Brief Information of the Compound and Protein
Compound Name
 Compound Info 
methyl 4-[[6-[[(2-propan-2-ylpyrazolo[1,5-a]pyridine-7-carbonyl)amino]methyl]-3-azabicyclo[3.1.0]hexan-3-yl]methyl]piperidine-1-carboxylate
    Show/Hide
 PubChem ID
CID: 145978067
Canonical SMILES
COC(=O)N1CCC(CN2CC3C(CNC(=O)c4cccc5cc(nn45)C(C)C)C3C2)CC1
    Show/Hide
Compound Formula C25H35N5O3
Compound Structure
Protein Name
 Protein Info 
5-hydroxytryptamine receptor 4
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
>
Small molecule receptor (family A GPCR)
>
Monoamine receptor
>
Serotonin receptor
Uniprot ID
Q13639
Gene Name
HTR4
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO
 Cell Line Info 
Cricetulus griseus (Chinese hamster)  1
1
EC50 = 8.4 nM
   TI
   LI
   LO
   TS