General Information of the Protein
Protein ID
PT06254
Protein Name
Probable G-protein coupled receptor 34
Gene Name
GPR34
Sequence
MRSHTITMTTTSVSSWPYSSHRMRFITNHSDQPPQNFSATPNVTTCPMDEKLLSTVLTTSYSVIFIVGLVGNIIALYVFLGIHRKRNSIQIYLLNVAIADLLLIFCLPFRIMYHINQNKWTLGVILCKVVGTLFYMNMYISIILLGFISLDRYIKINRSIQQRKAITTKQSIYVCCIVWMLALGGFLTMIILTLKKGGHNSTMCFHYRDKHNAKGEAIFNFILVVMFWLIFLLIILSYIKIGKNLLRISKRRSKFPNSGKYATTARNSFIVLIIFTICFVPYHAFRFIYISSQLNVSSCYWKEIVHKTNEIMLVLSSFNSCLDPVMYFLMSSNIRKIMCQLLFRRFQGEPSRSESTSEFKPGYSLHDTSVAVKIQSSSKST
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Organism
Homo sapiens, Human
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
Function
G-protein-coupled receptor of lysophosphatidylserine (LysoPS) that plays different roles in immune response (PubMed:16460680). Acts a damage-sensing receptor that triggers tissue repair upon recognition of dying neutrophils (By similarity). Mechanistically, apoptotic neutrophils release lysophosphatydilserine that are recognized by type 3 innate lymphoid cells (ILC3s) via GPR34, which activates downstream PI3K-AKT and RAS-ERK signaling pathways leading to STAT3 activation and IL-22 production (By similarity). Plays an important role in microglial function, controlling morphology and phagocytosis (By similarity).
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Uniprot ID
Primary ID:
Q9UPC5

Secondarily ID:
O95853
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Ensembl ID
ENSG00000171659
HGNC ID
HGNC:4490
Subcellular Location
Cell membrane
Map of Molecular Bioactivity Related to the Protein
Map of Molecular Bioactivity Related to the Protein

Protein
Cell Line
Compound

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Protein
Cell Line ID: CL000011 , CHO
 Cell Line Info 
Compound ID Compound Name Compound Formula
CP0850736
 Compound Info 
N-{[7-(4-Chlorophenyl)imidazo[1,2-a]pyridin-2-yl]carbonyl}-O-(4-methylbenzyl)tyrosine
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C31H26ClN3O4
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0850737
 Compound Info 
O-Benzyl-N-{[6-(2-chlorophenyl)imidazo[1,2-a]pyridin-2-yl]carbonyl}tyrosine
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C30H24ClN3O4
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0850738
 Compound Info 
O-Benzyl-N-{[6-(phenylethynyl)imidazo[1,2-b]pyridazin-2-yl]carbonyl}tyrosine
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C37H28N4O4
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0853136
 Compound Info 
O-Benzyl-N-{[5-(4-chlorophenyl)-3-methyl-1-benzofuran-2-yl]carbonyl}tyrosine
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C32H26ClNO5
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0853137
 Compound Info 
N-{[5-(4-Chlorophenyl)-1-benzothiophene-2-yl]carbonyl}-O-(4-fluorobenzyl)tyrosine
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C31H23ClFNO4S
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
   TI
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   TS
CP0853138
 Compound Info 
N-{[6-(4-Chlorophenyl)-3-methyl-1-benzofuran-2-yl]carbonyl}-O-(3-furylmethyl)-L-tyrosine
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C30H24ClNO6
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
   TI
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   LO
   TS
CP0853139
 Compound Info 
5-(4-Chlorophenyl)-2-({[4-(2,3-dihydro-1H-inden-2-yloxy)phenyl]acetyl}amino)indan-2-carboxylic acid
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C33H28ClNO4
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
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CP0859362
 Compound Info 
(2S)-[4-(Benzyloxy)phenyl]({[6-(4-chlorophenyl)-3-methyl-1-benzofuran-2-yl]carbonyl}amino)acetic acid
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C31H24ClNO5
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0864604
 Compound Info 
O-Benzyl-N-{[6-(4-chlorophenyl)-1H-indol-2-yl]carbonyl}tyrosine
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C31H25ClN2O4
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0864620
 Compound Info 
O-Benzyl-N-({6-[(E)-2-phenylethenyl]-1H-benzimidazol-2-yl}carbonyl)tyrosine
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C32H27N3O4
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
   TI
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   TS
CP0864621
 Compound Info 
O-(4-Fluorobenzyl)-N-{[5-(4-propoxyphenyl)-1-benzothiophene-2-yl]carbonyl}tyrosine
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C34H30FNO5S
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
   TI
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   TS
CP0864719
 Compound Info 
2-[({4-[(2-Aminobenzyl)oxy]phenyl}acetyl)amino]-5-(4-chlorophenyl)indan-2-carboxylic acid
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C31H27ClN2O4
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
   TI
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   TS
CP0864720
 Compound Info 
5-(5-Chloro-2-thienyl)-2-[({4-[4-fluorobenzyl)oxy]phenyl}acetyl)amino]indan-2-carboxylic acid
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C29H23ClFNO4S
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
   TI
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   TS
CP0866322
 Compound Info 
O--Benzyl-N-{[7-(4-chlorophenyl)imidazo[1,2-a]pyridin-2-yl]carbonyl}-L-tyrosine
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C30H24ClN3O4
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
   TI
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CP0866323
 Compound Info 
O-Benzyl-N-{[7-(4-chlorophenyl)imidazo[1,2-a]pyridin-2-yl]carbonyl}-N-methyltyrosine
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C31H26ClN3O4
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
   TI
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CP0866324
 Compound Info 
N-{[7-(4-Chlorophenyl)imidazo[1,2-a]pyridin-2-yl]carbonyl}-O-(4-fluorobenzyl)tyrosine
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C30H23ClFN3O4
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
   TI
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CP0867858
 Compound Info 
O-Benzyl-N-{[6-(benzylthio)imidazo[1,2-b]pyridazine-2-yl]carbonyl}tyrosine
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C30H26N4O4S
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
   TI
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CP0867859
 Compound Info 
O-Benzyl-N-({8-[(4-chlorobenzyl)oxy]imidazo[1,2-a]pyridin-2-yl}carbonyl)tyrosine
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C31H26ClN3O5
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
   TI
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CP0867860
 Compound Info 
O-Benzyl-N-{[2-(4-chlorophenyl)imidazo[1,2-a]pyridin-6-yl]carbonyl}tyrosine
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C30H24ClN3O4
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
   TI
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CP0867861
 Compound Info 
N-[2-[4-(Benzyloxy)phenyl]-1-(1H-tetrazol-5-yl)ethyl]-6-(4-chlorophenyl)imidazo[1,2-b]pyridazine-2-carboxamide
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C29H23ClN8O2
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
   TI
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CP0867862
 Compound Info 
O-Benzyl-N-{[6-(4-chlorophenyl)imidazo[1,2-a]pyridin-2-yl]carbonyl}-N-methyltyrosine
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C31H26ClN3O4
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0867863
 Compound Info 
N-{[6-(4-Chlorophenyl)imidazo[1,2-a]pyridin-2-yl]carbonyl}-O-(2-fluorobenzyl)tyrosine
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C30H23ClFN3O4
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0869104
 Compound Info 
O-Benzyl-N-({6-[(E)-2-(4-chlorophenyl)ethenyl]imidazo[1,2-b]pyridazin-2-yl}carbonyl)tyrosine
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C31H25ClN4O4
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0870073
 Compound Info 
O-Benzyl-N-{[5-(4-chlorophenyl)-1-benzothiophene-2-yl]carbonyl}tyrosine
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C31H24ClNO4S
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0873872
 Compound Info 
N-{[6-(4-Chlorophenyl)-1-benzofuran-2-yl]carbonyl}-O-(4-methylbenzyl)tyrosine
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C32H26ClNO5
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0873873
 Compound Info 
N-{[6-(4-Chlorophenyl)-1-benzofuran-2-yl]carbonyl}-O-(4-fluorobenzyl)tyrosine
   Show/Hide
C31H23ClFNO5
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
   TI
   LI
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CP0873874
 Compound Info 
O-Benzyl-N-{[7-(4-chlorophenyl)-2H-thiochromene-3-yl]carbonyl}tyrosine
   Show/Hide
C32H26ClNO4S
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0873875
 Compound Info 
O-Benzyl-N-{[5-(phenylethynyl)-1-benzothiophene-2-yl]carbonyl}tyrosine
   Show/Hide
C33H25NO4S
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
   TI
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CP0873876
 Compound Info 
5-(2-Chlorophenyl)-2-[({4-[(4-fluorobenzyl)oxy]phenyl}acetyl)amino]indan-2-carboxylic acid
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C31H25ClFNO4
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
   TI
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CP0873877
 Compound Info 
O-Benzyl-N-{[6-(4-chlorophenyl)-3-methyl-1-benzofuran-2-yl]carbonyl}-L-tyrosine
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C32H26ClNO5
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
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CP0877363
 Compound Info 
5-(4-Chlorophenyl)-2-{[(4-phenoxyphenyl)acetyl]amino)indan-2-carboxylic acid
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C30H24ClNO4
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
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CP0895831
 Compound Info 
2-(([4-(Benzyloxy)phenyl]acetyl}amino)-5-(4-chlorophenyl)indan-2-carboxylic acid
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C31H26ClNO4
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
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CP0899812
 Compound Info 
2-(([4-(1,3-Benzothiazol-2-yloxy)phenyl]acetyl}amino)-5-(4-chlorophenyl)indan-2-carboxylic acid
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C31H23ClN2O4S
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
   TI
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CP0899866
 Compound Info 
O-Benzyl-N-{[5-(4-chlorophenyl)-1H-indol-2-yl]carbonyl}tyrosine
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C31H25ClN2O4
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
   TI
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CP0899867
 Compound Info 
N-{[6-(4-Chlorophenyl)-1-benzofuran-2-yl]carbonyl}-O-(3-fluorobenzyl)tyrosine
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C31H23ClFNO5
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
   TI
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CP0903281
 Compound Info 
5-(4-Chlorophenyl)-2-{[(4-fluorobenzyl)sulfonyl]amino}indan-2-carboxylic acid
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C23H19ClFNO4S
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
   TI
   LI
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CP0903282
 Compound Info 
O-Benzyl-N-{[7-(4-chlorophenyl)imidazo[1,2-a]pyridin-2-yl]carbonyl}tyrosine
   Show/Hide
C30H24ClN3O4
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
   TI
   LI
   LO
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CP0903815
 Compound Info 
N-[3-Amino-5-(4-chlorophenyl)-1-benzofuran-2-yl]carbonyl)-O-benzyltyrosine
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C31H25ClN2O5
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0931113
 Compound Info 
O-Benzyl-N-{[6-(4-chlorophenyl)-1-methyl-1H-indole-2-yl]carbonyl}tyrosine
   Show/Hide
C32H27ClN2O4
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
   TI
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   LO
   TS
CP0931114
 Compound Info 
N-{[3-Amino-6-(4-chlorophenyl)-1-benzofuran-2-yl]carbonyl}-O-benzyltyrosine
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C31H25ClN2O5
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
   TI
   LI
   LO
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CP0931115
 Compound Info 
O-Benzyl-N-{[6-(4-chlorophenyl)-2-oxo-1,2-dihydroquinolin-3-yl]carbonyl}tyrosine
   Show/Hide
C32H25ClN2O5
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
   TI
   LI
   LO
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CP0931116
 Compound Info 
5-(3-Chlorophenyl)-2-[({4-[(4-fluorobenzyl)oxy]phenyl}acetyl)amino]indan-2-carboxylic acid
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C31H25ClFNO4
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
   TI
   LI
   LO
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CP0931117
 Compound Info 
5-(4-Chlorophenyl)-2-({[4-(3-thienylmethoxy)phenyl]acetyl}amino)indan-2-carboxylic acid
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C29H24ClNO4S
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
   TI
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CP0950996
 Compound Info 
N-{[6-(4-Chlorophenyl)imidazo[1,2-a]pyridin-2-yl]carbonyl}-N-{4-[(4-fluorobenzyl)oxy]benzyl}glycine
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C30H23ClFN3O4
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
   TI
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CP0950997
 Compound Info 
N-{[6-(4-Chlorophenyl)imidazo[1,2-a]pyridin-2-yl]carbonyl}-O-(4-fluorobenzyl)tyrosine
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C30H23ClFN3O4
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
   TI
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CP0952124
 Compound Info 
N-{[7-(4-Chlorophenyl)imidazo[1,2-a]pyridin-2-yl]carbonyl}-O-(2-fluorobenzyl)tyrosine
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C30H25ClFN3O4
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
   TI
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CP0952125
 Compound Info 
N-{[6-(4-Chlorophenyl)imidazo[1,2-a]pyridin-2-yl]carbonyl}-O-(3-thienylmethyl)-L-tyrosine
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C28H22ClN3O4S
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
   TI
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CP0952126
 Compound Info 
O-Benzyl-N-[(2E)-3-(4'-chlorobiphenyl-4-yl)propa-2-enoyl]tyrosine
   Show/Hide
C31H26ClNO4
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
   TI
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CP0952127
 Compound Info 
O-Benzyl-N-{[5-(4-chlorophenyl)-1-methyl-1H-indol-2-yl]carbonyl}tyrosine
   Show/Hide
C32H27ClN2O4
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
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CP0952216
 Compound Info 
O-Benzyl-N-{[6-(4-chlorophenyl)-1-benzofuran-2-yl]carbonyl}tyrosine
   Show/Hide
C31H24ClNO5
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
   TI
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CP0952217
 Compound Info 
O-Benzyl-N-{[6-(4-chlorophenyl)-1-benzothiophene-2-yl]carbonyl}tyrosine
   Show/Hide
C31H24ClNO4S
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
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CP0952218
 Compound Info 
2-[({4-[(3-Aminobenzyl)oxy]phenyl}acetyl)amino]-5-(4-chlorophenyl)indan-2-carboxylic acid
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C31H27ClN2O4
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
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CP0952219
 Compound Info 
N-{[6-(4-Chlorophenyl)-3-methyl-1-benzofuran-2-yl]carbonyl}-O-(3-thienylmethyl)-L-tyrosine
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C30H24ClNO5S
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
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CP0952855
 Compound Info 
O-Benzyl-N-{[5-(4-chlorophenyl)-1-benzofuran-2-yl]carbonyl}tyrosine
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C31H24ClNO5
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
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CP0952987
 Compound Info 
O-Benzyl-N-{[6-(4-chlorophenyl)-1H-benzimidazol-2-yl]carbonyl}tyrosine
   Show/Hide
C30H24ClN3O4
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
   TI
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CP0953611
 Compound Info 
N-[2-[4-(Benzyloxy)phenyl]-1-(1H-tetrazol-5-yl)ethyl]-6-(4-chlorophenyl)imidazo[1,2-a]pyridine-2-carboxamide
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C30H24ClN7O2
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
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CP0953984
 Compound Info 
O-Benzyl-N-{[6-(2-phenethyl)imidazo[1,2-a]pyridin-2-yl]carbonyl}tyrosine
   Show/Hide
C32H29N3O4
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
   TI
   LI
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CP0953986
 Compound Info 
O-Benzyl-N-{[6-(2-fluorophenyl)imidazo[1,2-a]pyridin-2-yl]carbonyl}tyrosine
   Show/Hide
C30H24FN3O4
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
   TI
   LI
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CP0953987
 Compound Info 
O-Benzyl-N-{[5-(4-chlorophenyl)imidazo[1,2-a]pyridin-2-yl]carbonyl}tyrosine
   Show/Hide
C30H24ClN3O4
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
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CP0953988
 Compound Info 
O-Benzyl-N-{[6-(4-chlorophenyl)imidazo[1,2-b]pyridazin-2-yl]carbonyl}tyrosine
   Show/Hide
C29H23ClN4O4
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
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CP0953989
 Compound Info 
O-Benzyl-N-[(2E)-3-(4'-chlorobiphenyl-3-yl)propa-2-enoyl]tyrosine
   Show/Hide
C31H26ClNO4
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
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CP0953990
 Compound Info 
N-{[6-(4-Chlorophenyl)-1H-benzimidazol-2-yl]carbonyl}-O-(4-fluorobenzyl)tyrosine
   Show/Hide
C30H23ClFN3O4
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
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CP0954257
 Compound Info 
O-Benzyl-N-{[6-(4-isopropoxyphenyl)imidazo[1,2-a]pyridin-2-yl]carbonyl}tyrosine
   Show/Hide
C33H31N3O5
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
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CP0954258
 Compound Info 
O-Benzyl-N-({6-[(E)-2-(4-chlorophenyl)ethenyl]imidazo[1,2-a]pyridin-2-yl}carbonyl)tyrosine
   Show/Hide
C32H26ClN3O4
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0954259
 Compound Info 
O-Benzyl-N-{[6-(4-chlorophenyl)-5-methylimidazo[1,2-a]pyridin-2-yl]carbonyl}tyrosine
   Show/Hide
C31H26ClN3O4
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
   TI
   LI
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   TS
CP0954260
 Compound Info 
O-Benzyl-N-alpha-{[6-(4-chlorophenyl)imidazo[1,2-a]pyridin-2-yl]carbonyl}-N-(methylsulfonyl)tyrosinamide
   Show/Hide
C31H27ClN4O5S
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
   TI
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CP0967263
 Compound Info 
N-{[7-(4-Chlorophenyl)imidazo[1,2-a]pyridin-2-yl]carbonyl}-O-(4-cyanobenzyl)tyrosine
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C31H23ClN4O4
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0967264
 Compound Info 
O-(4-Fluorobenzyl)-N-{[7-(phenylethyl)imidazo[1,2-a]pyridin-2-yl]carbonyl}tyrosine
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C32H24FN3O4
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0967265
 Compound Info 
O-Benzyl-N-{[3-chloro-6-(4-chlorophenyl)imidazo[1,2-a]pyridin-2-yl]carbonyl}tyrosine
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C30H23Cl2N3O4
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0967266
 Compound Info 
N-{[6-(4-Chlorophenyl)imidazo[1,2-a]pyridin-2-yl]carbonyl}-O-(3-fluorobenzyl)tyrosine
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C30H23ClFN3O4
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0967642
 Compound Info 
5-(4-Chlorophenyl)-2(4({4-[(4-fluorobenzyl)oxy]phenyl}acetyl)amino)indan-2-carboxylic acid
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C31H25ClFNO4
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0967643
 Compound Info 
N-{[7-(4-Chlorophenyl)imidazo[1,2-a]pyridin-2-yl]carbonyl}-O-(3-fluorobenzyl)tyrosine
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C30H23ClFN3O4
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0967645
 Compound Info 
O-Benzyl-N-({6-[(E)-2-(4-methylphenyl)ethenyl]imidazo[1,2-a]pyridin-2-yl}carbonyl)tyrosine
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C33H29N3O4
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0967646
 Compound Info 
O-Benzyl-N-{[6-(4-chlorophenyl)-8-methylimidazo[1,2-a]pyridin-2-yl]carbonyl}tyrosine
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C31H26ClN3O4
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0967647
 Compound Info 
O-Benzyl-N-{[7-(4-chlorophenyl)pyrazolo[1,5-a]pyrimidin-2-yl]carbonyl}tyrosine
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C29H23ClN4O4
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0967648
 Compound Info 
4-(Benzylamino)-N-([6-(4-chlorophenyl)imidazo[1,2-a]pyridin-2-yl]carbonyl)phenylalanine
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C30H25ClN4O3
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0967958
 Compound Info 
O-(4-Chlorobenzyl)-N-{[7-(4-chlorophenyl)imidazo[1,2-a]pyridin-2-yl]carbonyl}tyrosine
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C30H23Cl2N3O4
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0968252
 Compound Info 
N-{[7-(4-Chlorophenyl)imidazo[1,2-a]pyridin-2-yl]carbonyl}-O-(4-ethylbenzyl)tyrosine
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C32H28ClN3O4
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0968253
 Compound Info 
O-Benzyl-N-{[6-(4-chlorophenyl)imidazo[1,2-a]pyridin-2-yl]carbonyl}tyrosine
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C30H24ClN3O4
  1
1
IC50 <= 1000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
Cell Line ID: CL000050 , HEK293-A
 Cell Line Info 
Clinical Information about the Protein
Target 1 ( G-protein coupled receptor 34 (GPR34) )
Target Type Literature-reported Target