Brief Information of the Cell Line and Protein
Cell Line ID: CL000011 , CHO
Synonyms
Chinese Hamster Ovary
CHO-ori
Category Spontaneously immortalized cell line
Organism
Cricetulus griseus (Chinese hamster)
Cellosaurus ID
CVCL_0213
Protein ID: PT01462 , Bromodomain-containing protein 4
Gene Name BRD4
Organism Homo sapiens, Human
Protein Classification Epigenetic regulator
Uniprot ID O60885
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000011  Protein ID: PT01462
 
Compound ID Compound Name Compound Formula
CP0500065
US9125915, compound 17
   Show/Hide
C20H20ClN5O2S
 1
1
IC50 = 12.8 nM
   TI
   LI
   LO
   TS
CP0461553
US9125915, compound 13
   Show/Hide
C20H20ClN5OS
 1
1
IC50 = 17.3 nM
   TI
   LI
   LO
   TS
CP0346525
US9125915, compound 6
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C20H19ClN4O2S
 1
1
IC50 = 18.2 nM
   TI
   LI
   LO
   TS
CP0513413
US9125915, compound 14
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C21H22ClN5O2S
 1
1
IC50 = 21 nM
   TI
   LI
   LO
   TS
CP0545648
US9125915, compound 10
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C29H29N5O3S
 1
1
IC50 = 47.1 nM
   TI
   LI
   LO
   TS
CP0518845
US9125915, compound 5
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C19H16Cl2N4O2S
 1
1
IC50 = 54.2 nM
   TI
   LI
   LO
   TS
CP0461577
US9125915, compound 3
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C26H26N6O2S
 1
1
IC50 = 54.9 nM
   TI
   LI
   LO
   TS
CP0538882
US9125915, compound 9
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C27H27N5O2S
 1
1
IC50 = 73.6 nM
   TI
   LI
   LO
   TS
CP0461578
US9125915, compound 4
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C26H22F3N5O3S
 1
1
IC50 = 77.2 nM
   TI
   LI
   LO
   TS
CP0538883
US9125915, compound 12
   Show/Hide
C24H21ClN6OS
 1
1
IC50 = 107.8 nM
   TI
   LI
   LO
   TS
CP0518846
US9125915, compound 7
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C27H26N4O4S
 1
1
IC50 = 113 nM
   TI
   LI
   LO
   TS
CP0545651
US9125915, compound 16
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C25H23ClN6O2S
 1
1
IC50 = 116.4 nM
   TI
   LI
   LO
   TS
CP0518847
US9125915, compound 15
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C25H23ClN6OS
 1
1
IC50 = 119.8 nM
   TI
   LI
   LO
   TS
CP0468377
US9125915, compound 2
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C28H26N6O2S
 1
1
IC50 = 121.2 nM
   TI
   LI
   LO
   TS
CP0500064
US9125915, compound 8
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C26H25N5O2S
 1
1
IC50 = 123.5 nM
   TI
   LI
   LO
   TS
CP0518252
US9125915, compound 18
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C25H23ClN6O2S
 1
1
IC50 = 146.8 nM
   TI
   LI
   LO
   TS
CP0545650
US9125915, compound 11
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C28H28FN5O2S
 1
1
IC50 = 225.3 nM
   TI
   LI
   LO
   TS