Brief Information of the Cell Line and Protein
Cell Line ID: CL000011 , CHO
Synonyms
Chinese Hamster Ovary
CHO-ori
Category Spontaneously immortalized cell line
Organism
Cricetulus griseus (Chinese hamster)
Cellosaurus ID
CVCL_0213
Protein ID: PT01877 , P2Y purinoceptor 1
Gene Name P2RY1
Organism Homo sapiens, Human
Protein Classification Membrane receptor
Uniprot ID P47900
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000011  Protein ID: PT01877
 
Compound ID Compound Name Compound Formula
CP0477009
butyl 4-[2-[[5-[2-[(2S)-2-(cyclobutylcarbamoyl)pyrrolidin-1-yl]-2-oxoethoxy]-1-phenylpyrazole-3-carbonyl]amino]acetyl]piperazine-1-carboxylate
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C32H43N7O7
 1
1
Ki > 20000 nM
   TI
   LI
   LO
   TS
CP0488032
(4S)-4-[[5-[2-[(2S)-2-(cyclobutylcarbamoyl)pyrrolidin-1-yl]-2-oxoethoxy]-1-phenylpyrazole-3-carbonyl]amino]-5-(4-ethoxycarbonylpiperazin-1-yl)-5-oxopentanoic acid
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C33H43N7O9
 1
1
Ki > 20000 nM
   TI
   LI
   LO
   TS
CP0500086
(4S)-4-[[5-(1-ethoxycarbonylcyclobutyl)oxy-1-phenylpyrazole-3-carbonyl]amino]-5-(4-ethoxycarbonylpiperazin-1-yl)-5-oxopentanoic acid
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C29H37N5O9
 1
1
Ki > 20000 nM
   TI
   LI
   LO
   TS