| Compound ID |
Compound Name |
Compound Formula |
|
CP0437055
|
2-[1-[4-[[(2S)-7-fluoro-4-methyl-2,3-dihydro-1,4-benzoxazin-2-yl]methoxy]benzoyl]-2-methylindol-4-yl]acetic acid
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|
C28H25FN2O5
|
2
|
| 1 |
IC50 = 0.81 nM
|
|
|
| 2 |
Ki = 5.3 nM
|
|
|
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CP0400679
|
2-[2-methyl-1-[4-[[(2S)-4-methyl-2,3-dihydro-1,4-benzoxazin-2-yl]methoxy]benzoyl]indol-4-yl]acetic acid
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|
C28H26N2O5
|
2
|
| 1 |
IC50 = 1.2 nM
|
|
|
| 2 |
Ki = 3.5 nM
|
|
|
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CP0485482
|
2-[2-methyl-1-[4-[[(2R)-4-methyl-2,3-dihydro-1,4-benzoxazin-2-yl]methoxy]benzoyl]indol-4-yl]acetic acid
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|
C28H26N2O5
|
2
|
| 1 |
IC50 = 10 nM
|
|
|
| 2 |
Ki = 170 nM
|
|
|
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CP0439527
|
2-[1-[4-[[(3R)-2,3-dihydro-1,4-benzodioxin-3-yl]methoxy]benzoyl]-2-methylindol-4-yl]acetic acid
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|
C27H23NO6
|
2
|
| 1 |
IC50 = 30 nM
|
|
|
| 2 |
Ki = 10 nM
|
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CP0451828
|
2-[1-[4-(2,3-dihydro-1-benzofuran-2-ylmethoxy)benzoyl]-2-methylindol-4-yl]acetic acid
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|
C27H23NO5
|
2
|
| 1 |
IC50 = 30 nM
|
|
|
| 2 |
Ki = 20 nM
|
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|
|
CP0486394
|
2-[1-[4-(3,4-dihydro-2H-chromen-2-ylmethoxy)benzoyl]-2-methylindol-4-yl]acetic acid
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|
C28H25NO5
|
2
|
| 1 |
IC50 = 30 nM
|
|
|
| 2 |
Ki = 50 nM
|
|
|
|
CP0486387
|
2-[1-[4-(1,3-benzodioxol-2-ylmethoxy)benzoyl]-2-methylindol-4-yl]acetic acid
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|
C26H21NO6
|
2
|
| 1 |
IC50 = 50 nM
|
|
|
| 2 |
Ki = 30 nM
|
|
|
|
CP0086399
|
2-[6-chloro-2-[4-(4-ethylphenyl)benzoyl]-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
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|
C28H25ClN2O3
|
1
|
| 1 |
IC50 = 120 nM
|
|
|
|
CP0374553
|
2-[2-methyl-1-[4-(2-phenoxyethoxy)benzoyl]indol-4-yl]acetic acid
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|
C26H23NO5
|
2
|
| 1 |
IC50 = 250 nM
|
|
|
| 2 |
Ki = 290 nM
|
|
|
|
CP0442380
|
2-[1-[4-[[(3S)-2,3-dihydro-1,4-benzodioxin-3-yl]methoxy]benzoyl]-2-methylindol-4-yl]acetic acid
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|
C27H23NO6
|
2
|
| 1 |
IC50 = 270 nM
|
|
|
| 2 |
Ki = 130 nM
|
|
|
|
CP0156868
|
2-[6-chloro-8-fluoro-2-(naphthalene-1-carbonyl)-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
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|
C24H18ClFN2O3
|
1
|
| 1 |
IC50 = 310 nM
|
|
|
|
CP0042410
|
2-[8-chloro-2-(naphthalene-1-carbonyl)-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
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|
C24H19ClN2O3
|
1
|
| 1 |
IC50 = 690 nM
|
|
|
|
CP0042409
|
2-[2-[4-(4-ethylphenyl)benzoyl]-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
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|
C28H26N2O3
|
1
|
| 1 |
IC50 = 780 nM
|
|
|
|
CP0055416
|
2-[2-(naphthalene-1-carbonyl)-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
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|
C24H20N2O3
|
1
|
| 1 |
IC50 = 780 nM
|
|
|
|
CP0087804
|
ACT-129968
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|
C24H19FN2O3
|
1
|
| 1 |
IC50 = 1290 nM
|
|
|
|
CP0261961
|
2-[2-(naphthalene-1-carbonyl)-8-(trifluoromethyl)-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
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|
C25H19F3N2O3
|
1
|
| 1 |
IC50 = 2200 nM
|
|
|
|
CP0130562
|
2-[8-methyl-2-(naphthalene-1-carbonyl)-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
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|
C25H22N2O3
|
1
|
| 1 |
IC50 = 2700 nM
|
|
|
|
CP0055418
|
2-[6-chloro-2-(3-chlorobenzoyl)-8-fluoro-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
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|
C20H15Cl2FN2O3
|
1
|
| 1 |
IC50 = 4100 nM
|
|
|
|
CP0050067
|
2-[2-[(5-acetyl-2-methoxyphenyl)methylsulfanyl]benzimidazol-1-yl]acetic acid
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|
C19H18N2O4S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0115424
|
2-[2-[[5-(butylcarbamoyl)-2-methoxyphenyl]methylsulfanyl]-5-fluorobenzimidazol-1-yl]acetic acid
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|
C22H24FN3O4S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0126760
|
2-[2-[(5-acetyl-2-methoxyphenyl)methylsulfanyl]-5-fluorobenzimidazol-1-yl]acetic acid
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|
C19H17FN2O4S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0154070
|
2-[2-[[5-(2,3-dihydroindole-1-carbonyl)-2-methoxyphenyl]methylsulfanyl]-5-fluorobenzimidazol-1-yl]acetic acid
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|
C26H22FN3O4S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0045673
|
2-[2-(3-chlorobenzoyl)-8-fluoro-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
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|
C20H16ClFN2O3
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0055420
|
2-[2-(3-chlorobenzoyl)-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
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|
C20H17ClN2O3
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0055873
|
2-[8-fluoro-2-[2-(1H-indol-3-yl)acetyl]-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
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|
C23H20FN3O3
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
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CP0055874
|
2-[8-fluoro-2-(thiophene-2-carbonyl)-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
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|
C18H15FN2O3S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0055877
|
2-[2-benzoyl-8-(trifluoromethyl)-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
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|
C21H17F3N2O3
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0070143
|
2-(2-benzoyl-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl)acetic acid
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|
C20H18N2O3
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
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CP0083568
|
2-[8-fluoro-2-(3-naphthalen-1-ylpropanoyl)-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
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|
C26H23FN2O3
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
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CP0086409
|
2-[8-fluoro-2-(2-naphthalen-1-ylacetyl)-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
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|
C25H21FN2O3
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
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CP0445860
|
2-[1-[4-(3,4-dihydro-2H-chromen-3-ylmethoxy)benzoyl]-2-methylindol-4-yl]acetic acid
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|
C28H25NO5
|
1
|
| 1 |
Ki = 390 nM
|
|
|
|
CP0391849
|
2-[1-(2,5-dichlorophenyl)sulfonyl-5-fluoro-2-methylindol-3-yl]acetic acid
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|
C17H12Cl2FNO4S
|
1
|
| 1 |
Ki = 1872 nM
|
|
|
|
CP0378076
|
(1-Benzenesulfonyl-5-fluoro-2-methyl-1H-indol-3-yl)-acetic acid
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|
C17H14FNO4S
|
1
|
| 1 |
Ki = 4860 nM
|
|
|
|
CP0498276
|
2-[5-fluoro-1-(3-fluorophenyl)sulfonyl-2-methylindol-3-yl]acetic acid
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|
C17H13F2NO4S
|
1
|
| 1 |
Ki = 6890 nM
|
|
|
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CP0391851
|
2-[5-fluoro-1-(4-methoxyphenyl)sulfonyl-2-methylindol-3-yl]acetic acid
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|
C18H16FNO5S
|
1
|
| 1 |
Ki = 7710 nM
|
|
|
|
CP0378230
|
2-[1-(4-chlorophenyl)sulfonyl-5-fluoro-2-methylindol-3-yl]acetic acid
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|
C17H13ClFNO4S
|
1
|
| 1 |
Ki = 8460 nM
|
|
|
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CP0259564
|
2-[5-fluoro-2-methyl-1-(4-methylsulfonylphenyl)sulfonylindol-3-yl]acetic acid
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|
C18H16FNO6S2
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
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CP0446446
|
2-[5-fluoro-2-methyl-1-(4-methylphenyl)sulfonylindol-3-yl]acetic acid
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|
C18H16FNO4S
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
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CP0456427
|
2-(1-butylsulfonyl-5-fluoro-2-methylindol-3-yl)acetic acid
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|
C15H18FNO4S
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
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CP0485411
|
2-[1-(1,2-dimethylimidazol-4-yl)sulfonyl-5-fluoro-2-methylindol-3-yl]acetic acid
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|
C16H16FN3O4S
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
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CP0503860
|
2-[5-fluoro-1-(4-fluorophenyl)sulfonyl-2-methylindol-3-yl]acetic acid
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|
C17H13F2NO4S
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
