| Compound ID |
Compound Name |
Compound Formula |
|
CP0845571
|
(S)-5-(3-(1-(2-fluoroethylamino)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)-2-isopropoxybenzonitrile
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|
C23H23FN4O2
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0845573
|
(R)-2-(N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)sulfamoyl)acetic acid
Show/Hide
|
C23H22N4O6S
|
1
|
| 1 |
EC50 < 0.05 nM
|
|
|
|
CP0845575
|
(S)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-2-(4-hydroxypiperidin-1-yl)-2-oxoethanesulfonamide
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|
C28H31N5O6S
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0845577
|
(S)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)morpholine-4-carboxamide
Show/Hide
|
C26H27N5O4
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0845578
|
(R)-1-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-ylcarbamoyl)piperidine-4-carboxylic acid
Show/Hide
|
C28H29N5O5
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0845579
|
2-isopropoxy-5-(3-(1-(piperazin-1-yl)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)benzonitrile
Show/Hide
|
C25H27N5O2
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0845580
|
(R)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-l,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-2-hydroxyethanesulfonamide
Show/Hide
|
C23H24N4O5S
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0848222
|
methyl 1-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)azetidine-3-carboxylate
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|
C26H26N4O4
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0851368
|
(S)-N-((S)-4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-3-hydroxypyrrolidine-1-carboxamide
Show/Hide
|
C26H27N5O4
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0852162
|
5-(3-((R)-1-(2-((R)-3-hydroxypyrrolidin-1-yl)-2-oxoethylamino)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)-2-isopropoxybenzonitrile
Show/Hide
|
C27H29N5O4
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0861101
|
(R)-2-(azetidin-1-yl)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)ethanesulfonamide
Show/Hide
|
C26H29N5O4S
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0861102
|
(S)-3-(N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)sulfamoyl)propanoic acid
Show/Hide
|
C24H24N4O6S
|
1
|
| 1 |
EC50 < 0.05 nM
|
|
|
|
CP0861105
|
(S)-N-((R)-4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-3-hydroxypyrrolidine-1-carboxamide
Show/Hide
|
C26H27N5O4
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0861108
|
5-(3-(1-(4-hydroxypiperidin-1-yl)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)-2-isopropoxybenzonitrile
Show/Hide
|
C26H28N4O3
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0861109
|
(S)-4-(5-(4-isopropoxy-3-(trifluoromethyl)phenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-ol
Show/Hide
|
C21H19F3N2O3
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0861110
|
(R)-2-((R)-4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-ylamino)propanoic acid
Show/Hide
|
C24H24N4O4
|
1
|
| 1 |
EC50 < 0.05 nM
|
|
|
|
CP0861111
|
(R)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)methanesulfonamide
Show/Hide
|
C22H22N4O4S
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0861112
|
(R)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-2-(dimethylamino)ethanesulfonamide
Show/Hide
|
C25H29N5O4S
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0864437
|
(R)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-2-(2-hydroxyethylamino)ethanesulfonamide
Show/Hide
|
C25H29N5O5S
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0864439
|
(R)-N-((S)-4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-3-hydroxypiperidine-1-carboxamide
Show/Hide
|
C27H29N5O4
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0864440
|
(R)-3-amino-N-((R)-4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)pyrrolidine-1-carboxamide
Show/Hide
|
C26H28N6O3
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0864442
|
(R)-2-hydroxyethyl 4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-ylcarbamate
Show/Hide
|
C24H24N4O5
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0864443
|
(S)-2-(1-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-ylcarbamoyl)piperidin-4-yl)acetic acid
Show/Hide
|
C29H31N5O5
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0864449
|
5-(3-((R)-1-(((S)-1-hydroxypropan-2-yl)amino)-2,3-dihydro-1H-inden-4-yl)-l,2,4-oxadiazo1-5-yl)-2-isopropoxybenzonitrile
Show/Hide
|
C24H26N4O3
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0864457
|
(R)-2-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-ylamino)-N-methylacetamide
Show/Hide
|
C24H25N5O3
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0864458
|
5-(3-((R)-1-(((R)-1-hydroxypropan-2-yl)amino)-2,3-dihydro-1H-inden-4-yl)-l,2,4-oxadiazo1-5-yl)-2-isopropoxybenzonitrile
Show/Hide
|
C24H26N4O3
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0867140
|
(R)-5-(3-(1-hydroxy-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)-2-isopropoxybenzonitrile
Show/Hide
|
C21H19N3O3
|
1
|
| 1 |
EC50 < 0.05 nM
|
|
|
|
CP0869378
|
(S)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-2-(3-hydroxyazetidin-1-yl)-2-oxoethanesulfonamide
Show/Hide
|
C26H27N5O6S
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0869391
|
(R)-2-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-ylamino)acetamide
Show/Hide
|
C23H23N5O3
|
1
|
| 1 |
EC50 < 0.05 nM
|
|
|
|
CP0869393
|
(S)-5-(3-(1-hydroxy-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)-2-isopropoxybenzonitrile
Show/Hide
|
C21H19N3O3
|
1
|
| 1 |
EC50 < 0.05 nM
|
|
|
|
CP0869396
|
(R)-5-(3-(1-((2-fluoroethyl)amino)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazo1-5-yl)-2-isopropoxybenzonitrile
Show/Hide
|
C23H23FN4O2
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0871093
|
(S)-1-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-N,N-dimethylazetidine-3-carboxamide
Show/Hide
|
C27H29N5O3
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0873126
|
(R)-2-ethoxy-5-(3-(1-hydroxy-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)benzonitrile
Show/Hide
|
C20H17N3O3
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0873127
|
5-(3-(1-(4-(2-hydroxyethyl)piperazin-1-yl)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)-2-isopropoxybenzonitrile
Show/Hide
|
C27H31N5O3
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0873133
|
(S)-2-isopropoxy-5-(3-(1-(methylamino)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)benzonitrile
Show/Hide
|
C22H22N4O2
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0873146
|
5-(3-(1-(2-aminoethylamino)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)-2-isopropoxybenzonitrile
Show/Hide
|
C23H25N5O2
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0873690
|
3-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-ylamino)propanoic acid
Show/Hide
|
C24H24N4O4
|
1
|
| 1 |
EC50 < 0.05 nM
|
|
|
|
CP0873691
|
(S)-4-(5-(4-ethoxy-3-(trifluoromethyl)phenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-ol
Show/Hide
|
C20H17F3N2O3
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0873695
|
(R)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)acetamide
Show/Hide
|
C23H22N4O3
|
1
|
| 1 |
EC50 < 0.05 nM
|
|
|
|
CP0873698
|
(R)-2-(N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)sulfamoyl)-N,N-dimethylacetamide
Show/Hide
|
C25H27N5O5S
|
1
|
| 1 |
EC50 < 0.05 nM
|
|
|
|
CP0873699
|
(R)-1-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-N,N-dimethylazetidine-3-carboxamide
Show/Hide
|
C27H29N5O3
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0873700
|
(R)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)morpholine-4-carboxamide
Show/Hide
|
C26H27N5O4
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0875568
|
(R)-2-isopropoxy-5-(3-(1-(2-oxo-2-(pyrrolidin-1-yl)ethylamino)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)benzonitrile
Show/Hide
|
C27H29N5O3
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0875571
|
(R)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-3-hydroxypropane-1-sulfonamide
Show/Hide
|
C24H26N4O5S
|
1
|
| 1 |
EC50 < 0.05 nM
|
|
|
|
CP0875580
|
(S)-2-((4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)(methyl)amino)acetic acid
Show/Hide
|
C24H24N4O4
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0875581
|
(S)-5-(3-(1-((2-hydroxyethyl)(methyl)amino)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)-2-isopropoxybenzonitrile
Show/Hide
|
C24H26N4O3
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0883362
|
(R)-5-(3-(1-(bis(2-hydroxyethyl)amino)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)-2-isopropoxybenzonitrile
Show/Hide
|
C25H28N4O4
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0883363
|
(S)-5-(3-(1-(2,2-difluoroethylamino)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)-2-isopropoxybenzonitrile
Show/Hide
|
C23H22F2N4O2
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0883364
|
(R)-2-isopropoxy-5-(3-(1-(methylamino)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)benzonitrile
Show/Hide
|
C22H22N4O2
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0883365
|
(S)-2-isopropoxy-5-(3-(1-(propylamino)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)benzonitrile
Show/Hide
|
C24H26N4O2
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0883366
|
(S)-5-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-ylamino)pentanoic acid
Show/Hide
|
C26H28N4O4
|
1
|
| 1 |
EC50 < 0.05 nM
|
|
|
|
CP0883369
|
(S)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-4-(hydroxymethyl)piperidine-1-carboxamide
Show/Hide
|
C28H31N5O4
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0906137
|
(R)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-2-(3-hydroxyazetidin-1-yl)-2-oxoethanesulfonamide
Show/Hide
|
C26H27N5O6S
|
1
|
| 1 |
EC50 < 0.05 nM
|
|
|
|
CP0906138
|
(S)-1-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-N-methylazetidine-3-carboxamide
Show/Hide
|
C26H27N5O3
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0906139
|
(S)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)piperazine-1-carboxamide
Show/Hide
|
C26H28N6O3
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0906142
|
(S)-methyl 2-(1-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-ylcarbamoyl)piperidin-4-yl)acetate
Show/Hide
|
C30H33N5O5
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0906143
|
(R)-N-((R)-4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-3-hydroxypyrrolidine-1-carboxamide
Show/Hide
|
C26H27N5O4
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0906144
|
(R)-methyl 1-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-ylcarbamoyl)piperidine-4-carboxylate
Show/Hide
|
C29H31N5O5
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0906146
|
(S)-1-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)guanidine
Show/Hide
|
C22H22N6O2
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0906173
|
(R)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)cyclopropanesulfonamide
Show/Hide
|
C24H24N4O4S
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0906174
|
(S)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)cyclopropanesulfonamide
Show/Hide
|
C24H24N4O4S
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0906179
|
(S)-methyl 3-(N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)sulfamoyl)propanoate
Show/Hide
|
C25H26N4O6S
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0906183
|
5-(3-(1-((R)-2,3-dihydroxypropylamino)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)-2-isopropoxybenzonitrile
Show/Hide
|
C24H26N4O4
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0906185
|
(R)-4-(5-(3,4-diethoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-ol
Show/Hide
|
C21H22N2O4
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0906186
|
(R)-2-amino-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)acetamide
Show/Hide
|
C23H23N5O3
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0906188
|
(R)-5-(3-(1-(3-hydroxyazetidin-1-yl)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazo1-5-yl)-2-isopropoxybenzonitrile
Show/Hide
|
C24H24N4O3
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0906196
|
5-(3-((R)-1-(2-((S)-3-hydroxypyrrolidin-1-yl)-2-oxoethylamino)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)-2-isopropoxybenzonitrile
Show/Hide
|
C27H29N5O4
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0906198
|
(S)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-2-(dimethylamino)acetamide
Show/Hide
|
C25H27N5O3
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0919536
|
(R)-3-((4-(5-(3-cyano-4-isopropoxyphenyl)-l,2,4-oxadiazo1-3-yl)-2,3-dihydro-1H-inden-1-yl)amino)propanoic acid
Show/Hide
|
C24H24N4O4
|
1
|
| 1 |
EC50 < 0.05 nM
|
|
|
|
CP0919537
|
(S)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-2-(methylamino)ethanesulfonamide
Show/Hide
|
C24H27N5O4S
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0919540
|
(S)-2-(azetidin-1-yl)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-2-oxoethanesulfonamide
Show/Hide
|
C26H27N5O5S
|
1
|
| 1 |
EC50 < 0.05 nM
|
|
|
|
CP0919542
|
(R)-N-((S)-4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-3-hydroxypyrrolidine-1-carboxamide
Show/Hide
|
C26H27N5O4
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0919543
|
(S)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-4-hydroxypiperidine-1-carboxamide
Show/Hide
|
C27H29N5O4
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0933050
|
(R)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-2-ethoxyethanesulfonamide
Show/Hide
|
C25H28N4O5S
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0933052
|
(S)-2-(N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)sulfamoyl)-N-methylacetamide
Show/Hide
|
C24H25N5O5S
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0933055
|
(R)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-l,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)sulfamide
Show/Hide
|
C21H21N5O4S
|
1
|
| 1 |
EC50 < 0.05 nM
|
|
|
|
CP0933078
|
(S)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-2-hydroxy-N-methylacetamide
Show/Hide
|
C24H24N4O4
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0946700
|
(S)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-2-hydroxyacetamide
Show/Hide
|
C23H22N4O4
|
1
|
| 1 |
EC50 < 0.05 nM
|
|
|
|
CP0946701
|
(S)-methyl 4-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-ylamino)butanoate
Show/Hide
|
C26H28N4O4
|
1
|
| 1 |
EC50 < 0.05 nM
|
|
|
|
CP0946703
|
(S)-2-hydroxyethyl 4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-ylcarbamate
Show/Hide
|
C24H24N4O5
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0946716
|
rac-methyl 3-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-ylamino)propanoate
Show/Hide
|
C25H26N4O4
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0946717
|
N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-2-methoxyacetamide
Show/Hide
|
C24H24N4O4
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0946719
|
5-(3-(1-((1,3-dihydroxypropan-2-yl)amino)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)-2-iso-propoxybenzonitrile
Show/Hide
|
C23H24N4O4
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0946723
|
(S)-5-(3-(1-(ethylamino)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)-2-isopropoxybenzonitrile
Show/Hide
|
C23H24N4O2
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0946725
|
(R)-5-(3-(1-(ethyl(2-hydroxyethyl)amino)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)-2-isopropoxybenzonitrile
Show/Hide
|
C25H28N4O3
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0946727
|
(S)-3-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-1,1-dimethylurea
Show/Hide
|
C24H25N5O3
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0946728
|
(R)-2-isopropoxy-5-(3-(1-((2-(methylsulfonyl)ethyl)amino)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)benzonitrile
Show/Hide
|
C24H26N4O4S
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0946730
|
(R)-2-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-ylamino)-N-(2-hydroxyethyl)acetamide
Show/Hide
|
C25H27N5O4
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0946731
|
(S)-2-isopropoxy-5-(3-(1-(thiazol-5-ylmethylamino)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)benzonitrile
Show/Hide
|
C25H23N5O2S
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0946732
|
(S)-2-(N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)sulfamoyl)acetamide
Show/Hide
|
C23H23N5O5S
|
1
|
| 1 |
EC50 < 0.05 nM
|
|
|
|
CP0947296
|
(S)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)acetamide
Show/Hide
|
C23H22N4O3
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0947297
|
(R)-methyl(4-(5-(3-cyano-4-isopropoxyphenyl)-l,2,4-oxadiazol-3-y1)-2,3-dihydro-1H-inden-1-yl)carbamate
Show/Hide
|
C23H22N4O4
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0947298
|
(S)-methyl 4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-ylcarbamate
Show/Hide
|
C23H22N4O4
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0947299
|
(R)-2-isopropoxy-5-(3-(1-(2-oxooxazolidin-3-yl)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)benzonitrile
Show/Hide
|
C24H22N4O4
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0947300
|
(S)-2-isopropoxy-5-(3-(1-(2-oxooxazolidin-3-yl)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)benzonitrile
Show/Hide
|
C24H22N4O4
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0947301
|
(R)-2-(azetidin-1-yl)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-2-oxoethanesulfonamide
Show/Hide
|
C26H27N5O5S
|
1
|
| 1 |
EC50 < 0.05 nM
|
|
|
|
CP0947302
|
(S)-methyl 1-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-ylcarbamoyl)piperidine-4-carboxylate
Show/Hide
|
C29H31N5O5
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0947303
|
(S)-1-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-ylcarbamoyl)piperidine-4-carboxylic acid
Show/Hide
|
C28H29N5O5
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0949438
|
2-isopropoxy-5-(3-(1-(2-(methylsulfonyl)ethylamino)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)benzonitrile
Show/Hide
|
C24H26N4O4S
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0949439
|
2-((4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)amino)-N-methylethanesulfonamide
Show/Hide
|
C24H27N5O4S
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0949440
|
5-(3-((S)-1-(((R)-1-hydroxypropan-2-yl)amino)-2,3-dihydro-1H-inden-4-yl)-l,2,4-oxadiazo1-5-yl)-2-isopropoxybenzonitrile
Show/Hide
|
C24H26N4O3
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0949762
|
(S)-4-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-ylamino)butanoic acid
Show/Hide
|
C25H26N4O4
|
1
|
| 1 |
EC50 < 0.05 nM
|
|
|
|
CP0949766
|
5-(3-(1-((S)-2,3-dihydroxypropylamino)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)-2-isopropoxybenzonitrile
Show/Hide
|
C24H26N4O4
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0949767
|
5-(3-(1-((S)-2-hydroxypropylamino)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)-2-isopropoxybenzonitrile
Show/Hide
|
C24H26N4O3
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0949776
|
(R)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-2-morpholino-2-oxoethanesulfonamide
Show/Hide
|
C27H29N5O6S
|
1
|
| 1 |
EC50 < 0.05 nM
|
|
|
|
CP0949777
|
(R)-2-(N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)sulfamoyl)-N-methylacetamide
Show/Hide
|
C24H25N5O5S
|
1
|
| 1 |
EC50 < 0.05 nM
|
|
|
|
CP0950215
|
(S)-2-(N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)sulfamoyl)-N,N-dimethylacetamide
Show/Hide
|
C25H27N5O5S
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0950217
|
(R)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-2-(dimethylamino)acetamide
Show/Hide
|
C25H27N5O3
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0955060
|
2-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-ylamino)ethyl acetate
Show/Hide
|
C25H26N4O4
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0955065
|
(R)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-l,2,4-oxadiazo1-3-yl)-2,3-dihydro-1H-inden-1-yl)-2-hydroxyacetamide
Show/Hide
|
C23H22N4O4
|
1
|
| 1 |
EC50 < 0.05 nM
|
|
|
|
CP0955067
|
(S)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazo1-3-yl)-2,3-dihydro-1H-inden-1-yl)methanesulfonamide
Show/Hide
|
C22H22N4O4S
|
1
|
| 1 |
EC50 < 0.05 nM
|
|
|
|
CP0958194
|
(R)-2-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-ylamino)acetic acid
Show/Hide
|
C23H22N4O4
|
1
|
| 1 |
EC50 < 0.05 nM
|
|
|
|
CP0958195
|
(S)-5-(3-(1-(3-hydroxyazetidin-1-yl)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)-2-isopropoxybenzonitrile
Show/Hide
|
C24H24N4O3
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0958197
|
(S)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-2-morpholino-2-oxoethanesulfonamide
Show/Hide
|
C27H29N5O6S
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0958198
|
(S)-1-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)azetidine-3-carboxylic acid
Show/Hide
|
C25H24N4O4
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0961368
|
(S)-2-(N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)sulfamoyl)acetic acid
Show/Hide
|
C23H22N4O6S
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0963597
|
(R)-2-(N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)sulfamoyl)acetamide
Show/Hide
|
C23H23N5O5S
|
1
|
| 1 |
EC50 < 0.05 nM
|
|
|
|
CP0963598
|
(R)-1-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)azetidine-3-carboxylic acid
Show/Hide
|
C25H24N4O4
|
1
|
| 1 |
EC50 < 0.05 nM
|
|
|
|
CP0964204
|
methyl 5-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-ylamino)pentanoate
Show/Hide
|
C27H30N4O4
|
1
|
| 1 |
EC50 < 0.05 nM
|
|
|
|
CP0964206
|
N-((R)-4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-2-((R)-3-hydroxypyrrolidin-1-yl)ethanesulfonamide
Show/Hide
|
C27H31N5O5S
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0964207
|
(R)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-2-(3-hydroxyazetidin-1-yl)ethanesulfonamide
Show/Hide
|
C26H29N5O5S
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0966078
|
(S)-4-(5-(3,4-diethoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-ol
Show/Hide
|
C21H22N2O4
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0966079
|
(S)-2-((R)-4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-ylamino)propanoic acid
Show/Hide
|
C24H24N4O4
|
1
|
| 1 |
EC50 < 0.05 nM
|
|
|
|
CP0966080
|
(S)-2-isopropoxy-5-(3-(1-(2-methoxyethylamino)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)benzonitrile
Show/Hide
|
C24H26N4O3
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0966082
|
(S)-2-isopropoxy-5-(3-(1-(2-(methylsulfonyl)ethylamino)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)benzonitrile
Show/Hide
|
C24H26N4O4S
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0966787
|
N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-2-ethoxyacetamide
Show/Hide
|
C25H26N4O4
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0966789
|
(R)-2-isopropoxy-5-(3-(1-(2-morpholino-2-oxoethylamino)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)benzonitrile
Show/Hide
|
C27H29N5O4
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0966790
|
(S)-2-ethoxy-5-(3-(1-hydroxy-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)benzonitrile
Show/Hide
|
C20H17N3O3
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0967385
|
1-(4-(5-(3-cyano-4-isopropoxyphenyl)-l,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)azetidine-3-carboxylic acid
Show/Hide
|
C25H24N4O4
|
1
|
| 1 |
EC50 < 0.05 nM
|
|
|
|
CP0967388
|
(R)-5-(3-(1-(2-(azetidin-1-yl)-2-oxoethylamino)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)-2-isopropoxybenzonitrile
Show/Hide
|
C26H27N5O3
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
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CP0967392
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5-(3-cyano-4-isopropoxy-phenyl)-3-[(1S)-1-(sulfamoylamino)indan-4-yl]-1,2,4-oxadiazole
Show/Hide
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C21H21N5O4S
|
1
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| 1 |
EC50 < 0.05 nM
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CP0967394
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(S)-N-((S)-4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-3-hydroxypiperidine-1-carboxamide
Show/Hide
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C27H29N5O4
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1
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| 1 |
EC50 = 0.05 nM
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|
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CP0906147
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(S)-2-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazo1-3-yl)-2,3-dihydro-1H-inden-1-ylamino)-N,N-dimethylacetamide
Show/Hide
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C25H27N5O3
|
1
|
| 1 |
EC50 = 0.09 nM
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CP0906148
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(R)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-2-meth-oxyethanesulfonamide
Show/Hide
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C24H26N4O5S
|
1
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| 1 |
EC50 = 0.09 nM
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CP0848223
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(S)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-3-hydroxyazetidine-1-carboxamide
Show/Hide
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C25H25N5O4
|
1
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| 1 |
EC50 = 0.1 nM
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CP0861106
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(S)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-2-hydroxyethanesulfonamide
Show/Hide
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C23H24N4O5S
|
1
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| 1 |
EC50 = 0.1 nM
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CP0873702
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(R)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-l,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-3-hydroxyazetidine-1-carboxamide
Show/Hide
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C25H25N5O4
|
1
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| 1 |
EC50 = 0.1 nM
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CP0848219
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(R)-2-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazo1-3-yl)-2,3-dihydro-1H-inden-1-ylamino)-N,N-dimethylacetamide hydrochloride
Show/Hide
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C25H28ClN5O3
|
1
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| 1 |
EC50 = 0.13 nM
|
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CP0248629
|
Ozanimod
Show/Hide
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C23H24N4O3
|
1
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| 1 |
EC50 = 0.16 nM
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CP0861107
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(+/-)-4-(5-(3,4,diethoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-ol
Show/Hide
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C21H22N2O4
|
1
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| 1 |
EC50 = 0.16 nM
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CP0883372
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(R)-5-(3-(1-(2-hydroxyethylamino)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazo1-5-yl)-2-isopropoxybenzonitrile
Show/Hide
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C23H24N4O3
|
1
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| 1 |
EC50 = 0.16 nM
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CP0883375
|
(R)-5-(3-(1-amino-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)-2-isopropoxy-benzonitrile hydrochloride
Show/Hide
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C21H21ClN4O2
|
1
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| 1 |
EC50 = 0.17 nM
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CP0871098
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(S)-5-(3-(1-amino-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)-2-isopropoxybenzonitrile
Show/Hide
|
C21H20N4O2
|
1
|
| 1 |
EC50 = 0.19 nM
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|
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CP0845581
|
(S)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-2-methoxyethanesulfonamide
Show/Hide
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C24H26N4O5S
|
1
|
| 1 |
EC50 = 0.36 nM
|
|
|
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CP0845572
|
N-((S)-4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-2-((S)-3-hydroxypyrrolidin-1-yl)ethanesulfonamide
Show/Hide
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C27H31N5O5S
|
1
|
| 1 |
EC50 = 0.5 nM
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|
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CP0845576
|
(S)-5-(3-(1-(dimethylamino)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)-2-isopropoxybenzonitrile
Show/Hide
|
C23H24N4O2
|
1
|
| 1 |
EC50 = 0.5 nM
|
|
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CP0848218
|
(R)-2-isopropoxy-5-(3-(1-(2-methoxyethylamino)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)benzonitrile
Show/Hide
|
C24H26N4O3
|
1
|
| 1 |
EC50 = 0.5 nM
|
|
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CP0848221
|
(S)-5-(3-(1-(benzylamino)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)-2-isopropoxybenzonitrile
Show/Hide
|
C28H26N4O2
|
1
|
| 1 |
EC50 = 0.5 nM
|
|
|
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CP0848224
|
(R)-2-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-ylamino)-N,N-diethylacetamide
Show/Hide
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C27H31N5O3
|
1
|
| 1 |
EC50 = 0.5 nM
|
|
|
|
CP0852163
|
(S)-5-(3-(1-(((1H-imidazol-2-yl)methyl)amino)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)-2-isobutoxybenzonitrile
Show/Hide
|
C25H24N6O2
|
1
|
| 1 |
EC50 = 0.5 nM
|
|
|
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CP0852164
|
N-((R)-4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-2-((S)-3-hydroxypyrrolidin-1-yl)ethanesulfonamide
Show/Hide
|
C27H31N5O5S
|
1
|
| 1 |
EC50 = 0.5 nM
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|
|
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CP0861103
|
(S)-3-amino-N-((R)-4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)pyrrolidine-1-carboxamide
Show/Hide
|
C26H28N6O3
|
1
|
| 1 |
EC50 = 0.5 nM
|
|
|
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CP0861104
|
(R)-methyl 2-(1-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-ylcarbamoyl)piperidin-4-yl)acetate
Show/Hide
|
C30H33N5O5
|
1
|
| 1 |
EC50 = 0.5 nM
|
|
|
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CP0864434
|
2-isopropoxy-5-(3-((S)-1-(((2R,3S,4R)-2,3,4,5-tetrahydroxypentyl)amino)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)benzonitrile
Show/Hide
|
C26H30N4O6
|
1
|
| 1 |
EC50 = 0.5 nM
|
|
|
|
CP0864435
|
(R)-2-isopropoxy-5-(3-(1-(2-oxo-2-(piperidin-1-yl)ethylamino)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)benzonitrile
Show/Hide
|
C28H31N5O3
|
1
|
| 1 |
EC50 = 0.5 nM
|
|
|
|
CP0864436
|
(S)-2-isopropoxy-5-(3-(1-((4-methyl-1H-imidazol-2-yl)methylamino)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)benzonitrile
Show/Hide
|
C26H26N6O2
|
1
|
| 1 |
EC50 = 0.5 nM
|
|
|
|
CP0864438
|
(S)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)methane sulfonamide
Show/Hide
|
C28H29N5O3
|
1
|
| 1 |
EC50 = 0.5 nM
|
|
|
|
CP0864441
|
(S)-3-amino-N-((S)-4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)pyrrolidine-1-carboxamide
Show/Hide
|
C26H28N6O3
|
1
|
| 1 |
EC50 = 0.5 nM
|
|
|
|
CP0869392
|
(R)-4-(5-(4-ethoxy-3-(trifluoromethyl)phenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-ol
Show/Hide
|
C20H17F3N2O3
|
1
|
| 1 |
EC50 = 0.5 nM
|
|
|
|
CP0873077
|
(R)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-N-(2-hydroxyethyl)acetamide
Show/Hide
|
C25H26N4O4
|
1
|
| 1 |
EC50 = 0.5 nM
|
|
|
|
CP0873078
|
(R)-2-((4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)(methyl)amino)-N,N-dimethylacetamide
Show/Hide
|
C26H29N5O3
|
1
|
| 1 |
EC50 = 0.5 nM
|
|
|
|
CP0873082
|
(S)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-2-morpholinoethanesulfonamide
Show/Hide
|
C27H31N5O5S
|
1
|
| 1 |
EC50 = 0.5 nM
|
|
|
|
CP0873119
|
5-(3-(1-((1-hydroxy-2-methylpropan-2-yl)amino)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)-2-isopropoxybenzonitrile
Show/Hide
|
C25H28N4O3
|
1
|
| 1 |
EC50 = 0.5 nM
|
|
|
|
CP0873128
|
2-isopropoxy-5-(3-(1-(2-morpholinoethylamino)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)benzonitrile
Show/Hide
|
C27H31N5O3
|
1
|
| 1 |
EC50 = 0.5 nM
|
|
|
|
CP0873130
|
(R)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-2-(methylamino)ethanesulfonamide
Show/Hide
|
C24H27N5O4S
|
1
|
| 1 |
EC50 = 0.5 nM
|
|
|
|
CP0873132
|
5-(3-(1-((2-hydroxyethyl)amino)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)-2-isobutoxybenzonitrile
Show/Hide
|
C24H26N4O3
|
1
|
| 1 |
EC50 = 0.5 nM
|
|
|
|
CP0873147
|
(R)-5-(3-(1-(2-hydroxy-2-methylpropylamino)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)-2-isopropoxybenzonitrile
Show/Hide
|
C25H28N4O3
|
1
|
| 1 |
EC50 = 0.5 nM
|
|
|
|
CP0873688
|
2-isopropoxy-5-(3-(1-(2-(pyrrolidin-1-yl)ethylamino)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)benzonitrile
Show/Hide
|
C27H31N5O2
|
1
|
| 1 |
EC50 = 0.5 nM
|
|
|
|
CP0873689
|
5-(3-(1-((R)-3-hydroxypyrrolidin-1-yl)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)-2-isopropoxybenzonitrile
Show/Hide
|
C25H26N4O3
|
1
|
| 1 |
EC50 = 0.5 nM
|
|
|
|
CP0873692
|
(R)-4-(5-(4-isopropoxy-3-(trifluoromethyl)phenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-ol
Show/Hide
|
C21H19F3N2O3
|
1
|
| 1 |
EC50 = 0.5 nM
|
|
|
|
CP0873696
|
(R)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-2-(pyrrolidin-1-yl)ethanesulfonamide
Show/Hide
|
C27H31N5O4S
|
1
|
| 1 |
EC50 = 0.5 nM
|
|
|
|
CP0873697
|
N-((S)-4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-2-((R)-3-hydroxypyrrolidin-1-yl)ethanesulfonamide
Show/Hide
|
C27H31N5O5S
|
1
|
| 1 |
EC50 = 0.5 nM
|
|
|
|
CP0875570
|
(R)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-2-(piperidin-1-yl)ethanesulfonamide
Show/Hide
|
C28H33N5O4S
|
1
|
| 1 |
EC50 = 0.5 nM
|
|
|
|
CP0883356
|
5-(3-(1-(2-(diethylamino)ethylamino)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)-2-isopropoxybenzonitrile
Show/Hide
|
C27H33N5O2
|
1
|
| 1 |
EC50 = 0.5 nM
|
|
|
|
CP0883361
|
(R)-5-(3-(1-amino-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-y1)-2-(cyclopropylmethoxy)benzonitrile
Show/Hide
|
C22H20N4O2
|
1
|
| 1 |
EC50 = 0.5 nM
|
|
|
|
CP0883367
|
(R)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)piperazine-1-carboxamide
Show/Hide
|
C26H28N6O3
|
1
|
| 1 |
EC50 = 0.5 nM
|
|
|
|
CP0906140
|
(R)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-4-(hydroxymethyl)piperidine-1-carboxamide
Show/Hide
|
C28H31N5O4
|
1
|
| 1 |
EC50 = 0.5 nM
|
|
|
|
CP0906141
|
(R)-3-amino-N-((S)-4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)pyrrolidine-1-carboxamide
Show/Hide
|
C26H28N6O3
|
1
|
| 1 |
EC50 = 0.5 nM
|
|
|
|
CP0906145
|
(R)-N-((S)-4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-3-(dimethylamino)pyrrolidine-1-carboxamide
Show/Hide
|
C28H32N6O3
|
1
|
| 1 |
EC50 = 0.5 nM
|
|
|
|
CP0906176
|
(S)-2-(azetidin-1-yl)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)ethanesulfonamide
Show/Hide
|
C26H29N5O4S
|
1
|
| 1 |
EC50 = 0.5 nM
|
|
|
|
CP0906177
|
(R)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-2-(4-hydroxypiperidin-1-yl)ethanesulfonamide
Show/Hide
|
C28H33N5O5S
|
1
|
| 1 |
EC50 = 0.5 nM
|
|
|
|
CP0906178
|
(R)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-2-(piperazin-1-yl)ethanesulfonamide
Show/Hide
|
C27H32N6O4S
|
1
|
| 1 |
EC50 = 0.5 nM
|
|
|
|
CP0919539
|
(S)-2-isopropoxy-5-(3-(1-((3-methyl-1H-pyrazol-5-yl)methylamino)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)benzonitrile
Show/Hide
|
C26H26N6O2
|
1
|
| 1 |
EC50 = 0.5 nM
|
|
|
|
CP0919541
|
(R)-N-((R)-4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-3-hydroxypiperidine-1-carboxamide
Show/Hide
|
C27H29N5O4
|
1
|
| 1 |
EC50 = 0.5 nM
|
|
|
|
CP0930893
|
2-isopropoxy-5-(3-(1-morpholino-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)benzonitrile
Show/Hide
|
C25H26N4O3
|
1
|
| 1 |
EC50 = 0.5 nM
|
|
|
|
CP0933051
|
(S)-methyl 3-(N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)sulfamoyl)-2,2-dimethylpropanoate
Show/Hide
|
C27H30N4O6S
|
1
|
| 1 |
EC50 = 0.5 nM
|
|
|
|
CP0933053
|
(S)-N-((R)-4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-3-(dimethylamino)pyrrolidine-1-carboxamide
Show/Hide
|
C28H32N6O3
|
1
|
| 1 |
EC50 = 0.5 nM
|
|
|
|
CP0933061
|
2-isopropoxy-5-(3-(1-(2-(methylamino)ethylamino)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)benzonitrile
Show/Hide
|
C24H27N5O2
|
1
|
| 1 |
EC50 = 0.5 nM
|
|
|
|
CP0933071
|
(S)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazo1-3-yl)-2,3-dihydro-1H-inden-1-yl)-2-(dimethylamino)ethanesulfonamide
Show/Hide
|
C25H29N5O4S
|
1
|
| 1 |
EC50 = 0.5 nM
|
|
|
|
CP0933072
|
(R)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)benzenesulfonamide
Show/Hide
|
C27H24N4O4S
|
1
|
| 1 |
EC50 = 0.5 nM
|
|
|
|
CP0933073
|
(R)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-1-phenylmethanesulfonamide
Show/Hide
|
C28H26N4O4S
|
1
|
| 1 |
EC50 = 0.5 nM
|
|
|
|
CP0933079
|
(R)-5-(3-(1-((2-hydroxyethyl)(methyl)amino)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)-2-isopropoxybenzonitrile
Show/Hide
|
C24H26N4O3
|
1
|
| 1 |
EC50 = 0.5 nM
|
|
|
|
CP0946702
|
(R)-ethyl 4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-ylcarbamate
Show/Hide
|
C24H24N4O4
|
1
|
| 1 |
EC50 = 0.5 nM
|
|
|
|
CP0946704
|
(S)-5-(3-(1-((1H-benzo[d]imidazol-2-yl)methylamino)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)-2-isopropoxybenzonitrile
Show/Hide
|
C29H26N6O2
|
1
|
| 1 |
EC50 = 0.5 nM
|
|
|
|
CP0946715
|
5-(3-(1-((S)-3-hydroxypyrrolidin-1-yl)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)-2-isopropoxybenzonitrile
Show/Hide
|
C25H26N4O3
|
1
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| 1 |
EC50 = 0.5 nM
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CP0946718
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(R)-4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl acetate
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C23H21N3O4
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1
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| 1 |
EC50 = 0.5 nM
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CP0946720
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(S)-2-isopropoxy-5-(3-(1-(isopropylamino)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)benzonitrile
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C24H26N4O2
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1
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| 1 |
EC50 = 0.5 nM
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CP0946722
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(R)-2-(4-(5-(3-bromo-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-ylamino)ethanol
Show/Hide
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C22H24BrN3O3
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1
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| 1 |
EC50 = 0.5 nM
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CP0946724
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(R)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-N-(2-hydroxyethyl)methanesulfonamide
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C24H26N4O5S
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1
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| 1 |
EC50 = 0.5 nM
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CP0946729
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(R)-5-(3-(1-(2-(aziridin-1-yl)-2-oxoethylamino)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)-2-isopropoxybenzonitrile
Show/Hide
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C25H25N5O3
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1
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| 1 |
EC50 = 0.5 nM
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CP0949768
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(S)-4-(5-(4-ethoxy-3-nitrophenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-ol
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C19H17N3O5
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1
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| 1 |
EC50 = 0.5 nM
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CP0949769
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2-isopropoxy-5-(3-(1-(tetrahydro-2H-pyran-4-ylamino)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)benzonitrile
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C26H28N4O3
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1
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| 1 |
EC50 = 0.5 nM
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CP0949778
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(R)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-4-hydroxypiperidine-1-carboxamide
Show/Hide
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C27H29N5O4
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1
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| 1 |
EC50 = 0.5 nM
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CP0949779
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(S)-N-((S)-4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-3-(dimethylamino)pyrrolidine-1-carboxamide
Show/Hide
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C28H32N6O3
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1
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| 1 |
EC50 = 0.5 nM
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CP0949780
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(S)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-4-(dimethylamino)piperidine-1-carboxamide
Show/Hide
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C29H34N6O3
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1
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| 1 |
EC50 = 0.5 nM
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CP0949830
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(R)-4-(5-(4-isopropoxy-3-(methylsulfonyl)phenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-amine
Show/Hide
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C21H23N3O4S
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1
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| 1 |
EC50 = 0.5 nM
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CP0955061
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5-(3-((S)-1-(((S)-1-hydroxypropan-2-yl)amino)-2,3-dihydro-1H-inden-4-yl)-l,2,4-oxadiazo1-5-yl)-2-isopropoxybenzonitrile
Show/Hide
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C24H26N4O3
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1
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| 1 |
EC50 = 0.5 nM
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CP0955063
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(R)-4-(5-(4-ethoxy-3-nitrophenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-ol
Show/Hide
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C19H17N3O5
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1
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| 1 |
EC50 = 0.5 nM
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CP0955066
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(R)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-2-(pyrrolidin-1-yl)acetamide
Show/Hide
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C27H29N5O3
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1
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| 1 |
EC50 = 0.5 nM
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CP0955068
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(S)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)ethanesulfonamide
Show/Hide
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C23H24N4O4S
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1
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| 1 |
EC50 = 0.5 nM
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CP0955069
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(R)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-2-methylpropane-1-sulfonamide
Show/Hide
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C25H28N4O4S
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1
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| 1 |
EC50 = 0.5 nM
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CP0955070
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(R)-5-(3-(1-amino-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)-2-ethoxybenzonitrile
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C20H18N4O2
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1
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| 1 |
EC50 = 0.5 nM
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CP0955071
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(R)-2-((4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)(ethyl)amino)-N,N-dimethylacetamide
Show/Hide
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C27H31N5O3
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1
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| 1 |
EC50 = 0.5 nM
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CP0955072
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(R)-2-isopropoxy-5-(3-(1-(2-(4-methylpiperazin-1-yl)-2-oxoethylamino)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)benzonitrile
Show/Hide
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C28H32N6O3
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1
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| 1 |
EC50 = 0.5 nM
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CP0955074
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(R)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-2-morpholinoethanesulfonamide
Show/Hide
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C27H31N5O5S
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1
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| 1 |
EC50 = 0.5 nM
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CP0958205
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(R)-5-(3-(1-(2,2-difluoroethylamino)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)-2-isopropoxybenzonitrile
Show/Hide
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C23H22F2N4O2
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1
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| 1 |
EC50 = 0.5 nM
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CP0962595
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(S)-N-((R)-4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-3-hydroxypiperidine-1-carboxamide
Show/Hide
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C27H29N5O4
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1
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| 1 |
EC50 = 0.5 nM
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CP0964205
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(R)-5-(3-(1-(benzylamino)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)-2-isopropoxybenzonitrile
Show/Hide
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C28H26N4O2
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1
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| 1 |
EC50 = 0.5 nM
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CP0964210
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5-(3-(1-((R)-2-hydroxypropylamino)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)-2-isopropoxybenzonitrile
Show/Hide
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C24H26N4O3
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1
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| 1 |
EC50 = 0.5 nM
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CP0966786
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5-(3-(1-((S)-3-aminopyrrolidin-1-yl)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)-2-isopropoxybenzonitrile
Show/Hide
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C25H27N5O2
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1
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| 1 |
EC50 = 0.5 nM
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CP0966788
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2-((R)-4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-ylamino)-N,N-dimethylpropanamide
Show/Hide
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C26H29N5O3
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1
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| 1 |
EC50 = 0.5 nM
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CP0967389
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(S)-ethyl 4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-ylcarbamate
Show/Hide
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C24H24N4O4
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1
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| 1 |
EC50 = 0.5 nM
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CP0967390
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(R)-2-(1-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-ylcarbamoyl)piperidin-4-yl)acetic acid
Show/Hide
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C29H31N5O5
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1
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| 1 |
EC50 = 0.5 nM
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CP0967391
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(R)-N-((R)-4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-3-(dimethylamino)pyrrolidine-1-carboxamide
Show/Hide
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C28H32N6O3
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1
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| 1 |
EC50 = 0.5 nM
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CP0871095
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(+/-)-2-((4-(5-(3,4,diethoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)amino)ethanol
Show/Hide
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C23H27N3O4
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1
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| 1 |
EC50 = 2.88 nM
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CP0848220
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2-hydroxy-5-(3-(1-((2-hydroxyethyl)amino)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)benzonitrile
Show/Hide
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C20H18N4O3
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1
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| 1 |
EC50 > 5 nM
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CP0861113
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(R)-4-(N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)sulfamoyl)benzoic acid
Show/Hide
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C28H24N4O6S
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1
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| 1 |
EC50 > 5 nM
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CP0864456
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2-isopropoxy-5-(3-(1-(piperidin-1-yl)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)benzonitrile
Show/Hide
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C26H28N4O2
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1
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| 1 |
EC50 > 5 nM
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CP0869394
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(R)-4-(5-(3-chloro-4-isopropoxyphenyl)-1,2,4-oxadiazo1-3-yl)-2,3-dihydro-1H-inden-1-amine
Show/Hide
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C20H20ClN3O2
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1
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| 1 |
EC50 > 5 nM
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CP0869395
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2-isopropoxy-5-(3-((S)-1-((S)-1-phenylethylamino)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)benzonitrile
Show/Hide
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C29H28N4O2
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1
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| 1 |
EC50 > 5 nM
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CP0873129
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2-isopropoxy-5-(3-(1-(2-(piperidin-1-yl)ethylamino)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)benzonitrile
Show/Hide
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C28H33N5O2
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1
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| 1 |
EC50 > 5 nM
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CP0873131
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(R)-3-(3-(1-amino-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazo1-5-yl)-5-(trifluoromethoxy)benzonitrile
Show/Hide
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C19H13F3N4O2
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1
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| 1 |
EC50 > 5 nM
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CP0873693
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rac-5-(3-(1-(2-hydroxyethylamino)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)-2-(2-methoxyethoxy)benzonitrile
Show/Hide
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C23H24N4O4
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1
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| 1 |
EC50 > 5 nM
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CP0873694
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2-(2-cyano-4-(3-(1-(2-hydroxyethylamino)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)phenoxy)acetic acid
Show/Hide
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C22H20N4O5
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1
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| 1 |
EC50 > 5 nM
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CP0875569
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(R)-2-isopropoxy-5-(3-(1-(2-oxo-2-(piperazin-1-yl)ethylamino)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)benzonitrile
Show/Hide
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C27H30N6O3
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1
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| 1 |
EC50 > 5 nM
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CP0883357
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2-isopropoxy-5-(3-(1-(piperidin-4-ylamino)-2,3-dihydro-4H-inden-4-yl)-1,2,4-oxadiazol-5-yl)benzonitrile
Show/Hide
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C26H29N5O2
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1
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| 1 |
EC50 > 5 nM
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CP0906184
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(R)-4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl pivalate
Show/Hide
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C26H27N3O4
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1
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| 1 |
EC50 > 5 nM
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CP0906190
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(R)-4-(3-(1-amino-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)-2-isopropoxybenzonitri1e
Show/Hide
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C21H20N4O2
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1
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| 1 |
EC50 > 5 nM
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CP0906191
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2-cyano-4-(3-(1-(2-hydroxyethylamino)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)phenyl isobutyrate
Show/Hide
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C24H24N4O4
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1
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| 1 |
EC50 > 5 nM
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CP0906192
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(S)-5-(3-(1-(2-(dimethylamino)-2-oxoethylamino)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)-2-isopropoxybenzamide
Show/Hide
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C25H29N5O4
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1
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| 1 |
EC50 > 5 nM
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CP0906194
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(R)-4-bromo-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)benzamide
Show/Hide
|
C28H23BrN4O3
|
1
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| 1 |
EC50 > 5 nM
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CP0919538
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(R)-4-(5-(4-isopropoxyphenyl)-1,2,4-oxadiazo1-3-yl)-2,3-dihydro-1H-inden-1-amine
Show/Hide
|
C20H21N3O2
|
1
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| 1 |
EC50 > 5 nM
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CP0919544
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2-isopropoxy-5-(3-((R)-1-((R)-1-phenylethylamino)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)benzonitrile
Show/Hide
|
C29H28N4O2
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1
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| 1 |
EC50 > 5 nM
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CP0933054
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(R)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-4-(dimethylamino)piperidine-1-carboxamide
Show/Hide
|
C29H34N6O3
|
1
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| 1 |
EC50 > 5 nM
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CP0933074
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(R)-3-(3-(1-amino-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazo1-5-yl)benzonitrie
Show/Hide
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C18H14N4O
|
1
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| 1 |
EC50 > 5 nM
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CP0946721
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(R)-3-(3-(1-amino-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazo1-5-yl)-5-isopropoxybenzonitrile
Show/Hide
|
C21H20N4O2
|
1
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| 1 |
EC50 > 5 nM
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CP0946726
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(R)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)-N-(2-hydroxyethyl)benzenesulfonamide
Show/Hide
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C29H28N4O5S
|
1
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| 1 |
EC50 > 5 nM
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CP0947294
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(R)-N-(4-(N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)sulfamoyl)phenyl)acetamide
Show/Hide
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C29H27N5O5S
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1
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| 1 |
EC50 > 5 nM
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CP0955059
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2-isopropoxy-5-(3-(1-(2-(piperazin-1-yl)ethylamino)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)benzonitrile
Show/Hide
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C27H32N6O2
|
1
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| 1 |
EC50 > 5 nM
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CP0955064
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5-(3-(1-(cyclohexylamino)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)-2-isopropoxybenzonitrile
Show/Hide
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C27H30N4O2
|
1
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| 1 |
EC50 > 5 nM
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CP0958196
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2-((S)-2,3-dihydroxypropoxy)-5-(3-(1-(2-hydroxyethylamino)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)benzonitrile
Show/Hide
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C23H24N4O5
|
1
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| 1 |
EC50 > 5 nM
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CP0964209
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5-(3-(1-((R)-3-aminopyrrolidin-1-yl)-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)-2-isopropoxybenzonitrile
Show/Hide
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C25H27N5O2
|
1
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| 1 |
EC50 > 5 nM
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CP0967387
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(R)-3-(3-(1-amino-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)-4-isopropoxybenzonitrile
Show/Hide
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C21H20N4O2
|
1
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| 1 |
EC50 > 5 nM
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