| Compound ID |
Compound Name |
Compound Formula |
|
CP0531310
|
US9428456, 1.224
Show/Hide
|
C24H28ClFN4O2
|
1
|
| 1 |
EC50 = 0.4 nM
|
|
|
|
CP0572248
|
US9428456, 1.217
Show/Hide
|
C25H30ClN3O2
|
1
|
| 1 |
EC50 = 0.4 nM
|
|
|
|
CP0554776
|
US9428456, 1.223
Show/Hide
|
C24H30FN3O2
|
1
|
| 1 |
EC50 = 0.5 nM
|
|
|
|
CP0561184
|
US9428456, 1.229
Show/Hide
|
C24H29F3N4O2
|
1
|
| 1 |
EC50 = 0.5 nM
|
|
|
|
CP0483904
|
US9428456, 1.210
Show/Hide
|
C25H29F3N4O2
|
1
|
| 1 |
EC50 = 0.6 nM
|
|
|
|
CP0483906
|
US9428456, 1.227
Show/Hide
|
C24H28Cl2N4O2
|
1
|
| 1 |
EC50 = 0.6 nM
|
|
|
|
CP0515162
|
US9428456, 4.020
Show/Hide
|
C23H29FN4O2
|
1
|
| 1 |
EC50 = 0.6 nM
|
|
|
|
CP0531308
|
US9428456, 1.208
Show/Hide
|
C25H29F3N4O2
|
1
|
| 1 |
EC50 = 0.6 nM
|
|
|
|
CP0576503
|
US9428456, 1.339
Show/Hide
|
C23H29ClN4O2
|
1
|
| 1 |
EC50 = 0.6 nM
|
|
|
|
CP0483899
|
US9428456, 1.340
Show/Hide
|
C23H28ClFN4O2
|
1
|
| 1 |
EC50 = 0.7 nM
|
|
|
|
CP0483908
|
US9428456, 2.003
Show/Hide
|
C23H28ClN3O2
|
1
|
| 1 |
EC50 = 0.8 nM
|
|
|
|
CP0512939
|
US9428456, 1.207
Show/Hide
|
C24H29FN4O2
|
1
|
| 1 |
EC50 = 0.8 nM
|
|
|
|
CP0531328
|
US9428456, 1.225
Show/Hide
|
C25H28ClF3N4O2
|
1
|
| 1 |
EC50 = 0.8 nM
|
|
|
|
CP0574004
|
US9428456, 1.057
Show/Hide
|
C25H31FN4O2
|
1
|
| 1 |
EC50 = 0.8 nM
|
|
|
|
CP0576500
|
US9428456, 1.338
Show/Hide
|
C24H31ClN4O2
|
1
|
| 1 |
EC50 = 0.8 nM
|
|
|
|
CP0515747
|
US9428456, 1.206
Show/Hide
|
C25H30FN3O2
|
1
|
| 1 |
EC50 = 0.9 nM
|
|
|
|
CP0539536
|
US9428456, 2.001
Show/Hide
|
C25H30ClN3O2
|
1
|
| 1 |
EC50 = 0.9 nM
|
|
|
|
CP0544301
|
US9428456, 1.235
Show/Hide
|
C27H32N4O2
|
1
|
| 1 |
EC50 = 0.9 nM
|
|
|
|
CP0554102
|
US9428456, 1.219
Show/Hide
|
C25H29ClFN3O2
|
1
|
| 1 |
EC50 = 0.9 nM
|
|
|
|
CP0557226
|
US9428456, 1.344
Show/Hide
|
C23H29BrN4O2
|
1
|
| 1 |
EC50 = 0.9 nM
|
|
|
|
CP0572240
|
US9428456, 1.081
Show/Hide
|
C26H34N4O2
|
1
|
| 1 |
EC50 = 0.9 nM
|
|
|
|
CP0578092
|
US9428456, 1.260
Show/Hide
|
C25H39N3O2
|
1
|
| 1 |
EC50 = 0.9 nM
|
|
|
|
CP0402526
|
US9428456, 1.085
Show/Hide
|
C25H31BrN4O2
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0402528
|
US9428456, 1.209
Show/Hide
|
C24H29ClN4O2
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0466187
|
US9428456, 1.271
Show/Hide
|
C26H33N3O2
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0472283
|
US9428456, 1.341
Show/Hide
|
C25H31F3N4O2
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0472284
|
US9428456, 1.094
Show/Hide
|
C25H31ClN4O2
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0478603
|
US9428456, 1.295
Show/Hide
|
C25H31F3N4O2
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0512918
|
US9428456, 1.078
Show/Hide
|
C25H31ClN4O2
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0516919
|
US9428456, 2.009
Show/Hide
|
C24H30ClN3O2
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0518668
|
US9428456, 1.345
Show/Hide
|
C24H29F3N4O3
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0530647
|
US9428456, 2.004
Show/Hide
|
C24H30ClN3O2
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0531305
|
US9428456, 1.311
Show/Hide
|
C27H37N3O2
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0539504
|
US9428456, 2.007
Show/Hide
|
C24H28ClN3O2
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0539541
|
US9428456, 2.094
Show/Hide
|
C23H27F3N4O2
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0554103
|
US9428456, 1.220
Show/Hide
|
C25H28ClF3N4O2
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0554403
|
US9428456, 4.006
Show/Hide
|
C24H29FN4O3
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0554410
|
US9428456, 1.258
Show/Hide
|
C25H32ClN3O2
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0555973
|
US9428456, 1.309
Show/Hide
|
C27H35N3O2
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0559168
|
US9428456, 1.245
Show/Hide
|
C25H31Cl2N3O2
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0561183
|
US9428456, 1.228
Show/Hide
|
C24H29F3N4O2
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0561910
|
US9428456, 1.230
Show/Hide
|
C24H29F3N4O2
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0563163
|
US9428456, 1.300
Show/Hide
|
C25H32FN3O2
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0563165
|
US9428456, 1.346
Show/Hide
|
C25H31F3N4O3
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0566414
|
US9428456, 1.221
Show/Hide
|
C28H31ClN4O2
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0572262
|
US9428456, 1.269
Show/Hide
|
C27H36ClN3O2
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0574002
|
US9428456, 1.039
Show/Hide
|
C25H32N4O2
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0574007
|
US9428456, 1.061
Show/Hide
|
C26H34N4O2
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0574109
|
US9428456, 1.343
Show/Hide
|
C24H30ClFN4O2
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0576975
|
US9428456, 1.002
Show/Hide
|
C26H31F3N4O2
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0413225
|
US9428456, 1.031
Show/Hide
|
C27H35N3O3
|
1
|
| 1 |
EC50 = 2 nM
|
|
|
|
CP0451614
|
US9428456, 1.154
Show/Hide
|
C27H36N4O2
|
1
|
| 1 |
EC50 = 2 nM
|
|
|
|
CP0483894
|
US9428456, 1.310
Show/Hide
|
C27H34ClN3O2
|
1
|
| 1 |
EC50 = 2 nM
|
|
|
|
CP0483895
|
US9428456, 2.095
Show/Hide
|
C24H29F3N4O2
|
1
|
| 1 |
EC50 = 2 nM
|
|
|
|
CP0483905
|
US9428456, 1.215
Show/Hide
|
C24H29FN4O2
|
1
|
| 1 |
EC50 = 2 nM
|
|
|
|
CP0483909
|
US9428456, 2.006
Show/Hide
|
C23H26ClN3O2
|
1
|
| 1 |
EC50 = 2 nM
|
|
|
|
CP0483925
|
US9428456, 1.129
Show/Hide
|
C26H31F2N3O2
|
1
|
| 1 |
EC50 = 2 nM
|
|
|
|
CP0486853
|
US9428456, 1.273
Show/Hide
|
C25H32FN3O2
|
1
|
| 1 |
EC50 = 2 nM
|
|
|
|
CP0495296
|
US9428456, 4.025
Show/Hide
|
C24H31ClN4O3
|
1
|
| 1 |
EC50 = 2 nM
|
|
|
|
CP0507480
|
US9428456, 1.001
Show/Hide
|
C26H32ClN3O2
|
1
|
| 1 |
EC50 = 2 nM
|
|
|
|
CP0512947
|
US9428456, 2.071
Show/Hide
|
C24H29F3N4O2
|
1
|
| 1 |
EC50 = 2 nM
|
|
|
|
CP0512948
|
US9428456, 1.326
Show/Hide
|
C26H33F3N4O2
|
1
|
| 1 |
EC50 = 2 nM
|
|
|
|
CP0512952
|
US9428456, 1.301
Show/Hide
|
C25H31F3N4O2
|
1
|
| 1 |
EC50 = 2 nM
|
|
|
|
CP0515159
|
US9428456, 1.233
Show/Hide
|
C27H32N4O2
|
1
|
| 1 |
EC50 = 2 nM
|
|
|
|
CP0516305
|
US9428456, 1.234
Show/Hide
|
C26H31N5O2
|
1
|
| 1 |
EC50 = 2 nM
|
|
|
|
CP0516309
|
US9428456, 1.254
Show/Hide
|
C25H30ClF2N3O2
|
1
|
| 1 |
EC50 = 2 nM
|
|
|
|
CP0531311
|
US9428456, 2.014
Show/Hide
|
C26H30ClF2N3O2
|
1
|
| 1 |
EC50 = 2 nM
|
|
|
|
CP0537198
|
US9428456, 1.218
Show/Hide
|
C25H28ClF3N4O2
|
1
|
| 1 |
EC50 = 2 nM
|
|
|
|
CP0539497
|
US9428456, 1.272
Show/Hide
|
C28H37N3O2
|
1
|
| 1 |
EC50 = 2 nM
|
|
|
|
CP0539844
|
US9428456, 1.019
Show/Hide
|
C26H31F2N3O2
|
1
|
| 1 |
EC50 = 2 nM
|
|
|
|
CP0544303
|
US9428456, 1.248
Show/Hide
|
C25H31ClFN3O2
|
1
|
| 1 |
EC50 = 2 nM
|
|
|
|
CP0544396
|
US9428456, 1.249
Show/Hide
|
C26H31ClF3N3O2
|
1
|
| 1 |
EC50 = 2 nM
|
|
|
|
CP0544403
|
US9428456, 1.212
Show/Hide
|
C25H29F3N4O2
|
1
|
| 1 |
EC50 = 2 nM
|
|
|
|
CP0547472
|
US9428456, 1.267
Show/Hide
|
C27H35N3O2
|
1
|
| 1 |
EC50 = 2 nM
|
|
|
|
CP0552288
|
US9428456, 1.268
Show/Hide
|
C27H33Cl2N3O2
|
1
|
| 1 |
EC50 = 2 nM
|
|
|
|
CP0552302
|
US9428456, 1.205
Show/Hide
|
C22H25FN4O2
|
1
|
| 1 |
EC50 = 2 nM
|
|
|
|
CP0554094
|
US9428456, 1.141
Show/Hide
|
C24H31N5O2
|
1
|
| 1 |
EC50 = 2 nM
|
|
|
|
CP0554098
|
US9428456, 1.157
Show/Hide
|
C24H30ClN5O2
|
1
|
| 1 |
EC50 = 2 nM
|
|
|
|
CP0554111
|
US9428456, 1.006
Show/Hide
|
C24H31N5O2
|
1
|
| 1 |
EC50 = 2 nM
|
|
|
|
CP0555928
|
US9428456, 4.021
Show/Hide
|
C24H31FN4O3
|
1
|
| 1 |
EC50 = 2 nM
|
|
|
|
CP0556711
|
US9428456, 1.168
Show/Hide
|
C26H33ClN4O2
|
1
|
| 1 |
EC50 = 2 nM
|
|
|
|
CP0557234
|
US9428456, 1.261
Show/Hide
|
C24H34N4O2S
|
1
|
| 1 |
EC50 = 2 nM
|
|
|
|
CP0561185
|
US9428456, 1.247
Show/Hide
|
C25H31ClFN3O2
|
1
|
| 1 |
EC50 = 2 nM
|
|
|
|
CP0563248
|
US9428456, 1.142
Show/Hide
|
C25H33N5O2
|
1
|
| 1 |
EC50 = 2 nM
|
|
|
|
CP0564202
|
US9428456, 4.017
Show/Hide
|
C24H28F4N4O2
|
1
|
| 1 |
EC50 = 2 nM
|
|
|
|
CP0566252
|
US9428456, 1.033
Show/Hide
|
C26H32ClN3O2
|
1
|
| 1 |
EC50 = 2 nM
|
|
|
|
CP0572249
|
US9428456, 1.226
Show/Hide
|
C25H31ClN4O2
|
1
|
| 1 |
EC50 = 2 nM
|
|
|
|
CP0572258
|
US9428456, 1.156
Show/Hide
|
C26H32FN3O2
|
1
|
| 1 |
EC50 = 2 nM
|
|
|
|
CP0574111
|
US9428456, 1.067
Show/Hide
|
C25H31ClN4O2
|
1
|
| 1 |
EC50 = 2 nM
|
|
|
|
CP0413227
|
US9428456, 1.275
Show/Hide
|
C25H31F3N4O2
|
1
|
| 1 |
EC50 = 3 nM
|
|
|
|
CP0423964
|
US9428456, 1.100
Show/Hide
|
C27H35N3O2
|
1
|
| 1 |
EC50 = 3 nM
|
|
|
|
CP0472289
|
US9428456, 2.031
Show/Hide
|
C22H23ClF3N3O2
|
1
|
| 1 |
EC50 = 3 nM
|
|
|
|
CP0483907
|
US9428456, 2.002
Show/Hide
|
C21H24ClN3O2
|
1
|
| 1 |
EC50 = 3 nM
|
|
|
|
CP0486749
|
US9428456, 1.222
Show/Hide
|
C28H31ClN4O2
|
1
|
| 1 |
EC50 = 3 nM
|
|
|
|
CP0495278
|
US9428456, 1.355
Show/Hide
|
C24H29N5O2S
|
1
|
| 1 |
EC50 = 3 nM
|
|
|
|
CP0495292
|
US9428456, 2.059
Show/Hide
|
C25H34N4O2
|
1
|
| 1 |
EC50 = 3 nM
|
|
|
|
CP0515681
|
US9428456, 1.211
Show/Hide
|
C28H32N4O2
|
1
|
| 1 |
EC50 = 3 nM
|
|
|
|
CP0515746
|
US9428456, 1.199
Show/Hide
|
C23H26FN3O2
|
1
|
| 1 |
EC50 = 3 nM
|
|
|
|
CP0518671
|
US9428456, 1.092
Show/Hide
|
C26H34N4O3
|
1
|
| 1 |
EC50 = 3 nM
|
|
|
|
CP0531304
|
US9428456, 1.303
Show/Hide
|
C25H32FN3O2
|
1
|
| 1 |
EC50 = 3 nM
|
|
|
|
CP0531309
|
US9428456, 1.213
Show/Hide
|
C28H32N4O2
|
1
|
| 1 |
EC50 = 3 nM
|
|
|
|
CP0537319
|
US9428456, 1.232
Show/Hide
|
C26H31N5O2
|
1
|
| 1 |
EC50 = 3 nM
|
|
|
|
CP0537320
|
US9428456, 1.240
Show/Hide
|
C26H34N4O2
|
1
|
| 1 |
EC50 = 3 nM
|
|
|
|
CP0539539
|
US9428456, 2.092
Show/Hide
|
C24H29F3N4O3
|
1
|
| 1 |
EC50 = 3 nM
|
|
|
|
CP0539852
|
US9428456, 1.079
Show/Hide
|
C26H35N3O2
|
1
|
| 1 |
EC50 = 3 nM
|
|
|
|
CP0544302
|
US9428456, 1.246
Show/Hide
|
C25H31Cl2N3O2
|
1
|
| 1 |
EC50 = 3 nM
|
|
|
|
CP0544397
|
US9428456, 1.250
Show/Hide
|
C26H30Cl2F3N3O2
|
1
|
| 1 |
EC50 = 3 nM
|
|
|
|
CP0548103
|
US9428456, 3.008
Show/Hide
|
C22H28FN3O2S
|
1
|
| 1 |
EC50 = 3 nM
|
|
|
|
CP0552301
|
US9428456, 1.201
Show/Hide
|
C23H28N4O2
|
1
|
| 1 |
EC50 = 3 nM
|
|
|
|
CP0554091
|
US9428456, 1.025
Show/Hide
|
C27H34ClN3O2
|
1
|
| 1 |
EC50 = 3 nM
|
|
|
|
CP0554411
|
US9428456, 2.039
Show/Hide
|
C24H32N4O2
|
1
|
| 1 |
EC50 = 3 nM
|
|
|
|
CP0554414
|
US9428456, 4.016
Show/Hide
|
C26H30F4N4O2
|
1
|
| 1 |
EC50 = 3 nM
|
|
|
|
CP0555570
|
US9428456, 1.014
Show/Hide
|
C26H33N3O2
|
1
|
| 1 |
EC50 = 3 nM
|
|
|
|
CP0561272
|
US9428456, 4.007
Show/Hide
|
C23H29FN4O3
|
1
|
| 1 |
EC50 = 3 nM
|
|
|
|
CP0563162
|
US9428456, 1.299
Show/Hide
|
C25H34N4O2
|
1
|
| 1 |
EC50 = 3 nM
|
|
|
|
CP0564194
|
US9428456, 1.118
Show/Hide
|
C27H34FN3O2
|
1
|
| 1 |
EC50 = 3 nM
|
|
|
|
CP0566346
|
US9428456, 4.024
Show/Hide
|
C23H29ClN4O3
|
1
|
| 1 |
EC50 = 3 nM
|
|
|
|
CP0566349
|
US9428456, 1.251
Show/Hide
|
C26H30Cl2F3N3O2
|
1
|
| 1 |
EC50 = 3 nM
|
|
|
|
CP0572265
|
US9428456, 1.281
Show/Hide
|
C25H33N3O2S
|
1
|
| 1 |
EC50 = 3 nM
|
|
|
|
CP0577275
|
US9428456, 1.353
Show/Hide
|
C25H30N4O2S
|
1
|
| 1 |
EC50 = 3 nM
|
|
|
|
CP0577353
|
US9428456, 2.083
Show/Hide
|
C27H33F3N4O2
|
1
|
| 1 |
EC50 = 3 nM
|
|
|
|
CP0577886
|
US9428456, 1.077
Show/Hide
|
C25H31ClN4O2
|
1
|
| 1 |
EC50 = 3 nM
|
|
|
|
CP0423965
|
US9428456, 1.111
Show/Hide
|
C28H37N3O2
|
1
|
| 1 |
EC50 = 4 nM
|
|
|
|
CP0423966
|
US9428456, 1.238
Show/Hide
|
C25H30F3N3O2
|
1
|
| 1 |
EC50 = 4 nM
|
|
|
|
CP0426351
|
US9428456, 1.237
Show/Hide
|
C25H30F3N3O2
|
1
|
| 1 |
EC50 = 4 nM
|
|
|
|
CP0483901
|
US9428456, 1.082
Show/Hide
|
C26H34N4O2
|
1
|
| 1 |
EC50 = 4 nM
|
|
|
|
CP0483913
|
US9428456, 3.009
Show/Hide
|
C22H28FN3O2S
|
1
|
| 1 |
EC50 = 4 nM
|
|
|
|
CP0483922
|
US9428456, 1.012
Show/Hide
|
C24H31N3O2S
|
1
|
| 1 |
EC50 = 4 nM
|
|
|
|
CP0495277
|
US9428456, 4.005
Show/Hide
|
C25H31FN4O3
|
1
|
| 1 |
EC50 = 4 nM
|
|
|
|
CP0495279
|
US9428456, 2.102
Show/Hide
|
C25H31F3N4O2
|
1
|
| 1 |
EC50 = 4 nM
|
|
|
|
CP0495284
|
US9428456, 1.253
Show/Hide
|
C25H30Cl2FN3O2
|
1
|
| 1 |
EC50 = 4 nM
|
|
|
|
CP0495285
|
US9428456, 1.259
Show/Hide
|
C25H33N3O2
|
1
|
| 1 |
EC50 = 4 nM
|
|
|
|
CP0512953
|
US9428456, 1.306
Show/Hide
|
C25H32FN3O3
|
1
|
| 1 |
EC50 = 4 nM
|
|
|
|
CP0515161
|
US9428456, 1.252
Show/Hide
|
C25H30Cl2FN3O2
|
1
|
| 1 |
EC50 = 4 nM
|
|
|
|
CP0516937
|
US9428456, 2.010
Show/Hide
|
C26H32ClN3O2
|
1
|
| 1 |
EC50 = 4 nM
|
|
|
|
CP0537317
|
US9428456, 1.123
Show/Hide
|
C27H34FN3O3
|
1
|
| 1 |
EC50 = 4 nM
|
|
|
|
CP0539552
|
US9428456, 1.023
Show/Hide
|
C27H35N3O3
|
1
|
| 1 |
EC50 = 4 nM
|
|
|
|
CP0544306
|
US9428456, 8.001
Show/Hide
|
C23H31N5O2
|
1
|
| 1 |
EC50 = 4 nM
|
|
|
|
CP0548078
|
US9428456, 1.117
Show/Hide
|
C27H34FN3O2
|
1
|
| 1 |
EC50 = 4 nM
|
|
|
|
CP0548085
|
US9428456, 1.322
Show/Hide
|
C22H29N5O2
|
1
|
| 1 |
EC50 = 4 nM
|
|
|
|
CP0554059
|
US9428456, 2.068
Show/Hide
|
C21H23F3N4O2
|
1
|
| 1 |
EC50 = 4 nM
|
|
|
|
CP0554405
|
US9428456, 1.101
Show/Hide
|
C27H35N3O2
|
1
|
| 1 |
EC50 = 4 nM
|
|
|
|
CP0555970
|
US9428456, 1.304
Show/Hide
|
C25H31F3N4O3
|
1
|
| 1 |
EC50 = 4 nM
|
|
|
|
CP0561151
|
US9428456, 1.035
Show/Hide
|
C28H37N3O3
|
1
|
| 1 |
EC50 = 4 nM
|
|
|
|
CP0563247
|
US9428456, 1.131
Show/Hide
|
C26H31ClFN3O2
|
1
|
| 1 |
EC50 = 4 nM
|
|
|
|
CP0565142
|
US9428456, 2.069
Show/Hide
|
C22H25F3N4O2
|
1
|
| 1 |
EC50 = 4 nM
|
|
|
|
CP0566345
|
US9428456, 2.104
Show/Hide
|
C27H36N4O2
|
1
|
| 1 |
EC50 = 4 nM
|
|
|
|
CP0577278
|
US9428456, 1.241
Show/Hide
|
C25H34N4O2
|
1
|
| 1 |
EC50 = 4 nM
|
|
|
|
CP0577348
|
US9428456, 1.028
Show/Hide
|
C28H33N3O3
|
1
|
| 1 |
EC50 = 4 nM
|
|
|
|
CP0577716
|
US9428456, 1.102
Show/Hide
|
C26H32FN3O2
|
1
|
| 1 |
EC50 = 4 nM
|
|
|
|
CP0472290
|
US9428456, 2.032
Show/Hide
|
C26H32ClN3O3
|
1
|
| 1 |
EC50 = 5 nM
|
|
|
|
CP0472294
|
US9428456, 1.018
Show/Hide
|
C27H39N3O2
|
1
|
| 1 |
EC50 = 5 nM
|
|
|
|
CP0472295
|
US9428456, 1.143
Show/Hide
|
C28H34ClN3O3
|
1
|
| 1 |
EC50 = 5 nM
|
|
|
|
CP0472296
|
US9428456, 1.147
Show/Hide
|
C28H36N4O2
|
1
|
| 1 |
EC50 = 5 nM
|
|
|
|
CP0507484
|
US9428456, 1.029
Show/Hide
|
C29H37N3O2
|
1
|
| 1 |
EC50 = 5 nM
|
|
|
|
CP0515757
|
US9428456, 1.140
Show/Hide
|
C26H31Cl2N3O2
|
1
|
| 1 |
EC50 = 5 nM
|
|
|
|
CP0516306
|
US9428456, 1.244
Show/Hide
|
C25H31Cl2N3O2
|
1
|
| 1 |
EC50 = 5 nM
|
|
|
|
CP0537316
|
US9428456, 1.115
Show/Hide
|
C27H34FN3O2
|
1
|
| 1 |
EC50 = 5 nM
|
|
|
|
CP0544295
|
US9428456, 1.097
Show/Hide
|
C28H37N3O2
|
1
|
| 1 |
EC50 = 5 nM
|
|
|
|
CP0548080
|
US9428456, 1.128
Show/Hide
|
C26H31F2N3O2
|
1
|
| 1 |
EC50 = 5 nM
|
|
|
|
CP0552303
|
US9428456, 2.005
Show/Hide
|
C23H28ClN3O3
|
1
|
| 1 |
EC50 = 5 nM
|
|
|
|
CP0554407
|
US9428456, 1.121
Show/Hide
|
C27H34ClN3O2
|
1
|
| 1 |
EC50 = 5 nM
|
|
|
|
CP0554408
|
US9428456, 1.124
Show/Hide
|
C27H34FN3O3
|
1
|
| 1 |
EC50 = 5 nM
|
|
|
|
CP0559167
|
US9428456, 1.236
Show/Hide
|
C27H31ClN4O2
|
1
|
| 1 |
EC50 = 5 nM
|
|
|
|
CP0561147
|
US9428456, 2.081
Show/Hide
|
C25H31F3N4O2
|
1
|
| 1 |
EC50 = 5 nM
|
|
|
|
CP0565138
|
US9428456, 1.148
Show/Hide
|
C28H36FN3O2
|
1
|
| 1 |
EC50 = 5 nM
|
|
|
|
CP0566319
|
US9428456, 1.105
Show/Hide
|
C27H32F3N3O2
|
1
|
| 1 |
EC50 = 5 nM
|
|
|
|
CP0572243
|
US9428456, 1.095
Show/Hide
|
C27H32F3N3O3
|
1
|
| 1 |
EC50 = 5 nM
|
|
|
|
CP0572260
|
US9428456, 1.160
Show/Hide
|
C26H31Cl2N3O2
|
1
|
| 1 |
EC50 = 5 nM
|
|
|
|
CP0574005
|
US9428456, 1.058
Show/Hide
|
C26H31F3N4O2
|
1
|
| 1 |
EC50 = 5 nM
|
|
|
|
CP0576498
|
US9428456, 1.282
Show/Hide
|
C24H30ClN3O2S
|
1
|
| 1 |
EC50 = 5 nM
|
|
|
|
CP0577276
|
US9428456, 1.104
Show/Hide
|
C27H32F3N3O2
|
1
|
| 1 |
EC50 = 5 nM
|
|
|
|
CP0578214
|
US9428456, 1.046
Show/Hide
|
C24H32N4O2
|
1
|
| 1 |
EC50 = 5 nM
|
|
|
|
CP0402527
|
US9428456, 1.090
Show/Hide
|
C25H30Cl2N4O2
|
1
|
| 1 |
EC50 = 6 nM
|
|
|
|
CP0413222
|
US9428456, 1.007
Show/Hide
|
C30H35N3O2
|
1
|
| 1 |
EC50 = 6 nM
|
|
|
|
CP0413226
|
US9428456, 1.138
Show/Hide
|
C26H31Cl2N3O2
|
1
|
| 1 |
EC50 = 6 nM
|
|
|
|
CP0478604
|
US9428456, 1.296
Show/Hide
|
C25H31F3N4O3
|
1
|
| 1 |
EC50 = 6 nM
|
|
|
|
CP0486852
|
US9428456, 1.270
Show/Hide
|
C25H32ClN3O3
|
1
|
| 1 |
EC50 = 6 nM
|
|
|
|
CP0495283
|
US9428456, 1.119
Show/Hide
|
C27H34FN3O2
|
1
|
| 1 |
EC50 = 6 nM
|
|
|
|
CP0512955
|
US9428456, 2.093
Show/Hide
|
C24H29F3N4O3
|
1
|
| 1 |
EC50 = 6 nM
|
|
|
|
CP0516312
|
US9428456, 2.046
Show/Hide
|
C25H32N4O2
|
1
|
| 1 |
EC50 = 6 nM
|
|
|
|
CP0531303
|
US9428456, 1.302
Show/Hide
|
C25H34N4O2
|
1
|
| 1 |
EC50 = 6 nM
|
|
|
|
CP0539535
|
US9428456, 1.321
Show/Hide
|
C25H32FN3O3
|
1
|
| 1 |
EC50 = 6 nM
|
|
|
|
CP0548087
|
US9428456, 2.087
Show/Hide
|
C25H31F3N4O2
|
1
|
| 1 |
EC50 = 6 nM
|
|
|
|
CP0548088
|
US9428456, 2.091
Show/Hide
|
C24H29F3N4O3
|
1
|
| 1 |
EC50 = 6 nM
|
|
|
|
CP0554409
|
US9428456, 1.242
Show/Hide
|
C24H29F3N4O2
|
1
|
| 1 |
EC50 = 6 nM
|
|
|
|
CP0561182
|
US9428456, 1.116
Show/Hide
|
C27H34FN3O2
|
1
|
| 1 |
EC50 = 6 nM
|
|
|
|
CP0561270
|
US9428456, 2.056
Show/Hide
|
C24H32N4O2
|
1
|
| 1 |
EC50 = 6 nM
|
|
|
|
CP0572261
|
US9428456, 1.266
Show/Hide
|
C26H33N3O3
|
1
|
| 1 |
EC50 = 6 nM
|
|
|
|
CP0572264
|
US9428456, 1.276
Show/Hide
|
C25H31F3N4O2
|
1
|
| 1 |
EC50 = 6 nM
|
|
|
|
CP0574116
|
US9428456, 2.008
Show/Hide
|
C27H32ClN3O2
|
1
|
| 1 |
EC50 = 6 nM
|
|
|
|
CP0576497
|
US9428456, 1.278
Show/Hide
|
C24H31ClN4O2
|
1
|
| 1 |
EC50 = 6 nM
|
|
|
|
CP0576969
|
US9428456, 2.070
Show/Hide
|
C25H31F3N4O2
|
1
|
| 1 |
EC50 = 6 nM
|
|
|
|
CP0578546
|
US9428456, 1.103
Show/Hide
|
C26H32FN3O2
|
1
|
| 1 |
EC50 = 6 nM
|
|
|
|
CP0472193
|
US9428456, 1.049
Show/Hide
|
C23H30N4O3
|
1
|
| 1 |
EC50 = 7 nM
|
|
|
|
CP0507485
|
US9428456, 1.133
Show/Hide
|
C26H31ClFN3O2
|
1
|
| 1 |
EC50 = 7 nM
|
|
|
|
CP0516918
|
US9428456, 1.216
Show/Hide
|
C25H29F3N4O2
|
1
|
| 1 |
EC50 = 7 nM
|
|
|
|
CP0544398
|
US9428456, 1.068
Show/Hide
|
C26H31F3N4O2
|
1
|
| 1 |
EC50 = 7 nM
|
|
|
|
CP0547467
|
US9428456, 1.011
Show/Hide
|
C27H35N3O2
|
1
|
| 1 |
EC50 = 7 nM
|
|
|
|
CP0555968
|
US9428456, 1.182
Show/Hide
|
C27H36N4O2
|
1
|
| 1 |
EC50 = 7 nM
|
|
|
|
CP0555972
|
US9428456, 1.305
Show/Hide
|
C25H34N4O3
|
1
|
| 1 |
EC50 = 7 nM
|
|
|
|
CP0556165
|
US9428456, 1.056
Show/Hide
|
C25H31FN4O2
|
1
|
| 1 |
EC50 = 7 nM
|
|
|
|
CP0561181
|
US9428456, 1.113
Show/Hide
|
C28H37N3O2
|
1
|
| 1 |
EC50 = 7 nM
|
|
|
|
CP0561241
|
US9428456, 1.187
Show/Hide
|
C27H33F3N4O2
|
1
|
| 1 |
EC50 = 7 nM
|
|
|
|
CP0561267
|
US9428456, 1.257
Show/Hide
|
C23H35N3O2
|
1
|
| 1 |
EC50 = 7 nM
|
|
|
|
CP0572254
|
US9428456, 1.135
Show/Hide
|
C27H31F4N3O2
|
1
|
| 1 |
EC50 = 7 nM
|
|
|
|
CP0576965
|
US9428456, 1.130
Show/Hide
|
C26H31ClFN3O2
|
1
|
| 1 |
EC50 = 7 nM
|
|
|
|
CP0577351
|
US9428456, 2.075
Show/Hide
|
C24H31N3O2S
|
1
|
| 1 |
EC50 = 7 nM
|
|
|
|
CP0495282
|
US9428456, 1.107
Show/Hide
|
C27H32N4O2
|
1
|
| 1 |
EC50 = 8 nM
|
|
|
|
CP0512942
|
US9428456, 1.134
Show/Hide
|
C27H31F4N3O2
|
1
|
| 1 |
EC50 = 8 nM
|
|
|
|
CP0516314
|
US9428456, 4.014
Show/Hide
|
C24H32N4O3
|
1
|
| 1 |
EC50 = 8 nM
|
|
|
|
CP0531306
|
US9428456, 1.312
Show/Hide
|
C26H34ClN3O2
|
1
|
| 1 |
EC50 = 8 nM
|
|
|
|
CP0539498
|
US9428456, 1.337
Show/Hide
|
C26H33N3O2
|
1
|
| 1 |
EC50 = 8 nM
|
|
|
|
CP0539503
|
US9428456, 1.348
Show/Hide
|
C24H29F3N4O3
|
1
|
| 1 |
EC50 = 8 nM
|
|
|
|
CP0548077
|
US9428456, 1.110
Show/Hide
|
C28H37N3O2
|
1
|
| 1 |
EC50 = 8 nM
|
|
|
|
CP0553289
|
US9428456, 1.164
Show/Hide
|
C27H34ClN3O2
|
1
|
| 1 |
EC50 = 8 nM
|
|
|
|
CP0554060
|
US9428456, 1.328
Show/Hide
|
C26H34FN3O2
|
1
|
| 1 |
EC50 = 8 nM
|
|
|
|
CP0554095
|
US9428456, 1.146
Show/Hide
|
C27H33N5O2
|
1
|
| 1 |
EC50 = 8 nM
|
|
|
|
CP0559169
|
US9428456, 2.057
Show/Hide
|
C25H34N4O2
|
1
|
| 1 |
EC50 = 8 nM
|
|
|
|
CP0572289
|
US9428456, 4.019
Show/Hide
|
C24H31FN4O2
|
1
|
| 1 |
EC50 = 8 nM
|
|
|
|
CP0576495
|
US9428456, 1.137
Show/Hide
|
C26H31Cl2N3O2
|
1
|
| 1 |
EC50 = 8 nM
|
|
|
|
CP0577717
|
US9428456, 2.040
Show/Hide
|
C25H34N4O2
|
1
|
| 1 |
EC50 = 8 nM
|
|
|
|
CP0531469
|
US9428456, 4.013
Show/Hide
|
C25H32N4O3
|
1
|
| 1 |
EC50 = 9 nM
|
|
|
|
CP0554061
|
US9428456, 1.043
Show/Hide
|
C27H41N3O2
|
1
|
| 1 |
EC50 = 9 nM
|
|
|
|
CP0554682
|
US9428456, 2.033
Show/Hide
|
C29H30ClN3O2
|
1
|
| 1 |
EC50 = 9 nM
|
|
|
|
CP0572239
|
US9428456, 1.075
Show/Hide
|
C26H33ClN4O3
|
1
|
| 1 |
EC50 = 9 nM
|
|
|
|
CP0572263
|
US9428456, 1.274
Show/Hide
|
C25H31F3N4O2
|
1
|
| 1 |
EC50 = 9 nM
|
|
|
|
CP0451613
|
US9428456, 1.153
Show/Hide
|
C28H32F5N3O2
|
1
|
| 1 |
EC50 = 10 nM
|
|
|
|
CP0495293
|
US9428456, 2.060
Show/Hide
|
C26H34N4O2
|
1
|
| 1 |
EC50 = 10 nM
|
|
|
|
CP0512941
|
US9428456, 1.132
Show/Hide
|
C26H31ClFN3O2
|
1
|
| 1 |
EC50 = 10 nM
|
|
|
|
CP0518675
|
US9428456, 1.151
Show/Hide
|
C26H39N3O2
|
1
|
| 1 |
EC50 = 10 nM
|
|
|
|
CP0518678
|
US9428456, 1.055
Show/Hide
|
C26H34N4O2
|
1
|
| 1 |
EC50 = 10 nM
|
|
|
|
CP0531532
|
US9428456, 4.012
Show/Hide
|
C26H34N4O3
|
1
|
| 1 |
EC50 = 10 nM
|
|
|
|
CP0539538
|
US9428456, 2.086
Show/Hide
|
C25H31F3N4O2
|
1
|
| 1 |
EC50 = 10 nM
|
|
|
|
CP0548079
|
US9428456, 1.125
Show/Hide
|
C28H37N3O4
|
1
|
| 1 |
EC50 = 10 nM
|
|
|
|
CP0561156
|
US9428456, 1.166
Show/Hide
|
C27H34FN3O2
|
1
|
| 1 |
EC50 = 10 nM
|
|
|
|
CP0572238
|
US9428456, 1.069
Show/Hide
|
C26H34N4O3
|
1
|
| 1 |
EC50 = 10 nM
|
|
|
|
CP0572253
|
US9428456, 1.024
Show/Hide
|
C27H34ClN3O2
|
1
|
| 1 |
EC50 = 10 nM
|
|
|
|
CP0572257
|
US9428456, 1.152
Show/Hide
|
C27H41N3O2
|
1
|
| 1 |
EC50 = 10 nM
|
|
|
|
CP0516315
|
US9428456, 4.018
Show/Hide
|
C26H33FN4O2
|
1
|
| 1 |
EC50 = 11 nM
|
|
|
|
CP0572241
|
US9428456, 1.083
Show/Hide
|
C27H36N4O2
|
1
|
| 1 |
EC50 = 11 nM
|
|
|
|
CP0495281
|
US9428456, 1.098
Show/Hide
|
C29H39N3O2
|
1
|
| 1 |
EC50 = 12 nM
|
|
|
|
CP0512950
|
US9428456, 1.050
Show/Hide
|
C26H32ClN3O2
|
1
|
| 1 |
EC50 = 12 nM
|
|
|
|
CP0518680
|
US9428456, 1.169
Show/Hide
|
C26H34N4O2
|
1
|
| 1 |
EC50 = 12 nM
|
|
|
|
CP0548083
|
US9428456, 2.038
Show/Hide
|
C23H30N4O2
|
1
|
| 1 |
EC50 = 12 nM
|
|
|
|
CP0554406
|
US9428456, 1.106
Show/Hide
|
C27H32N4O2
|
1
|
| 1 |
EC50 = 12 nM
|
|
|
|
CP0557228
|
US9428456, 1.091
Show/Hide
|
C25H30Cl2N4O2
|
1
|
| 1 |
EC50 = 12 nM
|
|
|
|
CP0576967
|
US9428456, 1.155
Show/Hide
|
C26H31F3N4O2
|
1
|
| 1 |
EC50 = 12 nM
|
|
|
|
CP0413262
|
US9428456, 3.013
Show/Hide
|
C22H30N4O2S
|
1
|
| 1 |
EC50 = 13 nM
|
|
|
|
CP0495288
|
US9428456, 2.041
Show/Hide
|
C24H30N4O2
|
1
|
| 1 |
EC50 = 13 nM
|
|
|
|
CP0563164
|
US9428456, 1.318
Show/Hide
|
C25H32FN3O2
|
1
|
| 1 |
EC50 = 13 nM
|
|
|
|
CP0564193
|
US9428456, 1.114
Show/Hide
|
C27H34FN3O2
|
1
|
| 1 |
EC50 = 13 nM
|
|
|
|
CP0565143
|
US9428456, 1.038
Show/Hide
|
C23H31N5O2
|
1
|
| 1 |
EC50 = 13 nM
|
|
|
|
CP0572250
|
US9428456, 2.013
Show/Hide
|
C25H30ClN3O3
|
1
|
| 1 |
EC50 = 13 nM
|
|
|
|
CP0578548
|
US9428456, 4.011
Show/Hide
|
C25H31F3N4O2
|
1
|
| 1 |
EC50 = 13 nM
|
|
|
|
CP0512944
|
US9428456, 1.158
Show/Hide
|
C25H32ClN3O2S
|
1
|
| 1 |
EC50 = 14 nM
|
|
|
|
CP0544400
|
US9428456, 1.080
Show/Hide
|
C25H32N4O3
|
1
|
| 1 |
EC50 = 14 nM
|
|
|
|
CP0572259
|
US9428456, 1.159
Show/Hide
|
C27H34ClN3O3
|
1
|
| 1 |
EC50 = 14 nM
|
|
|
|
CP0472287
|
US9428456, 2.026
Show/Hide
|
C28H30ClN3O3
|
1
|
| 1 |
EC50 = 15 nM
|
|
|
|
CP0512289
|
US9428456, 1.122
Show/Hide
|
C28H37N3O3
|
1
|
| 1 |
EC50 = 15 nM
|
|
|
|
CP0513452
|
US9428456, 1.197
Show/Hide
|
C26H35N5O2
|
1
|
| 1 |
EC50 = 15 nM
|
|
|
|
CP0518670
|
US9428456, 1.089
Show/Hide
|
C25H29Cl2FN4O2
|
1
|
| 1 |
EC50 = 15 nM
|
|
|
|
CP0531302
|
US9428456, 1.189
Show/Hide
|
C29H43N5O2
|
1
|
| 1 |
EC50 = 15 nM
|
|
|
|
CP0539532
|
US9428456, 1.185
Show/Hide
|
C26H35N5O2
|
1
|
| 1 |
EC50 = 15 nM
|
|
|
|
CP0553287
|
US9428456, 1.265
Show/Hide
|
C26H34N4O2
|
1
|
| 1 |
EC50 = 15 nM
|
|
|
|
CP0561146
|
US9428456, 2.080
Show/Hide
|
C25H31F3N4O2
|
1
|
| 1 |
EC50 = 15 nM
|
|
|
|
CP0572285
|
US9428456, 2.036
Show/Hide
|
C24H25ClN4O2
|
1
|
| 1 |
EC50 = 15 nM
|
|
|
|
CP0486836
|
US9428456, 1.347
Show/Hide
|
C25H31F3N4O3
|
1
|
| 1 |
EC50 = 16 nM
|
|
|
|
CP0518676
|
US9428456, 1.332
Show/Hide
|
C26H33F3N4O2
|
1
|
| 1 |
EC50 = 16 nM
|
|
|
|
CP0529365
|
US9428456, 1.200
Show/Hide
|
C22H25ClN4O2
|
1
|
| 1 |
EC50 = 16 nM
|
|
|
|
CP0576974
|
US9428456, 4.002
Show/Hide
|
C24H31FN4O2
|
1
|
| 1 |
EC50 = 16 nM
|
|
|
|
CP0495280
|
US9428456, 2.103
Show/Hide
|
C25H34N4O2
|
1
|
| 1 |
EC50 = 17 nM
|
|
|
|
CP0518673
|
US9428456, 1.009
Show/Hide
|
C27H35N3O3
|
1
|
| 1 |
EC50 = 17 nM
|
|
|
|
CP0561149
|
US9428456, 1.334
Show/Hide
|
C26H34FN3O2
|
1
|
| 1 |
EC50 = 17 nM
|
|
|
|
CP0561239
|
US9428456, 1.047
Show/Hide
|
C28H37N3O3
|
1
|
| 1 |
EC50 = 17 nM
|
|
|
|
CP0561911
|
US9428456, 1.239
Show/Hide
|
C25H30F3N3O2
|
1
|
| 1 |
EC50 = 17 nM
|
|
|
|
CP0578569
|
US9428456, 2.025
Show/Hide
|
C27H27Cl2N3O2
|
1
|
| 1 |
EC50 = 17 nM
|
|
|
|
CP0507482
|
US9428456, 1.005
Show/Hide
|
C24H32N4O3
|
1
|
| 1 |
EC50 = 18 nM
|
|
|
|
CP0512949
|
US9428456, 1.034
Show/Hide
|
C28H37N3O2
|
1
|
| 1 |
EC50 = 18 nM
|
|
|
|
CP0518681
|
US9428456, 1.170
Show/Hide
|
C25H33N5O2
|
1
|
| 1 |
EC50 = 18 nM
|
|
|
|
CP0547473
|
US9428456, 1.277
Show/Hide
|
C24H31FN4O2
|
1
|
| 1 |
EC50 = 18 nM
|
|
|
|
CP0576494
|
US9428456, 1.030
Show/Hide
|
C30H38N4O2
|
1
|
| 1 |
EC50 = 18 nM
|
|
|
|
CP0472195
|
US9428456, 1.313
Show/Hide
|
C25H32FN3O2
|
1
|
| 1 |
EC50 = 19 nM
|
|
|
|
CP0478605
|
US9428456, 1.298
Show/Hide
|
C25H32FN3O3
|
1
|
| 1 |
EC50 = 19 nM
|
|
|
|
CP0518679
|
US9428456, 1.064
Show/Hide
|
C26H34N4O2
|
1
|
| 1 |
EC50 = 19 nM
|
|
|
|
CP0531307
|
US9428456, 2.088
Show/Hide
|
C26H33F3N4O2
|
1
|
| 1 |
EC50 = 19 nM
|
|
|
|
CP0544296
|
US9428456, 1.099
Show/Hide
|
C27H35N3O2
|
1
|
| 1 |
EC50 = 19 nM
|
|
|
|
CP0576847
|
US9428456, 4.015
Show/Hide
|
C25H34N4O3
|
1
|
| 1 |
EC50 = 19 nM
|
|
|
|
CP0578093
|
US9428456, 2.048
Show/Hide
|
C26H34N4O2
|
1
|
| 1 |
EC50 = 19 nM
|
|
|
|
CP0512940
|
US9428456, 1.013
Show/Hide
|
C26H34N4O2
|
1
|
| 1 |
EC50 = 20 nM
|
|
|
|
CP0531312
|
US9428456, 2.022
Show/Hide
|
C26H27ClN4O2
|
1
|
| 1 |
EC50 = 20 nM
|
|
|
|
CP0566320
|
US9428456, 2.043
Show/Hide
|
C24H30N4O2
|
1
|
| 1 |
EC50 = 20 nM
|
|
|
|
CP0576846
|
US9428456, 4.009
Show/Hide
|
C24H28F4N4O2
|
1
|
| 1 |
EC50 = 20 nM
|
|
|
|
CP0516938
|
US9428456, 2.020
Show/Hide
|
C29H30ClN3O2
|
1
|
| 1 |
EC50 = 21 nM
|
|
|
|
CP0554794
|
US9428456, 1.335
Show/Hide
|
C21H31N3O2
|
1
|
| 1 |
EC50 = 21 nM
|
|
|
|
CP0572284
|
US9428456, 1.112
Show/Hide
|
C28H37N3O2
|
1
|
| 1 |
EC50 = 21 nM
|
|
|
|
CP0515756
|
US9428456, 1.139
Show/Hide
|
C26H31Cl2N3O2
|
1
|
| 1 |
EC50 = 22 nM
|
|
|
|
CP0483931
|
US9428456, 1.165
Show/Hide
|
C27H35N3O2
|
1
|
| 1 |
EC50 = 23 nM
|
|
|
|
CP0555569
|
US9428456, 1.003
Show/Hide
|
C25H32N4O2
|
1
|
| 1 |
EC50 = 23 nM
|
|
|
|
CP0555941
|
US9428456, 1.193
Show/Hide
|
C25H33N5O2
|
1
|
| 1 |
EC50 = 23 nM
|
|
|
|
CP0486835
|
US9428456, 3.001
Show/Hide
|
C25H31FN4O2
|
1
|
| 1 |
EC50 = 24 nM
|
|
|
|
CP0513450
|
US9428456, 1.088
Show/Hide
|
C27H38N6O2
|
1
|
| 1 |
EC50 = 24 nM
|
|
|
|
CP0483924
|
US9428456, 1.020
Show/Hide
|
C25H39N3O2
|
1
|
| 1 |
EC50 = 25 nM
|
|
|
|
CP0518674
|
US9428456, 1.150
Show/Hide
|
C24H35N3O2
|
1
|
| 1 |
EC50 = 25 nM
|
|
|
|
CP0577885
|
US9428456, 1.167
Show/Hide
|
C28H37N3O3
|
1
|
| 1 |
EC50 = 25 nM
|
|
|
|
CP0419342
|
US9428456, 1.076
Show/Hide
|
C27H33N5O2
|
1
|
| 1 |
EC50 = 26 nM
|
|
|
|
CP0518683
|
US9428456, 1.173
Show/Hide
|
C29H36F3N3O2
|
1
|
| 1 |
EC50 = 26 nM
|
|
|
|
CP0544305
|
US9428456, 2.065
Show/Hide
|
C24H29F3N4O3
|
1
|
| 1 |
EC50 = 26 nM
|
|
|
|
CP0554413
|
US9428456, 2.050
Show/Hide
|
C25H32N4O2
|
1
|
| 1 |
EC50 = 26 nM
|
|
|
|
CP0577350
|
US9428456, 1.161
Show/Hide
|
C29H36ClN3O2
|
1
|
| 1 |
EC50 = 26 nM
|
|
|
|
CP0554412
|
US9428456, 2.044
Show/Hide
|
C26H32F2N4O2
|
1
|
| 1 |
EC50 = 27 nM
|
|
|
|
CP0478606
|
US9428456, 3.011
Show/Hide
|
C23H30ClN3O2S
|
1
|
| 1 |
EC50 = 28 nM
|
|
|
|
CP0531531
|
US9428456, 2.062
Show/Hide
|
C24H30N4O2
|
1
|
| 1 |
EC50 = 28 nM
|
|
|
|
CP0554104
|
US9428456, 3.007
Show/Hide
|
C25H31ClN4O2
|
1
|
| 1 |
EC50 = 28 nM
|
|
|
|
CP0554404
|
US9428456, 2.096
Show/Hide
|
C23H30N4O2
|
1
|
| 1 |
EC50 = 28 nM
|
|
|
|
CP0555455
|
US9428456, 1.172
Show/Hide
|
C27H36N4O2
|
1
|
| 1 |
EC50 = 28 nM
|
|
|
|
CP0566267
|
US9428456, 1.327
Show/Hide
|
C26H36N4O2
|
1
|
| 1 |
EC50 = 28 nM
|
|
|
|
CP0413223
|
US9428456, 1.017
Show/Hide
|
C25H37N3O2
|
1
|
| 1 |
EC50 = 29 nM
|
|
|
|
CP0518669
|
US9428456, 1.350
Show/Hide
|
C27H34N4O4
|
1
|
| 1 |
EC50 = 29 nM
|
|
|
|
CP0554415
|
US9428456, 5.001
Show/Hide
|
C22H27F3N6O2
|
1
|
| 1 |
EC50 = 29 nM
|
|
|
|
CP0577888
|
US9428456, 2.024
Show/Hide
|
C24H25ClN4O2S
|
1
|
| 1 |
EC50 = 32 nM
|
|
|
|
CP0552291
|
US9428456, 1.288
Show/Hide
|
C25H34N4O2
|
1
|
| 1 |
EC50 = 33 nM
|
|
|
|
CP0574010
|
US9428456, 1.184
Show/Hide
|
C27H36N4O2
|
1
|
| 1 |
EC50 = 33 nM
|
|
|
|
CP0413233
|
US9428456, 1.349
Show/Hide
|
C25H32N4O4
|
1
|
| 1 |
EC50 = 34 nM
|
|
|
|
CP0547474
|
US9428456, 1.283
Show/Hide
|
C28H39N3O2S
|
1
|
| 1 |
EC50 = 34 nM
|
|
|
|
CP0554092
|
US9428456, 1.032
Show/Hide
|
C30H41N3O2
|
1
|
| 1 |
EC50 = 34 nM
|
|
|
|
CP0566253
|
US9428456, 1.037
Show/Hide
|
C27H34ClN3O2
|
1
|
| 1 |
EC50 = 34 nM
|
|
|
|
CP0542739
|
US9428456, 1.008
Show/Hide
|
C27H33N5O2
|
1
|
| 1 |
EC50 = 35 nM
|
|
|
|
CP0566348
|
US9428456, 1.120
Show/Hide
|
C27H34ClN3O2
|
1
|
| 1 |
EC50 = 35 nM
|
|
|
|
CP0576501
|
US9428456, 1.036
Show/Hide
|
C30H41N3O2
|
1
|
| 1 |
EC50 = 35 nM
|
|
|
|
CP0483897
|
US9428456, 3.004
Show/Hide
|
C25H31ClN4O2
|
1
|
| 1 |
EC50 = 36 nM
|
|
|
|
CP0537193
|
US9428456, 1.316
Show/Hide
|
C25H31F3N4O2
|
1
|
| 1 |
EC50 = 36 nM
|
|
|
|
CP0537318
|
US9428456, 1.127
Show/Hide
|
C26H31F2N3O2
|
1
|
| 1 |
EC50 = 36 nM
|
|
|
|
CP0557225
|
US9428456, 2.089
Show/Hide
|
C25H29F3N4O2
|
1
|
| 1 |
EC50 = 36 nM
|
|
|
|
CP0572242
|
US9428456, 1.087
Show/Hide
|
C24H31N5O2
|
1
|
| 1 |
EC50 = 36 nM
|
|
|
|
CP0576971
|
US9428456, 1.052
Show/Hide
|
C30H39N3O2
|
1
|
| 1 |
EC50 = 36 nM
|
|
|
|
CP0555925
|
US9428456, 2.097
Show/Hide
|
C24H29ClFN3O2
|
1
|
| 1 |
EC50 = 37 nM
|
|
|
|
CP0566271
|
US9428456, 1.177
Show/Hide
|
C28H34F3N3O2
|
1
|
| 1 |
EC50 = 37 nM
|
|
|
|
CP0554100
|
US9428456, 1.084
Show/Hide
|
C29H39N5O2
|
1
|
| 1 |
EC50 = 39 nM
|
|
|
|
CP0577347
|
US9428456, 1.021
Show/Hide
|
C29H34N4O2
|
1
|
| 1 |
EC50 = 39 nM
|
|
|
|
CP0512966
|
US9428456, 1.004
Show/Hide
|
C29H41N3O2S
|
1
|
| 1 |
EC50 = 40 nM
|
|
|
|
CP0519671
|
US9428456, 2.019
Show/Hide
|
C30H32ClN3O2
|
1
|
| 1 |
EC50 = 40 nM
|
|
|
|
CP0539553
|
US9428456, 1.053
Show/Hide
|
C25H32N4O2
|
1
|
| 1 |
EC50 = 40 nM
|
|
|
|
CP0544297
|
US9428456, 1.109
Show/Hide
|
C28H37N3O2
|
1
|
| 1 |
EC50 = 40 nM
|
|
|
|
CP0544399
|
US9428456, 1.070
Show/Hide
|
C26H33ClN4O2
|
1
|
| 1 |
EC50 = 40 nM
|
|
|
|
CP0572244
|
US9428456, 1.096
Show/Hide
|
C28H38N4O2
|
1
|
| 1 |
EC50 = 40 nM
|
|
|
|
CP0518677
|
US9428456, 1.054
Show/Hide
|
C31H42N4O2
|
1
|
| 1 |
EC50 = 41 nM
|
|
|
|
CP0576973
|
US9428456, 3.010
Show/Hide
|
C23H30ClN3O2S
|
1
|
| 1 |
EC50 = 41 nM
|
|
|
|
CP0486839
|
US9428456, 1.027
Show/Hide
|
C28H34N4O2
|
1
|
| 1 |
EC50 = 42 nM
|
|
|
|
CP0507486
|
US9428456, 1.136
Show/Hide
|
C28H31F6N3O2
|
1
|
| 1 |
EC50 = 43 nM
|
|
|
|
CP0561152
|
US9428456, 1.041
Show/Hide
|
C30H41N3O2
|
1
|
| 1 |
EC50 = 43 nM
|
|
|
|
CP0561245
|
US9428456, 1.066
Show/Hide
|
C25H31ClN4O2
|
1
|
| 1 |
EC50 = 44 nM
|
|
|
|
CP0574119
|
US9428456, 3.012
Show/Hide
|
C22H30N4O2S
|
1
|
| 1 |
EC50 = 44 nM
|
|
|
|
CP0495286
|
US9428456, 2.035
Show/Hide
|
C27H28ClN3O2
|
1
|
| 1 |
EC50 = 45 nM
|
|
|
|
CP0566272
|
US9428456, 1.319
Show/Hide
|
C25H31F3N4O3
|
1
|
| 1 |
EC50 = 45 nM
|
|
|
|
CP0478607
|
US9428456, 4.001
Show/Hide
|
C26H33FN4O2
|
1
|
| 1 |
EC50 = 46 nM
|
|
|
|
CP0561246
|
US9428456, 2.015
Show/Hide
|
C27H34ClN3O2
|
1
|
| 1 |
EC50 = 46 nM
|
|
|
|
CP0566269
|
US9428456, 1.048
Show/Hide
|
C30H35N3O2
|
1
|
| 1 |
EC50 = 46 nM
|
|
|
|
CP0554101
|
US9428456, 1.204
Show/Hide
|
C22H25FN4O2
|
1
|
| 1 |
EC50 = 47 nM
|
|
|
|
CP0555976
|
US9428456, 1.320
Show/Hide
|
C25H34N4O3
|
1
|
| 1 |
EC50 = 48 nM
|
|
|
|
CP0406789
|
US9428456, 1.290
Show/Hide
|
C25H34N4O2
|
1
|
| 1 |
EC50 = 49 nM
|
|
|
|
CP0516316
|
US9428456, 2.106
Show/Hide
|
C27H33F3N4O2
|
1
|
| 1 |
EC50 = 49 nM
|
|
|
|
CP0548086
|
US9428456, 1.324
Show/Hide
|
C23H30ClN5O2
|
1
|
| 1 |
EC50 = 51 nM
|
|
|
|
CP0553290
|
US9428456, 1.180
Show/Hide
|
C26H33ClN4O2
|
1
|
| 1 |
EC50 = 51 nM
|
|
|
|
CP0483903
|
US9428456, 1.203
Show/Hide
|
C23H28N4O2
|
1
|
| 1 |
EC50 = 56 nM
|
|
|
|
CP0518657
|
US9428456, 3.006
Show/Hide
|
C25H31FN4O2
|
1
|
| 1 |
EC50 = 56 nM
|
|
|
|
CP0518656
|
US9428456, 3.005
Show/Hide
|
C25H31FN4O2
|
1
|
| 1 |
EC50 = 57 nM
|
|
|
|
CP0531468
|
US9428456, 4.010
Show/Hide
|
C27H33F3N4O2
|
1
|
| 1 |
EC50 = 57 nM
|
|
|
|
CP0566270
|
US9428456, 1.062
Show/Hide
|
C26H35N5O4
|
1
|
| 1 |
EC50 = 57 nM
|
|
|
|
CP0576499
|
US9428456, 1.333
Show/Hide
|
C26H36N4O2
|
1
|
| 1 |
EC50 = 57 nM
|
|
|
|
CP0576972
|
US9428456, 3.002
Show/Hide
|
C25H31ClN4O2
|
1
|
| 1 |
EC50 = 57 nM
|
|
|
|
CP0517249
|
US9428456, 4.004
Show/Hide
|
C25H34N4O2
|
1
|
| 1 |
EC50 = 59 nM
|
|
|
|
CP0561244
|
US9428456, 1.065
Show/Hide
|
C26H34N4O2
|
1
|
| 1 |
EC50 = 59 nM
|
|
|
|
CP0483900
|
US9428456, 1.074
Show/Hide
|
C25H31ClN4O2
|
1
|
| 1 |
EC50 = 60 nM
|
|
|
|
CP0544294
|
US9428456, 2.099
Show/Hide
|
C25H29F3N4O2
|
1
|
| 1 |
EC50 = 60 nM
|
|
|
|
CP0572287
|
US9428456, 2.055
Show/Hide
|
C22H28N4O2
|
1
|
| 1 |
EC50 = 60 nM
|
|
|
|
CP0519511
|
US9428456, 7.001
Show/Hide
|
C23H31N5O2
|
1
|
| 1 |
EC50 = 62 nM
|
|
|
|
CP0547479
|
US9428456, 1.331
Show/Hide
|
C26H34FN3O2
|
1
|
| 1 |
EC50 = 62 nM
|
|
|
|
CP0512951
|
US9428456, 1.191
Show/Hide
|
C27H36N4O2
|
1
|
| 1 |
EC50 = 64 nM
|
|
|
|
CP0531300
|
US9428456, 1.178
Show/Hide
|
C28H34N4O2
|
1
|
| 1 |
EC50 = 64 nM
|
|
|
|
CP0559170
|
US9428456, 2.061
Show/Hide
|
C26H34N4O2
|
1
|
| 1 |
EC50 = 64 nM
|
|
|
|
CP0576502
|
US9428456, 1.323
Show/Hide
|
C22H29N5O2
|
1
|
| 1 |
EC50 = 66 nM
|
|
|
|
CP0516313
|
US9428456, 2.047
Show/Hide
|
C24H30N4O2
|
1
|
| 1 |
EC50 = 67 nM
|
|
|
|
CP0537204
|
US9428456, 1.010
Show/Hide
|
C29H34N4O2
|
1
|
| 1 |
EC50 = 68 nM
|
|
|
|
CP0555977
|
US9428456, 2.085
Show/Hide
|
C26H36N4O2
|
1
|
| 1 |
EC50 = 68 nM
|
|
|
|
CP0547477
|
US9428456, 2.074
Show/Hide
|
C22H29N3O2S
|
1
|
| 1 |
EC50 = 70 nM
|
|
|
|
CP0564195
|
US9428456, 1.126
Show/Hide
|
C28H37N3O4
|
1
|
| 1 |
EC50 = 70 nM
|
|
|
|
CP0544293
|
US9428456, 1.352
Show/Hide
|
C25H33N3O4S
|
1
|
| 1 |
EC50 = 71 nM
|
|
|
|
CP0566321
|
US9428456, 4.008
Show/Hide
|
C26H30F4N4O2
|
1
|
| 1 |
EC50 = 71 nM
|
|
|
|
CP0472192
|
US9428456, 1.144
Show/Hide
|
C28H38N4O2
|
1
|
| 1 |
EC50 = 73 nM
|
|
|
|
CP0512954
|
US9428456, 1.317
Show/Hide
|
C25H34N4O2
|
1
|
| 1 |
EC50 = 76 nM
|
|
|
|
CP0483923
|
US9428456, 1.015
Show/Hide
|
C31H37N3O2
|
1
|
| 1 |
EC50 = 78 nM
|
|
|
|
CP0572234
|
US9428456, 1.179
Show/Hide
|
C28H34N4O2
|
1
|
| 1 |
EC50 = 78 nM
|
|
|
|
CP0574003
|
US9428456, 1.042
Show/Hide
|
C28H37N3O3
|
1
|
| 1 |
EC50 = 79 nM
|
|
|
|
CP0554097
|
US9428456, 1.149
Show/Hide
|
C23H33N3O2
|
1
|
| 1 |
EC50 = 81 nM
|
|
|
|
CP0565141
|
US9428456, 1.293
Show/Hide
|
C22H27ClN4O2S
|
1
|
| 1 |
EC50 = 81 nM
|
|
|
|
CP0495287
|
US9428456, 2.037
Show/Hide
|
C23H28N4O2
|
1
|
| 1 |
EC50 = 82 nM
|
|
|
|
CP0555966
|
US9428456, 1.336
Show/Hide
|
C20H29N3O2
|
1
|
| 1 |
EC50 = 83 nM
|
|
|
|
CP0531301
|
US9428456, 1.186
Show/Hide
|
C31H42N6O2
|
1
|
| 1 |
EC50 = 86 nM
|
|
|
|
CP0539534
|
US9428456, 1.308
Show/Hide
|
C28H35F3N4O2
|
1
|
| 1 |
EC50 = 87 nM
|
|
|
|
CP0561145
|
US9428456, 2.077
Show/Hide
|
C25H33N3O2S
|
1
|
| 1 |
EC50 = 87 nM
|
|
|
|
CP0576845
|
US9428456, 2.064
Show/Hide
|
C25H31F3N4O3
|
1
|
| 1 |
EC50 = 87 nM
|
|
|
|
CP0512945
|
US9428456, 1.264
Show/Hide
|
C23H31N5O2
|
1
|
| 1 |
EC50 = 90 nM
|
|
|
|
CP0561913
|
US9428456, 2.063
Show/Hide
|
C25H32N4O2
|
1
|
| 1 |
EC50 = 92 nM
|
|
|
|
CP0572246
|
US9428456, 1.198
Show/Hide
|
C26H35N5O2
|
1
|
| 1 |
EC50 = 92 nM
|
|
|
|
CP0572286
|
US9428456, 2.051
Show/Hide
|
C26H34N4O2
|
1
|
| 1 |
EC50 = 96 nM
|
|
|
|
CP0572252
|
US9428456, 1.022
Show/Hide
|
C29H34N4O2
|
1
|
| 1 |
EC50 = 97 nM
|
|
|
|
CP0555969
|
US9428456, 1.297
Show/Hide
|
C25H34N4O3
|
1
|
| 1 |
EC50 = 98 nM
|
|
|
|
CP0574009
|
US9428456, 1.183
Show/Hide
|
C27H33F3N4O2
|
1
|
| 1 |
EC50 = 98 nM
|
|
|
|
CP0544300
|
US9428456, 1.231
Show/Hide
|
C24H29F3N4O2
|
1
|
| 1 |
EC50 = 99 nM
|
|
|
|
CP0572235
|
US9428456, 1.192
Show/Hide
|
C28H38N4O2
|
1
|
| 1 |
EC50 = 102 nM
|
|
|
|
CP0512287
|
US9428456, 1.354
Show/Hide
|
C26H32N4O2S
|
1
|
| 1 |
EC50 = 108 nM
|
|
|
|
CP0495290
|
US9428456, 2.054
Show/Hide
|
C24H28F2N4O2
|
1
|
| 1 |
EC50 = 109 nM
|
|
|
|
CP0514669
|
US9428456, 1.214
Show/Hide
|
C25H29F3N4O2
|
1
|
| 1 |
EC50 = 109 nM
|
|
|
|
CP0565140
|
US9428456, 1.289
Show/Hide
|
C24H32N4O2
|
1
|
| 1 |
EC50 = 113 nM
|
|
|
|
CP0451615
|
US9428456, 1.262
Show/Hide
|
C24H34N4O2S
|
1
|
| 1 |
EC50 = 120 nM
|
|
|
|
CP0470693
|
US9428456, 2.082
Show/Hide
|
C26H33F3N4O2
|
1
|
| 1 |
EC50 = 121 nM
|
|
|
|
CP0554112
|
US9428456, 1.016
Show/Hide
|
C23H35N3O2
|
1
|
| 1 |
EC50 = 121 nM
|
|
|
|
CP0577281
|
US9428456, 2.052
Show/Hide
|
C24H29FN4O2
|
1
|
| 1 |
EC50 = 121 nM
|
|
|
|
CP0565144
|
US9428456, 1.051
Show/Hide
|
C24H33N5O2
|
1
|
| 1 |
EC50 = 130 nM
|
|
|
|
CP0483927
|
US9428456, 1.291
Show/Hide
|
C27H36N4O2
|
1
|
| 1 |
EC50 = 134 nM
|
|
|
|
CP0574117
|
US9428456, 2.016
Show/Hide
|
C28H36ClN3O2
|
1
|
| 1 |
EC50 = 134 nM
|
|
|
|
CP0961328
|
US9428456, 1.190
Show/Hide
|
C28H35N5O2
|
1
|
| 1 |
EC50 = 134 nM
|
|
|
|
CP0516311
|
US9428456, 1.255
Show/Hide
|
C24H37N3O3
|
1
|
| 1 |
EC50 = 137 nM
|
|
|
|
CP0554099
|
US9428456, 1.263
Show/Hide
|
C23H31N5O2
|
1
|
| 1 |
EC50 = 143 nM
|
|
|
|
CP0529359
|
US9428456, 1.314
Show/Hide
|
C25H34N4O2
|
1
|
| 1 |
EC50 = 145 nM
|
|
|
|
CP0572247
|
US9428456, 1.202
Show/Hide
|
C23H28N4O2
|
1
|
| 1 |
EC50 = 145 nM
|
|
|
|
CP0574008
|
US9428456, 1.181
Show/Hide
|
C27H36N4O2
|
1
|
| 1 |
EC50 = 148 nM
|
|
|
|
CP0556712
|
US9428456, 1.093
Show/Hide
|
C27H33N5O2
|
1
|
| 1 |
EC50 = 149 nM
|
|
|
|
CP0572233
|
US9428456, 1.171
Show/Hide
|
C26H34N4O2
|
1
|
| 1 |
EC50 = 150 nM
|
|
|
|
CP0515759
|
US9428456, 2.073
Show/Hide
|
C20H25N3O2S
|
1
|
| 1 |
EC50 = 155 nM
|
|
|
|
CP0566268
|
US9428456, 1.329
Show/Hide
|
C26H33F3N4O2
|
1
|
| 1 |
EC50 = 159 nM
|
|
|
|
CP0423963
|
US9428456, 2.100
Show/Hide
|
C26H31ClFN3O2
|
1
|
| 1 |
EC50 = 161 nM
|
|
|
|
CP0530648
|
US9428456, 2.023
Show/Hide
|
C26H27ClN4O2
|
1
|
| 1 |
EC50 = 162 nM
|
|
|
|
CP0574107
|
US9428456, 3.003
Show/Hide
|
C25H31FN4O2
|
1
|
| 1 |
EC50 = 167 nM
|
|
|
|
CP0519510
|
US9428456, 4.023
Show/Hide
|
C25H34N4O3
|
1
|
| 1 |
EC50 = 173 nM
|
|
|
|
CP0539845
|
US9428456, 1.176
Show/Hide
|
C26H34N4O2
|
1
|
| 1 |
EC50 = 173 nM
|
|
|
|
CP0423271
|
US9428456, 1.351
Show/Hide
|
C25H33N3O4S
|
1
|
| 1 |
EC50 = 176 nM
|
|
|
|
CP0572245
|
US9428456, 1.195
Show/Hide
|
C25H33N5O2
|
1
|
| 1 |
EC50 = 176 nM
|
|
|
|
CP0531326
|
US9428456, 1.175
Show/Hide
|
C29H39N3O4
|
1
|
| 1 |
EC50 = 181 nM
|
|
|
|
CP0576968
|
US9428456, 1.287
Show/Hide
|
C23H30N4O2
|
1
|
| 1 |
EC50 = 181 nM
|
|
|
|
CP0413224
|
US9428456, 1.026
Show/Hide
|
C29H36N4O2
|
1
|
| 1 |
EC50 = 182 nM
|
|
|
|
CP0566410
|
US9428456, 1.071
Show/Hide
|
C29H41N5O2
|
1
|
| 1 |
EC50 = 182 nM
|
|
|
|
CP0547476
|
US9428456, 2.072
Show/Hide
|
C19H23N3O2S
|
1
|
| 1 |
EC50 = 188 nM
|
|
|
|
CP0512288
|
US9428456, 2.098
Show/Hide
|
C23H27F3N4O2
|
1
|
| 1 |
EC50 = 193 nM
|
|
|
|
CP0555975
|
US9428456, 1.315
Show/Hide
|
C25H31F3N4O2
|
1
|
| 1 |
EC50 = 193 nM
|
|
|
|
CP0548084
|
US9428456, 2.053
Show/Hide
|
C24H29FN4O2
|
1
|
| 1 |
EC50 = 195 nM
|
|
|
|
CP0563166
|
US9428456, 4.003
Show/Hide
|
C27H36N4O2
|
1
|
| 1 |
EC50 = 197 nM
|
|
|
|
CP0413228
|
US9428456, 1.285
Show/Hide
|
C24H32N6O2
|
1
|
| 1 |
EC50 = 199 nM
|
|
|
|
CP0539533
|
US9428456, 1.188
Show/Hide
|
C30H41N5O2
|
1
|
| 1 |
EC50 = 215 nM
|
|
|
|
CP0512967
|
US9428456, 1.342
Show/Hide
|
C23H36N4O2
|
1
|
| 1 |
EC50 = 216 nM
|
|
|
|
CP0561247
|
US9428456, 2.021
Show/Hide
|
C26H27ClN4O2
|
1
|
| 1 |
EC50 = 218 nM
|
|
|
|
CP0554681
|
US9428456, 2.017
Show/Hide
|
C29H32ClN3O2
|
1
|
| 1 |
EC50 = 219 nM
|
|
|
|
CP0548082
|
US9428456, 1.256
Show/Hide
|
C22H33N3O3
|
1
|
| 1 |
EC50 = 222 nM
|
|
|
|
CP0565139
|
US9428456, 1.284
Show/Hide
|
C24H29F3N6O2
|
1
|
| 1 |
EC50 = 223 nM
|
|
|
|
CP0495291
|
US9428456, 2.058
Show/Hide
|
C24H32N4O3
|
1
|
| 1 |
EC50 = 224 nM
|
|
|
|
CP0577352
|
US9428456, 2.079
Show/Hide
|
C27H35F3N4O2
|
1
|
| 1 |
EC50 = 226 nM
|
|
|
|
CP0516318
|
US9428456, 4.022
Show/Hide
|
C24H32N4O3
|
1
|
| 1 |
EC50 = 234 nM
|
|
|
|
CP0553288
|
US9428456, 1.063
Show/Hide
|
C26H34N4O2
|
1
|
| 1 |
EC50 = 237 nM
|
|
|
|
CP0554777
|
US9428456, 2.011
Show/Hide
|
C26H32ClN3O3
|
1
|
| 1 |
EC50 = 241 nM
|
|
|
|
CP0515760
|
US9428456, 2.078
Show/Hide
|
C26H33F3N4O2
|
1
|
| 1 |
EC50 = 257 nM
|
|
|
|
CP0572236
|
US9428456, 1.325
Show/Hide
|
C25H31F3N4O3
|
1
|
| 1 |
EC50 = 262 nM
|
|
|
|
CP0547475
|
US9428456, 1.286
Show/Hide
|
C22H27F3N6O2
|
1
|
| 1 |
EC50 = 265 nM
|
|
|
|
CP0547478
|
US9428456, 1.330
Show/Hide
|
C26H36N4O2
|
1
|
| 1 |
EC50 = 285 nM
|
|
|
|
CP0564200
|
US9428456, 2.049
Show/Hide
|
C25H30F2N4O2
|
1
|
| 1 |
EC50 = 300 nM
|
|
|
|
CP0472194
|
US9428456, 1.194
Show/Hide
|
C28H39N5O2S
|
1
|
| 1 |
EC50 = 303 nM
|
|
|
|
CP0539537
|
US9428456, 2.084
Show/Hide
|
C25H32N4O2
|
1
|
| 1 |
EC50 = 304 nM
|
|
|
|
CP0483910
|
US9428456, 2.018
Show/Hide
|
C32H32ClN3O2
|
1
|
| 1 |
EC50 = 349 nM
|
|
|
|
CP0554069
|
US9428456, 1.307
Show/Hide
|
C28H38N4O2
|
1
|
| 1 |
EC50 = 350 nM
|
|
|
|
CP0419341
|
US9428456, 1.073
Show/Hide
|
C29H39N5O3
|
1
|
| 1 |
EC50 = 371 nM
|
|
|
|
CP0483930
|
US9428456, 1.163
Show/Hide
|
C25H32ClN3O2S
|
1
|
| 1 |
EC50 = 386 nM
|
|
|
|
CP0539499
|
US9428456, 1.059
Show/Hide
|
C26H31F3N4O2
|
1
|
| 1 |
EC50 = 393 nM
|
|
|
|
CP0483911
|
US9428456, 2.028
Show/Hide
|
C28H30ClN3O3
|
1
|
| 1 |
EC50 = 394 nM
|
|
|
|
CP0577280
|
US9428456, 2.045
Show/Hide
|
C24H27N5O2
|
1
|
| 1 |
EC50 = 402 nM
|
|
|
|
CP0495294
|
US9428456, 2.067
Show/Hide
|
C26H33F3N4O3
|
1
|
| 1 |
EC50 = 406 nM
|
|
|
|
CP0561242
|
US9428456, 1.294
Show/Hide
|
C22H29N5O2S
|
1
|
| 1 |
EC50 = 408 nM
|
|
|
|
CP0515758
|
US9428456, 1.280
Show/Hide
|
C25H32FN3O3
|
1
|
| 1 |
EC50 = 409 nM
|
|
|
|
CP0512946
|
US9428456, 1.279
Show/Hide
|
C24H28BrF3N4O2
|
1
|
| 1 |
EC50 = 420 nM
|
|
|
|
CP0572255
|
US9428456, 1.145
Show/Hide
|
C27H31F4N3O2
|
1
|
| 1 |
EC50 = 425 nM
|
|
|
|
CP0561271
|
US9428456, 2.066
Show/Hide
|
C28H35F3N4O3
|
1
|
| 1 |
EC50 = 431 nM
|
|
|
|
CP0577889
|
US9428456, 2.029
Show/Hide
|
C27H27Cl2N3O2
|
1
|
| 1 |
EC50 = 433 nM
|
|
|
|
CP0516939
|
US9428456, 2.027
Show/Hide
|
C27H27Cl2N3O2
|
1
|
| 1 |
EC50 = 442 nM
|
|
|
|
CP0419314
|
US9428456, 1.072
Show/Hide
|
C30H42N6O2
|
1
|
| 1 |
EC50 = 471 nM
|
|
|
|
CP0530644
|
US9428456, 1.196
Show/Hide
|
C30H43N5O2
|
1
|
| 1 |
EC50 = 491 nM
|
|
|
|
CP0555980
|
US9428456, 1.086
Show/Hide
|
C25H33N5O2
|
1
|
| 1 |
EC50 = 527 nM
|
|
|
|
CP0516935
|
US9428456, 2.034
Show/Hide
|
C27H27ClF3N3O3
|
1
|
| 1 |
EC50 = 533 nM
|
|
|
|
CP0470694
|
US9428456, 1.174
Show/Hide
|
C26H33ClN4O2
|
1
|
| 1 |
EC50 = 559 nM
|
|
|
|
CP0561266
|
US9428456, 1.108
Show/Hide
|
C28H37N3O2
|
1
|
| 1 |
EC50 = 633 nM
|
|
|
|
CP0566266
|
US9428456, 2.076
Show/Hide
|
C25H27N3O2S
|
1
|
| 1 |
EC50 = 780 nM
|
|
|
|
CP0483912
|
US9428456, 2.030
Show/Hide
|
C28H30ClN3O3
|
1
|
| 1 |
EC50 = 832 nM
|
|
|
|
CP0539853
|
US9428456, 2.012
Show/Hide
|
C30H40ClN3O2
|
1
|
| 1 |
EC50 = 1050 nM
|
|
|
|
CP0531324
|
US9428456, 1.044
Show/Hide
|
C23H31N5O2
|
1
|
| 1 |
EC50 = 1240 nM
|
|
|
|
CP0577354
|
US9428456, 1.040
Show/Hide
|
C23H31N5O2
|
1
|
| 1 |
EC50 = 1260 nM
|
|
|
|
CP0556164
|
US9428456, 1.045
Show/Hide
|
C29H37N5O2
|
1
|
| 1 |
EC50 = 2490 nM
|
|
|
|
CP0561240
|
US9428456, 1.162
Show/Hide
|
C26H31Cl2N3O2
|
1
|
| 1 |
EC50 = 2780 nM
|
|
|
