(3-methoxypropyl)-3-azabicyclo[3.1.0]hexan-6-yl]methyl]-1-propan-2-ylimidazo[1,5-a]pyridine-3-carboxamide
Show/Hide
|
C21H30N4O2
|
1
|
1 |
EC50 = 13.6 nM
|
|
|
CP0545823
|
N-[[3-(3-methoxypropyl)-3-azabicyclo[3.1.0]hexan-6-yl]methyl]-2-propan-2-ylimidazo[1,2-a]pyridine-8-carboxamide
Show/Hide
|
C21H30N4O2
|
1
|
1 |
EC50 = 13.8 nM
|
|
|
CP0385052
|
N-[1-(cyclobutylmethyl)piperidin-4-yl]-3-propan-2-ylimidazo[1,5-a]pyridine-1-carboxamide
Show/Hide
|
C21H30N4O
|
1
|
1 |
EC50 = 15.5 nM
|
|
|
CP0414038
|
N-[[3-(2-hydroxy-2-methylpropyl)-3-azabicyclo[3.1.0]hexan-6-yl]methyl]-2-propan-2-ylimidazo[1,2-a]pyridine-8-carboxamide
Show/Hide
|
C21H30N4O2
|
1
|
1 |
EC50 = 17 nM
|
|
|
CP0406997
|
N-[[(1S,5R)-3-cyclobutyl-3-azabicyclo[3.1.0]hexan-6-yl]methyl]-3-propan-2-ylimidazo[1,5-a]pyridine-1-carboxamide
Show/Hide
|
C21H28N4O
|
1
|
1 |
EC50 = 18 nM
|
|
|
CP0429687
|
N-[[(1S,5R)-3-(2-fluoro-2-methylpropyl)-3-azabicyclo[3.1.0]hexan-6-yl]methyl]-3-propan-2-ylimidazo[1,5-a]pyridine-1-carboxamide
Show/Hide
|
C21H29FN4O
|
1
|
1 |
EC50 = 18 nM
|
|
|
CP0538418
|
3-propan-2-yl-N-[[(1S,5R)-3-propan-2-yl-3-azabicyclo[3.1.0]hexan-6-yl]methyl]imidazo[1,5-a]pyridine-1-carboxamide
Show/Hide
|
C20H28N4O
|
1
|
1 |
EC50 = 18.3 nM
|
|
|
CP0380293
|
N-[[(1R,5S)-3-(3-methoxy-2,2-dimethylpropyl)-3-azabicyclo[3.1.0]hexan-6-yl]methyl]-3-propan-2-ylimidazo[1,5-a]pyridine-1-carboxamide
Show/Hide
|
C23H34N4O2
|
1
|
1 |
EC50 = 19.8 nM
|
|
|
CP0429688
|
N-[[(1S,5R)-3-(oxan-4-yl)-3-azabicyclo[3.1.0]hexan-6-yl]methyl]-3-propan-2-ylimidazo[1,5-a]pyridine-1-carboxamide
Show/Hide
|
C22H30N4O2
|
1
|
1 |
EC50 = 20.7 nM
|
|
|
CP0120561
|
N-[[(1R,5S)-3-(3-methoxypropyl)-3-azabicyclo[3.1.0]hexan-6-yl]methyl]-3-propan-2-ylimidazo[1,5-a]pyridine-1-carboxamide
Show/Hide
|
C21H30N4O2
|
1
|
1 |
EC50 = 22 nM
|
|
|
CP0462777
|
N-[1-(oxolan-3-ylmethyl)piperidin-4-yl]-3-propan-2-ylimidazo[1,5-a]pyridine-1-carboxamide
Show/Hide
|
C21H30N4O2
|
1
|
1 |
EC50 = 25 nM
|
|
|
CP0456851
|
N-[[(1S,5R)-3-(oxan-4-ylmethyl)-3-azabicyclo[3.1.0]hexan-6-yl]methyl]-3-propan-2-ylimidazo[1,5-a]pyridine-1-carboxamide
Show/Hide
|
C23H32N4O2
|
1
|
1 |
EC50 = 31 nM
|
|
|
CP0385050
|
N-[[(1S,5R)-3-(2-hydroxy-2-methylpropyl)-3-azabicyclo[3.1.0]hexan-6-yl]methyl]-3-propan-2-ylimidazo[1,5-a]pyridine-1-carboxamide
Show/Hide
|
C21H30N4O2
|
1
|
1 |
EC50 = 34 nM
|
|
|
CP0414036
|
2-propan-2-yl-N-[(3-propan-2-yl-3-azabicyclo[3.1.0]hexan-6-yl)methyl]imidazo[1,2-a]pyridine-8-carboxamide
Show/Hide
|
C20H28N4O
|
1
|
1 |
EC50 = 34.2 nM
|
|
|
CP0542700
|
N-[[3-(oxan-4-yl)-3-azabicyclo[3.1.0]hexan-6-yl]methyl]-2-propan-2-ylimidazo[1,2-a]pyridine-8-carboxamide
Show/Hide
|
C22H30N4O2
|
1
|
1 |
EC50 = 36 nM
|
|
|
CP0429689
|
N-[8-(2-hydroxy-2-methylpropyl)-8-azabicyclo[3.2.1]octan-3-yl]-3-propan-2-ylimidazo[1,5-a]pyridine-1-carboxamide
Show/Hide
|
C22H32N4O2
|
1
|
1 |
EC50 = 39 nM
|
|
|
CP0385053
|
N-[1-(2-hydroxy-2-methylpropyl)piperidin-4-yl]-3-propan-2-ylimidazo[1,5-a]pyridine-1-carboxamide
Show/Hide
|
C20H30N4O2
|
1
|
1 |
EC50 = 40 nM
|
|
|
CP0429649
|
N-[1-(3-methoxypropyl)piperidin-4-yl]-3-propan-2-ylimidazo[1,5-a]pyridine-1-carboxamide
Show/Hide
|
C20H30N4O2
|
1
|
1 |
EC50 = 40 nM
|
|
|
CP0542703
|
N-[[1-(oxan-4-yl)piperidin-4-yl]methyl]-1-propan-2-ylimidazo[1,5-a]pyridine-3-carboxamide
Show/Hide
|
C22H32N4O2
|
1
|
1 |
EC50 = 42 nM
|
|
|
CP0385049
|
N-[1-(3-methoxy-2,2-dimethylpropyl)piperidin-4-yl]-3-propan-2-ylimidazo[1,5-a]pyridine-1-carboxamide
Show/Hide
|
C22H34N4O2
|
1
|
1 |
EC50 = 47 nM
|
|
|
CP0545825
|
1-propan-2-yl-N-[(1-propan-2-ylpiperidin-4-yl)methyl]imidazo[1,5-a]pyridine-3-carboxamide
Show/Hide
|
C20H30N4O
|
1
|
1 |
EC50 = 48 nM
|
|
|
CP0380219
|
N-[1-(oxan-4-yl)piperidin-4-yl]-3-propan-2-ylimidazo[1,5-a]pyridine-1-carboxamide
Show/Hide
|
C21H30N4O2
|
1
|
1 |
EC50 = 49 nM
|
|
|
CP0486594
|
N-[1-(cyclopropylmethyl)piperidin-4-yl]-3-propan-2-ylimidazo[1,5-a]pyridine-1-carboxamide
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|
C20H28N4O
|
1
|
1 |
EC50 = 49 nM
|
|
|
CP0575191
|
N-(1-ethylpiperidin-4-yl)-3-propan-2-ylimidazo[1,5-a]pyridine-1-carboxamide
Show/Hide
|
C18H26N4O
|
1
|
1 |
EC50 = 50 nM
|
|
|
CP0456854
|
N-[[4-methyl-1-(oxan-4-ylmethyl)piperidin-4-yl]methyl]-3-propan-2-ylimidazo[1,5-a]pyridine-1-carboxamide
Show/Hide
|
C24H36N4O2
|
1
|
1 |
EC50 = 53 nM
|
|
|
CP0469612
|
2-(1-propan-2-ylpiperidin-4-yl)-5-(2-propan-2-ylpyrazolo[1,5-a]pyridin-7-yl)-1,3,4-oxadiazole
Show/Hide
|
C20H27N5O
|
1
|
1 |
EC50 = 54 nM
|
|
|
CP0385054
|
N-[[4-hydroxy-1-(oxan-4-ylmethyl)piperidin-4-yl]methyl]-3-propan-2-ylimidazo[1,5-a]pyridine-1-carboxamide
Show/Hide
|
C23H34N4O3
|
1
|
1 |
EC50 = 56.7 nM
|
|
|
CP0240582
|
Prx-03140
Show/Hide
|
C19H27N3O3S
|
1
|
1 |
EC50 = 58 nM
|
|
|
CP0538687
|
N-[[1-(3-methoxypropyl)piperidin-4-yl]methyl]-1-propan-2-ylimidazo[1,5-a]pyridine-3-carboxamide
Show/Hide
|
C21H32N4O2
|
1
|
1 |
EC50 = 65 nM
|
|
|
CP0456855
|
N-[[4-hydroxy-1-(2-hydroxy-2-methylpropyl)piperidin-4-yl]methyl]-3-propan-2-ylimidazo[1,5-a]pyridine-1-carboxamide
Show/Hide
|
C21H32N4O3
|
1
|
1 |
EC50 = 72.3 nM
|
|
|
CP0410418
|
N-[[1-(oxan-4-ylmethyl)piperidin-4-yl]methyl]-2-propan-2-yl-[1,2,4]triazolo[1,5-a]pyridine-8-carboxamide
Show/Hide
|
C22H33N5O2
|
1
|
1 |
EC50 = 79 nM
|
|
|
CP0380212
|
N-[8-[(4-hydroxyoxan-4-yl)methyl]-8-azabicyclo[3.2.1]octan-3-yl]-3-propan-2-ylimidazo[1,5-a]pyridine-1-carboxamide
Show/Hide
|
C24H34N4O3
|
1
|
1 |
EC50 = 88 nM
|
|
|
CP0549058
|
2-propan-2-yl-N-[(1-propan-2-ylpiperidin-4-yl)methyl]pyrazolo[1,5-a]pyridine-7-carboxamide
Show/Hide
|
C20H30N4O
|
1
|
1 |
EC50 = 98 nM
|
|
|
CP0526732
|
N-[[3-(oxan-4-ylmethyl)-3-azabicyclo[3.1.0]hexan-6-yl]methyl]-2-propan-2-ylimidazo[1,2-a]pyridine-8-carboxamide
Show/Hide
|
C23H32N4O2
|
1
|
1 |
EC50 = 114 nM
|
|
|
CP0407003
|
N-[1-(2-fluoro-2-methylpropyl)piperidin-4-yl]-3-propan-2-ylimidazo[1,5-a]pyridine-1-carboxamide
Show/Hide
|
C20H29FN4O
|
1
|
1 |
EC50 = 132 nM
|
|
|
CP0407004
|
N-[1-[(4-hydroxyoxan-4-yl)methyl]piperidin-4-yl]-3-propan-2-ylimidazo[1,5-a]pyridine-1-carboxamide
Show/Hide
|
C22H32N4O3
|
1
|
1 |
EC50 = 144 nM
|
|
|
CP0486595
|
N-[1-(2-methoxyethyl)piperidin-4-yl]-3-propan-2-ylimidazo[1,5-a]pyridine-1-carboxamide
Show/Hide
|
C19H28N4O2
|
1
|
1 |
EC50 = 144 nM
|
|
|
CP0429648
|
N-[1-[(4-fluorooxan-4-yl)methyl]piperidin-4-yl]-3-propan-2-ylimidazo[1,5-a]pyridine-1-carboxamide
Show/Hide
|
C22H31FN4O2
|
1
|
1 |
EC50 = 196 nM
|
|
|
CP0390035
|
3-chloro-N-[[3-(oxan-4-yl)-3-azabicyclo[3.1.0]hexan-6-yl]methyl]-2-propan-2-ylpyrazolo[1,5-a]pyridine-7-carboxamide
Show/Hide
|
C22H29ClN4O2
|
1
|
1 |
EC50 = 291 nM
|
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CP0385055
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N-[[4-hydroxy-1-(3-methoxypropyl)piperidin-4-yl]methyl]-3-propan-2-ylimidazo[1,5-a]pyridine-1-carboxamide
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C21H32N4O3
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1
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1 |
EC50 = 315.7 nM
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CP0406492
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N-[[4-(oxan-4-yl)morpholin-2-yl]methyl]-3-propan-2-ylimidazo[1,5-a]pyridine-1-carboxamide
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C21H30N4O3
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1
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1 |
EC50 = 467 nM
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CP0525751
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2-[1-(oxan-4-ylmethyl)piperidin-4-yl]-5-(1-propan-2-ylimidazo[1,5-a]pyridin-3-yl)-1,3,4-oxadiazole
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C23H31N5O2
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1
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1 |
EC50 = 484 nM
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CP0429632
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2-(3-propan-2-ylimidazo[1,5-a]pyridin-1-yl)-5-(1-propan-2-ylpiperidin-4-yl)-1,3,4-oxadiazole
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C20H27N5O
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1
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1 |
EC50 = 500 nM
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CP0417322
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2-[1-(cyclobutylmethyl)piperidin-4-yl]-5-(3-propan-2-ylimidazo[1,5-a]pyridin-1-yl)-1,3,4-oxadiazole
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C22H29N5O
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1
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1 |
EC50 = 520 nM
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CP0466629
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2-[1-(oxan-4-ylmethyl)piperidin-4-yl]-5-(2-propan-2-ylimidazo[1,2-a]pyridin-8-yl)-1,3,4-oxadiazole
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C23H31N5O2
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1
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1 |
EC50 = 598 nM
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CP0395413
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N-[[4-fluoro-1-(3-methoxypropyl)piperidin-4-yl]methyl]-3-propan-2-ylimidazo[1,5-a]pyridine-1-carboxamide
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C21H31FN4O2
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1
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1 |
EC50 = 633 nM
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CP0410447
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2-[1-(3-methoxypropyl)piperidin-4-yl]-5-(2-propan-2-ylimidazo[1,2-a]pyridin-8-yl)-1,3,4-oxadiazole
Show/Hide
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C21H29N5O2
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1
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1 |
EC50 = 687 nM
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CP0429631
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2-[1-(3-methoxypropyl)piperidin-4-yl]-5-(3-propan-2-ylimidazo[1,5-a]pyridin-1-yl)-1,3,4-oxadiazole
Show/Hide
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C21H29N5O2
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1
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1 |
EC50 = 736 nM
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CP0390899
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2-(1-propan-2-ylimidazo[1,5-a]pyridin-3-yl)-5-(1-propan-2-ylpiperidin-4-yl)-1,3,4-oxadiazole
Show/Hide
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C20H27N5O
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1
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1 |
EC50 = 758 nM
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CP0542702
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2-[1-(3-methoxypropyl)piperidin-4-yl]-5-(1-propan-2-ylimidazo[1,5-a]pyridin-3-yl)-1,3,4-oxadiazole
Show/Hide
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C21H29N5O2
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1
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1 |
EC50 = 796 nM
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CP0429633
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2-(1-cyclobutylpiperidin-4-yl)-5-(3-propan-2-ylimidazo[1,5-a]pyridin-1-yl)-1,3,4-oxadiazole
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C21H27N5O
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1
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1 |
EC50 = 840 nM
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CP0417320
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2-[1-(cyclopropylmethyl)piperidin-4-yl]-5-(3-propan-2-ylimidazo[1,5-a]pyridin-1-yl)-1,3,4-oxadiazole
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C21H27N5O
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1
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1 |
EC50 = 857 nM
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CP0385051
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N-[3-(oxan-4-ylmethyl)-3-azabicyclo[3.1.0]hexan-6-yl]-3-propan-2-ylimidazo[1,5-a]pyridine-1-carboxamide
Show/Hide
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C22H30N4O2
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1
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1 |
EC50 = 1061 nM
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CP0545899
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3-chloro-N-[[1-(3-methoxypropyl)piperidin-4-yl]methyl]-2-propan-2-ylimidazo[1,2-a]pyridine-8-carboxamide
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C21H31ClN4O2
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1
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1 |
EC50 = 1090 nM
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CP0564099
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N-[[4-fluoro-1-(oxan-4-ylmethyl)piperidin-4-yl]methyl]-3-propan-2-ylimidazo[1,5-a]pyridine-1-carboxamide
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C23H33FN4O2
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1
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1 |
EC50 = 1358 nM
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CP0467812
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N-[[1-(3-methoxypropyl)piperidin-4-yl]methyl]-2-propan-2-yl-[1,2,4]triazolo[1,5-a]pyridine-8-carboxamide
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C20H31N5O2
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1
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1 |
EC50 = 1941 nM
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CP0538688
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N-[[1-(3-methoxypropyl)piperidin-4-yl]methyl]-2-propan-2-yl-[1,2,4]triazolo[1,5-a]pyridine-5-carboxamide
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C20H31N5O2
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1
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1 |
EC50 = 1941 nM
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CP0462774
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N-[(4-cyclobutylmorpholin-2-yl)methyl]-3-propan-2-ylimidazo[1,5-a]pyridine-1-carboxamide
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C20H28N4O2
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1
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1 |
EC50 = 2247 nM
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CP0395410
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N-[3-(3-methoxypropyl)-3-azabicyclo[3.1.0]hexan-6-yl]-3-propan-2-ylimidazo[1,5-a]pyridine-1-carboxamide
Show/Hide
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C20H28N4O2
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1
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1 |
EC50 > 10000 nM
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CP0406999
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N-[3-(2-hydroxy-2-methylpropyl)-3-azabicyclo[3.1.0]hexan-6-yl]-3-propan-2-ylimidazo[1,5-a]pyridine-1-carboxamide
Show/Hide
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C20H28N4O2
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1
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1 |
EC50 > 10000 nM
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CP0390002
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3-chloro-N-[[1-(3-methoxypropyl)piperidin-4-yl]methyl]-2-propan-2-ylpyrazolo[1,5-a]pyridine-7-carboxamide
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C21H31ClN4O2
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1
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1 |
EC50 > 10000 nM
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CP0545909
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3-chloro-N-[[3-(3-methoxypropyl)-3-azabicyclo[3.1.0]hexan-6-yl]methyl]-2-propan-2-ylimidazo[1,2-a]pyridine-8-carboxamide
Show/Hide
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C21H29ClN4O2
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1
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1 |
EC50 > 10000 nM
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CP0549489
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N-[[1-(oxan-4-ylmethyl)piperidin-4-yl]methyl]-2-propan-2-yl-[1,2,4]triazolo[1,5-a]pyridine-5-carboxamide
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C22H33N5O2
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1
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1 |
EC50 > 10000 nM
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CP0559962
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2-propan-2-yl-N-[(1-propan-2-ylpiperidin-4-yl)methyl]-[1,2,4]triazolo[1,5-a]pyridine-5-carboxamide
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C19H29N5O
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1
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1 |
EC50 > 10000 nM
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CP0559963
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3-chloro-N-[[3-(3-methoxypropyl)-3-azabicyclo[3.1.0]hexan-6-yl]methyl]-2-propan-2-ylpyrazolo[1,5-a]pyridine-7-carboxamide
Show/Hide
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C21H29ClN4O2
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1
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1 |
EC50 > 10000 nM
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CP0123097
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3H-GR113808
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C19H27N3O4S
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3
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1 |
IC50 = 0.21 nM
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2 |
Ki = 0.5 nM
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3 |
Ki = 0.7 nM
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CP0046314
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4-[2-[4-[(2-methylpyrrolo[3,4-c]quinolin-4-yl)oxymethyl]piperidin-1-yl]ethyl]benzoic acid
Show/Hide
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C27H29N3O3
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1
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1 |
IC50 = 2.8 nM
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CP0046312
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4-[2-[4-[[(1-propan-2-ylindazole-3-carbonyl)amino]methyl]piperidin-1-yl]ethyl]benzoic acid
Show/Hide
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C26H32N4O3
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1
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1 |
IC50 = 9.8 nM
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CP0170456
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3-chloro-1-(4-fluoro benzenesulfonyl)-5-(4-methylpiperazin-1-yl-methyl)-1H-indole
Show/Hide
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C20H21ClFN3O2S
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1
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1 |
IC50 > 10000 nM
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CP0212171
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1-(2-Bromo benzenesulfonyl)-5-(4-ethylpiperazin-1-yl-methyl)-1H-indole
Show/Hide
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C21H24BrN3O2S
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1
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1 |
IC50 > 10000 nM
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CP0376851
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6-fluoro-N-[[1-[(4-hydroxyoxan-4-yl)methyl]piperidin-4-yl]methyl]-2-oxo-3-propan-2-ylbenzimidazole-1-carboxamide
Show/Hide
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C23H33FN4O4
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1
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1 |
Ki = 4.9 nM
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CP0395625
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6-fluoro-N-[[1-[(4-hydroxyoxan-4-yl)methyl]piperidin-4-yl]methyl]-3,3-dimethyl-2-oxoindole-1-carboxamide
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C23H32FN3O4
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1
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1 |
Ki = 6.3 nM
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CP0913714
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2-(4-{4-[N-(3-{4-[3-(N-{3-[(1-{2-[(4-amino-5-chloro-2-methoxyphenyl)carbonyloxy]ethyl}piperidin-4-yl)carbamoyl]propyl}-2,2-dimethylpropanamido)propyl]phenyl}propyl)-2,2-dimethylpropanamido]butanamido}piperidin-1-yl)ethyl 4-amino-5-chloro-2-methoxybenzoate
Show/Hide
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C60H88Cl2N8O12
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1
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1 |
Ki = 10 nM
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