| Compound ID |
Compound Name |
Compound Formula |
|
CP0410312
|
4-[2-[(2R)-2-[(E,3S)-3-hydroxy-4-[3-(pyridin-2-ylmethoxy)phenyl]but-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]butanoic acid
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|
C26H32N2O5S
|
1
|
| 1 |
EC50 = 0.61 nM
|
|
|
|
CP0387595
|
2-[2-[(2R)-2-[(E,3S)-3-hydroxy-4-(3-methylphenyl)but-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]-1,3-thiazole-4-carboxylic acid
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|
C21H24N2O4S2
|
1
|
| 1 |
EC50 = 0.79 nM
|
|
|
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CP0395230
|
4-[2-[(1R,2R)-2-[(E,3S)-3-hydroxy-4-[3-(methoxymethyl)phenyl]but-1-enyl]-5-oxocyclopentyl]ethylsulfanyl]butanoic acid
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|
C23H32O5S
|
1
|
| 1 |
EC50 = 1.1 nM
|
|
|
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CP0395226
|
4-[2-[(2R)-2-[(E,3S)-3-hydroxy-4-[3-(methoxymethyl)phenyl]but-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]butanoic acid
Show/Hide
|
C22H31NO5S
|
1
|
| 1 |
EC50 = 1.3 nM
|
|
|
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CP0224474
|
4-(2-((1R,2R,3R)-3-hydroxy-2-((S,E)-3-hydroxy-4-(3-(methoxymethyl)phenyl)but-1-enyl)-5-oxocyclopentyl)ethylthio)butanoic acid
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|
C23H32O6S
|
1
|
| 1 |
EC50 = 1.4 nM
|
|
|
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CP0378129
|
2-[2-[(2R)-2-[(E,3S)-3-hydroxy-4-[3-(6-methyl-1,3-benzoxazol-2-yl)phenyl]but-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]-1,3-thiazole-4-carboxylic acid
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|
C28H27N3O5S2
|
1
|
| 1 |
EC50 = 1.6 nM
|
|
|
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CP0401107
|
4-[2-[(4S)-4-[(E,3S)-4-(3-ethylphenyl)-3-hydroxybut-1-enyl]-2-oxo-1,3-thiazolidin-3-yl]ethylsulfanyl]butanoic acid
Show/Hide
|
C21H29NO4S2
|
1
|
| 1 |
EC50 = 1.9 nM
|
|
|
|
CP0378148
|
2-[2-[(2R)-2-[(E,3S)-4-[3-(1,3-benzoxazol-2-yl)phenyl]-3-hydroxybut-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C27H25N3O5S2
|
1
|
| 1 |
EC50 = 2.2 nM
|
|
|
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CP0431080
|
4-[2-[(4S)-4-[(E,3S)-3-hydroxy-4-[3-(methoxymethyl)phenyl]but-1-enyl]-2-oxo-1,3-thiazolidin-3-yl]ethylsulfanyl]butanoic acid
Show/Hide
|
C21H29NO5S2
|
1
|
| 1 |
EC50 = 2.4 nM
|
|
|
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CP0410231
|
4-[2-[(2R)-2-[(E,3S)-4-[3-(1,3-benzothiazol-2-yl)phenyl]-3-hydroxybut-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]butanoic acid
Show/Hide
|
C27H30N2O4S2
|
1
|
| 1 |
EC50 = 3.2 nM
|
|
|
|
CP0388033
|
4-[2-[(4S)-4-[(E,3S)-3-hydroxy-4-[3-(trifluoromethyl)phenyl]but-1-enyl]-2-oxo-1,3-thiazolidin-3-yl]ethylsulfanyl]butanoic acid
Show/Hide
|
C20H24F3NO4S2
|
1
|
| 1 |
EC50 = 4.3 nM
|
|
|
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CP0388032
|
4-[2-[(4S)-4-[(E,3S)-3-hydroxy-4-phenylbut-1-enyl]-2-oxo-1,3-thiazolidin-3-yl]ethylsulfanyl]butanoic acid
Show/Hide
|
C19H25NO4S2
|
1
|
| 1 |
EC50 = 4.8 nM
|
|
|
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CP0410311
|
2-[2-[(2R)-2-[(E,3S)-4-[3-(5-chloro-1,3-benzoxazol-2-yl)phenyl]-3-hydroxybut-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C27H24ClN3O5S2
|
1
|
| 1 |
EC50 = 4.9 nM
|
|
|
|
CP0423877
|
2-[2-[(2R)-2-[(E,3S)-4-[3-(1-benzofuran-2-yl)phenyl]-3-hydroxybut-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C28H26N2O5S2
|
1
|
| 1 |
EC50 = 5.3 nM
|
|
|
|
CP0427837
|
4-[2-[(4S)-4-[(E,3S)-4-(3-fluorophenyl)-3-hydroxybut-1-enyl]-2-oxo-1,3-thiazolidin-3-yl]ethylsulfanyl]butanoic acid
Show/Hide
|
C19H24FNO4S2
|
1
|
| 1 |
EC50 = 5.7 nM
|
|
|
|
CP0378128
|
4-[2-[(2R)-2-[(E,3S)-3-hydroxy-4-(3-methylphenyl)but-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]butanoic acid
Show/Hide
|
C21H29NO4S
|
1
|
| 1 |
EC50 = 5.7 nM
|
|
|
|
CP0431204
|
4-[2-[(4S)-4-[(E,3S)-3-hydroxy-4-(3-propylphenyl)but-1-enyl]-2-oxo-1,3-thiazolidin-3-yl]ethylsulfanyl]butanoic acid
Show/Hide
|
C22H31NO4S2
|
1
|
| 1 |
EC50 = 6.1 nM
|
|
|
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CP0480109
|
4-[2-[(2R)-2-[(E,3S)-4-[3-(1-benzofuran-2-yl)phenyl]-3-hydroxybut-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]butanoic acid
Show/Hide
|
C28H31NO5S
|
1
|
| 1 |
EC50 = 7 nM
|
|
|
|
CP0400839
|
7-[(2R)-2-[(E,3S)-3-hydroxy-4-[3-(methoxymethyl)phenyl]but-1-enyl]-5-sulfanylidenepyrrolidin-1-yl]heptanoic acid
Show/Hide
|
C23H33NO4S
|
1
|
| 1 |
EC50 = 7.3 nM
|
|
|
|
CP0391384
|
4-[2-[(2R)-2-[(E,3S)-3-hydroxy-4-(3-methylphenyl)but-1-enyl]-5-sulfanylidenepyrrolidin-1-yl]ethylsulfanyl]butanoic acid
Show/Hide
|
C21H29NO3S2
|
1
|
| 1 |
EC50 = 7.7 nM
|
|
|
|
CP0410241
|
2-[2-[(2R)-2-[(E,3S)-4-[3-(5,7-dimethyl-1,3-benzoxazol-2-yl)phenyl]-3-hydroxybut-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C29H29N3O5S2
|
1
|
| 1 |
EC50 = 7.7 nM
|
|
|
|
CP0410233
|
2-[2-[(2R)-2-[(E,3S)-3-hydroxy-4-(3-phenylphenyl)but-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C26H26N2O4S2
|
1
|
| 1 |
EC50 = 8 nM
|
|
|
|
CP0410240
|
2-[2-[(2R)-2-[(E,3S)-3-hydroxy-4-[3-(5-methyl-1,3-benzoxazol-2-yl)phenyl]but-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C28H27N3O5S2
|
1
|
| 1 |
EC50 = 8.8 nM
|
|
|
|
CP0391383
|
7-[(2R)-2-[(E,3S)-4-(3-ethylphenyl)-3-hydroxybut-1-enyl]-5-sulfanylidenepyrrolidin-1-yl]heptanoic acid
Show/Hide
|
C23H33NO3S
|
1
|
| 1 |
EC50 = 9.4 nM
|
|
|
|
CP0410235
|
2-[2-[(2R)-2-[(E,3S)-4-[3-(5-chloro-1,3-benzothiazol-2-yl)phenyl]-3-hydroxybut-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C27H24ClN3O4S3
|
1
|
| 1 |
EC50 = 9.7 nM
|
|
|
|
CP0400838
|
7-[(2R)-2-[(E,3S)-3-hydroxy-4-[3-(trifluoromethyl)phenyl]but-1-enyl]-5-sulfanylidenepyrrolidin-1-yl]heptanoic acid
Show/Hide
|
C22H28F3NO3S
|
1
|
| 1 |
EC50 = 10 nM
|
|
|
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CP0395231
|
4-[2-[(4S)-4-[(E,3S)-3-hydroxy-4-[3-(trifluoromethyl)phenyl]but-1-enyl]-2-oxo-1,3-oxazolidin-3-yl]ethylsulfanyl]butanoic acid
Show/Hide
|
C20H24F3NO5S
|
1
|
| 1 |
EC50 = 12 nM
|
|
|
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CP0410237
|
2-[2-[(2R)-2-[(E,3S)-4-[3-(1,3-benzothiazol-2-yl)phenyl]-3-hydroxybut-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C27H25N3O4S3
|
1
|
| 1 |
EC50 = 13 nM
|
|
|
|
CP0432929
|
4-[2-[(2R)-2-[(E,3S)-4-[3-(1,3-benzoxazol-2-yl)phenyl]-3-hydroxybut-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]butanoic acid
Show/Hide
|
C27H30N2O5S
|
1
|
| 1 |
EC50 = 13 nM
|
|
|
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CP0403544
|
7-[(2R)-2-[(E,3S)-3-hydroxy-4-[3-(methoxymethyl)phenyl]but-1-enyl]-5-oxopyrrolidin-1-yl]heptanoic acid
Show/Hide
|
C23H33NO5
|
1
|
| 1 |
EC50 = 15 nM
|
|
|
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CP0378130
|
2-[2-[(2R)-2-[(E,3S)-3-hydroxy-4-[3-(4-methylphenyl)phenyl]but-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C27H28N2O4S2
|
1
|
| 1 |
EC50 = 15 nM
|
|
|
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CP0410234
|
2-[2-[(2R)-2-[(E,3S)-3-hydroxy-4-[3-(4-methoxyphenyl)phenyl]but-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C27H28N2O5S2
|
1
|
| 1 |
EC50 = 15 nM
|
|
|
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CP0400837
|
4-[2-[(4S)-4-[(E,3S)-4-(3-ethylphenyl)-3-hydroxybut-1-enyl]-2-oxo-1,3-oxazolidin-3-yl]ethylsulfanyl]butanoic acid
Show/Hide
|
C21H29NO5S
|
1
|
| 1 |
EC50 = 18 nM
|
|
|
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CP0423860
|
4-[2-[(2R)-2-[(E,3S)-3-hydroxy-4-[3-(pyridin-3-ylmethoxy)phenyl]but-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]butanoic acid
Show/Hide
|
C26H32N2O5S
|
1
|
| 1 |
EC50 = 19 nM
|
|
|
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CP0410239
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2-[2-[(2R)-2-[(E,3S)-4-[3-(3,4-dimethylphenyl)phenyl]-3-hydroxybut-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C28H30N2O4S2
|
1
|
| 1 |
EC50 = 21 nM
|
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CP0388030
|
4-[2-[(4S)-4-[(E,3S)-4-(3-chlorophenyl)-3-hydroxybut-1-enyl]-2-oxo-1,3-oxazolidin-3-yl]ethylsulfanyl]butanoic acid
Show/Hide
|
C19H24ClNO5S
|
1
|
| 1 |
EC50 = 23 nM
|
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CP0401106
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4-[2-[(4S)-4-[(E,3S)-3-hydroxy-4-[3-(methoxymethyl)phenyl]but-1-enyl]-2-oxo-1,3-oxazolidin-3-yl]ethylsulfanyl]butanoic acid
Show/Hide
|
C21H29NO6S
|
1
|
| 1 |
EC50 = 24 nM
|
|
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CP0388031
|
7-[(2R)-2-[(E,3S)-4-(3-fluorophenyl)-3-hydroxybut-1-enyl]-5-sulfanylidenepyrrolidin-1-yl]heptanoic acid
Show/Hide
|
C21H28FNO3S
|
1
|
| 1 |
EC50 = 26 nM
|
|
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CP0392256
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7-[(2R)-2-[(E,3S)-3-hydroxy-4-(3-propylphenyl)but-1-enyl]-5-sulfanylidenepyrrolidin-1-yl]heptanoic acid
Show/Hide
|
C24H35NO3S
|
1
|
| 1 |
EC50 = 27 nM
|
|
|
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CP0410236
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2-[2-[(2R)-2-[(E,3S)-4-[3-(4-chlorophenyl)phenyl]-3-hydroxybut-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C26H25ClN2O4S2
|
1
|
| 1 |
EC50 = 27 nM
|
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CP0410238
|
4-[2-[(2R)-2-[(E,3S)-4-[3-(1,3-dihydroisoindol-2-yl)phenyl]-3-hydroxybut-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]butanoic acid
Show/Hide
|
C28H34N2O4S
|
1
|
| 1 |
EC50 = 28 nM
|
|
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CP0410310
|
2-[2-[(2R)-2-[(E,3S)-3-hydroxy-4-[3-(4-methyl-1,3-benzoxazol-2-yl)phenyl]but-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C28H27N3O5S2
|
1
|
| 1 |
EC50 = 28 nM
|
|
|
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CP0388034
|
7-[(2R)-2-[(E,3S)-3-hydroxy-4-phenylbut-1-enyl]-5-sulfanylidenepyrrolidin-1-yl]heptanoic acid
Show/Hide
|
C21H29NO3S
|
1
|
| 1 |
EC50 = 29 nM
|
|
|
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CP0427503
|
4-[2-[(4S)-4-[(E,3S)-3-hydroxy-4-(3-methylphenyl)but-1-enyl]-2-oxo-1,3-oxazolidin-3-yl]ethylsulfanyl]butanoic acid
Show/Hide
|
C20H27NO5S
|
1
|
| 1 |
EC50 = 33 nM
|
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CP0401105
|
4-[2-[(4S)-4-[(E,3S)-4-(3-fluorophenyl)-3-hydroxybut-1-enyl]-2-oxo-1,3-oxazolidin-3-yl]ethylsulfanyl]butanoic acid
Show/Hide
|
C19H24FNO5S
|
1
|
| 1 |
EC50 = 35 nM
|
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CP0403545
|
4-[2-[(4S)-4-[(E,3S)-3-hydroxy-4-phenylbut-1-enyl]-2-oxo-1,3-oxazolidin-3-yl]ethylsulfanyl]butanoic acid
Show/Hide
|
C19H25NO5S
|
1
|
| 1 |
EC50 = 36 nM
|
|
|
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CP0410232
|
4-[2-[(2R)-2-[(E,3S)-3-hydroxy-4-[3-(pyridin-4-ylmethoxy)phenyl]but-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]butanoic acid
Show/Hide
|
C26H32N2O5S
|
1
|
| 1 |
EC50 = 46 nM
|
|
|
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CP0423862
|
4-[2-[(2R)-2-[(E,3S)-3-hydroxy-4-(3-phenylphenyl)but-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]butanoic acid
Show/Hide
|
C26H31NO4S
|
1
|
| 1 |
EC50 = 52 nM
|
|
|
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CP0416072
|
4-[2-[(2R)-2-[(E,3S)-3-hydroxy-4-[3-(1H-indol-5-yl)phenyl]but-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]butanoic acid
Show/Hide
|
C28H32N2O4S
|
1
|
| 1 |
EC50 = 85 nM
|
|
|
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CP0378146
|
4-[2-[(2R)-2-[(E,3S)-3-hydroxy-4-(3-pyridin-2-ylphenyl)but-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]butanoic acid
Show/Hide
|
C25H30N2O4S
|
1
|
| 1 |
EC50 = 86 nM
|
|
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CP0388029
|
4-[2-[(4S)-4-[(E,3S)-3-hydroxy-4-(3-propylphenyl)but-1-enyl]-2-oxo-1,3-oxazolidin-3-yl]ethylsulfanyl]butanoic acid
Show/Hide
|
C22H31NO5S
|
1
|
| 1 |
EC50 = 93 nM
|
|
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CP0423859
|
4-[2-[(2R)-2-[(E,3S)-3-hydroxy-4-(3-naphthalen-2-ylphenyl)but-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]butanoic acid
Show/Hide
|
C30H33NO4S
|
1
|
| 1 |
EC50 = 96 nM
|
|
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CP0400840
|
4-[2-[(4S)-4-[(E,3S)-3-hydroxy-4-[3-(trifluoromethoxy)phenyl]but-1-enyl]-2-oxo-1,3-oxazolidin-3-yl]ethylsulfanyl]butanoic acid
Show/Hide
|
C20H24F3NO6S
|
1
|
| 1 |
EC50 = 160 nM
|
|
|
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CP0410313
|
2-[2-[(2R)-2-[(E,3S)-4-[3-(2,4-dimethylphenyl)phenyl]-3-hydroxybut-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C28H30N2O4S2
|
1
|
| 1 |
EC50 = 160 nM
|
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CP0463502
|
4-[2-[(4S)-4-[(E,3S)-3-hydroxy-4-(3-phenylphenyl)but-1-enyl]-2-oxo-1,3-oxazolidin-3-yl]ethylsulfanyl]butanoic acid
Show/Hide
|
C25H29NO5S
|
1
|
| 1 |
EC50 = 450 nM
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CP0387597
|
2-[2-[(2R)-2-[(E,3S)-3-hydroxy-4-(3-naphthalen-2-ylphenyl)but-1-enyl]-5-oxopyrrolidin-1-yl]ethylsulfanyl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C30H28N2O4S2
|
1
|
| 1 |
EC50 = 480 nM
|
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|
