| Compound ID |
Compound Name |
Compound Formula |
|
CP0387595
|
2-[2-[(2R)-2-[(E,3S)-3-hydroxy-4-(3-methylphenyl)but-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C21H24N2O4S2
|
1
|
| 1 |
EC50 = 90 nM
|
|
|
|
CP0410236
|
2-[2-[(2R)-2-[(E,3S)-4-[3-(4-chlorophenyl)phenyl]-3-hydroxybut-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C26H25ClN2O4S2
|
1
|
| 1 |
EC50 = 260 nM
|
|
|
|
CP0378130
|
2-[2-[(2R)-2-[(E,3S)-3-hydroxy-4-[3-(4-methylphenyl)phenyl]but-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C27H28N2O4S2
|
1
|
| 1 |
EC50 = 380 nM
|
|
|
|
CP0410239
|
2-[2-[(2R)-2-[(E,3S)-4-[3-(3,4-dimethylphenyl)phenyl]-3-hydroxybut-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C28H30N2O4S2
|
1
|
| 1 |
EC50 = 1400 nM
|
|
|
|
CP0423877
|
2-[2-[(2R)-2-[(E,3S)-4-[3-(1-benzofuran-2-yl)phenyl]-3-hydroxybut-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C28H26N2O5S2
|
1
|
| 1 |
EC50 = 1500 nM
|
|
|
|
CP0378148
|
2-[2-[(2R)-2-[(E,3S)-4-[3-(1,3-benzoxazol-2-yl)phenyl]-3-hydroxybut-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C27H25N3O5S2
|
1
|
| 1 |
EC50 = 1600 nM
|
|
|
|
CP0410233
|
2-[2-[(2R)-2-[(E,3S)-3-hydroxy-4-(3-phenylphenyl)but-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C26H26N2O4S2
|
1
|
| 1 |
EC50 = 1800 nM
|
|
|
|
CP0410237
|
2-[2-[(2R)-2-[(E,3S)-4-[3-(1,3-benzothiazol-2-yl)phenyl]-3-hydroxybut-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C27H25N3O4S3
|
1
|
| 1 |
EC50 = 2700 nM
|
|
|
|
CP0378129
|
2-[2-[(2R)-2-[(E,3S)-3-hydroxy-4-[3-(6-methyl-1,3-benzoxazol-2-yl)phenyl]but-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C28H27N3O5S2
|
1
|
| 1 |
EC50 = 3200 nM
|
|
|
|
CP0410234
|
2-[2-[(2R)-2-[(E,3S)-3-hydroxy-4-[3-(4-methoxyphenyl)phenyl]but-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C27H28N2O5S2
|
1
|
| 1 |
EC50 = 4600 nM
|
|
|
|
CP0410310
|
2-[2-[(2R)-2-[(E,3S)-3-hydroxy-4-[3-(4-methyl-1,3-benzoxazol-2-yl)phenyl]but-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C28H27N3O5S2
|
1
|
| 1 |
EC50 = 8500 nM
|
|
|
|
CP0387597
|
2-[2-[(2R)-2-[(E,3S)-3-hydroxy-4-(3-naphthalen-2-ylphenyl)but-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C30H28N2O4S2
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0410235
|
2-[2-[(2R)-2-[(E,3S)-4-[3-(5-chloro-1,3-benzothiazol-2-yl)phenyl]-3-hydroxybut-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C27H24ClN3O4S3
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0410240
|
2-[2-[(2R)-2-[(E,3S)-3-hydroxy-4-[3-(5-methyl-1,3-benzoxazol-2-yl)phenyl]but-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C28H27N3O5S2
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0410241
|
2-[2-[(2R)-2-[(E,3S)-4-[3-(5,7-dimethyl-1,3-benzoxazol-2-yl)phenyl]-3-hydroxybut-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C29H29N3O5S2
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0410311
|
2-[2-[(2R)-2-[(E,3S)-4-[3-(5-chloro-1,3-benzoxazol-2-yl)phenyl]-3-hydroxybut-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C27H24ClN3O5S2
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0410313
|
2-[2-[(2R)-2-[(E,3S)-4-[3-(2,4-dimethylphenyl)phenyl]-3-hydroxybut-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C28H30N2O4S2
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
