| Compound ID |
Compound Name |
Compound Formula |
|
CP0389427
|
N-[(S)-(3-fluoropyridin-2-yl)-[3-fluoro-4-(trifluoromethyl)phenyl]methyl]-6-oxo-1H-pyridine-3-carboxamide
Show/Hide
|
C19H12F5N3O2
|
1
|
| 1 |
IC50 = 5 nM
|
|
|
|
CP0389434
|
6-oxo-N-[(S)-[4-(trifluoromethyl)phenyl]-[3-(trifluoromethyl)pyridin-2-yl]methyl]-1H-pyridine-3-carboxamide
Show/Hide
|
C20H13F6N3O2
|
1
|
| 1 |
IC50 = 6 nM
|
|
|
|
CP0389437
|
4-hydroxy-N-[(S)-[4-(trifluoromethyl)phenyl]-[3-(trifluoromethyl)pyridin-2-yl]methyl]benzamide
Show/Hide
|
C21H14F6N2O2
|
1
|
| 1 |
IC50 = 8 nM
|
|
|
|
CP0365159
|
(4R)-8-chloro-4-hydroxy-N-[4-(trifluoromethoxy)phenyl]spiro[3,4-dihydrochromene-2,4'-piperidine]-1'-carboxamide
Show/Hide
|
C21H20ClF3N2O4
|
1
|
| 1 |
IC50 = 8.9 nM
|
|
|
|
CP0476724
|
N-[(S)-(3-fluoropyridin-2-yl)-[3-fluoro-4-(trifluoromethoxy)phenyl]methyl]-6-oxo-1H-pyridine-3-carboxamide
Show/Hide
|
C19H12F5N3O3
|
1
|
| 1 |
IC50 = 9 nM
|
|
|
|
CP0375227
|
(4R)-8-fluoro-4-hydroxy-N-[4-(trifluoromethoxy)phenyl]spiro[3,4-dihydrochromene-2,4'-piperidine]-1'-carboxamide
Show/Hide
|
C21H20F4N2O4
|
1
|
| 1 |
IC50 = 9.5 nM
|
|
|
|
CP0389429
|
N-[(S)-(3-fluoropyridin-2-yl)-[4-(trifluoromethyl)phenyl]methyl]-6-oxo-1H-pyridine-3-carboxamide
Show/Hide
|
C19H13F4N3O2
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0466273
|
6-[[(S)-[4-(trifluoromethyl)phenyl]-[3-(trifluoromethyl)pyridin-2-yl]methyl]carbamoyl]pyridine-3-carboxylic acid
Show/Hide
|
C21H13F6N3O3
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0219345
|
6-[[(S)-(3-fluoropyridin-2-yl)-[3-fluoro-4-(trifluoromethoxy)phenyl]methyl]carbamoyl]pyridine-3-carboxylic acid
Show/Hide
|
C20H12F5N3O4
|
1
|
| 1 |
IC50 = 13 nM
|
|
|
|
CP0845991
|
(+/-)-8-Chloro-4-hydroxy-N-[4-(trifluoromethoxy)phenyl]-3,4-dihydro-1'H-spiro[chromene-2,4'-piperidine]-1'-carboxamide
Show/Hide
|
C21H20ClF3N2O4
|
1
|
| 1 |
IC50 = 13.3 nM
|
|
|
|
CP0396486
|
6-methoxy-N-[(S)-[4-(trifluoromethyl)phenyl]-[3-(trifluoromethyl)pyridin-2-yl]methyl]pyridine-3-carboxamide
Show/Hide
|
C21H15F6N3O2
|
1
|
| 1 |
IC50 = 15 nM
|
|
|
|
CP0375224
|
(4R)-8-bromo-4-hydroxy-N-[4-(trifluoromethoxy)phenyl]spiro[3,4-dihydrochromene-2,4'-piperidine]-1'-carboxamide
Show/Hide
|
C21H20BrF3N2O4
|
1
|
| 1 |
IC50 = 16.6 nM
|
|
|
|
CP0389426
|
N-[(S)-[4-(trifluoromethyl)phenyl]-[3-(trifluoromethyl)pyridin-2-yl]methyl]quinoline-7-carboxamide
Show/Hide
|
C24H15F6N3O
|
1
|
| 1 |
IC50 = 18 nM
|
|
|
|
CP0566817
|
8-bromo-N-[4-(trifluoromethyl)phenyl]spiro[3,4-dihydrochromene-2,4'-piperidine]-1'-carboxamide
Show/Hide
|
C21H20BrF3N2O2
|
1
|
| 1 |
IC50 = 18.9 nM
|
|
|
|
CP0390976
|
N-[(S)-[3-fluoro-4-(trifluoromethyl)phenyl]-[3-(trifluoromethyl)pyridin-2-yl]methyl]quinoline-7-carboxamide
Show/Hide
|
C24H14F7N3O
|
1
|
| 1 |
IC50 = 19 nM
|
|
|
|
CP0873823
|
(+/-)-8-Bromo-4-hydroxy-N-[4-(trifluoromethoxy)phenyl]-3,4-dihydro-1'H-spiro[chromene-2,4'-piperidine]-1'-carboxamide
Show/Hide
|
C21H20BrF3N2O4
|
1
|
| 1 |
IC50 = 19.5 nM
|
|
|
|
CP0446361
|
4-[[(S)-(3-fluoropyridin-2-yl)-[3-fluoro-4-(trifluoromethoxy)phenyl]methyl]carbamoyl]benzoic acid
Show/Hide
|
C21H13F5N2O4
|
1
|
| 1 |
IC50 = 20 nM
|
|
|
|
CP0553575
|
N-[(S)-[4-(trifluoromethyl)phenyl]-[3-(trifluoromethyl)pyridin-2-yl]methyl]quinoline-6-carboxamide
Show/Hide
|
C24H15F6N3O
|
1
|
| 1 |
IC50 = 20 nM
|
|
|
|
CP0466390
|
N-[(S)-[4-(trifluoromethoxy)phenyl]-[3-(trifluoromethyl)pyridin-2-yl]methyl]quinoline-7-carboxamide
Show/Hide
|
C24H15F6N3O2
|
1
|
| 1 |
IC50 = 22 nM
|
|
|
|
CP0963723
|
(+/-)-8-Fluoro-4-hydroxy-N-[4-(trifluoromethoxy)phenyl]-3,4-dihydro-1'H-spiro[chromene-2,4'-piperidine]-1'-carboxamide
Show/Hide
|
C21H20F4N2O4
|
1
|
| 1 |
IC50 = 22.5 nM
|
|
|
|
CP0390975
|
4-cyano-N-[(S)-[4-(trifluoromethyl)phenyl]-[3-(trifluoromethyl)pyridin-2-yl]methyl]benzamide
Show/Hide
|
C22H13F6N3O
|
1
|
| 1 |
IC50 = 27 nM
|
|
|
|
CP0396485
|
N-[(S)-[3-fluoro-4-(trifluoromethyl)phenyl]-[3-(trifluoromethyl)pyridin-2-yl]methyl]benzamide
Show/Hide
|
C21H13F7N2O
|
1
|
| 1 |
IC50 = 27 nM
|
|
|
|
CP0396484
|
N-[(S)-[4-(trifluoromethyl)phenyl]-[3-(trifluoromethyl)pyridin-2-yl]methyl]pyridine-3-carboxamide
Show/Hide
|
C20H13F6N3O
|
1
|
| 1 |
IC50 = 35 nM
|
|
|
|
CP0539003
|
8-chloro-N-[4-(trifluoromethoxy)phenyl]spiro[3,4-dihydrochromene-2,4'-piperidine]-1'-carboxamide
Show/Hide
|
C21H20ClF3N2O3
|
1
|
| 1 |
IC50 = 41.1 nM
|
|
|
|
CP0539002
|
8-bromo-4-hydroxy-N-[4-(trifluoromethyl)phenyl]spiro[3,4-dihydrochromene-2,4'-piperidine]-1'-carboxamide
Show/Hide
|
C21H20BrF3N2O3
|
1
|
| 1 |
IC50 = 44.5 nM
|
|
|
|
CP0375226
|
(4S)-8-chloro-4-hydroxy-N-[4-(trifluoromethoxy)phenyl]spiro[3,4-dihydrochromene-2,4'-piperidine]-1'-carboxamide
Show/Hide
|
C21H20ClF3N2O4
|
1
|
| 1 |
IC50 = 46.3 nM
|
|
|
|
CP0484709
|
8-chloro-N-[4-(trifluoromethyl)phenyl]spiro[3,4-dihydrochromene-2,4'-piperidine]-1'-carboxamide
Show/Hide
|
C21H20ClF3N2O2
|
1
|
| 1 |
IC50 = 48.5 nM
|
|
|
|
CP0390973
|
1-[(S)-[4-(trifluoromethyl)phenyl]-[3-(trifluoromethyl)pyridin-2-yl]methyl]-3-[(2S)-1,1,1-trifluoropropan-2-yl]urea
Show/Hide
|
C18H14F9N3O
|
1
|
| 1 |
IC50 = 51 nM
|
|
|
|
CP0466391
|
1-[(S)-(3-bromopyridin-2-yl)-[4-(trifluoromethyl)phenyl]methyl]-3-[(2S)-1,1,1-trifluoropropan-2-yl]urea
Show/Hide
|
C17H14BrF6N3O
|
1
|
| 1 |
IC50 = 59 nM
|
|
|
|
CP0375225
|
(4S)-8-bromo-4-hydroxy-N-[4-(trifluoromethoxy)phenyl]spiro[3,4-dihydrochromene-2,4'-piperidine]-1'-carboxamide
Show/Hide
|
C21H20BrF3N2O4
|
1
|
| 1 |
IC50 = 60 nM
|
|
|
|
CP0429060
|
8-chloro-4-hydroxy-N-[4-(trifluoromethyl)phenyl]spiro[3,4-dihydrochromene-2,4'-piperidine]-1'-carboxamide
Show/Hide
|
C21H20ClF3N2O3
|
1
|
| 1 |
IC50 = 65.9 nM
|
|
|
|
CP0389435
|
N-[(S)-quinolin-3-yl-[3-(trifluoromethyl)pyridin-2-yl]methyl]quinoline-7-carboxamide
Show/Hide
|
C26H17F3N4O
|
1
|
| 1 |
IC50 = 75 nM
|
|
|
|
CP0466259
|
N-[(S)-(4-methylphenyl)-[3-(trifluoromethyl)pyridin-2-yl]methyl]quinoline-7-carboxamide
Show/Hide
|
C24H18F3N3O
|
1
|
| 1 |
IC50 = 75 nM
|
|
|
|
CP0429061
|
8-fluoro-4-hydroxy-N-[4-(trifluoromethyl)phenyl]spiro[3,4-dihydrochromene-2,4'-piperidine]-1'-carboxamide
Show/Hide
|
C21H20F4N2O3
|
1
|
| 1 |
IC50 = 90.1 nM
|
|
|
|
CP0390978
|
N-[(S)-(3-methylphenyl)-[3-(trifluoromethyl)pyridin-2-yl]methyl]quinoline-7-carboxamide
Show/Hide
|
C24H18F3N3O
|
1
|
| 1 |
IC50 = 92 nM
|
|
|
|
CP0375228
|
(4S)-8-fluoro-4-hydroxy-N-[4-(trifluoromethoxy)phenyl]spiro[3,4-dihydrochromene-2,4'-piperidine]-1'-carboxamide
Show/Hide
|
C21H20F4N2O4
|
1
|
| 1 |
IC50 = 94 nM
|
|
|
|
CP0555772
|
N-[(S)-(4-methoxyphenyl)-[3-(trifluoromethyl)pyridin-2-yl]methyl]quinoline-7-carboxamide
Show/Hide
|
C24H18F3N3O2
|
1
|
| 1 |
IC50 = 95 nM
|
|
|
|
CP0375230
|
8-fluoro-N-[4-(trifluoromethyl)phenyl]spiro[3,4-dihydrochromene-2,4'-piperidine]-1'-carboxamide
Show/Hide
|
C21H20F4N2O2
|
1
|
| 1 |
IC50 = 97.3 nM
|
|
|
|
CP0541835
|
8-bromo-4-oxo-N-[4-(trifluoromethoxy)phenyl]spiro[3H-chromene-2,4'-piperidine]-1'-carboxamide
Show/Hide
|
C21H18BrF3N2O4
|
1
|
| 1 |
IC50 = 107.3 nM
|
|
|
|
CP0390979
|
N-[(S)-[3-fluoro-4-(trifluoromethyl)phenyl]-[2-(trifluoromethyl)phenyl]methyl]quinoline-7-carboxamide
Show/Hide
|
C25H15F7N2O
|
1
|
| 1 |
IC50 = 109 nM
|
|
|
|
CP0541836
|
8-chloro-4-oxo-N-[4-(trifluoromethoxy)phenyl]spiro[3H-chromene-2,4'-piperidine]-1'-carboxamide
Show/Hide
|
C21H18ClF3N2O4
|
1
|
| 1 |
IC50 = 111 nM
|
|
|
|
CP0426426
|
8-chloro-N-(6-fluoro-1,3-benzothiazol-2-yl)spiro[3,4-dihydrochromene-2,4'-piperidine]-1'-carboxamide
Show/Hide
|
C21H19ClFN3O2S
|
1
|
| 1 |
IC50 = 113.1 nM
|
|
|
|
CP0446362
|
1-[(S)-(3-fluoropyridin-2-yl)-[4-(trifluoromethyl)phenyl]methyl]-3-[(2S)-1,1,1-trifluoropropan-2-yl]urea
Show/Hide
|
C17H14F7N3O
|
1
|
| 1 |
IC50 = 119 nM
|
|
|
|
CP0548517
|
N-[(S)-(4-fluorophenyl)-[3-(trifluoromethyl)pyridin-2-yl]methyl]quinoline-7-carboxamide
Show/Hide
|
C23H15F4N3O
|
1
|
| 1 |
IC50 = 129 nM
|
|
|
|
CP0390977
|
N-[(S)-[3-(trifluoromethyl)phenyl]-[3-(trifluoromethyl)pyridin-2-yl]methyl]quinoline-7-carboxamide
Show/Hide
|
C24H15F6N3O
|
1
|
| 1 |
IC50 = 157 nM
|
|
|
|
CP0414937
|
8-chloro-N-[2-chloro-4-(trifluoromethyl)phenyl]spiro[3,4-dihydrochromene-2,4'-piperidine]-1'-carboxamide
Show/Hide
|
C21H19Cl2F3N2O2
|
1
|
| 1 |
IC50 = 177.8 nM
|
|
|
|
CP0407038
|
8-fluoro-4-oxo-N-[4-(trifluoromethoxy)phenyl]spiro[3H-chromene-2,4'-piperidine]-1'-carboxamide
Show/Hide
|
C21H18F4N2O4
|
1
|
| 1 |
IC50 = 182.1 nM
|
|
|
|
CP0414936
|
8-chloro-4-oxo-N-[4-(trifluoromethyl)phenyl]spiro[3H-chromene-2,4'-piperidine]-1'-carboxamide
Show/Hide
|
C21H18ClF3N2O3
|
1
|
| 1 |
IC50 = 230.4 nM
|
|
|
|
CP0489781
|
8-chloro-N-[4-(trifluoromethyl)-1,3-thiazol-2-yl]spiro[3,4-dihydrochromene-2,4'-piperidine]-1'-carboxamide
Show/Hide
|
C18H17ClF3N3O2S
|
1
|
| 1 |
IC50 = 265.8 nM
|
|
|
|
CP0429063
|
N-[4-(trifluoromethyl)phenyl]spiro[3,4-dihydrochromene-2,4'-piperidine]-1'-carboxamide
Show/Hide
|
C21H21F3N2O2
|
1
|
| 1 |
IC50 = 280.7 nM
|
|
|
|
CP0426427
|
8-chloro-N-(4-methylphenyl)spiro[3,4-dihydrochromene-2,4'-piperidine]-1'-carboxamide
Show/Hide
|
C21H23ClN2O2
|
1
|
| 1 |
IC50 = 289.6 nM
|
|
|
|
CP0429062
|
8-fluoro-4-oxo-N-[4-(trifluoromethyl)phenyl]spiro[3H-chromene-2,4'-piperidine]-1'-carboxamide
Show/Hide
|
C21H18F4N2O3
|
1
|
| 1 |
IC50 = 295.2 nM
|
|
|
|
CP0476725
|
N-[(S)-cyclohexyl-[3-(trifluoromethyl)pyridin-2-yl]methyl]quinoline-7-carboxamide
Show/Hide
|
C23H22F3N3O
|
1
|
| 1 |
IC50 = 301 nM
|
|
|
|
CP0466371
|
N-[(S)-[4-(trifluoromethyl)phenyl]-[4-(trifluoromethyl)pyridin-3-yl]methyl]quinoline-7-carboxamide
Show/Hide
|
C24H15F6N3O
|
1
|
| 1 |
IC50 = 311 nM
|
|
|
|
CP0493064
|
N-[(S)-phenyl-[3-(trifluoromethyl)pyridin-2-yl]methyl]quinoline-7-carboxamide
Show/Hide
|
C23H16F3N3O
|
1
|
| 1 |
IC50 = 389 nM
|
|
|
|
CP0552668
|
quinolin-6-yl-[(1R)-1-[4-(trifluoromethyl)phenyl]-3,4-dihydro-1H-isoquinolin-2-yl]methanone
Show/Hide
|
C26H19F3N2O
|
1
|
| 1 |
IC50 = 390 nM
|
|
|
|
CP0566816
|
8-chloro-6-fluoro-N-[4-(trifluoromethyl)phenyl]spiro[3,4-dihydrochromene-2,4'-piperidine]-1'-carboxamide
Show/Hide
|
C21H19ClF4N2O2
|
1
|
| 1 |
IC50 = 457.2 nM
|
|
|
|
CP0375229
|
8-chloro-N-(4-cyanophenyl)spiro[3,4-dihydrochromene-2,4'-piperidine]-1'-carboxamide
Show/Hide
|
C21H20ClN3O2
|
1
|
| 1 |
IC50 = 543.7 nM
|
|
|
|
CP0426425
|
8-bromo-4-oxo-N-[4-(trifluoromethyl)phenyl]spiro[3H-chromene-2,4'-piperidine]-1'-carboxamide
Show/Hide
|
C21H18BrF3N2O3
|
1
|
| 1 |
IC50 = 656.9 nM
|
|
|
|
CP0541069
|
6-fluoro-N-[4-(trifluoromethyl)phenyl]spiro[3,4-dihydrochromene-2,4'-piperidine]-1'-carboxamide
Show/Hide
|
C21H20F4N2O2
|
1
|
| 1 |
IC50 = 666.9 nM
|
|
|
|
CP0446363
|
N-[(1S)-2-phenyl-1-[3-(trifluoromethyl)pyridin-2-yl]ethyl]quinoline-7-carboxamide
Show/Hide
|
C24H18F3N3O
|
1
|
| 1 |
IC50 = 1140 nM
|
|
|
|
CP0375231
|
N-phenylspiro[3,4-dihydrochromene-2,4'-piperidine]-1'-carboxamide
Show/Hide
|
C20H22N2O2
|
1
|
| 1 |
IC50 = 2423 nM
|
|
|
|
CP0019489
|
US9108905, 1
Show/Hide
|
C12H14FNO
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0262006
|
4-[3-(3-methoxypropoxy)phenyl]-2-sulfanylidene-3,4-dihydro-1H-indeno[1,2-d]pyrimidin-5-one
Show/Hide
|
C21H20N2O3S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0402704
|
US9186360, 85
Show/Hide
|
C21H15F4N5O3S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0402705
|
US9186360, 24
Show/Hide
|
C21H16ClFN4O3S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0412454
|
US9186360, 22
Show/Hide
|
C26H28N4O4S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0412557
|
US9186360, 21
Show/Hide
|
C22H16ClF3N4O3S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0412575
|
US9186360, 49
Show/Hide
|
C23H19F5N4O4S2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0412578
|
US9186360, 70
Show/Hide
|
C21H16F4N4O5S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0412582
|
US9186360, 18
Show/Hide
|
C22H16F4N4O3S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0412583
|
US9186360, 30
Show/Hide
|
C22H17ClF2N4O4S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0412586
|
US9186360, 75
Show/Hide
|
C24H24Cl2N4O5S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0412587
|
US9186360, 82
Show/Hide
|
C19H13F4N5O4S2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0412588
|
US9186360, 11
Show/Hide
|
C22H17F3N4O3S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0412589
|
US9186360, 14
Show/Hide
|
C24H24N4O3S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0412592
|
US9186360, 56
Show/Hide
|
C22H17F5N4O4S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0412617
|
US9186360, 17
Show/Hide
|
C23H22N4O3S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0412618
|
US9186360, 28
Show/Hide
|
C22H15F5N4O3S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0412619
|
US9186360, 39
Show/Hide
|
C20H17F3N6O3S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0413535
|
US9186360, 58
Show/Hide
|
C20H14F4N4O4S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0413536
|
US9186360, 77
Show/Hide
|
C19H12F5N5O3S2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0413540
|
US9186360, 69
Show/Hide
|
C21H16F4N4O4S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0413541
|
US9186360, 87
Show/Hide
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C21H14F5N5O3S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
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CP0419511
|
US9186360, 31
Show/Hide
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C22H15F5N4O3S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
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CP0419512
|
US9186360, 73
Show/Hide
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C21H16ClF3N4O5S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
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CP0419513
|
US9186360, 94
Show/Hide
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C21H18F5N6O7PS
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
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CP0419515
|
US9186360, 6
Show/Hide
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C22H20N4O3S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0419516
|
US9186360, 20
Show/Hide
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C22H16F4N4O3S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0423872
|
US9186360, 27
Show/Hide
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C21H16F2N4O3S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0441106
|
US9186360, 86
Show/Hide
|
C22H16F5N5O4S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0441108
|
US9186360, 95
Show/Hide
|
C27H27ClF3N5O7S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0441109
|
US9186360, 1
Show/Hide
|
C19H16BrN7O2S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0441110
|
US9186360, 4
Show/Hide
|
C21H16Cl2N4O3S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0441111
|
US9186360, 9
Show/Hide
|
C21H17ClN4O3S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0441112
|
US9186360, 19
Show/Hide
|
C22H16F4N4O3S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0441113
|
US9186360, 23
Show/Hide
|
C25H26N4O4S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0441114
|
US9186360, 25
Show/Hide
|
C21H16ClFN4O3S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0441115
|
US9186360, 41
Show/Hide
|
C20H16F4N6O4S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0441116
|
US9186360, 62
Show/Hide
|
C22H17F5N4O5S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0463397
|
US9186360, 3
Show/Hide
|
C21H17BrN4O3S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0463398
|
US9186360, 12
Show/Hide
|
C25H26N4O3S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0463399
|
US9186360, 15
Show/Hide
|
C21H16ClFN4O3S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0463400
|
US9186360, 16
Show/Hide
|
C22H18F3N5O3
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0463403
|
US9186360, 60
Show/Hide
|
C21H15ClF4N4O5S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0463405
|
US9186360, 48
Show/Hide
|
C22H18F4N4O4S2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0470141
|
US9186360, 67
Show/Hide
|
C21H16F4N4O4S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0470143
|
US9186360, 92
Show/Hide
|
C19H12F5N5O4S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0470699
|
US9186360, 68
Show/Hide
|
C21H16F4N4O5S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0470719
|
US9186360, 47
Show/Hide
|
C20H16Cl2N4O3S2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0472819
|
US9186360, 38
Show/Hide
|
C20H16F4N6O3S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0478201
|
US9186360, 34
Show/Hide
|
C20H16F3N5O4S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0478205
|
US9186360, 54
Show/Hide
|
C20H14F4N4O4S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0478206
|
US9186360, 63
Show/Hide
|
C21H16ClF3N4O5S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0478207
|
US9186360, 71
Show/Hide
|
C21H16ClF3N4O4S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0478208
|
US9186360, 79
Show/Hide
|
C19H13F4N5O3S2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0478209
|
US9186360, 83
Show/Hide
|
C19H13F4N5O3S2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0479347
|
US9186360, 32
Show/Hide
|
C23H17F5N4O4S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0479348
|
US9186360, 36
Show/Hide
|
C20H15F4N5O3S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0479349
|
US9186360, 37
Show/Hide
|
C23H24Cl2N6O4S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0479354
|
US9186360, 50
Show/Hide
|
C22H18F4N4O3S2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0482710
|
US9186360, 65
Show/Hide
|
C21H16F4N4O4S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0482711
|
US9186360, 62
Show/Hide
|
C25H26F2N4O5S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0482713
|
US9186360, 35
Show/Hide
|
C22H18Cl2F3N5O4S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0483920
|
US9186360, 33
Show/Hide
|
C22H15F5N4O3S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0485488
|
US9186360, 81
Show/Hide
|
C19H13F4N5O3S2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0489890
|
US9186360, 10
Show/Hide
|
C27H28N4O3S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0490192
|
US9186360, 88
Show/Hide
|
C21H15F4N5O4S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0490193
|
US9186360, 16
Show/Hide
|
C22H17F3N4O3S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0495054
|
US9186360, 26
Show/Hide
|
C22H17F3N4O4S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0495055
|
US9186360, 29
Show/Hide
|
C22H16F4N4O4S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0499846
|
US9186360, 78
Show/Hide
|
C19H13F4N5O3S2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0512070
|
US9186360, 57
Show/Hide
|
C21H15Cl2F3N4O5S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0512071
|
US9186360, 72
Show/Hide
|
C21H15F5N4O4S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0512072
|
US9186360, 61
Show/Hide
|
C21H16F4N4O4S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0512088
|
US9186360, 5
Show/Hide
|
C21H17IN4O3S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0512093
|
US9186360, 8
Show/Hide
|
C21H18ClN5O3
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0516824
|
US9186360, 93
Show/Hide
|
C22H19ClF3N4O9PS
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0516825
|
US9186360, 76
Show/Hide
|
C21H15F5N4O4S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0516826
|
US9186360, 53
Show/Hide
|
C23H22F2N4O5S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0518910
|
US9186360, 55
Show/Hide
|
C20H14F4N4O4S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0518928
|
US9186360, 59
Show/Hide
|
C20H14F4N4O4S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0518929
|
US9186360, 74
Show/Hide
|
C22H18ClF3N4O5S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0518944
|
US9186360, 2
Show/Hide
|
C23H25N7O2S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0519543
|
US9186360, 13
Show/Hide
|
C21H16F2N4O3S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0544901
|
US9186360, 64
Show/Hide
|
C21H15F5N4O4S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0544902
|
US9186360, 84
Show/Hide
|
C19H12F5N5O3S2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0548934
|
US9186360, 80
Show/Hide
|
C19H13ClF3N5O4S2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0466275
|
N-[(S)-pyridin-2-yl-[3-(trifluoromethyl)pyridin-2-yl]methyl]quinoline-7-carboxamide
Show/Hide
|
C22H15F3N4O
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0492710
|
N-[(R)-1,3-thiazol-2-yl-[3-(trifluoromethyl)pyridin-2-yl]methyl]quinoline-7-carboxamide
Show/Hide
|
C20H13F3N4OS
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0396611
|
N-[(S)-(2-methylphenyl)-[3-(trifluoromethyl)pyridin-2-yl]methyl]quinoline-7-carboxamide
Show/Hide
|
C24H18F3N3O
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0521618
|
US9186360, 46
Show/Hide
|
C23H20F4N4O3S2
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
