Brief Information of the Compound and Protein
Compound Name
methyl 4-[[(1S,5R)-6-[[(3-propan-2-ylimidazo[1,5-a]pyridine-1-carbonyl)amino]methyl]-3-azabicyclo[3.1.0]hexan-3-yl]methyl]piperidine-1-carboxylate
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Canonical SMILES
COC(=O)N1CCC(CN2C[C@H]3[C@H](CNC(=O)c4nc(C(C)C)n5ccccc45)[C@H]3C2)CC1
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Compound Formula C25H35N5O3
Compound Structure
Protein Name
5-hydroxytryptamine receptor 4
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Serotonin receptor
Uniprot ID
Q13639
Gene Name
HTR4
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
EC50 = 8.7 nM
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