Brief Information of the Cell Line and Protein
Cell Line ID: CL000011 , CHO
Synonyms
Chinese Hamster Ovary
CHO-ori
Category Spontaneously immortalized cell line
Organism
Cricetulus griseus (Chinese hamster)
Cellosaurus ID
CVCL_0213
Protein ID: PT01188 , Kappa-type opioid receptor
Gene Name OPRK1
Organism Cavia porcellus, Guinea pig
Protein Classification Membrane receptor
Uniprot ID P41144
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000011  Protein ID: PT01188
 
Compound ID Compound Name Compound Formula
CP0091844
BDBM50241435
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C75H126N24O15
 1
1
Ki = 0.31 nM
   TI
   LI
   LO
   TS
CP0056102
Analog of Dynorphin A
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C72H115N19O16
 1
1
Ki = 1.5 nM
   TI
   LI
   LO
   TS
CP0123441
Analog of Dynorphin A
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C71H113N19O16
 1
1
Ki = 2.5 nM
   TI
   LI
   LO
   TS
CP0151231
Analog of Dynorphin A
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C70H111N19O16
 1
1
Ki = 2.6 nM
   TI
   LI
   LO
   TS
CP0042625
Analog of Dynorphin A
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C73H119N21O17
 1
1
Ki = 8 nM
   TI
   LI
   LO
   TS
CP0267780
Analog of Dynorphin A
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C70H113N25O16
 1
1
Ki = 8 nM
   TI
   LI
   LO
   TS
CP0183020
Analog of Dynorphin A
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C72H117N25O16
 1
1
Ki = 12 nM
   TI
   LI
   LO
   TS
CP0267602
Analog of Dynorphin A
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C70H113N19O17
 1
1
Ki = 12 nM
   TI
   LI
   LO
   TS
CP0091810
Analog of Dynorphin A
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C71H115N25O16
 1
1
Ki = 14 nM
   TI
   LI
   LO
   TS
CP0274780
Analog of Dynorphin A
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C70H115N25O17
 1
1
Ki = 20 nM
   TI
   LI
   LO
   TS
CP0267761
Analog of Dynorphin A
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C77H128N24O17
 1
1
Ki = 28 nM
   TI
   LI
   LO
   TS
CP0303774
Analog of Dynorphin A
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C73H120N24O17
 1
1
Ki = 58 nM
   TI
   LI
   LO
   TS