| Compound ID |
Compound Name |
Compound Formula |
|
CP0155419
|
N-(2,3-dichlorophenyl)-2-[4-[6-(2-methylimidazol-1-yl)pyridin-3-yl]triazol-1-yl]acetamide
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|
C19H15Cl2N7O
|
2
|
| 1 |
EC50 = 2 nM
|
|
|
| 2 |
EC50 = 8 nM
|
|
|
|
CP0155420
|
N-(2,3-dichlorophenyl)-2-[4-[4-(2-methylimidazol-1-yl)phenyl]triazol-1-yl]acetamide
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|
C20H16Cl2N6O
|
2
|
| 1 |
EC50 = 3 nM
|
|
|
| 2 |
EC50 = 27 nM
|
|
|
|
CP0475865
|
N-(2,3-dichlorophenyl)-2-[4-(4-imidazol-1-ylphenyl)triazol-1-yl]acetamide
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|
C19H14Cl2N6O
|
2
|
| 1 |
EC50 = 3 nM
|
|
|
| 2 |
EC50 = 18 nM
|
|
|
|
CP0094466
|
N-(2,3-dichlorophenyl)-2-[4-[3-fluoro-4-(4-methylimidazol-1-yl)phenyl]triazol-1-yl]acetamide
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|
C20H15Cl2FN6O
|
2
|
| 1 |
EC50 = 9 nM
|
|
|
| 2 |
EC50 = 78 nM
|
|
|
|
CP0432996
|
N-(2,3-dichlorophenyl)-2-[4-[4-(4-methylimidazol-1-yl)phenyl]triazol-1-yl]acetamide
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|
C20H16Cl2N6O
|
2
|
| 1 |
EC50 = 12 nM
|
|
|
| 2 |
EC50 = 19 nM
|
|
|
|
CP0419296
|
N-(2,3-dichlorophenyl)-2-[4-[2-fluoro-4-(4-methylimidazol-1-yl)phenyl]triazol-1-yl]acetamide
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|
C20H15Cl2FN6O
|
2
|
| 1 |
EC50 = 19 nM
|
|
|
| 2 |
EC50 = 687 nM
|
|
|
|
CP0008174
|
2-[4-[3-methoxy-4-(4-methylimidazol-1-yl)phenyl]triazol-1-yl]-N-naphthalen-1-ylacetamide
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|
C25H22N6O2
|
2
|
| 1 |
EC50 = 23 nM
|
|
|
| 2 |
EC50 = 37 nM
|
|
|
|
CP0419292
|
N-(2,3-dichlorophenyl)-2-[4-[3-methoxy-4-(4-methylimidazol-1-yl)phenyl]triazol-1-yl]acetamide
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|
C21H18Cl2N6O2
|
2
|
| 1 |
EC50 = 36 nM
|
|
|
| 2 |
EC50 = 198 nM
|
|
|
|
CP0433029
|
N-(2,3-dimethylphenyl)-2-[4-[3-methoxy-4-(4-methylimidazol-1-yl)phenyl]triazol-1-yl]acetamide
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|
C23H24N6O2
|
1
|
| 1 |
EC50 = 80 nM
|
|
|
|
CP0419293
|
N-(2,3-dichlorophenyl)-2-methyl-2-[4-[4-(2-methylimidazol-1-yl)phenyl]triazol-1-yl]propanamide
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|
C22H20Cl2N6O
|
1
|
| 1 |
EC50 = 801 nM
|
|
|
|
CP0432997
|
N-(2,3-dichlorophenyl)-N-methyl-2-[4-[4-(2-methylimidazol-1-yl)phenyl]triazol-1-yl]acetamide
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|
C21H18Cl2N6O
|
1
|
| 1 |
EC50 > 20000 nM
|
|
|
|
CP0558267
|
N-(3-chloro-2-fluorophenyl)-7-pyridin-4-yl-3,5-dihydro-2H-1,4-benzoxazepine-4-carboxamide
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|
C21H17ClFN3O2
|
1
|
| 1 |
IC50 = 59 nM
|
|
|
|
CP0490372
|
N-(3-phenylphenyl)-7-pyridin-4-yl-3,5-dihydro-2H-1,4-benzoxazepine-4-carboxamide
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|
C27H23N3O2
|
1
|
| 1 |
IC50 = 62 nM
|
|
|
|
CP0421603
|
N-(3-cyanophenyl)-7-pyridin-4-yl-3,5-dihydro-2H-1,4-benzoxazepine-4-carboxamide
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|
C22H18N4O2
|
1
|
| 1 |
IC50 = 79 nM
|
|
|
|
CP0500791
|
N-(2-methoxyphenyl)-7-pyridin-4-yl-3,5-dihydro-2H-1,4-benzoxazepine-4-carboxamide
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|
C22H21N3O3
|
1
|
| 1 |
IC50 = 92 nM
|
|
|
|
CP0560535
|
7-pyridin-4-yl-N-[3-(trifluoromethyl)phenyl]-3,5-dihydro-2H-1,4-benzoxazepine-4-carboxamide
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|
C22H18F3N3O2
|
1
|
| 1 |
IC50 = 110 nM
|
|
|
|
CP0421600
|
N-(3,4-dichlorophenyl)-7-pyridin-4-yl-3,5-dihydro-2H-1,4-benzoxazepine-4-carboxamide
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|
C21H17Cl2N3O2
|
1
|
| 1 |
IC50 = 138 nM
|
|
|
|
CP0421602
|
N-(3-phenoxyphenyl)-7-pyridin-4-yl-3,5-dihydro-2H-1,4-benzoxazepine-4-carboxamide
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|
C27H23N3O3
|
1
|
| 1 |
IC50 = 146 nM
|
|
|
|
CP0466147
|
7-pyridin-4-yl-4-[[3-(trifluoromethyl)phenyl]methylsulfonyl]-3,5-dihydro-2H-1,4-benzoxazepine
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|
C22H19F3N2O3S
|
1
|
| 1 |
IC50 = 157 nM
|
|
|
|
CP0568468
|
N-(2,3-dichlorophenyl)-7-pyridin-4-yl-3,5-dihydro-2H-1,4-benzoxazepine-4-carboxamide
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|
C21H17Cl2N3O2
|
1
|
| 1 |
IC50 = 157 nM
|
|
|
|
CP0421597
|
N-(3,4-dichlorophenyl)-7-pyridin-4-yl-1,2,3,5-tetrahydro-1,4-benzodiazepine-4-carboxamide
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|
C21H18Cl2N4O
|
1
|
| 1 |
IC50 = 158 nM
|
|
|
|
CP0466150
|
N-(3-chlorophenyl)-7-pyridin-4-yl-3,5-dihydro-2H-1,4-benzoxazepine-4-carboxamide
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|
C21H18ClN3O2
|
1
|
| 1 |
IC50 = 164 nM
|
|
|
|
CP0466145
|
N-(3-methoxyphenyl)-7-quinolin-4-yl-3,5-dihydro-2H-1,4-benzoxazepine-4-carboxamide
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|
C26H23N3O3
|
1
|
| 1 |
IC50 = 216 nM
|
|
|
|
CP0560537
|
N-(3-methoxyphenyl)-7-pyridin-4-yl-3,5-dihydro-2H-1,4-benzoxazepine-4-carboxamide
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|
C22H21N3O3
|
1
|
| 1 |
IC50 = 305 nM
|
|
|
|
CP0560536
|
N-(3-fluorophenyl)-7-pyridin-4-yl-3,5-dihydro-2H-1,4-benzoxazepine-4-carboxamide
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|
C21H18FN3O2
|
1
|
| 1 |
IC50 = 413 nM
|
|
|
|
CP0500790
|
7-(2-aminopyridin-4-yl)-N-(3-cyanophenyl)-3,5-dihydro-2H-1,4-benzoxazepine-4-carboxamide
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|
C22H19N5O2
|
1
|
| 1 |
IC50 = 448 nM
|
|
|
|
CP0546100
|
N-(3-methoxyphenyl)-7-(3-methoxypyridin-4-yl)-3,5-dihydro-2H-1,4-benzoxazepine-4-carboxamide
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|
C23H23N3O4
|
1
|
| 1 |
IC50 = 486 nM
|
|
|
|
CP0421595
|
N-(3,4-dichlorophenyl)-8-pyridin-4-yl-1,3,4,5-tetrahydro-2-benzazepine-2-carboxamide
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|
C22H19Cl2N3O
|
1
|
| 1 |
IC50 = 590 nM
|
|
|
|
CP0564323
|
N-(2-fluorophenyl)-7-pyridin-4-yl-3,5-dihydro-2H-1,4-benzoxazepine-4-carboxamide
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|
C21H18FN3O2
|
1
|
| 1 |
IC50 = 604 nM
|
|
|
|
CP0466149
|
1-(7-pyridin-4-yl-3,5-dihydro-2H-1,4-benzoxazepin-4-yl)-2-[3-(trifluoromethyl)phenyl]ethanone
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|
C23H19F3N2O2
|
1
|
| 1 |
IC50 = 611 nM
|
|
|
|
CP0497286
|
N-(3-chloro-4-fluorophenyl)-7-pyridin-4-yl-3,5-dihydro-2H-1,4-benzoxazepine-4-carboxamide
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|
C21H17ClFN3O2
|
1
|
| 1 |
IC50 = 613 nM
|
|
|
|
CP0421604
|
N-phenyl-7-pyridin-4-yl-3,5-dihydro-2H-1,4-benzoxazepine-4-carboxamide
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|
C21H19N3O2
|
1
|
| 1 |
IC50 = 851 nM
|
|
|
|
CP0558266
|
N-(3,4-dichlorophenyl)-7-pyridin-4-yl-3,4-dihydro-1H-isoquinoline-2-carboxamide
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|
C21H17Cl2N3O
|
1
|
| 1 |
IC50 = 1050 nM
|
|
|
|
CP0485432
|
N-(3-methoxyphenyl)-7-(3-methylpyridin-4-yl)-3,5-dihydro-2H-1,4-benzoxazepine-4-carboxamide
Show/Hide
|
C23H23N3O3
|
1
|
| 1 |
IC50 = 1180 nM
|
|
|
|
CP0421599
|
N-(3,4-dichlorophenyl)-1-methyl-7-pyridin-4-yl-3,5-dihydro-2H-1,4-benzodiazepine-4-carboxamide
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|
C22H20Cl2N4O
|
1
|
| 1 |
IC50 = 2570 nM
|
|
|
|
CP0549438
|
N-(3-methoxyphenyl)-7-(2-methoxypyridin-4-yl)-3,5-dihydro-2H-1,4-benzoxazepine-4-carboxamide
Show/Hide
|
C23H23N3O4
|
1
|
| 1 |
IC50 = 2570 nM
|
|
|
|
CP0466148
|
N-(4-fluorophenyl)-7-pyridin-4-yl-3,5-dihydro-2H-1,4-benzoxazepine-4-carboxamide
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|
C21H18FN3O2
|
1
|
| 1 |
IC50 = 2610 nM
|
|
|
|
CP0546101
|
N-(3,4-dichlorophenyl)-6-pyridin-4-yl-2,3-dihydroindole-1-carboxamide
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|
C20H15Cl2N3O
|
1
|
| 1 |
IC50 = 2950 nM
|
|
|
|
CP0497287
|
1-butyl-N-(3,4-dichlorophenyl)-7-pyridin-4-yl-3,5-dihydro-2H-1,4-benzodiazepine-4-carboxamide
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|
C25H26Cl2N4O
|
1
|
| 1 |
IC50 = 4500 nM
|
|
|
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CP0421598
|
N-(3,4-dichlorophenyl)-5-pyridin-4-yl-1,3-dihydroisoindole-2-carboxamide
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|
C20H15Cl2N3O
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
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CP0421601
|
N-(3-methoxyphenyl)-N-methyl-7-pyridin-4-yl-3,5-dihydro-2H-1,4-benzoxazepine-4-carboxamide
Show/Hide
|
C23H23N3O3
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
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CP0466146
|
N-(3,4-dichlorophenyl)-7-pyridin-4-yl-3,4-dihydro-2H-quinoline-1-carboxamide
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|
C21H17Cl2N3O
|
1
|
| 1 |
IC50 > 20000 nM
|
|
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CP0466151
|
N-(4-methoxyphenyl)-7-pyridin-4-yl-3,5-dihydro-2H-1,4-benzoxazepine-4-carboxamide
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|
C22H21N3O3
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
