| Compound ID |
Compound Name |
Compound Formula |
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CP0094665
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(S)-3-[(S)-2-((S)-2-Acetylamino-3,3-diphenyl-propionylamino)-4-methyl-pentanoylamino]-N-((1S,2S)-1-{(1S,2S)-1-[(S)-1-carboxy-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-methyl-butylcarbamoyl}-2-methyl-butyl)-succinamic acid
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|
C50H65N7O10
|
1
|
| 1 |
IC50 = 20 nM
|
|
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CP0293980
|
(S)-N-((1S,2S)-1-{(1S,2S)-1-[(S)-1-Carboxy-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-methyl-butylcarbamoyl}-2-methyl-butyl)-3-{(S)-4-methyl-2-[(S)-2-(3-methyl-ureido)-3,3-diphenyl-propionylamino]-pentanoylamino}-succinamic acid
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|
C50H66N8O10
|
1
|
| 1 |
IC50 = 20 nM
|
|
|
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CP0080355
|
(S)-N-((1S,2S)-1-{(1S,2S)-1-[(S)-1-Carboxy-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-methyl-butylcarbamoyl}-2-methyl-butyl)-3-[(S)-2-((S)-3,3-diphenyl-2-propionylamino-propionylamino)-4-methyl-pentanoylamino]-succinamic acid
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|
C51H67N7O10
|
1
|
| 1 |
IC50 = 220 nM
|
|
|
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CP0307256
|
(S)-N-((1S,2S)-1-{(1S,2S)-1-[(S)-1-Carboxy-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-methyl-butylcarbamoyl}-2-methyl-butyl)-3-{(S)-2-[(S)-3,3-diphenyl-2-(2,2,2-trifluoro-acetylamino)-propionylamino]-4-methyl-pentanoylamino}-succinamic acid
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|
C50H62F3N7O10
|
1
|
| 1 |
IC50 = 290 nM
|
|
|
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CP0320424
|
(S)-3-[(S)-2-((S)-2-Benzoylamino-3,3-diphenyl-propionylamino)-4-methyl-pentanoylamino]-N-((1S,2S)-1-{(1S,2S)-1-[(S)-1-carboxy-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-methyl-butylcarbamoyl}-2-methyl-butyl)-succinamic acid
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|
C55H67N7O10
|
1
|
| 1 |
IC50 = 290 nM
|
|
|
|
CP0051768
|
(S)-N-((1S,2S)-1-{(1S,2S)-1-[(S)-1-Carboxy-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-methyl-butylcarbamoyl}-2-methyl-butyl)-3-{(S)-2-[(S)-2-(cyclohexanecarbonyl-amino)-3,3-diphenyl-propionylamino]-4-methyl-pentanoylamino}-succinamic acid
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|
C55H73N7O10
|
1
|
| 1 |
IC50 = 560 nM
|
|
|
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CP0046911
|
(S)-N-((1S,2S)-1-{(1S,2S)-1-[(S)-1-Carboxy-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-methyl-butylcarbamoyl}-2-methyl-butyl)-3-{(S)-2-[(S)-2-(2,2-dimethyl-propionylamino)-3,3-diphenyl-propionylamino]-4-methyl-pentanoylamino}-succinamic acid
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|
C53H71N7O10
|
1
|
| 1 |
IC50 = 890 nM
|
|
|
|
CP0152807
|
(S)-N-((1S,2S)-1-{(1S,2S)-1-[(S)-1-Carboxy-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-methyl-butylcarbamoyl}-2-methyl-butyl)-3-[(S)-2-((S)-2-methanesulfonylamino-3,3-diphenyl-propionylamino)-4-methyl-pentanoylamino]-succinamic acid
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|
C49H65N7O11S
|
1
|
| 1 |
IC50 = 1300 nM
|
|
|
|
CP0509991
|
(S)-N-((1S,2S)-1-{(1S,2S)-1-[(S)-1-Carboxy-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-methyl-butylcarbamoyl}-2-methyl-butyl)-3-((S)-2-{(S)-3,3-diphenyl-2-[(pyridine-3-carbonyl)-amino]-propionylamino}-4-methyl-pentanoylamino)-succinamic acid
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|
C54H66N8O10
|
1
|
| 1 |
IC50 = 2500 nM
|
|
|
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CP0048328
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(3S)-4-[[(2S,3S)-1-[[(2S,3S)-1-[[(1S)-1-carboxy-2-(1H-indol-3-yl)ethyl]amino]-3-methyl-1-oxopentan-2-yl]amino]-3-methyl-1-oxopentan-2-yl]amino]-3-[[(2S)-2-[[(2S)-3,3-diphenyl-2-(tricyclo[9.4.0.03,8]pentadeca-1(15),3,5,7,11,13-hexaene-2-carbonylamino)propanoyl]amino]-4-methylpentanoyl]amino]-4-oxobutanoic acid
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|
C64H75N7O10
|
1
|
| 1 |
IC50 = 3600 nM
|
|
|
|
CP0307091
|
3-(2-{2-[(Adamantane-1-carbonyl)-amino]-3,3-diphenyl-propionylamino}-4-methyl-pentanoylamino)-N-(1-{1-[1-carboxy-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-methyl-butylcarbamoyl}-2-methyl-butyl)-succinamic acid
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|
C59H77N7O10
|
1
|
| 1 |
IC50 = 4000 nM
|
|
|
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CP0168569
|
(S)-3-[(S)-2-((S)-2-Amino-3,3-diphenyl-propionylamino)-4-methyl-pentanoylamino]-N-((1S,2S)-1-{(1S,2S)-1-[(S)-1-carboxy-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-methyl-butylcarbamoyl}-2-methyl-butyl)-succinamic acid
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|
C48H63N7O9
|
1
|
| 1 |
IC50 = 9200 nM
|
|
|
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CP0135125
|
(S)-N-((1S,2S)-1-{(1S,2S)-1-[(S)-1-Carboxy-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-methyl-butylcarbamoyl}-2-methyl-butyl)-3-{(S)-2-[(S)-2-(3-cyclohexyl-ureido)-3,3-diphenyl-propionylamino]-4-methyl-pentanoylamino}-succinamic acid
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|
C55H74N8O10
|
1
|
| 1 |
IC50 = 9300 nM
|
|
|
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CP0319208
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(S)-N-((1S,2S)-1-{(1S,2S)-1-[(S)-1-Carboxy-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-methyl-butylcarbamoyl}-2-methyl-butyl)-3-[(S)-2-((S)-2-diphenylacetylamino-3,3-diphenyl-propionylamino)-4-methyl-pentanoylamino]-succinamic acid
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|
C62H73N7O10
|
1
|
| 1 |
IC50 = 9300 nM
|
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