| Compound ID |
Compound Name |
Compound Formula |
|
CP0442988
|
US8916594, I-017
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|
C17H23FN4O3S
|
1
|
| 1 |
IC50 = 0.81 nM
|
|
|
|
CP0442989
|
US8916594, I-029
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|
C17H22F2N4O3S
|
1
|
| 1 |
IC50 = 0.86 nM
|
|
|
|
CP0919380
|
(9S)-9-(2-Hydroxy-4,4-dimethyl-6-oxo-1-cyclohexen-1-yl)-3,3-dimethyl-2,3,4,9-tetrahydro-1H-xanthen-1-one
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|
C23H26O4
|
1
|
| 1 |
IC50 = 34 nM
|
|
|
|
CP0879964
|
9'-(6-Hydroxy-8-oxospiro[3.5]non-7-yl)-4',9'-dihydrospiro[cyclobutane-1,3'-xanthen]-1'(2'H)-one
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|
C25H26O4
|
1
|
| 1 |
IC50 = 45 nM
|
|
|
|
CP0879963
|
9'-(7-Hydroxy-9-oxospiro[4.5]dec-8-yl)-4',9'-dihydrospiro[cyclopentane-1,3'-xanthen]-1'(2'H)-one
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|
C27H30O4
|
1
|
| 1 |
IC50 = 58 nM
|
|
|
|
CP0659250
|
9-(2-hydroxy-4,4-dimethyl-6-oxocyclohex-1-enyl)-3,3-dimethyl-2,3,4,9-tetrahydro-1H-xanthen-1-one
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|
C23H26O4
|
1
|
| 1 |
IC50 = 61 nM
|
|
|
|
CP0926509
|
6-Fluoro-9-(2-hydroxy-4,4-dimethyl-6-oxocyclohexyl)-3,3-dimethyl-2,3,4,9-tetrahydro-1H-xanthen-1-one
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|
C23H25FO4
|
1
|
| 1 |
IC50 = 63 nM
|
|
|
|
CP0926508
|
5-Fluoro-9-(2-hydroxy-4,4-dimethyl-6-oxocyclohexyl)-3,3-dimethyl-2,3,4,9-tetrahydro-1H-xanthen-1-one
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|
C23H25FO4
|
1
|
| 1 |
IC50 = 73 nM
|
|
|
|
CP0915023
|
6-Bromo-9-(2-hydroxy-4,4-dimethyl-6-oxocyclohexyl)-3,3-dimethyl-2,3,4,9-tetrahydro-1H-xanthen-1-one
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|
C23H25BrO4
|
1
|
| 1 |
IC50 = 81 nM
|
|
|
|
CP0906863
|
6-Chloro-9-(2-hydroxy-4,4-dimethyl-6-oxocyclohexyl)-3,3-dimethyl-2,3,4,9-tetrahydro-1H-xanthen-1-one
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|
C23H25ClO4
|
1
|
| 1 |
IC50 = 82 nM
|
|
|
|
CP0926196
|
9-(4,4-Diethyl-2-hydroxy-6-oxocyclohexyl)-3,3-diethyl-2,3,4,9-tetrahydro-1H-xanthen-1-one
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|
C27H34O4
|
1
|
| 1 |
IC50 = 90 nM
|
|
|
|
CP0916038
|
9'-(2-Hydroxy-4-oxospiro[5.5]undec-3-yl)-4',9'-dihydrospiro[cyclohexane-1,3'-xanthen]-1'(2'H)-one
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|
C29H34O4
|
1
|
| 1 |
IC50 = 109 nM
|
|
|
|
CP0949784
|
9-(2-Hydroxy-4,4-dimethyl-6-oxocyclohexyl)-3,3,6-trimethyl-2,3,4,9-tetrahydro-1H-xanthen-1-one
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|
C24H28O4
|
1
|
| 1 |
IC50 = 111 nM
|
|
|
|
CP0845121
|
1-((R)-9-Amino-4-(2,2-diphenylacetamido)-1-(4-hydroxyphenyl)-3,11,15-trioxo-2,8,10,16-tetraazaoctadec-9-en-18-yl)-4-((E)-2-(1,2,3,5,6,7-hexahydropyrido[3,2,1-ij]quinolin-9-yl)ethenyl)-2,6-dimethylpyridinium-hydrotrifluoroacetate
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|
C57H65F3N8O7
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 5000 nM
|
|
|
|
CP0917054
|
(9R)-9-(2-hydroxy-4,4-dimethyl-6-oxocyclohex-1-enyl)-3,3-dimethyl-2,3,4,4a,9,9a-hexahydroxanthen-1-one
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|
C23H26O4
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0871818
|
3-((R)-9-Amino-4-(2,2-diphenylacetamido)-1-(4-hydroxyphenyl)-3,11,18-trioxo-2,8,10,12,17-pentaazahenicos-9-en-21-yl)-2-((1E,3E)-4-(4-(dimethylamino)phenyl)buta-1,3-enyl)benzo[d]thiazol-3-ium hydrotrifluoroacetate
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|
C57H64F3N9O7S
|
2
|
| 1 |
IC50 > 1000 nM
|
|
|
| 2 |
Ki > 400 nM
|
|
|
