| Compound ID |
Compound Name |
Compound Formula |
|
CP0165878
|
(2R)-N-[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]-1-(4-methylphenyl)sulfonylpiperidine-2-carboxamide
Show/Hide
|
C23H25N3O4S2
|
1
|
| 1 |
EC50 = 260 nM
|
|
|
|
CP0423690
|
(2R)-1-(4-chlorophenyl)sulfonyl-N-[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]piperidine-2-carboxamide
Show/Hide
|
C22H22ClN3O4S2
|
1
|
| 1 |
EC50 = 420 nM
|
|
|
|
CP0423684
|
N-[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]-4-(4-methylphenyl)sulfonylthiomorpholine-3-carboxamide
Show/Hide
|
C22H23N3O4S3
|
1
|
| 1 |
EC50 = 600 nM
|
|
|
|
CP0433948
|
(2R)-N-[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]-1-(4-propylphenyl)sulfonylpiperidine-2-carboxamide
Show/Hide
|
C25H29N3O4S2
|
1
|
| 1 |
EC50 = 700 nM
|
|
|
|
CP0453130
|
(2R)-1-(2-chlorophenyl)sulfonyl-N-[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]piperidine-2-carboxamide
Show/Hide
|
C22H22ClN3O4S2
|
1
|
| 1 |
EC50 = 730 nM
|
|
|
|
CP0437847
|
(2R)-1-(1,3-benzodioxol-5-ylsulfonyl)-N-[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]piperidine-2-carboxamide
Show/Hide
|
C23H23N3O6S2
|
1
|
| 1 |
EC50 = 780 nM
|
|
|
|
CP0423680
|
(2R)-1-(3-methoxyphenyl)sulfonyl-N-[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]piperidine-2-carboxamide
Show/Hide
|
C23H25N3O5S2
|
1
|
| 1 |
EC50 = 810 nM
|
|
|
|
CP0487671
|
(2R)-1-(3-cyanophenyl)sulfonyl-N-[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]piperidine-2-carboxamide
Show/Hide
|
C23H22N4O4S2
|
1
|
| 1 |
EC50 = 880 nM
|
|
|
|
CP0423679
|
(2R)-N-[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]-1-(3-methylphenyl)sulfonylpiperidine-2-carboxamide
Show/Hide
|
C23H25N3O4S2
|
1
|
| 1 |
EC50 = 890 nM
|
|
|
|
CP0433944
|
(2R)-N-[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]-1-[3-(trifluoromethyl)phenyl]sulfonylpiperidine-2-carboxamide
Show/Hide
|
C23H22F3N3O4S2
|
1
|
| 1 |
EC50 = 1000 nM
|
|
|
|
CP0453129
|
(2R)-1-(4-fluorophenyl)sulfonyl-N-[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]piperidine-2-carboxamide
Show/Hide
|
C22H22FN3O4S2
|
1
|
| 1 |
EC50 = 1030 nM
|
|
|
|
CP0523380
|
(2R)-1-(3-fluorophenyl)sulfonyl-N-[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]piperidine-2-carboxamide
Show/Hide
|
C22H22FN3O4S2
|
1
|
| 1 |
EC50 = 1160 nM
|
|
|
|
CP0433946
|
(2R)-N-[4-(1-benzofuran-5-yl)-1,3-thiazol-2-yl]-1-(4-methylphenyl)sulfonylpiperidine-2-carboxamide
Show/Hide
|
C24H23N3O4S2
|
1
|
| 1 |
EC50 = 1320 nM
|
|
|
|
CP0423682
|
(2R)-N-[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]-1-pyridin-3-ylsulfonylpiperidine-2-carboxamide
Show/Hide
|
C21H22N4O4S2
|
1
|
| 1 |
EC50 = 1360 nM
|
|
|
|
CP0423686
|
(2R)-N-[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]-1-(2-methylphenyl)sulfonylpiperidine-2-carboxamide
Show/Hide
|
C23H25N3O4S2
|
1
|
| 1 |
EC50 = 1380 nM
|
|
|
|
CP0379106
|
(2R)-1-(3-chlorophenyl)sulfonyl-N-[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]piperidine-2-carboxamide
Show/Hide
|
C22H22ClN3O4S2
|
1
|
| 1 |
EC50 = 1410 nM
|
|
|
|
CP0429461
|
(2R)-1-(benzenesulfonyl)-N-[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]piperidine-2-carboxamide
Show/Hide
|
C22H23N3O4S2
|
1
|
| 1 |
EC50 = 1470 nM
|
|
|
|
CP0379105
|
(2R)-1-(4-cyanophenyl)sulfonyl-N-[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]piperidine-2-carboxamide
Show/Hide
|
C23H22N4O4S2
|
1
|
| 1 |
EC50 = 1630 nM
|
|
|
|
CP0188691
|
1-(benzenesulfonyl)-N-[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]piperidine-2-carboxamide
Show/Hide
|
C22H23N3O4S2
|
1
|
| 1 |
EC50 = 1690 nM
|
|
|
|
CP0423689
|
(2R)-N-[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]-1-[4-(trifluoromethyl)phenyl]sulfonylpiperidine-2-carboxamide
Show/Hide
|
C23H22F3N3O4S2
|
1
|
| 1 |
EC50 = 1710 nM
|
|
|
|
CP0453126
|
(2R)-1-(2-methoxyphenyl)sulfonyl-N-[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]piperidine-2-carboxamide
Show/Hide
|
C23H25N3O5S2
|
1
|
| 1 |
EC50 = 1780 nM
|
|
|
|
CP0423687
|
(2R)-N-[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]-1-(4-propan-2-ylphenyl)sulfonylpiperidine-2-carboxamide
Show/Hide
|
C25H29N3O4S2
|
1
|
| 1 |
EC50 = 2590 nM
|
|
|
|
CP0433949
|
N-[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]-1-(4-methylphenyl)sulfonylpyrrolidine-2-carboxamide
Show/Hide
|
C22H23N3O4S2
|
1
|
| 1 |
EC50 = 2860 nM
|
|
|
|
CP0483283
|
N-[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]-4-(4-methylphenyl)sulfonylmorpholine-3-carboxamide
Show/Hide
|
C22H23N3O5S2
|
1
|
| 1 |
EC50 = 4380 nM
|
|
|
|
CP0423688
|
(2R)-N-[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]-1-[2-(trifluoromethyl)phenyl]sulfonylpiperidine-2-carboxamide
Show/Hide
|
C23H22F3N3O4S2
|
1
|
| 1 |
EC50 = 4740 nM
|
|
|
|
CP0379109
|
(2R)-1-(3-fluorobenzoyl)-N-[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]piperidine-2-carboxamide
Show/Hide
|
C23H22FN3O3S
|
1
|
| 1 |
EC50 = 6130 nM
|
|
|
|
CP0438914
|
(2R)-1-isoquinolin-1-ylsulfonyl-N-[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]piperidine-2-carboxamide
Show/Hide
|
C25H24N4O4S2
|
1
|
| 1 |
EC50 = 7970 nM
|
|
|
|
CP0423692
|
(2R)-1-benzoyl-N-[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]piperidine-2-carboxamide
Show/Hide
|
C23H23N3O3S
|
1
|
| 1 |
EC50 = 8160 nM
|
|
|
|
CP0514751
|
(2R)-N-[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]-2-[(4-methylphenyl)sulfonylamino]propanamide
Show/Hide
|
C20H21N3O4S2
|
1
|
| 1 |
EC50 = 12900 nM
|
|
|
|
CP0437850
|
(2R)-N-[5-(4-methoxyphenyl)-1,3-thiazol-2-yl]-1-(4-methylphenyl)sulfonylpiperidine-2-carboxamide
Show/Hide
|
C23H25N3O4S2
|
1
|
| 1 |
EC50 = 27400 nM
|
|
|
|
CP0379108
|
(2R)-1-(2-chloro-4-fluorophenyl)sulfonyl-N-[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]piperidine-2-carboxamide
Show/Hide
|
C22H21ClFN3O4S2
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0379110
|
N-[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]-3-[(4-methylphenyl)sulfonylamino]propanamide
Show/Hide
|
C20H21N3O4S2
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0379111
|
(2R)-N-[4-(4-fluorophenyl)-1,3-thiazol-2-yl]-1-(4-methylphenyl)sulfonylpiperidine-2-carboxamide
Show/Hide
|
C22H22FN3O3S2
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0423681
|
(2R)-1-(5-chloro-2-fluorophenyl)sulfonyl-N-[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]piperidine-2-carboxamide
Show/Hide
|
C22H21ClFN3O4S2
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0423683
|
N-[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]-1-(4-methylphenyl)sulfonylazetidine-2-carboxamide
Show/Hide
|
C21H21N3O4S2
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0423685
|
(2R)-N-[5-(1-benzofuran-5-yl)-1,3,4-thiadiazol-2-yl]-1-(4-methylphenyl)sulfonylpiperidine-2-carboxamide
Show/Hide
|
C23H22N4O4S2
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0423691
|
(2R)-1-(3-fluoro-2-methylphenyl)sulfonyl-N-[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]piperidine-2-carboxamide
Show/Hide
|
C23H24FN3O4S2
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0433945
|
(2R)-N-(1,3-benzothiazol-2-yl)-1-(4-methylphenyl)sulfonylpiperidine-2-carboxamide
Show/Hide
|
C20H21N3O3S2
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0433947
|
(2R)-N-[5-(4-methoxyphenyl)-1,3,4-thiadiazol-2-yl]-1-(4-methylphenyl)sulfonylpiperidine-2-carboxamide
Show/Hide
|
C22H24N4O4S2
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0437848
|
(2R)-1-[(4-chlorophenyl)methylsulfonyl]-N-[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]piperidine-2-carboxamide
Show/Hide
|
C23H24ClN3O4S2
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0437849
|
(2R)-N-[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]-3,3-dimethyl-2-[(4-methylphenyl)sulfonylamino]butanamide
Show/Hide
|
C23H27N3O4S2
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0438915
|
(3S)-N-[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]-1-(4-methylphenyl)sulfonylpiperidine-3-carboxamide
Show/Hide
|
C23H25N3O4S2
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0438916
|
(2R)-1-(4-chlorophenyl)sulfonyl-N-[5-(4-methoxyphenyl)-1,3,4-thiadiazol-2-yl]piperidine-2-carboxamide
Show/Hide
|
C21H21ClN4O4S2
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0453124
|
(2S)-1-(benzenesulfonyl)-N-[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]piperidine-2-carboxamide
Show/Hide
|
C22H23N3O4S2
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0480480
|
(2R)-1-(2,3-dichlorophenyl)sulfonyl-N-[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]piperidine-2-carboxamide
Show/Hide
|
C22H21Cl2N3O4S2
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0480484
|
N-[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]-1-(4-methylphenyl)sulfonylazepane-2-carboxamide
Show/Hide
|
C24H27N3O4S2
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0483280
|
(2R)-1-(4-methylphenyl)sulfonyl-N-[4-(4-methylphenyl)-1,3-thiazol-2-yl]piperidine-2-carboxamide
Show/Hide
|
C23H25N3O3S2
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0483281
|
(2R)-1-(4-methylphenyl)sulfonyl-N-[4-(4-nitrophenyl)-1,3-thiazol-2-yl]piperidine-2-carboxamide
Show/Hide
|
C22H22N4O5S2
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0483282
|
(2R)-1-(2-cyanophenyl)sulfonyl-N-[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]piperidine-2-carboxamide
Show/Hide
|
C23H22N4O4S2
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0487673
|
(2R)-N-[5-(1-benzofuran-5-yl)-1,3-thiazol-2-yl]-1-(4-methylphenyl)sulfonylpiperidine-2-carboxamide
Show/Hide
|
C24H23N3O4S2
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0514747
|
(2R)-1-[(2-chlorophenyl)methylsulfonyl]-N-[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]piperidine-2-carboxamide
Show/Hide
|
C23H24ClN3O4S2
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0523379
|
(2R)-1-(4-tert-butylphenyl)sulfonyl-N-[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]piperidine-2-carboxamide
Show/Hide
|
C26H31N3O4S2
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0526928
|
(2R)-1-(4-methylphenyl)sulfonyl-N-(4-phenyl-1,3-thiazol-2-yl)piperidine-2-carboxamide
Show/Hide
|
C22H23N3O3S2
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0526972
|
(2R)-N-[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]-1-(1-methylimidazol-4-yl)sulfonylpiperidine-2-carboxamide
Show/Hide
|
C20H23N5O4S2
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0526973
|
(2R)-N-[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]-1-(2-methylpyridin-3-yl)sulfonylpiperidine-2-carboxamide
Show/Hide
|
C22H24N4O4S2
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0526975
|
(2R)-N-[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]-3-methyl-2-[(4-methylphenyl)sulfonylamino]butanamide
Show/Hide
|
C22H25N3O4S2
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0526977
|
(2R)-1-(4-methylphenyl)sulfonyl-N-(1,3-thiazol-2-yl)piperidine-2-carboxamide
Show/Hide
|
C16H19N3O3S2
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0527019
|
(2R)-1-(4-methylphenyl)sulfonyl-N-[4-[4-(trifluoromethoxy)phenyl]-1,3-thiazol-2-yl]piperidine-2-carboxamide
Show/Hide
|
C23H22F3N3O4S2
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0531931
|
(2R)-1-(2-methoxybenzoyl)-N-[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]piperidine-2-carboxamide
Show/Hide
|
C24H25N3O4S
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0531933
|
N-[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]-1-(4-methylphenyl)sulfonylpiperazine-2-carboxamide
Show/Hide
|
C22H24N4O4S2
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0531934
|
(2R)-1-(4-methylphenyl)sulfonyl-N-[4-(4-propan-2-ylphenyl)-1,3-thiazol-2-yl]piperidine-2-carboxamide
Show/Hide
|
C25H29N3O3S2
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0531936
|
(2R)-N-[4-(4-chlorophenyl)-1,3-thiazol-2-yl]-1-(4-methylphenyl)sulfonylpiperidine-2-carboxamide
Show/Hide
|
C22H22ClN3O3S2
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0870546
|
N-(4-(4-methoxyphenyl)thiazol-2-yl)-1-tosylpiperidine-3-carboxamide
Show/Hide
|
C23H25N3O4S2
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0010522
|
(2S)-2-phenyl-N-(2-pyrrolidin-1-ylphenyl)butanamide
Show/Hide
|
C20H24N2O
|
1
|
| 1 |
IC50 = 2920 nM
|
|
|
