Compound ID |
Compound Name |
Compound Formula |
CP0420443
|
N'-[(2S)-1-[[(2S)-5-[[(E)-N'-(4-aminobutylcarbamoyl)carbamimidoyl]amino]-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-1-oxopentan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]-N-[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]octanediamide
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C85H132N26O17
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2
|
1 |
EC50 = 6.4 nM
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2 |
Ki = 1.2 nM
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CP0420444
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(2R,7R)-2,7-diamino-N,N'-bis[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]octanediamide
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C80H124N26O16
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4
|
1 |
EC50 = 6.9 nM
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|
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2 |
Ki = 0.18 nM
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3 |
Ki = 0.45 nM
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4 |
Ki = 2 nM
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CP0446417
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1229U91
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C110H170N34O24
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3
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1 |
EC50 = 8.5 nM
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2 |
Ki = 1.3 nM
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3 |
Ki = 1.6 nM
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CP0451146
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(4S)-5-[[(2S)-5-amino-1-[[(2S)-1-[[(2S)-1-[[(2S)-5-amino-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S,3S)-1-[[(2S)-4-amino-1-[[(2S)-1-[[(2S)-1-[[(2S,3R)-1-[[(2S)-1-[(2S)-2-[[(2S)-1-[[(2S)-1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]carbamoyl]pyrrolidin-1-yl]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-3-hydroxy-1-oxobutan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-4-methylsulfanyl-1-oxobutan-2-yl]amino]-1,4-dioxobutan-2-yl]amino]-3-methyl-1-oxopentan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-3-carboxy-1-oxopropan-2-yl]amino]-1-oxopropan-2-yl]amino]-1-oxopropan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-1,5-dioxopentan-2-yl]amino]-1-oxopropan-2-yl]amino]-4-methylsulfanyl-1-oxobutan-2-yl]amino]-1,5-dioxopentan-2-yl]amino]-4-[[(2S)-1-[(2S,3R)-2-[[(2S)-2-[[(2S)-4-amino-2-[[(2S)-2-[[2-[[(2S)-1-[(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-aminopropanoyl]pyrrolidine-2-carbonyl]amino]-4-methylpentanoyl]amino]-4-carboxybutanoyl]pyrrolidine-2-carbonyl]amino]-3-methylbutanoyl]amino]-3-(4-hydroxyphenyl)propanoyl]pyrrolidine-2-carbonyl]amino]acetyl]amino]-3-carboxypropanoyl]amino]-4-oxobutanoyl]amino]propanoyl]amino]-3-hydroxybutanoyl]pyrrolidine-2-carbonyl]amino]-5-oxopentanoic acid
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C185H287N53O54S2
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3
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1 |
EC50 = 9.7 nM
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2 |
Ki = 0.37 nM
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3 |
Ki = 0.65 nM
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CP0423824
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N-[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]-N'-[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-1-oxo-5-[[(E)-N'-[4-(propanoylamino)butylcarbamoyl]carbamimidoyl]amino]pentan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]octanediamide
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C88H136N26O18
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3
|
1 |
EC50 = 13 nM
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2 |
Ki = 0.66 nM
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3 |
Ki = 1.2 nM
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CP0529436
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(2S,7S)-2-amino-N,N'-bis[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]-7-(propanoylamino)octanediamide
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C83H128N26O17
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4
|
1 |
EC50 = 14 nM
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2 |
Ki = 0.32 nM
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3 |
Ki = 0.87 nM
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4 |
Ki = 6.3 nM
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CP0423825
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(2S,7S)-2,7-diamino-N,N'-bis[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]octanediamide
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C80H124N26O16
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3
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1 |
EC50 = 18 nM
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|
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2 |
Ki = 2.3 nM
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3 |
Ki = 17 nM
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CP0482449
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N,N'-bis[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]octanediamide
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C80H122N24O16
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2
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1 |
EC50 = 49 nM
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2 |
Ki = 3.5 nM
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CP0475519
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(2R,7R)-2-amino-N-[(2R)-1-[[(2R)-1-[[(2R)-1-[[(2R)-1-[[(2R)-1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]-N'-[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]-7-(propanoylamino)octanediamide
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C83H128N26O17
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2
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1 |
EC50 = 59 nM
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2 |
Ki = 2.8 nM
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CP0482448
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N'-[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]-N-[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-1-oxopropan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]octanediamide
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C77H115N21O16
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2
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1 |
EC50 = 290 nM
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2 |
Ki = 12 nM
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CP0446419
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N'-[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]-N-[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-1-oxopropan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]octanediamide
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|
C77H115N21O16
|
2
|
1 |
EC50 = 310 nM
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|
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2 |
Ki = 11 nM
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CP0489960
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N,N'-bis[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-1-oxopropan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]octanediamide
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C74H108N18O16
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2
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1 |
EC50 > 3000 nM
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2 |
Ki > 3000 nM
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CP0530735
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(2S)-2-amino-N,N'-bis[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-1-oxopropan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]octanediamide
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C74H109N19O16
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2
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1 |
EC50 > 3000 nM
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2 |
Ki > 3000 nM
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CP0845121
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1-((R)-9-Amino-4-(2,2-diphenylacetamido)-1-(4-hydroxyphenyl)-3,11,15-trioxo-2,8,10,16-tetraazaoctadec-9-en-18-yl)-4-((E)-2-(1,2,3,5,6,7-hexahydropyrido[3,2,1-ij]quinolin-9-yl)ethenyl)-2,6-dimethylpyridinium-hydrotrifluoroacetate
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C57H65F3N8O7
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2
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1 |
IC50 > 10000 nM
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2 |
Ki > 3000 nM
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CP0871818
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3-((R)-9-Amino-4-(2,2-diphenylacetamido)-1-(4-hydroxyphenyl)-3,11,18-trioxo-2,8,10,12,17-pentaazahenicos-9-en-21-yl)-2-((1E,3E)-4-(4-(dimethylamino)phenyl)buta-1,3-enyl)benzo[d]thiazol-3-ium hydrotrifluoroacetate
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C57H64F3N9O7S
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2
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1 |
IC50 > 1000 nM
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2 |
Ki > 500 nM
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CP0475520
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N-[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]-N'-[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-5-[[N-[4-(2,3-ditritiopropanoylamino)butylcarbamoyl]carbamimidoyl]amino]-1-oxopentan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]octanediamide
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C88H136N26O18
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1
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1 |
Kd = 0.67 nM
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|
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CP0904722
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[3H]-(2R,7R)-2-Amino-7-(propionylamino)octanedioyl-bis(Tyr-Arg-Leu-Arg-Tyr-amide)
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C83H128N26O17
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2
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1 |
Kd = 0.67 nM
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2 |
Kd = 9.8 nM
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CP0494526
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2,7-diamino-N,N'-bis[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]octanediamide
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C80H124N26O16
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2
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1 |
Kd = 0.67 nM
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2 |
Ki = 1.06 nM
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CP0875457
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Sub[-Tyr-Arg-Leu-Arg-Tyr-NH2]2
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C80H122N24O18
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1
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1 |
Ki = 0.05 nM
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|
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CP0487387
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(3S,12S,18S,27S)-9-N,24-N-bis[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]-3,18-bis[[(2S,3S)-2-amino-3-methylpentanoyl]amino]-2,6,11,17,21,26-hexaoxo-1,7,10,16,22,25-hexazatricyclo[25.3.0.012,16]triacontane-9,24-dicarboxamide
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C110H170N34O24
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1
|
1 |
Ki = 0.36 nM
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|
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CP0386806
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(2S)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-acetamido-5-carbamimidamidopentanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]-3-methylpentanoyl]amino]-N-[(2S)-1-[[(2S,3S)-1-[[(1R,3S)-3-[[(2S)-1-[[(1R,3S)-3-[[(2S)-1-[[(2S)-1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]carbamoyl]-2,2-dimethylcyclobutyl]amino]-5-carbamimidamido-1-oxopentan-2-yl]carbamoyl]-2,2-dimethylcyclobutyl]amino]-3-methyl-1-oxopentan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]butanediamide
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C80H127N25O16
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1
|
1 |
Ki = 0.53 nM
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|
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CP0403213
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(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-amino-1-hydroxy-3-(1H-indol-3-yl)propylidene]amino]-5-carbamimidamido-1-hydroxypentylidene]amino]-1-hydroxypentylidene]amino]-5-carbamimidamido-1-hydroxypentylidene]amino]-1-hydroxy-3-(4-hydroxyphenyl)propylidene]amino]-1-hydroxy-3-(1H-indol-3-yl)propylidene]amino]-5-carbamimidamido-1-hydroxypentylidene]amino]-1-hydroxypentylidene]amino]-5-carbamimidamido-1-hydroxypentylidene]amino]-1-hydroxy-3-(4-hydroxyphenyl)propylidene]amino]-1-hydroxy-3-(1H-indol-3-yl)propylidene]amino]-5-carbamimidamido-1-hydroxypentylidene]amino]-1-hydroxypentylidene]amino]-5-carbamimidamido-N-[(2S)-1-hydroxy-3-(4-hydroxyphenyl)-1-iminopropan-2-yl]pentanimidic acid
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C111H159N37O18
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1
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1 |
Ki = 3.9 nM
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CP0860001
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Adp[-Trp-Arg-Nva-Arg-Tyr-NH2]2
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C80H118N28O14
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1
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1 |
Ki = 4.2 nM
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CP0403212
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(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-amino-1-hydroxy-3-(1H-indol-3-yl)propylidene]amino]-5-carbamimidamido-1-hydroxypentylidene]amino]-1-hydroxypentylidene]amino]-5-carbamimidamido-1-hydroxypentylidene]amino]-1-hydroxy-3-(4-hydroxyphenyl)propylidene]amino]-1-hydroxy-3-(1H-indol-3-yl)propylidene]amino]-5-carbamimidamido-1-hydroxypentylidene]amino]-1-hydroxypentylidene]amino]-5-carbamimidamido-N-[(2S)-1-hydroxy-3-(4-hydroxyphenyl)-1-iminopropan-2-yl]pentanimidic acid
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C74H107N25O12
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1
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1 |
Ki = 5.3 nM
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|
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CP0434504
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(2S)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-acetamido-5-(diaminomethylideneamino)pentanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]-3-methylpentanoyl]amino]-N-[(2S)-1-[[(2S,3S)-1-[[(2S,3R)-1-[[(2S)-1-[[(1S,2R)-2-[[(2S)-1-[[(2S)-1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]carbamoyl]cyclopentyl]amino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-3-hydroxy-1-oxobutan-2-yl]amino]-3-methyl-1-oxopentan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]butanediamide
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C76H121N25O17
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1
|
1 |
Ki = 10 nM
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|
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CP0420154
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(2S)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-acetamido-5-carbamimidamidopentanoyl]amino]-5-carbamimidamidopentanoyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]-3-methylpentanoyl]amino]-N-[(2S)-1-[[(2S)-1-[[(2S,3R)-1-[[(2S)-1-[[(1S,2R)-2-[[(2S)-1-[[(2S)-1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]carbamoyl]cyclopentyl]amino]-5-carbamimidamido-1-oxopentan-2-yl]amino]-3-hydroxy-1-oxobutan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-1-oxohexan-2-yl]butanediamide
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C76H126N26O17
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1
|
1 |
Ki = 14 nM
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|
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CP0403214
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(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2R)-2-amino-3-[[(2R)-2-amino-3-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-1-oxopentan-2-yl]amino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-3-(1H-indol-3-yl)-1-oxopropan-2-yl]amino]-3-oxopropyl]disulfanyl]propanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]pentanoyl]amino]-N-[(2S)-1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]-5-(diaminomethylideneamino)pentanamide
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C80H118N28O14S2
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1
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1 |
Ki = 30 nM
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|
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CP0375160
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(2S)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-acetamido-5-carbamimidamidopentanoyl]amino]-3-(1H-imidazol-4-yl)propanoyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]-3-methylpentanoyl]amino]-N-[(2S)-1-[[(2S)-1-[[(1S,2R)-2-[[(2S)-1-[[(1S,2R)-2-[[(2S)-1-[[(2S)-1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]carbamoyl]cyclobutyl]amino]-5-carbamimidamido-1-oxopentan-2-yl]carbamoyl]cyclobutyl]amino]-5-carbamimidamido-1-oxopentan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]butanediamide
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C76H120N28O16
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1
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1 |
Ki = 35 nM
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CP0375161
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(2S)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-acetamido-5-(diaminomethylideneamino)pentanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]-3-methylpentanoyl]amino]-N-[(2S)-1-[[(2S,3S)-1-[[(1S,2R)-2-[[(2S)-1-[[(1S,2R)-2-[[(2S)-1-[[(2S)-1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]carbamoyl]cyclopentyl]amino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]carbamoyl]cyclopentyl]amino]-3-methyl-1-oxopentan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]butanediamide
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C78H123N25O16
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1
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1 |
Ki = 37 nM
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CP0420318
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(2S)-2-[[(2S)-2-[[(2S)-2-acetamido-3-(4-hydroxyphenyl)propanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]-N-[(2S)-1-[[(2S)-1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]-4-methylpentanamide
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C38H58N12O8
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2
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1 |
Ki = 50 nM
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2 |
Ki = 337 nM
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CP0375179
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(2S)-2-[[(2S)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-acetamido-5-carbamimidamidopentanoyl]amino]-5-carbamimidamidopentanoyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]-3-methylpentanoyl]amino]-4-amino-4-oxobutanoyl]amino]-N-[(2S)-1-[[(2S,3R)-1-[[(2S)-1-[[(1S,2R)-2-[[(2S)-1-[[(2S)-1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]carbamoyl]cyclobutyl]amino]-5-carbamimidamido-1-oxopentan-2-yl]amino]-3-hydroxy-1-oxobutan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]butanediamide
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C73H119N27O18
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1
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1 |
Ki = 70 nM
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CP0476460
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(2S)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-acetamido-5-carbamimidamidopentanoyl]amino]-3-(1H-imidazol-4-yl)propanoyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]-3-methylpentanoyl]amino]-N-[(2S)-1-[[(2S,3S)-1-[[(2S,3R)-1-[[(2S)-1-[[(1S,2R)-2-[[(2S)-1-[[(2S)-1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]carbamoyl]cyclobutyl]amino]-5-carbamimidamido-1-oxopentan-2-yl]amino]-3-hydroxy-1-oxobutan-2-yl]amino]-3-methyl-1-oxopentan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]butanediamide
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C75H119N25O17
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1
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1 |
Ki = 72 nM
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CP0375180
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(2S)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-acetamido-5-(diaminomethylideneamino)pentanoyl]amino]-5-carbamimidamidopentanoyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]-3-methylpentanoyl]amino]-N-[(2S)-1-[[(2S)-1-[[(2S,3R)-1-[[(2S)-1-[(2S)-2-[[(2S)-1-[[(2S)-1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]carbamoyl]pyrrolidin-1-yl]-5-carbamimidamido-1-oxopentan-2-yl]amino]-3-hydroxy-1-oxobutan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-1-oxohexan-2-yl]butanediamide
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C75H124N26O17
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1
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1 |
Ki = 75 nM
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CP0469093
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(2S)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-acetamido-5-carbamimidamidopentanoyl]amino]-5-carbamimidamidopentanoyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]-3-methylpentanoyl]amino]-N-[(2S)-1-[[(2S)-1-[[(2S,3R)-1-[[(2S)-1-[[(1S,2R)-2-[[(2S)-1-[[(2S)-1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]carbamoyl]cyclobutyl]amino]-5-carbamimidamido-1-oxopentan-2-yl]amino]-3-hydroxy-1-oxobutan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-1-oxohexan-2-yl]butanediamide
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C75H124N26O17
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1
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1 |
Ki = 93 nM
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CP0386811
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(1R,2S)-2-[[(2S)-2-[[(2S)-2-acetamido-3-(4-hydroxyphenyl)propanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]-N-[(2S)-1-[[(2S)-1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]cyclopentane-1-carboxamide
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C38H56N12O8
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1
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1 |
Ki = 105 nM
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CP0853428
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(R,R)-N,N-Bis[N-(N-{8-[4-diphenylacetylamino-4-(4-hydroxybenzylaminocarbonyl)butyl]amino-(amino)methyleneamino-carbonylamino-3,6-dioxaoctyl}-4-aminocarbonylbenzoyl)-2-aminoethyl]ethane-1,2-diamine tetra(hydrotrifluoroacetate)
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C92H113F3N18O18
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1
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1 |
Ki = 130 nM
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CP0529435
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1-N-[2-[2-[[4-[2-[2-[2-[[(E)-[amino-[[(4R)-4-[(2,2-diphenylacetyl)amino]-5-[(4-hydroxyphenyl)methylamino]-5-oxopentyl]amino]methylidene]carbamoyl]amino]ethoxy]ethoxy]ethylcarbamoyl]benzoyl]amino]ethyl-(2-aminoethyl)amino]ethyl]-4-N-[2-[2-[2-[[N-[(4R)-4-[(2,2-diphenylacetyl)amino]-5-[(4-hydroxyphenyl)methylamino]-5-oxopentyl]carbamimidoyl]carbamoylamino]ethoxy]ethoxy]ethyl]benzene-1,4-dicarboxamide
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C90H112N18O16
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3
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1 |
Ki = 150 nM
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2 |
Ki = 630 nM
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3 |
Ki = 660 nM
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CP0386808
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(2S)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-acetamido-5-carbamimidamidopentanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]-3-methylpentanoyl]amino]-N-[(2S)-1-[[(2S,3S)-1-[[(2S,3R)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]amino]-3-hydroxy-1-oxobutan-2-yl]amino]-3-methyl-1-oxopentan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]butanediamide
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C76H123N25O17
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1
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1 |
Ki = 157 nM
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CP0870060
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(R,R)-N,N-Bis[N-(N-{4-[4-diphenylacetylamino-4-(4-hydroxybenzylaminocarbonyl)butyl]amino-(amino)methyleneamino-carbonylaminobutyl}-4-aminocarbonylbenzoyl)-2-aminoethyl]ethane-1,2-diamine tetra(hydrotrifluoroacetate)
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C88H105F3N18O14
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1
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1 |
Ki = 210 nM
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CP0873884
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(S,S)-N,N-Bis[N-(N-{8-[4-diphenylacetylamino-4-(4-hydroxybenzylaminocarbonyl)butyl]amino-(amino)methyleneamino-carbonylamino-3,6-dioxaoctyl}-4-aminocarbonylbenzoyl)-2-aminoethyl]ethane-1,2-diamine tetra(hydrotrifluoroacetate)
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C92H113F3N18O18
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1
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1 |
Ki = 260 nM
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CP0903766
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(R,R)-N,N-Bis[N-(N-{6-[4-diphenylacetylamino-4-(4-hydroxybenzylaminocarbonyl)butyl]amino-(amino)methyleneamino-carbonylaminohexyl}-4-amino-4-oxo-butanoyl)-2-aminoethyl]ethane-1,2-diamine tetra(hydrotrifluoroacetate)
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C84H113F3N18O14
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1
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1 |
Ki = 270 nM
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CP0055951
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(4S)-5-[[(2S)-1-[[(2S)-1-[(2S)-2-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S,3S)-1-[[(2S)-4-amino-1-[[(2S)-1-[[(2S,3S)-1-[[(2S,3R)-1-[[(2S)-1-[[(2S)-5-amino-1-[[(2S)-1-[[(2S)-1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]amino]-1,5-dioxopentan-2-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]amino]-3-hydroxy-1-oxobutan-2-yl]amino]-3-methyl-1-oxopentan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-1,4-dioxobutan-2-yl]amino]-3-methyl-1-oxopentan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-3-(1H-imidazol-5-yl)-1-oxopropan-2-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-1-oxopropan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]amino]-1-oxopropan-2-yl]amino]-4-methylsulfanyl-1-oxobutan-2-yl]amino]-3-carboxy-1-oxopropan-2-yl]amino]-4-carboxy-1-oxobutan-2-yl]amino]-1-oxopropan-2-yl]carbamoyl]pyrrolidin-1-yl]-1-oxopropan-2-yl]amino]-3-carboxy-1-oxopropan-2-yl]amino]-4-[[2-[[(2S)-1-[(2S)-4-amino-2-[[(2S)-2-[[(2S)-1-[(2S)-6-amino-2-[[(2S)-2-[[(2S)-1-[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]pyrrolidine-2-carbonyl]amino]-3-hydroxypropanoyl]amino]hexanoyl]pyrrolidine-2-carbonyl]amino]-3-carboxypropanoyl]amino]-4-oxobutanoyl]pyrrolidine-2-carbonyl]amino]acetyl]amino]-5-oxopentanoic acid
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C189H285N55O57S
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1
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1 |
Ki = 282 nM
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CP0853471
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(R,R)-N,N-Bis{N-[N-(8-{4-diphenylacetylamino-4-[4-(ureidomethyl)benzylaminocarbonyl]butyl}amino-(amino)methyleneamino-carbonylamino-3,6-dioxaoctyl)-4-amino-4-oxo-butanoyl]-2-aminoethyl}ethane-1,2-diamine tetra(hydrotrifluoroacetate)
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C88H121F3N22O18
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1
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1 |
Ki = 290 nM
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CP0915112
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(R,R)-N,N-Bis[N-(N-{8-[4-diphenylacetylamino-4-(4-hydroxybenzylaminocarbonyl)butyl]amino-(amino)methyleneamino-carbonylamino-3,6-dioxaoctyl}-5-amino-5-oxopentanoyl)-2-aminoethyl]ethane-1,2-diamine tetra(hydrotrifluoroacetate)
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C86H117F3N18O18
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1
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1 |
Ki = 290 nM
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CP0853425
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(S,S)-N,N-Bis{N-[N-(8-{4-diphenylacetylamino-4-[4-(ureidomethyl)benzylaminocarbonyl]butyl}amino-(amino)methyleneamino-carbonylamino-3,6-dioxaoctyl)-4-amino-4-oxo-butanoyl]-2-aminoethyl}ethane-1,2-diamine tetra(hydrotrifluoroacetate)
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C88H121F3N22O18
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1
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1 |
Ki = 310 nM
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CP0486721
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N-[2-[2-aminoethyl-[2-[[5-[[N'-[(4R)-4-[(2,2-diphenylacetyl)amino]-5-[(4-hydroxyphenyl)methylamino]-5-oxopentyl]carbamimidoyl]amino]-5-oxopentanoyl]amino]ethyl]amino]ethyl]-N'-[N'-[(4R)-4-[(2,2-diphenylacetyl)amino]-5-[(4-hydroxyphenyl)methylamino]-5-oxopentyl]carbamimidoyl]pentanediamide
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C70H88N14O10
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1
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1 |
Ki = 390 nM
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CP0903765
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N1,N1'-(2,2'-(2-propionamidoethylazanediyl)bis(ethane-2,1-diyl))bis(N4-((R,Z)-9-amino-4-(2,2-diphenylacetamido)-1-(4-hydroxyphenyl)-3,11-dioxo-15,18-dioxa-2,8,10,12-tetraazaicos-9-en-20-yl)terephthalamide)tris(hydrotrifluoroacetate)
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C95H117F3N18O19
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1
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1 |
Ki = 410 nM
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CP0870337
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(R,R)-N,N-Bis[N-(N-{8-[4-diphenylacetylamino-4-(4-hydroxybenzylaminocarbonyl)butyl]amino-(amino)methyleneamino-carbonylamino-3,6-dioxaoctyl}-4-amino-4-oxobutanoyl)-2-aminoethyl]ethane-1,2-diamine tetra(hydrotrifluoroacetate)
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C84H113F3N18O18
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1
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1 |
Ki = 470 nM
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CP0375159
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(2S)-2-[[(2S)-2-[[(2S,3R)-2-acetamido-3-hydroxybutanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]-N-[(2S)-1-[[(2S)-1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]-4-methylpentanamide
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C33H56N12O8
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1
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1 |
Ki = 490 nM
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CP0395195
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(1R,2S)-2-[[(2S)-2-[[(2S,3R)-2-acetamido-3-hydroxybutanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]-N-[(2S)-1-[[(2S)-1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]cyclopentane-1-carboxamide
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C33H54N12O8
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1
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1 |
Ki = 509 nM
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CP0911606
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(R,R)-N,N-Bis[N-(N-{4-[4-diphenylacetylamino-4-(4-hydroxybenzylaminocarbonyl)butyl]amino-(amino)methyleneamino-carbonylaminobutyl}-6-amino-6-oxo-hexanoyl)-2-aminoethyl]ethane-1,2-diamine tetra(hydrotrifluoroacetate)
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C84H113F3N18O14
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1
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1 |
Ki = 550 nM
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CP0853466
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N-{N-[N-(6-{[(4R)-4-Diphenylacetylamino-4-(4-hydroxybenzylaminocarbonyl)butyl]amino-(amino)methylene-aminocarbonyl}aminohexyl)-4-amino-4-oxo-butanoyl]-2-aminoethyl}-N-(N-{N-[6-({(4S)-5-[2-(3,5-dioxo-1,2-diphenyl-1,2,4-triazolidin-4-yl)ethylamino]-5-oxo-4-[2-(1-{2-oxo-2-[4-(6-oxo-6,11-dihydro-5H-dibenzo[b,e]azepin-11-yl)piperazin-1-yl]ethyl}cyclopentyl)acetamido]pentyl}-amino-(amino)methylene-aminocarbonyl)aminohexyl]-aminocarbonylpropanoyl}-2-aminoethyl)ethane-1,2-diamine tetra(hydrotrifluoroacetate)
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C106H139F3N24O17
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1
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1 |
Ki = 910 nM
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CP0407120
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N,N'-bis[N'-[(4R)-4-[(2,2-diphenylacetyl)amino]-5-[(4-hydroxyphenyl)methylamino]-5-oxopentyl]carbamimidoyl]octanediamide
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C62H72N10O8
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1
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1 |
Ki = 2000 nM
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CP0852386
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(R,R)-N,N-Bis(N-{N-(N-[N-(4-{N-[2-diphenylacetylamino-2-(3-guanidinopropyl)acetyl]aminomethyl}benzyl)aminocarbonylaminobutyl]-aminocarbonylmethyl)-aminocarbonylpropanoyl}-2-aminoethyl)ethane-1,2-diamine tetra(hydrotrifluoroacetate)
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C86H117F3N22O14
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1
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1 |
Ki = 2200 nM
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CP0913286
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(S)-N1-{9-Amino-4-diphenylacetylamino-3,11-dioxo-1-[4-(ureidomethyl)phenyl]-2,8,10,12-tetraazatetradec-9-en-14-yl}-N4-{2-[2-(2-aminoethoxy)ethoxy]ethyl}succinamide bis(hydrotrifluoroacetate)
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C44H60F3N11O10
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1
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1 |
Ki = 3200 nM
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CP0887444
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(S)-N1-{9-Amino-4-diphenylacetylamino-3,11-dioxo-1-[4-(ureidomethyl)phenyl]-2,8,10,12-tetraazatetradec-9-en-14-yl}-N4-[2-(3-aminopropionylamino)ethyl]succinamidebis(hydrotrifluoroacetate)
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C43H57F3N12O9
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1
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1 |
Ki = 3300 nM
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CP0873882
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(R,R)-N,N-Bis(N-{N-[N-(4-{N-[2-diphenylacetylamino-2-(3-guanidinopro pyl)acetyl]aminomethyl}benzyl)aminocarbonylaminobutyl]-aminocarbonylbutanoyl}-2-aminoethyl)ethane-1,2-diamine tetra(hydrotrifluoroacetate)
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C84H115F3N20O12
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1
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1 |
Ki = 3500 nM
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CP0873885
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(S)-N1-{9-Amino-4-diphenylacetylamino-3,11,16,19-tetraoxo-1-[4-(ureidomethyl)phenyl]-2,8,10,12,15,20-hexaazadocos-9-en-22-yl}-N4-[2-(3-aminopropionylamino)ethyl]succinamide bis(hydrotrifluoroacetate)
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C49H67F3N14O11
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1
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1 |
Ki = 3500 nM
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CP0873886
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(S)-N1-(9-amino-4-(2,2-diphenylacetamido)-3,11-dioxo-1-(4-(ureidomethyl)phenyl)-2,8,10,12-tetraazatetradec-9-en-14-yl)-N4-(2-(2-(2-(3-aminopropoxy)ethoxy)ethoxy)ethyl)succinamide bis(hydrotrifluoroacetate)
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C47H66F3N11O11
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1
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1 |
Ki = 3700 nM
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CP0903995
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(R)-Nomega-(8-Guanidino-3,6-dioxaoctyl)aminocarbonyl-Nadiphenylacetyl-(4-hydroxy benzyl)argininamidebis(hydrotrifluoroacetate)
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C37H48F3N9O8
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1
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1 |
Ki = 3800 nM
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CP0856345
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(S)-N1-{9-Amino-4-diphenylacetylamino-3,11-dioxo-1-[4-(ureidomethyl)phenyl]-2,8,10,12-tetraazatetradec-9-en-14-yl}-N4-(2-aminoethyl)succinamidebis(hydrotrifluoroacetate)
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C40H52F3N11O8
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1
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1 |
Ki = 4100 nM
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CP0419095
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(R)-Nalpha-(2,2-diphenylacetyl)-N-(4-hydroxybenzyl)-N-omega-propanoylargininamide
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C30H35N5O4
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1
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1 |
Ki > 10000 nM
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CP0181598
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(R)-1-((5-(4-hydroxybenzylamino)-4-(2,2-diphenylacetamido)-5-oxopentylamino)(amino)methylene)-3-ethylurea
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C30H36N6O4
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1
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1 |
Ki > 10000 nM
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CP0382183
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(R)-ethyl 2-(3-((5-(4-hydroxybenzylamino)-4-(2,2-diphenylacetamido)-5-oxopentylamino)(amino)methylene)ureido)acetate
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C32H38N6O6
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1
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1 |
Ki > 10000 nM
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CP0382200
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(2R)-5-[[amino-[2-(propanoylamino)ethylcarbamoylamino]methylidene]amino]-2-[(2,2-diphenylacetyl)amino]-N-[(4-hydroxyphenyl)methyl]pentanamide;2,2,2-trifluoroacetic acid
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C37H43F6N7O9
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1
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1 |
Ki > 10000 nM
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CP0385636
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(2R)-5-[[amino-[(1-methyltriazol-4-yl)methylcarbamoylamino]methylidene]amino]-2-[(2,2-diphenylacetyl)amino]-N-[(4-hydroxyphenyl)methyl]pentanamide;2,2,2-trifluoroacetic acid
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C34H38F3N9O6
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1
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1 |
Ki > 10000 nM
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CP0403846
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ethyl 3-[[N'-[(4R)-4-[(2,2-diphenylacetyl)amino]-5-[(4-hydroxyphenyl)methylamino]-5-oxopentyl]carbamimidoyl]carbamoylamino]propanoate
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C33H40N6O6
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1
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1 |
Ki > 10000 nM
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CP0403847
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(2R)-5-[[amino-(2-aminoethylcarbamoylamino)methylidene]amino]-2-[(2,2-diphenylacetyl)amino]-N-[(4-hydroxyphenyl)methyl]pentanamide;2,2,2-trifluoroacetic acid
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C34H39F6N7O8
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1
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1 |
Ki > 10000 nM
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CP0334304
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(4S)-5-[[(2S)-5-amino-1-[[(2S)-1-[[(2S)-1-[[(2S)-5-amino-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S,3R)-1-[[(2S)-4-amino-1-[[(2S)-1-[[(2S)-1-[[(2S,3S)-1-[[(2S)-1-[(2S)-2-[[(2S)-1-[[(1S)-1-amino-2-(4-hydroxyphenyl)ethyl]amino]-5-carbamimidamido-1-oxopentan-2-yl]carbamoyl]pyrrolidin-1-yl]-5-carbamimidamido-1-oxopentan-2-yl]amino]-3-methyl-1-oxopentan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-4-methylsulfanyl-1-oxobutan-2-yl]amino]-1,4-dioxobutan-2-yl]amino]-3-hydroxy-1-oxobutan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-3-carboxy-1-oxopropan-2-yl]amino]-1-oxopropan-2-yl]amino]-1-oxopropan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-1,5-dioxopentan-2-yl]amino]-1-oxopropan-2-yl]amino]-4-methylsulfanyl-1-oxobutan-2-yl]amino]-1,5-dioxopentan-2-yl]amino]-4-[[(2S)-1-[(2S,3R)-2-[[(2S)-2-[[(2S)-4-amino-2-[[(2S)-2-[[2-[[(2S)-1-[(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-aminopropanoyl]pyrrolidine-2-carbonyl]amino]-4-methylpentanoyl]amino]-4-carboxybutanoyl]pyrrolidine-2-carbonyl]amino]-3-methylbutanoyl]amino]-3-(4-hydroxyphenyl)propanoyl]pyrrolidine-2-carbonyl]amino]acetyl]amino]-3-carboxypropanoyl]amino]-4-oxobutanoyl]amino]propanoyl]amino]-3-hydroxybutanoyl]pyrrolidine-2-carbonyl]amino]-5-oxopentanoic acid
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C184H287N53O53S2
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1
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1 |
Ki > 1000 nM
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CP0375162
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(2S)-2-[[(2S)-2-[[(2S,3R)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-acetamido-5-(diaminomethylideneamino)pentanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]-3-methylpentanoyl]amino]-4-amino-4-oxobutanoyl]amino]-4-methylpentanoyl]amino]-3-methylpentanoyl]amino]-3-hydroxybutanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]-N-[(2S)-1-[[(2S)-1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]pentanediamide
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C75H120N26O18
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1
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1 |
Ki > 1000 nM
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CP0429059
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(2S)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-acetamido-5-(diaminomethylideneamino)pentanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]-3-methylpentanoyl]amino]-N-[(2S)-1-[[(2S,3S)-1-[[(2S,3R)-1-[[(2S)-1-[[(1S,3R)-3-[[(2S)-1-[[(2S)-1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]carbamoyl]-2,2-dimethylcyclobutyl]amino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-3-hydroxy-1-oxobutan-2-yl]amino]-3-methyl-1-oxopentan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]butanediamide
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C77H123N25O17
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1
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1 |
Ki > 1000 nM
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CP0084655
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(R)-2-(2,2-diphenylacetamido)-5-guanidino-N-(4-hydroxybenzyl)pentanamide
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C27H31N5O3
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1
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1 |
Ki > 5000 nM
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CP0395455
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(R)-N-alpha-(2,2-Diphenylacetyl)-N-(4-ureidomethylbenzyl)argininamide
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C29H35N7O3
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1
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1 |
Ki > 5000 nM
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CP0429184
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(2S)-5-(diaminomethylideneamino)-2-[(2,2-diphenylacetyl)amino]-N-[(4-hydroxyphenyl)methyl]pentanamide
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C27H31N5O3
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1
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1 |
Ki > 5000 nM
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CP0853426
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(R)-Nalpha-Diphenylacetyl-[4-(4-aminobutylaminocarbonylaminomethyl)benzyl]argininamide bis(hydrotrifluoroacetate)
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C35H45F3N8O5
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1
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1 |
Ki > 5000 nM
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CP0856280
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(R)-N1-{9-Amino-4-diphenylacetylamino-3,11,16,19-tetraoxo-1-[4-(ureidomethyl)phenyl]-2,8,10,12,15,20-hexaazadocos-9-en-22-yl}-N4-[2-(3-aminopropionylamino)ethyl]succinamide bis(hydrotrifluoroacetate)
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C49H67F3N14O11
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1
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1 |
Ki > 5000 nM
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CP0856297
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(R)-Ndelta-(4-Aminobutyl)aminocarbonyl-Nalpha-diphenylacetyl-(4-ureidomethylbenzyl)ornithinamidetris(hydrotrifluoroacetate)
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C33H40F3N5O6
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1
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1 |
Ki > 5000 nM
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CP0856299
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(R)-Nomega-(8-Amino-3,6-dioxaoctyl)aminocarbonyl-Nalpha-diphenylacetyl-(4-hydroxy benzyl)argininamide bis(hydrotrifluoroacetate)
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C36H46F3N7O8
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1
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1 |
Ki > 5000 nM
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CP0856321
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(R)-N1-{9-Amino-4-diphenylacetylamino-3,11-dioxo-1-[4-(ureidomethyl)phenyl]-2,8,10,12-tetraazatetradec-9-en-14-yl}-N4-[2-(3-aminopropionylamino)ethyl]succinamidebis(hydrotrifluoroacetate)
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C43H57F3N12O9
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1
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1 |
Ki > 5000 nM
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CP0856323
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(S)-N1-{9-Amino-4-diphenylacetylamino-3,11,16,19-tetraoxo-1-[4-(ureidomethyl)phenyl]-2,8,10,12,15,20-hexaazadocos-9-en-22-yl}-N4-(2-aminoethyl)succinamide bis(hydrotrifluoroacetate)
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C46H62F3N13O10
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1
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1 |
Ki > 5000 nM
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CP0856324
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(R)-N1-(9-amino-4-(2,2-diphenylacetamido)-3,11-dioxo-1-(4-(ureidomethyl)phenyl)-2,8,10,12-tetraazatetradec-9-en-14-yl)-N4-(2-(2-(2-(3-aminopropoxy)ethoxy)ethoxy)ethyl)succinamide bis(hydrotrifluoroacetate)
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C47H66F3N11O11
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1
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1 |
Ki > 5000 nM
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CP0861468
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(R)-N1-{9-Amino-4-diphenylacetylamino-3,11,16,19-tetraoxo-1-[4-(ureidomethyl)phenyl]-2,8,10,12,15,20-hexaazadocos-9-en-22-yl}-N4-(2-aminoethyl)succinamide bis(hydrotrifluoroacetate)
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C46H62F3N13O10
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1
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1 |
Ki > 5000 nM
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CP0861469
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(R)-N1-{9-Amino-4-diphenylacetylamino-3,11-dioxo-1-[4-(ureidomethyl)phenyl]-2,8,10,12-tetraazatetradec-9-en-14-yl}-N4-{2-[2-(2-aminoethoxy)ethoxy]ethyl}succinamide bis(hydrotrifluoroacetate)
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C44H60F3N11O10
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1
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1 |
Ki > 5000 nM
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CP0861471
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(S)-Nomega-(8-Amino-3,6-dioxaoctyl)aminocarbonyl-Nalpha-diphenylacetyl-(4-ureidomethylbenzyl)argininamidebis(hydrotrifluoroacetate)
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C38H50F3N9O8
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1
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1 |
Ki > 5000 nM
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CP0861479
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(R)-N1-{9-Amino-4-diphenylacetylamino-3,11-dioxo-1-[4-(ureidomethyl)phenyl]-2,8,10,12-tetraazatetradec-9-en-14-yl}-N4-(2-aminoethyl)succinamide bis(hydrotrifluoroacetate)
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C40H52F3N11O8
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1
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1 |
Ki > 5000 nM
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CP0861485
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(R)-5-(2-(4-aminobutylcarbamoyl)guanidino)-2-(2,2-diphenylacetamido)-N-(4-hydroxybenzyl)pentanamide trifluoroacetate
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C34H42F3N7O6
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1
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1 |
Ki > 5000 nM
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CP0938240
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(R)-Nomega-(6-Aminohexyl)aminocarbonyl-Nalpha-diphenylacetyl-(4-ureidomethylbenzyl)argininamide bis(hydrotrifluoroacetate)
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C38H50F3N9O6
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1
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1 |
Ki > 5000 nM
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CP0201259
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(2R)-5-(diaminomethylideneamino)-N-[2-(3,5-dioxo-1,2-diphenyl-1,2,4-triazolidin-4-yl)ethyl]-2-[[2-[1-[2-oxo-2-[4-(6-oxo-5,11-dihydrobenzo[c][1]benzazepin-11-yl)piperazin-1-yl]ethyl]cyclopentyl]acetyl]amino]pentanamide
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C49H57N11O6
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1
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1 |
Ki > 7500 nM
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