Brief Information of the Cell Line and Protein
Cell Line ID: CL000011 , CHO
 Cell Line Info 
Synonyms
Chinese Hamster Ovary
CHO-ori
Category Spontaneously immortalized cell line
Organism
Cricetulus griseus (Chinese hamster)
Cellosaurus ID
CVCL_0213
Protein ID: PT01398 , Somatostatin receptor type 4
 Protein Info 
Gene Name SSTR4
Organism Homo sapiens, Human
Protein Classification Membrane receptor
Uniprot ID P31391
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000011
 Cell Line Info 
 Protein ID: PT01398
 Protein Info 
 
Compound ID Compound Name Compound Formula
CP0072718
 Compound Info 
3-[(1R,3R)-3-[5-(4-fluorophenyl)-1H-imidazol-2-yl]-1-(1-methylpyrazol-4-yl)-2,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-5-methyl-1,2,4-oxadiazole
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C27H23FN8O
  1
1
IC50 = 384 nM
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CP0237736
 Compound Info 
2-[(1R,3R)-3-[5-(4-fluorophenyl)-1H-imidazol-2-yl]-1-(1-methylpyrazol-4-yl)-2,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyridine-4-carboxylic acid
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C30H24FN7O2
  1
1
IC50 > 10000 nM
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CP0651917
 Compound Info 
5-((1R,3R)-1-(1-ethyl-1H-pyrazol-4-yl)-3-(4-(5-fluoropyridin-2-yl)-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol-1-yl)-3-methyl-1,3,4-oxadiazol-2(3H)-one
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C27H24FN9O2
  1
1
IC50 > 100000 nM
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CP0076698
 Compound Info 
(1R,3R)-1-(oxan-4-yl)-3-(5-phenyl-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole
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C25H26N4O
  1
1
IC50 > 1000 nM
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CP0432311
 Compound Info 
(4R,7S,10S,13S,16S,19S,22S,25S,28S,31S,34S,37R)-19,34-bis(4-aminobutyl)-31-(2-amino-2-oxoethyl)-37-[[2-[[(2S)-2-aminopropanoyl]amino]acetyl]amino]-13,25,28-tribenzyl-10,16-bis[(1R)-1-hydroxyethyl]-22-(1H-indol-3-ylmethyl)-7-methyl-6,9,12,15,18,21,24,27,30,33,36-undecaoxo-1,2-dithia-5,8,11,14,17,20,23,26,29,32,35-undecazacyclooctatriacontane-4-carboxamide
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C76H105N19O17S2
  1
1
Ki < 0.1 nM
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CP0430413
 Compound Info 
(4R,7S,10S,13S,16S,19S,22S,25S,28S,31S,34S,37R)-19,34-bis(4-aminobutyl)-37-[[2-[[(2S)-2-aminopropanoyl]amino]acetyl]amino]-13,25,28-tribenzyl-10,16-bis[(1R)-1-hydroxyethyl]-7-(hydroxymethyl)-22-(1H-indol-3-ylmethyl)-31-methyl-6,9,12,15,18,21,24,27,30,33,36-undecaoxo-1,2-dithia-5,8,11,14,17,20,23,26,29,32,35-undecazacyclooctatriacontane-4-carboxamide
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C75H104N18O17S2
  1
1
Ki < 0.1995 nM
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CP0485884
 Compound Info 
(4R,7S,10S,13S,16S,19S,22S,25S,28S,31S,34S,37R)-19,34-bis(4-aminobutyl)-31-(2-amino-2-oxoethyl)-37-[[(2S)-2-[[(2S)-2-aminopropanoyl]amino]propanoyl]amino]-13,25,28-tribenzyl-10,16-bis[(1R)-1-hydroxyethyl]-7-(hydroxymethyl)-22-(1H-indol-3-ylmethyl)-6,9,12,15,18,21,24,27,30,33,36-undecaoxo-1,2-dithia-5,8,11,14,17,20,23,26,29,32,35-undecazacyclooctatriacontane-4-carboxamide
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C77H107N19O18S2
  1
1
Ki < 0.1995 nM
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CP0398954
 Compound Info 
(4R,7S,10S,13S,16S,19S,22S,25S,28S,31S,34S,37R)-19-(4-aminobutyl)-31-(2-amino-2-oxoethyl)-37-[[2-[[(2S)-2-aminopropanoyl]amino]acetyl]amino]-13,25,28-tribenzyl-10,16-bis[(1R)-1-hydroxyethyl]-7-(hydroxymethyl)-22-(1H-indol-3-ylmethyl)-34-methyl-6,9,12,15,18,21,24,27,30,33,36-undecaoxo-1,2-dithia-5,8,11,14,17,20,23,26,29,32,35-undecazacyclooctatriacontane-4-carboxylic acid
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C73H97N17O19S2
  1
1
Ki < 0.3162 nM
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CP0049566
 Compound Info 
15-28-Somatostatin-28
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C76H104N18O19S2
  2
1
Ki = 0.59 nM
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2
Ki = 1.259 nM
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CP0406383
 Compound Info 
(4R,7S,10S,13S,16S,19S,22S,25S,28S,31S,34S,37R)-19,34-bis(4-aminobutyl)-31-(2-amino-2-oxoethyl)-37-[[2-[[(2S)-2-aminopropanoyl]amino]acetyl]amino]-13,25,28-tribenzyl-16-[(1R)-1-hydroxyethyl]-7-(hydroxymethyl)-22-(1H-indol-3-ylmethyl)-10-methyl-6,9,12,15,18,21,24,27,30,33,36-undecaoxo-1,2-dithia-5,8,11,14,17,20,23,26,29,32,35-undecazacyclooctatriacontane-4-carboxamide
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C75H103N19O17S2
  1
1
Ki < 0.631 nM
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CP0404159
 Compound Info 
(4R,7S,10S,13S,16S,19S,22S,25S,28S,31S,34S,37R)-19,34-bis(4-aminobutyl)-31-(2-amino-2-oxoethyl)-37-[[2-[[(2S)-2-aminopropanoyl]amino]acetyl]amino]-25,28-dibenzyl-10,16-bis[(1R)-1-hydroxyethyl]-7-(hydroxymethyl)-22-(1H-indol-3-ylmethyl)-13-methyl-6,9,12,15,18,21,24,27,30,33,36-undecaoxo-1,2-dithia-5,8,11,14,17,20,23,26,29,32,35-undecazacyclooctatriacontane-4-carboxamide
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C70H101N19O18S2
  1
1
Ki < 1 nM
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CP0460931
 Compound Info 
(4R,7S,10S,13S,16S,19S,22S,25S,28S,31S,34S,37R)-19,34-bis(4-aminobutyl)-31-(2-amino-2-oxoethyl)-37-[[2-[[(2S)-2-aminopropanoyl]amino]acetyl]amino]-13,28-dibenzyl-10,16-bis[(1R)-1-hydroxyethyl]-7-(hydroxymethyl)-22-(1H-indol-3-ylmethyl)-25-methyl-6,9,12,15,18,21,24,27,30,33,36-undecaoxo-1,2-dithia-5,8,11,14,17,20,23,26,29,32,35-undecazacyclooctatriacontane-4-carboxamide
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C70H101N19O18S2
  1
1
Ki < 1.995 nM
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CP0470520
 Compound Info 
(4R,7S,10R,13S,16R,19S,22R,25S,28R,31S,34R,37S)-19,34-bis(4-aminobutyl)-31-(2-amino-2-oxoethyl)-37-[[2-[[(2S)-2-aminopropanoyl]amino]acetyl]amino]-13,25,28-tribenzyl-16-[(1S)-1-hydroxyethyl]-10-[(1R)-1-hydroxyethyl]-7-(hydroxymethyl)-22-(1H-indol-3-ylmethyl)-6,9,12,15,18,21,24,27,30,33,36-undecaoxo-1,2-dithia-5,8,11,14,17,20,23,26,29,32,35-undecazacyclooctatriacontane-4-carboxylic acid
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C76H104N18O19S2
  1
1
Ki = 2 nM
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CP0404418
 Compound Info 
(4R,7S,10S,13S,16S,19S,22S,25S,28S,31S,34S,37R)-19,34-bis(4-aminobutyl)-31-(2-amino-2-oxoethyl)-37-[[2-[[(2S)-2-aminopropanoyl]amino]acetyl]amino]-13,25,28-tribenzyl-10-[(1R)-1-hydroxyethyl]-7-(hydroxymethyl)-22-(1H-indol-3-ylmethyl)-16-methyl-6,9,12,15,18,21,24,27,30,33,36-undecaoxo-1,2-dithia-5,8,11,14,17,20,23,26,29,32,35-undecazacyclooctatriacontane-4-carboxamide
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C75H103N19O17S2
  1
1
Ki < 3.981 nM
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CP0050675
 Compound Info 
(4R,7R,10S,13S,16S,19S,22S,25S,28S,31S,34S,37R)-37-{2-[(2S)-2-[(2S)-6-amino-2-[(2S)-2-[(2S)-2-[(2S)-2-{[(2S)-1-[(2S)-2-[(2S)-2-[(2S)-2-{[(2S)-1-[(2R)-2-[(2S)-2-[(2S)-2-[(2S)-2-[(2S)-2-amino-3-hydroxypropanamido]propanamido]-3-carbamoylpropanamido]-3-hydroxypropanamido]-3-carbamoylpropanoyl]pyrrolidin-2-yl]formamido}propanamido]-4-(methylsulfanyl)butanamido]propanoyl]pyrrolidin-2-yl]formamido}-5-carbamimidamidopentanamido]-4-carboxybutanamido]-5-carbamimidamidopentanamido]hexanamido]propanamido]a
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C137H207N41O39S3
  1
1
Ki = 5.4 nM
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CP0485165
 Compound Info 
(4R,7S,10S,13S,16S,19S,22S,25S,28S,31S,34S,37R)-19,34-bis(4-aminobutyl)-31-(2-amino-2-oxoethyl)-37-[[2-[[(2S)-2-aminopropanoyl]amino]acetyl]amino]-13,25-dibenzyl-10,16-bis[(1R)-1-hydroxyethyl]-7-(hydroxymethyl)-22-(1H-indol-3-ylmethyl)-28-methyl-6,9,12,15,18,21,24,27,30,33,36-undecaoxo-1,2-dithia-5,8,11,14,17,20,23,26,29,32,35-undecazacyclooctatriacontane-4-carboxamide
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C70H101N19O18S2
  1
1
Ki < 79.43 nM
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CP0375504
 Compound Info 
(5S,8S,11S,14R,17S,19aS)-11-(4-Amino-butyl)-5,17-dibenzyl-8-((R)-1-hydroxy-ethyl)-14-(1H-indol-3-ylmethyl)-tetradecahydro-3a,6,9,12,15,18-hexaaza-cyclopentacyclooctadecene-4,7,10,13,16,19-hexaone
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C44H54N8O7
  1
1
Ki < 100 nM
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CP0403937
 Compound Info 
CHEBI:72312
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C58H66N10O9
  1
1
Ki < 100 nM
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CP0403938
 Compound Info 
[(3S,6S,9S,12R,15S,18S,20R)-9-(4-aminobutyl)-3,15-dibenzyl-12-(1H-indol-3-ylmethyl)-2,5,8,11,14,17-hexaoxo-6-[(4-phenylmethoxyphenyl)methyl]-1,4,7,10,13,16-hexazabicyclo[16.3.0]henicosan-20-yl] N-[2-(dimethylamino)ethyl]carbamate
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C61H72N10O9
  1
1
Ki < 100 nM
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CP0406372
 Compound Info 
[(3S,6S,9S,12R,15S,18S,20R)-9-(4-aminobutyl)-3-benzyl-15-(1H-imidazol-5-ylmethyl)-12-(1H-indol-3-ylmethyl)-2,5,8,11,14,17-hexaoxo-6-[(4-phenylmethoxyphenyl)methyl]-1,4,7,10,13,16-hexazabicyclo[16.3.0]henicosan-20-yl] N-(2-aminoethyl)carbamate
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C56H66N12O9
  1
1
Ki < 100 nM
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CP0425318
 Compound Info 
[(3S,6S,9S,12R,15S,18S,20R)-9-(4-aminobutyl)-3-benzyl-15-[(4-hydroxyphenyl)methyl]-12-(1H-indol-3-ylmethyl)-2,5,8,11,14,17-hexaoxo-6-[(4-phenylmethoxyphenyl)methyl]-1,4,7,10,13,16-hexazabicyclo[16.3.0]henicosan-20-yl] N-(2-aminoethyl)carbamate
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C59H68N10O10
  1
1
Ki < 100 nM
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CP0375512
 Compound Info 
(4R,7S,10S,13R,16S,19R)-10-(4-aminobutyl)-N-[(2S)-1-amino-3-(1H-indol-3-yl)-1-oxopropan-2-yl]-19-[[(2R)-2-amino-3-phenylpropanoyl]amino]-16-[(4-hydroxyphenyl)methyl]-13-(1H-indol-3-ylmethyl)-6,9,12,15,18-pentaoxo-7-propan-2-yl-1,2-dithia-5,8,11,14,17-pentazacycloicosane-4-carboxamide
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C57H70N12O9S2
  1
1
Ki = 158.49 nM
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CP0416639
 Compound Info 
(3S,6S,9S,12R,15S,18S,20R)-9-(4-aminobutyl)-3,15-dibenzyl-20-hydroxy-12-(1H-indol-3-ylmethyl)-6-[(4-phenylmethoxyphenyl)methyl]-1,4,7,10,13,16-hexazabicyclo[16.3.0]henicosane-2,5,8,11,14,17-hexone
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C56H62N8O8
  1
1
Ki = 316.23 nM
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CP0463563
 Compound Info 
[(3S,6S,9S,12R,15S,18S,20R)-9-(4-aminobutyl)-3-benzyl-15-[3-(diaminomethylideneamino)propyl]-12-(1H-indol-3-ylmethyl)-2,5,8,11,14,17-hexaoxo-6-[(4-phenylmethoxyphenyl)methyl]-1,4,7,10,13,16-hexazabicyclo[16.3.0]henicosan-20-yl] N-(2-aminoethyl)carbamate
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C56H71N13O9
  1
1
Ki = 316.23 nM
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CP0492743
 Compound Info 
[(3S,6S,9S,12R,15S,18S,20R)-9-(4-aminobutyl)-3,15-dibenzyl-12-(1H-indol-3-ylmethyl)-2,5,8,11,14,17-hexaoxo-6-[(4-phenylmethoxyphenyl)methyl]-1,4,7,10,13,16-hexazabicyclo[16.3.0]henicosan-20-yl] N-(2-aminoethyl)carbamate
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C59H68N10O9
  1
1
Ki = 501.19 nM
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CP0861120
 Compound Info 
Cpa-cyclo(DCys-Pal-DTrp-Lys-NMeThr-Cys)-Nal-NH2
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C58H69ClN12O9S2
  1
1
Ki = 575 nM
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CP0375513
 Compound Info 
[(3S,6S,9S,12R,15S,18S,20R)-9-(4-aminobutyl)-3,15-dibenzyl-12-(1H-indol-3-ylmethyl)-2,5,8,11,14,17-hexaoxo-6-[(4-phenylmethoxyphenyl)methyl]-1,4,7,10,13,16-hexazabicyclo[16.3.0]henicosan-20-yl] N-(5-aminopentyl)carbamate
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C62H74N10O9
  1
1
Ki = 630.96 nM
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CP0136960
 Compound Info 
(4R,7S,10S,13R,16S,19S)-10-(4-aminobutyl)-19-[[(2S)-2-amino-3-(4-chlorophenyl)propanoyl]amino]-N-[(2S)-1-amino-3-naphthalen-2-yl-1-oxopropan-2-yl]-7-[(1R)-1-hydroxyethyl]-16-[(4-hydroxyphenyl)methyl]-13-(1H-indol-3-ylmethyl)-6,9,12,15,18-pentaoxo-1,2-dithia-5,8,11,14,17-pentazacycloicosane-4-carboxamide
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C58H68ClN11O10S2
  1
1
Ki = 1000 nM
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CP0845116
 Compound Info 
Cpa-cyclo(DCys-Pal-DTrp-Dab-Thr-Cys)-Nal-NH2
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C55H63ClN12O9S2
  1
1
Ki = 1000 nM
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CP0847290
 Compound Info 
Cpa-cyclo(DCys-Pal-DTrp-DDap-Thr-Cys)-Nal-NH2
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C54H61ClN12O9S2
  1
1
Ki = 1000 nM
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CP0847340
 Compound Info 
Cpa-cyclo(DCys-Pal-DTrp-Lys-Thr-Cys)-Nal-NH2
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C57H67ClN12O9S2
  1
1
Ki = 1000 nM
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CP0847417
 Compound Info 
Cpa-cyclo(DCys-Pal-DTrp-NMeLys-Thr-Cys)-DTrp-NH2
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C56H68ClN13O9S2
  1
1
Ki = 1000 nM
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CP0847584
 Compound Info 
Cpa-cyclo(DCys-Pal-NMeDTrp-Lys-Thr-Cys)-Nal-NH2
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C58H69ClN12O9S2
  1
1
Ki = 1000 nM
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CP0858062
 Compound Info 
Cpa-cyclo(DCys-Pal-DTrp-NMeLys-Thr-Cys)-Nal-NH2
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C58H69ClN12O9S2
  1
1
Ki = 1000 nM
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CP0859471
 Compound Info 
Cpa-cyclo(DCys-Pal-DTrp-Lys-Thr-Cys)-NMeNal-NH2
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C58H69ClN12O9S2
  1
1
Ki = 1000 nM
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CP0862999
 Compound Info 
Cpa-cyclo(DCys-Pal-DTrp-Lys-NMeThr-Cys)-Nal-NH2
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C58H69ClN12O9S2
  1
1
Ki = 1000 nM
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CP0880603
 Compound Info 
Cpa-cyclo(NMeDCys-Pal-DTrp-Lys-Thr-Cys)-Dip-NHMe
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C61H73ClN12O9S2
  1
1
Ki = 1000 nM
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CP0880716
 Compound Info 
Pal-cyclo(DCys-Pal-DTrp-NMeLys-Thr-Cys)-DTrp-NH2
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C55H68N14O9S2
  1
1
Ki = 1000 nM
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CP0886292
 Compound Info 
Cpa-cyclo(NMeDCys-Pal-DTrp-Lys-Thr-Cys)-Nal-NH2
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C59H72N12O9S2
  1
1
Ki = 1000 nM
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CP0888162
 Compound Info 
Cpa-cyclo(DCys-NMePal-DTrp-Lys-Thr-Cys)-Nal-NH2
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C58H69ClN12O9S2
  1
1
Ki = 1000 nM
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CP0902700
 Compound Info 
Nal-cyclo(DCys-Pal-DTrp-NMeLys-Thr-Cys)-DTrp-NH2
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C60H71N13O9S2
  1
1
Ki = 1000 nM
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CP0912534
 Compound Info 
Cpa-cyclo(DCys-Pal-NMeDTrp-NMeLys-Thr-Cys)-Nal-NH2
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C59H71ClN12O9S2
  1
1
Ki = 1000 nM
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CP0917823
 Compound Info 
NMeCpa-cyclo(DCys-Pal-DTrp-Lys-Thr-Cys)-Nal-NH2
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C58H69ClN12O9S2
  1
1
Ki = 1000 nM
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CP0854677
 Compound Info 
Tfm-cyclo(DCys-Pal-DTrp-NMeLys-Thr-Cys)-Nal-NH2
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C59H69F3N12O9S2
  1
1
Ki = 1246 nM
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CP0487505
 Compound Info 
4-Chloro-N-[(R)-2-(1H-indol-3-yl)-1-(4-phenyl-1H-imidazol-2-yl)-ethyl]-benzamidine
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C26H22ClN5
  1
1
Ki = 3840 nM
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CP0421312
 Compound Info 
N'-[(1R)-2-(1H-indol-3-yl)-1-(5-phenyl-1H-imidazol-2-yl)ethyl]-4-(trifluoromethoxy)benzenecarboximidamide
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C27H22F3N5O
  1
1
Ki = 3970 nM
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CP0421355
 Compound Info 
N'-[(1R)-2-(1H-indol-3-yl)-1-(5-phenyl-1H-imidazol-2-yl)ethyl]-4-methoxybenzenecarboximidamide
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C27H25N5O
  1
1
Ki = 5010 nM
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CP0415095
 Compound Info 
N'-[(1R)-2-(1H-indol-3-yl)-1-(5-phenyl-1H-imidazol-2-yl)ethyl]ethanimidamide
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C21H21N5
  1
1
Ki = 5920 nM
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CP0404417
 Compound Info 
N'-[(1R)-2-(1H-indol-3-yl)-1-(5-phenyl-1H-imidazol-2-yl)ethyl]-4-(trifluoromethyl)benzenecarboximidamide
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C27H22F3N5
  1
1
Ki = 6660 nM
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CP0392901
 Compound Info 
N'-[(1R)-2-(1H-indol-3-yl)-1-(5-phenyl-1H-imidazol-2-yl)ethyl]benzenecarboximidamide
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C26H23N5
  1
1
Ki = 7090 nM
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CP0376599
 Compound Info 
1-tert-Butyl-3-[(R)-2-(1H-indol-3-yl)-1-(4-phenyl-1H-imidazol-2-yl)-ethyl]-urea
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C24H27N5O
  1
1
Ki > 10000 nM
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CP0377054
 Compound Info 
4-tert-Butyl-N-[(R)-2-(1H-indol-3-yl)-1-(4-phenyl-1H-imidazol-2-yl)-ethyl]-benzamidine
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C30H31N5
  1
1
Ki > 10000 nM
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CP0382365
 Compound Info 
tert-butyl N-[(1R)-2-(1H-indol-3-yl)-1-(5-phenyl-1H-imidazol-2-yl)ethyl]carbamate
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C24H26N4O2
  1
1
Ki > 10000 nM
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CP0395005
 Compound Info 
1-(2,4-Difluoro-phenyl)-3-[(R)-2-(1H-indol-3-yl)-1-(4-phenyl-1H-imidazol-2-yl)-ethyl]-urea
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C26H21F2N5O
  1
1
Ki > 10000 nM
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CP0430098
 Compound Info 
N-[(1R)-2-(1H-indol-3-yl)-1-(5-phenyl-1H-imidazol-2-yl)ethyl]-2-[3-(trifluoromethyl)phenyl]acetamide
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C28H23F3N4O
  1
1
Ki > 10000 nM
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CP0495082
 Compound Info 
2,4-Difluoro-N-[(R)-2-(1H-indol-3-yl)-1-(4-phenyl-1H-imidazol-2-yl)-ethyl]-benzamidine
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C26H21F2N5
  1
1
Ki > 10000 nM
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CP0049568
 Compound Info 
(4R,7S,10S,13R,16S,19R)-10-(4-aminobutyl)-19-[[(2R)-2-amino-3-phenylpropanoyl]amino]-16-benzyl-N-[(2S,3R)-1,3-dihydroxybutan-2-yl]-7-[(1R)-1-hydroxyethyl]-13-(1H-indol-3-ylmethyl)-6,9,12,15,18-pentaoxo-1,2-dithia-5,8,11,14,17-pentazacycloicosane-4-carboxamide
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C49H66N10O10S2
  1
1
Ki < 1000 nM
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CP0151093
 Compound Info 
(3S,6S,9S,12R,15S,18S)-9-(4-Amino-butyl)-3-benzyl-15-(4-hydroxy-benzyl)-12-(1H-indol-3-ylmethyl)-6-isopropyl-1,18-dimethyl-1,4,7,10,13,16hexaaza-cyclooctadecane-2,5,8,11,14,17-hexaone
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C44H56N8O7
  1
1
Ki < 1000 nM
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CP0375444
 Compound Info 
3-(2-Naphtyl)-D-Ala-L-Cys(1)-L-Tyr-D-Trp-L-Lys-L-Val-L-Cys(1)-L-Thr-NH2
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C54H69N11O10S2
  1
1
Ki < 1000 nM
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CP0375876
 Compound Info 
(4R,7S,10S,13S,16S,19S,22S,25S,28S,31S,34S,37R)-19,34-bis(4-aminobutyl)-31-(2-amino-2-oxoethyl)-37-[[2-[[(2S)-2-aminopropanoyl]amino]acetyl]amino]-13,25,28-tribenzyl-10,16-bis[(1R)-1-hydroxyethyl]-7-(hydroxymethyl)-22-methyl-6,9,12,15,18,21,24,27,30,33,36-undecaoxo-1,2-dithia-5,8,11,14,17,20,23,26,29,32,35-undecazacyclooctatriacontane-4-carboxamide
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C68H100N18O18S2
  1
1
Ki < 1000 nM
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CP0412492
 Compound Info 
(3S,6S,9S,12R,15S,18S,20R)-9-(4-aminobutyl)-3,15-dibenzyl-20-hydroxy-6-[(1R)-1-hydroxyethyl]-12-(1H-indol-3-ylmethyl)-1,4,7,10,13,16-hexazabicyclo[16.3.0]henicosane-2,5,8,11,14,17-hexone
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C44H54N8O8
  1
1
Ki < 1000 nM
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CP0425316
 Compound Info 
(4R,7S,10S,13S,16S,19S,22S,25S,28S,31S,34S,37R)-34-(4-aminobutyl)-31-(2-amino-2-oxoethyl)-37-[[2-[[(2S)-2-aminopropanoyl]amino]acetyl]amino]-13,25,28-tribenzyl-10,16-bis[(1R)-1-hydroxyethyl]-7-(hydroxymethyl)-22-(1H-indol-3-ylmethyl)-19-methyl-6,9,12,15,18,21,24,27,30,33,36-undecaoxo-1,2-dithia-5,8,11,14,17,20,23,26,29,32,35-undecazacyclooctatriacontane-4-carboxamide
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C73H98N18O18S2
  1
1
Ki < 1000 nM
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