Brief Information of the Compound and Protein
Compound Name
4-Amino-5-chloro-2,3-dihydro-benzofuran-7-carboxylic acid [1-(3-methoxy-propyl)-piperidin-4-yl]-amide
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PubChem ID
CID: 3052762
SID: 14803834
Canonical SMILES
COCCCN1CCC(CC1)NC(=O)c1cc(Cl)c(N)c2CCOc12
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Compound Formula C18H26ClN3O3
Compound Structure
Protein Name
5-hydroxytryptamine receptor 4
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Serotonin receptor
Uniprot ID
Q13639
Gene Name
HTR4
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
EC50 = 5.2 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 EC50 = 26 nM
2 Ki = 2.512 nM