| Compound ID |
Compound Name |
Compound Formula |
|
CP0227731
|
2-[3-cyclopropyl-5-ethyl-1-[[4-[[4-(trifluoromethyl)benzoyl]amino]phenyl]methyl]pyrazol-4-yl]acetic acid
Show/Hide
|
C25H24F3N3O3
|
1
|
| 1 |
Ki = 0.1 nM
|
|
|
|
CP0410550
|
US8791272, 2.50
Show/Hide
|
C25H24F3N3O3
|
1
|
| 1 |
Ki = 0.1 nM
|
|
|
|
CP0426616
|
US8791272, 3.9
Show/Hide
|
C24H25Cl2N3O4
|
1
|
| 1 |
Ki = 0.1 nM
|
|
|
|
CP0443055
|
US8791272, 17.1
Show/Hide
|
C25H26F3N3O3
|
1
|
| 1 |
Ki = 0.1 nM
|
|
|
|
CP0463988
|
US8791272, 3.12
Show/Hide
|
C28H29N3O4
|
1
|
| 1 |
Ki = 0.1 nM
|
|
|
|
CP0506869
|
US8791272, 2.42
Show/Hide
|
C29H31N3O3
|
1
|
| 1 |
Ki = 0.1 nM
|
|
|
|
CP0499877
|
US9206164, 19
Show/Hide
|
C27H26N4O2
|
1
|
| 1 |
Ki = 0.1 nM
|
|
|
|
CP0415259
|
US8791272, 2.41
Show/Hide
|
C26H28F3N3O3
|
1
|
| 1 |
Ki = 0.2 nM
|
|
|
|
CP0463973
|
US8791272, 2.53
Show/Hide
|
C23H22F3N3O3
|
1
|
| 1 |
Ki = 0.2 nM
|
|
|
|
CP0500375
|
US8791272, 2.40
Show/Hide
|
C25H27Cl2N3O3
|
1
|
| 1 |
Ki = 0.2 nM
|
|
|
|
CP0531854
|
US8791272, 2.14
Show/Hide
|
C27H27N3O3
|
1
|
| 1 |
Ki = 0.2 nM
|
|
|
|
CP0555325
|
US8791272, 1.15
Show/Hide
|
C25H29N3O3
|
1
|
| 1 |
Ki = 0.2 nM
|
|
|
|
CP0563977
|
US8791272, 2.1
Show/Hide
|
C24H24F3N3O3
|
1
|
| 1 |
Ki = 0.2 nM
|
|
|
|
CP0475771
|
US9206164, 20
Show/Hide
|
C24H23F3N4O2
|
1
|
| 1 |
Ki = 0.2 nM
|
|
|
|
CP0508931
|
US9206164, 68
Show/Hide
|
C27H32N4O2
|
1
|
| 1 |
Ki = 0.2 nM
|
|
|
|
CP0540939
|
US9206164, 16
Show/Hide
|
C23H22Cl2N4O2
|
1
|
| 1 |
Ki = 0.2 nM
|
|
|
|
CP0469786
|
US8791272, 2.6
Show/Hide
|
C23H23Cl2N3O3
|
1
|
| 1 |
Ki = 0.25 nM
|
|
|
|
CP0463987
|
US8791272, 3.3
Show/Hide
|
C24H27N3O4
|
1
|
| 1 |
Ki = 0.3 nM
|
|
|
|
CP0546817
|
US8791272, 7.5
Show/Hide
|
C26H25N3O3
|
1
|
| 1 |
Ki = 0.3 nM
|
|
|
|
CP0406816
|
US9206164, 106
Show/Hide
|
C24H24ClFN4O2
|
1
|
| 1 |
Ki = 0.3 nM
|
|
|
|
CP0418105
|
US9206164, 45
Show/Hide
|
C23H23ClN4O2
|
1
|
| 1 |
Ki = 0.3 nM
|
|
|
|
CP0488848
|
US9206164, 4
Show/Hide
|
C23H20F3N3O2
|
1
|
| 1 |
Ki = 0.3 nM
|
|
|
|
CP0495822
|
US9206164, 28
Show/Hide
|
C23H22BrClN4O2
|
1
|
| 1 |
Ki = 0.3 nM
|
|
|
|
CP0555331
|
US8791272, 2.37
Show/Hide
|
C25H28ClN3O3
|
1
|
| 1 |
Ki = 0.4 nM
|
|
|
|
CP0419326
|
US9206164, 65
Show/Hide
|
C23H22Cl2N4O2
|
1
|
| 1 |
Ki = 0.4 nM
|
|
|
|
CP0488703
|
US9206164, 87
Show/Hide
|
C23H22BrFN4O2
|
1
|
| 1 |
Ki = 0.4 nM
|
|
|
|
CP0557881
|
US9206164, 27
Show/Hide
|
C23H22ClFN4O2
|
1
|
| 1 |
Ki = 0.4 nM
|
|
|
|
CP0443138
|
US8791272, 2.52
Show/Hide
|
C23H22F3N3O3
|
1
|
| 1 |
Ki = 0.5 nM
|
|
|
|
CP0463971
|
US8791272, 2.21
Show/Hide
|
C27H31N3O3
|
1
|
| 1 |
Ki = 0.5 nM
|
|
|
|
CP0500379
|
US8791272, 9.27
Show/Hide
|
C24H22ClF4N3O3
|
1
|
| 1 |
Ki = 0.5 nM
|
|
|
|
CP0546677
|
US8791272, 3.4
Show/Hide
|
C22H21Cl2N3O4
|
1
|
| 1 |
Ki = 0.5 nM
|
|
|
|
CP0406808
|
US9206164, 55
Show/Hide
|
C24H25ClN4O2
|
1
|
| 1 |
Ki = 0.5 nM
|
|
|
|
CP0418101
|
US9206164, 5
Show/Hide
|
C23H19F4N3O2
|
1
|
| 1 |
Ki = 0.5 nM
|
|
|
|
CP0464851
|
US9206164, 80
Show/Hide
|
C23H22ClFN4O2
|
1
|
| 1 |
Ki = 0.5 nM
|
|
|
|
CP0488699
|
US9206164, 33
Show/Hide
|
C25H28N4O2
|
1
|
| 1 |
Ki = 0.5 nM
|
|
|
|
CP0506921
|
US8791272, 7.15
Show/Hide
|
C21H18Cl3N3O3
|
1
|
| 1 |
Ki = 0.6 nM
|
|
|
|
CP0544509
|
US8791272, 2.49
Show/Hide
|
C25H26ClN3O3
|
1
|
| 1 |
Ki = 0.6 nM
|
|
|
|
CP0548676
|
US8791272, 2.46
Show/Hide
|
C25H26ClN3O3
|
1
|
| 1 |
Ki = 0.6 nM
|
|
|
|
CP0561773
|
US8791272, 3.7
Show/Hide
|
C26H25N3O4
|
1
|
| 1 |
Ki = 0.6 nM
|
|
|
|
CP0464850
|
US9206164, 76
Show/Hide
|
C23H21ClF2N4O2
|
1
|
| 1 |
Ki = 0.6 nM
|
|
|
|
CP0463970
|
US8791272, 2.17
Show/Hide
|
C24H26BrN3O3
|
1
|
| 1 |
Ki = 0.7 nM
|
|
|
|
CP0531855
|
US8791272, 2.36
Show/Hide
|
C27H30F3N3O3
|
1
|
| 1 |
Ki = 0.7 nM
|
|
|
|
CP0499867
|
US9206164, 11
Show/Hide
|
C24H19F6N3O2
|
1
|
| 1 |
Ki = 0.7 nM
|
|
|
|
CP0508934
|
US9206164, 92
Show/Hide
|
C21H20FN5O3
|
1
|
| 1 |
Ki = 0.7 nM
|
|
|
|
CP0518177
|
US9206164, 104
Show/Hide
|
C23H21Cl2FN4O2
|
1
|
| 1 |
Ki = 0.7 nM
|
|
|
|
CP0546813
|
US8791272, 2.5
Show/Hide
|
C23H24ClN3O3
|
1
|
| 1 |
Ki = 0.75 nM
|
|
|
|
CP0426556
|
US8791272, 2.33
Show/Hide
|
C27H35N3O3
|
1
|
| 1 |
Ki = 0.8 nM
|
|
|
|
CP0463990
|
US8791272, 7.8
Show/Hide
|
C22H19ClF3N3O3
|
1
|
| 1 |
Ki = 0.8 nM
|
|
|
|
CP0565193
|
US8791272, 2.10
Show/Hide
|
C26H21Cl2N3O3
|
1
|
| 1 |
Ki = 0.8 nM
|
|
|
|
CP0418107
|
US9206164, 84
Show/Hide
|
C23H21F3N4O2
|
1
|
| 1 |
Ki = 0.8 nM
|
|
|
|
CP0464836
|
US9206164, 18
Show/Hide
|
C25H22N4O2
|
1
|
| 1 |
Ki = 0.8 nM
|
|
|
|
CP0475233
|
US9206164, 1
Show/Hide
|
C22H20ClN3O2
|
1
|
| 1 |
Ki = 0.8 nM
|
|
|
|
CP0574886
|
US9206164, 6
Show/Hide
|
C22H19ClFN3O2
|
1
|
| 1 |
Ki = 0.8 nM
|
|
|
|
CP0555707
|
US8791272, 9.13
Show/Hide
|
C24H23ClF3N3O3
|
1
|
| 1 |
Ki = 0.9 nM
|
|
|
|
CP0556280
|
US8791272, 7.11
Show/Hide
|
C23H22ClN3O3
|
1
|
| 1 |
Ki = 0.9 nM
|
|
|
|
CP0470646
|
US9206164, 97
Show/Hide
|
C25H27FN4O2
|
1
|
| 1 |
Ki = 0.9 nM
|
|
|
|
CP0500374
|
US8791272, 2.38
Show/Hide
|
C26H30ClN3O3
|
1
|
| 1 |
Ki = 1 nM
|
|
|
|
CP0413240
|
US9206164, 66
Show/Hide
|
C21H18Cl2N4O2
|
1
|
| 1 |
Ki = 1 nM
|
|
|
|
CP0464849
|
US9206164, 75
Show/Hide
|
C24H25FN4O3
|
1
|
| 1 |
Ki = 1 nM
|
|
|
|
CP0574821
|
US9206164, 82
Show/Hide
|
C23H22F2N4O2
|
1
|
| 1 |
Ki = 1 nM
|
|
|
|
CP0424190
|
US8791272, 2.2
Show/Hide
|
C24H26ClN3O3
|
1
|
| 1 |
Ki = 1.1 nM
|
|
|
|
CP0474696
|
US8791272, 1.14
Show/Hide
|
C23H22ClN3O3
|
1
|
| 1 |
Ki = 1.1 nM
|
|
|
|
CP0563981
|
US8791272, 7.17
Show/Hide
|
C22H19F4N3O3
|
1
|
| 1 |
Ki = 1.1 nM
|
|
|
|
CP0464842
|
US9206164, 54
Show/Hide
|
C22H21ClN4O2
|
1
|
| 1 |
Ki = 1.1 nM
|
|
|
|
CP0488701
|
US9206164, 50
Show/Hide
|
C23H22F2N4O2
|
1
|
| 1 |
Ki = 1.1 nM
|
|
|
|
CP0488704
|
US9206164, 101
Show/Hide
|
C23H21F3N4O2
|
1
|
| 1 |
Ki = 1.1 nM
|
|
|
|
CP0518173
|
US9206164, 43
Show/Hide
|
C23H22F2N4O2
|
1
|
| 1 |
Ki = 1.1 nM
|
|
|
|
CP0506868
|
US8791272, 2.11
Show/Hide
|
C27H22F3N3O3
|
1
|
| 1 |
Ki = 1.2 nM
|
|
|
|
CP0532387
|
US8791272, 7.6
Show/Hide
|
C21H19Cl2N3O3
|
1
|
| 1 |
Ki = 1.2 nM
|
|
|
|
CP0470644
|
US9206164, 74
Show/Hide
|
C23H22F2N4O2
|
1
|
| 1 |
Ki = 1.2 nM
|
|
|
|
CP0499878
|
US9206164, 32
Show/Hide
|
C21H19BrN4O2
|
1
|
| 1 |
Ki = 1.2 nM
|
|
|
|
CP0425126
|
US8791272, 7.13
Show/Hide
|
C25H22ClN3O3
|
1
|
| 1 |
Ki = 1.3 nM
|
|
|
|
CP0426613
|
US8791272, 2.4
Show/Hide
|
C24H27N3O3
|
1
|
| 1 |
Ki = 1.3 nM
|
|
|
|
CP0488401
|
US8791272, 2.8
Show/Hide
|
C30H25N3O3
|
1
|
| 1 |
Ki = 1.3 nM
|
|
|
|
CP0463914
|
US9206164, 39
Show/Hide
|
C24H26N4O3
|
1
|
| 1 |
Ki = 1.3 nM
|
|
|
|
CP0463915
|
US9206164, 79
Show/Hide
|
C23H24FN5O3
|
1
|
| 1 |
Ki = 1.3 nM
|
|
|
|
CP0464844
|
US9206164, 58
Show/Hide
|
C24H26N4O2
|
1
|
| 1 |
Ki = 1.3 nM
|
|
|
|
CP0514980
|
US9206164, 56
Show/Hide
|
C23H23FN4O2
|
1
|
| 1 |
Ki = 1.3 nM
|
|
|
|
CP0518176
|
US9206164, 83
Show/Hide
|
C24H25FN4O2
|
1
|
| 1 |
Ki = 1.3 nM
|
|
|
|
CP0557194
|
US8791272, 2.15
Show/Hide
|
C25H29N3O3
|
1
|
| 1 |
Ki = 1.4 nM
|
|
|
|
CP0464837
|
US9206164, 21
Show/Hide
|
C22H19F3N4O2
|
1
|
| 1 |
Ki = 1.4 nM
|
|
|
|
CP0499879
|
US9206164, 57
Show/Hide
|
C22H22BrN5O2
|
1
|
| 1 |
Ki = 1.5 nM
|
|
|
|
CP0412331
|
US8791272, 18.1
Show/Hide
|
C20H18Cl2N4O3
|
1
|
| 1 |
Ki = 1.6 nM
|
|
|
|
CP0415258
|
US8791272, 2.39
Show/Hide
|
C25H29N3O3
|
1
|
| 1 |
Ki = 1.6 nM
|
|
|
|
CP0506920
|
US8791272, 7.14
Show/Hide
|
C23H21ClF3N3O3
|
1
|
| 1 |
Ki = 1.6 nM
|
|
|
|
CP0402519
|
US9206164, 94
Show/Hide
|
C21H18BrFN4O2
|
1
|
| 1 |
Ki = 1.6 nM
|
|
|
|
CP0418104
|
US9206164, 42
Show/Hide
|
C22H22ClN5O2
|
1
|
| 1 |
Ki = 1.7 nM
|
|
|
|
CP0518175
|
US9206164, 67
Show/Hide
|
C23H23FN4O2
|
1
|
| 1 |
Ki = 1.7 nM
|
|
|
|
CP0472591
|
US8791272, 2.48
Show/Hide
|
C28H27N3O3
|
1
|
| 1 |
Ki = 1.8 nM
|
|
|
|
CP0546888
|
US8791272, 2.9
Show/Hide
|
C27H22F3N3O3
|
1
|
| 1 |
Ki = 1.8 nM
|
|
|
|
CP0406817
|
US9206164, 109
Show/Hide
|
C22H20ClFN4O2
|
1
|
| 1 |
Ki = 1.8 nM
|
|
|
|
CP0472590
|
US8791272, 2.22
Show/Hide
|
C23H23BrClN3O3
|
1
|
| 1 |
Ki = 1.9 nM
|
|
|
|
CP0571112
|
US8791272, 7.21
Show/Hide
|
C23H22FN3O3
|
1
|
| 1 |
Ki = 1.9 nM
|
|
|
|
CP0475772
|
US9206164, 24
Show/Hide
|
C21H19ClN4O2
|
1
|
| 1 |
Ki = 1.9 nM
|
|
|
|
CP0406815
|
US9206164, 102
Show/Hide
|
C21H17ClF2N4O2
|
1
|
| 1 |
Ki = 2.1 nM
|
|
|
|
CP0426618
|
US8791272, 7.4
Show/Hide
|
C22H21Cl2N3O3
|
1
|
| 1 |
Ki = 2.2 nM
|
|
|
|
CP0476981
|
US8791272, 7.20
Show/Hide
|
C25H22FN3O3
|
1
|
| 1 |
Ki = 2.2 nM
|
|
|
|
CP0488702
|
US9206164, 51
Show/Hide
|
C24H26N4O2
|
1
|
| 1 |
Ki = 2.2 nM
|
|
|
|
CP0546814
|
US8791272, 2.12
Show/Hide
|
C30H25N3O3
|
1
|
| 1 |
Ki = 2.3 nM
|
|
|
|
CP0441623
|
US9206164, 108
Show/Hide
|
C21H18ClFN4O2
|
1
|
| 1 |
Ki = 2.3 nM
|
|
|
|
CP0464834
|
US9206164, 15
Show/Hide
|
C23H24N4O2
|
1
|
| 1 |
Ki = 2.3 nM
|
|
|
|
CP0478765
|
US9206164, 53
Show/Hide
|
C21H18ClFN4O2
|
1
|
| 1 |
Ki = 2.3 nM
|
|
|
|
CP0565194
|
US8791272, 7.18
Show/Hide
|
C21H18Cl2FN3O3
|
1
|
| 1 |
Ki = 2.4 nM
|
|
|
|
CP0410653
|
US8791272, 1.29
Show/Hide
|
C25H27N3O3
|
1
|
| 1 |
Ki = 2.5 nM
|
|
|
|
CP0450076
|
US8791272, 1.7
Show/Hide
|
C25H23N3O3
|
1
|
| 1 |
Ki = 2.5 nM
|
|
|
|
CP0463991
|
US8791272, 7.9
Show/Hide
|
C23H24ClN3O3
|
1
|
| 1 |
Ki = 2.5 nM
|
|
|
|
CP0550364
|
US8791272, 1.17
Show/Hide
|
C23H24BrN3O3
|
1
|
| 1 |
Ki = 2.5 nM
|
|
|
|
CP0441626
|
US9206164, 111
Show/Hide
|
C22H18F4N4O2
|
1
|
| 1 |
Ki = 2.5 nM
|
|
|
|
CP0464848
|
US9206164, 73
Show/Hide
|
C21H17Cl2FN4O2
|
1
|
| 1 |
Ki = 2.5 nM
|
|
|
|
CP0472353
|
US8791272, 1.8
Show/Hide
|
C21H19Cl2N3O3
|
1
|
| 1 |
Ki = 2.6 nM
|
|
|
|
CP0500373
|
US8791272, 2.32
Show/Hide
|
C22H29N3O3
|
1
|
| 1 |
Ki = 2.6 nM
|
|
|
|
CP0546691
|
US8791272, 10.1
Show/Hide
|
C20H20FN3O4S
|
1
|
| 1 |
Ki = 2.6 nM
|
|
|
|
CP0413241
|
US9206164, 81
Show/Hide
|
C24H22FN5O2
|
1
|
| 1 |
Ki = 2.6 nM
|
|
|
|
CP0549871
|
US9206164, 89
Show/Hide
|
C22H21BrFN5O2
|
1
|
| 1 |
Ki = 2.6 nM
|
|
|
|
CP0546702
|
US8791272, 1.11
Show/Hide
|
C23H22F3N3O3
|
1
|
| 1 |
Ki = 2.7 nM
|
|
|
|
CP0520318
|
US8791272, 2.24
Show/Hide
|
C23H23BrClN3O3
|
1
|
| 1 |
Ki = 2.8 nM
|
|
|
|
CP0555329
|
US8791272, 2.18
Show/Hide
|
C23H31N3O3
|
1
|
| 1 |
Ki = 2.8 nM
|
|
|
|
CP0472588
|
US8791272, 1.1
Show/Hide
|
C22H20F3N3O3
|
1
|
| 1 |
Ki = 2.9 nM
|
|
|
|
CP0546890
|
US8791272, 2.13
Show/Hide
|
C26H21Cl2N3O3
|
1
|
| 1 |
Ki = 2.9 nM
|
|
|
|
CP0476982
|
US8791272, 9.6
Show/Hide
|
C22H19ClF3N3O3
|
1
|
| 1 |
Ki = 3 nM
|
|
|
|
CP0546826
|
US8791272, 9.14
Show/Hide
|
C23H23BrFN3O3
|
1
|
| 1 |
Ki = 3.1 nM
|
|
|
|
CP0555327
|
US8791272, 1.25
Show/Hide
|
C26H25N3O3
|
1
|
| 1 |
Ki = 3.1 nM
|
|
|
|
CP0546818
|
US8791272, 7.7
Show/Hide
|
C22H21Cl2N3O3
|
1
|
| 1 |
Ki = 3.4 nM
|
|
|
|
CP0556284
|
US8791272, 2.3
Show/Hide
|
C23H25N3O3
|
1
|
| 1 |
Ki = 3.4 nM
|
|
|
|
CP0463967
|
US8791272, 1.6
Show/Hide
|
C21H20ClN3O3
|
1
|
| 1 |
Ki = 3.5 nM
|
|
|
|
CP0544511
|
US8791272, 2.51
Show/Hide
|
C28H27N3O3
|
1
|
| 1 |
Ki = 3.5 nM
|
|
|
|
CP0550369
|
US8791272, 7.16
Show/Hide
|
C23H21F4N3O3
|
1
|
| 1 |
Ki = 3.5 nM
|
|
|
|
CP0557195
|
US8791272, 3.11
Show/Hide
|
C24H26BrN3O4
|
1
|
| 1 |
Ki = 3.5 nM
|
|
|
|
CP0546518
|
US8791272, 2.26
Show/Hide
|
C27H26BrN3O3
|
1
|
| 1 |
Ki = 3.6 nM
|
|
|
|
CP0419328
|
US9206164, 91
Show/Hide
|
C22H21FN4O2
|
1
|
| 1 |
Ki = 3.7 nM
|
|
|
|
CP0475773
|
US9206164, 34
Show/Hide
|
C24H23N5O2
|
1
|
| 1 |
Ki = 3.7 nM
|
|
|
|
CP0443043
|
US8791272, 3.1
Show/Hide
|
C22H23N3O4
|
1
|
| 1 |
Ki = 3.8 nM
|
|
|
|
CP0555326
|
US8791272, 1.16
Show/Hide
|
C22H22BrN3O3
|
1
|
| 1 |
Ki = 3.9 nM
|
|
|
|
CP0415254
|
US8791272, 1.34
Show/Hide
|
C25H31N3O3
|
1
|
| 1 |
Ki = 4 nM
|
|
|
|
CP0450078
|
US8791272, 1.13
Show/Hide
|
C23H23N3O3
|
1
|
| 1 |
Ki = 4 nM
|
|
|
|
CP0546828
|
US8791272, 9.23
Show/Hide
|
C26H26N4O3
|
1
|
| 1 |
Ki = 4 nM
|
|
|
|
CP0506872
|
US8791272, 2.6
Show/Hide
|
C25H23N3O4
|
1
|
| 1 |
Ki = 4.2 nM
|
|
|
|
CP0499866
|
US9206164, 3
Show/Hide
|
C22H20ClN3O2
|
1
|
| 1 |
Ki = 4.2 nM
|
|
|
|
CP0466593
|
US8791272, 2.34
Show/Hide
|
C20H27N3O3
|
1
|
| 1 |
Ki = 4.3 nM
|
|
|
|
CP0557164
|
US8791272, 2.27
Show/Hide
|
C27H33N3O3
|
1
|
| 1 |
Ki = 4.3 nM
|
|
|
|
CP0565188
|
US8791272, 17.2
Show/Hide
|
C25H26F3N3O3
|
1
|
| 1 |
Ki = 4.3 nM
|
|
|
|
CP0450080
|
US8791272, 7.12
Show/Hide
|
C23H24ClN3O3
|
1
|
| 1 |
Ki = 4.7 nM
|
|
|
|
CP0506873
|
US8791272, 3.13
Show/Hide
|
C22H22ClN3O4
|
1
|
| 1 |
Ki = 4.7 nM
|
|
|
|
CP0301754
|
2-[1-[[4-[[4-chloro-3-(trifluoromethyl)phenyl]methoxy]phenyl]methyl]-3,5-diethylpyrazol-4-yl]acetic acid
Show/Hide
|
C24H24ClF3N2O3
|
1
|
| 1 |
Ki = 4.8 nM
|
|
|
|
CP0450131
|
US8791272, 9.12
Show/Hide
|
C23H23ClFN3O3
|
1
|
| 1 |
Ki = 4.8 nM
|
|
|
|
CP0418103
|
US9206164, 41
Show/Hide
|
C22H22N4O2
|
1
|
| 1 |
Ki = 4.8 nM
|
|
|
|
CP0418106
|
US9206164, 47
Show/Hide
|
C21H18F2N4O2
|
1
|
| 1 |
Ki = 4.9 nM
|
|
|
|
CP0415255
|
US8791272, 2.31
Show/Hide
|
C21H27N3O3
|
1
|
| 1 |
Ki = 5 nM
|
|
|
|
CP0550110
|
US8791272, 13.12
Show/Hide
|
C25H27F3N2O4
|
1
|
| 1 |
Ki = 5 nM
|
|
|
|
CP0549872
|
US9206164, 95
Show/Hide
|
C22H21ClFN5O2
|
1
|
| 1 |
Ki = 5.1 nM
|
|
|
|
CP0574822
|
US9206164, 105
Show/Hide
|
C21H17F3N4O2
|
1
|
| 1 |
Ki = 5.1 nM
|
|
|
|
CP0469788
|
US8791272, 3.10
Show/Hide
|
C24H26ClN3O4
|
1
|
| 1 |
Ki = 5.2 nM
|
|
|
|
CP0443142
|
US8791272, 7.10
Show/Hide
|
C21H20ClN3O3
|
1
|
| 1 |
Ki = 5.5 nM
|
|
|
|
CP0566706
|
US9206164, 77
Show/Hide
|
C21H17F3N4O2
|
1
|
| 1 |
Ki = 5.5 nM
|
|
|
|
CP0506712
|
US9206164, 36
Show/Hide
|
C21H18F2N4O2
|
1
|
| 1 |
Ki = 5.6 nM
|
|
|
|
CP0536382
|
US8791272, 1.23
Show/Hide
|
C25H22ClN3O3
|
1
|
| 1 |
Ki = 5.7 nM
|
|
|
|
CP0413244
|
US9206164, 96
Show/Hide
|
C22H21FN4O3
|
1
|
| 1 |
Ki = 5.7 nM
|
|
|
|
CP0450079
|
US8791272, 2.19
Show/Hide
|
C24H26BrN3O3
|
1
|
| 1 |
Ki = 5.8 nM
|
|
|
|
CP0546520
|
US8791272, 2.3
Show/Hide
|
C21H29N3O3
|
1
|
| 1 |
Ki = 5.8 nM
|
|
|
|
CP0563982
|
US8791272, 7.19
Show/Hide
|
C22H21ClFN3O3
|
1
|
| 1 |
Ki = 5.8 nM
|
|
|
|
CP0426615
|
US8791272, 2.23
Show/Hide
|
C25H29N3O3
|
1
|
| 1 |
Ki = 6.1 nM
|
|
|
|
CP0459872
|
US8791272, 2.29
Show/Hide
|
C29H35N3O3
|
1
|
| 1 |
Ki = 6.3 nM
|
|
|
|
CP0475775
|
US9206164, 86
Show/Hide
|
C21H18F2N4O2
|
1
|
| 1 |
Ki = 6.5 nM
|
|
|
|
CP0548685
|
US8791272, 9.16
Show/Hide
|
C23H23BrFN3O3
|
1
|
| 1 |
Ki = 6.7 nM
|
|
|
|
CP0476983
|
US8791272, 9.11
Show/Hide
|
C23H23ClFN3O3
|
1
|
| 1 |
Ki = 7.1 nM
|
|
|
|
CP0450077
|
US8791272, 1.10
Show/Hide
|
C23H25N3O3
|
1
|
| 1 |
Ki = 7.4 nM
|
|
|
|
CP0488700
|
US9206164, 38
Show/Hide
|
C20H18BrN5O2
|
1
|
| 1 |
Ki = 7.4 nM
|
|
|
|
CP0425130
|
US8791272, 9.7
Show/Hide
|
C22H22ClN3O3
|
1
|
| 1 |
Ki = 7.5 nM
|
|
|
|
CP0406809
|
US9206164, 59
Show/Hide
|
C22H22N4O3
|
1
|
| 1 |
Ki = 7.6 nM
|
|
|
|
CP0383803
|
US8791272, 1.4
Show/Hide
|
C22H23N3O3
|
1
|
| 1 |
Ki = 7.7 nM
|
|
|
|
CP0450132
|
US8791272, 9.21
Show/Hide
|
C29H35N3O3
|
1
|
| 1 |
Ki = 7.8 nM
|
|
|
|
CP0464847
|
US9206164, 71
Show/Hide
|
C21H19FN4O2
|
1
|
| 1 |
Ki = 8.5 nM
|
|
|
|
CP0555639
|
US8791272, 9.3
Show/Hide
|
C21H19Cl2N3O3
|
1
|
| 1 |
Ki = 8.7 nM
|
|
|
|
CP0464841
|
US9206164, 52
Show/Hide
|
C21H19FN4O2
|
1
|
| 1 |
Ki = 8.7 nM
|
|
|
|
CP0442542
|
US8791272, 2.45
Show/Hide
|
C32H24F3N3O3
|
1
|
| 1 |
Ki = 8.9 nM
|
|
|
|
CP0546682
|
US8791272, 3.14
Show/Hide
|
C22H22FN3O4
|
1
|
| 1 |
Ki = 8.9 nM
|
|
|
|
CP0463969
|
US8791272, 1.27
Show/Hide
|
C21H19BrClN3O3
|
1
|
| 1 |
Ki = 9.3 nM
|
|
|
|
CP0418108
|
US9206164, 99
Show/Hide
|
C21H18F2N4O2
|
1
|
| 1 |
Ki = 9.7 nM
|
|
|
|
CP0464845
|
US9206164, 63
Show/Hide
|
C22H22N4O2
|
1
|
| 1 |
Ki = 10 nM
|
|
|
|
CP0500376
|
US8791272, 2.44
Show/Hide
|
C35H27N3O3
|
1
|
| 1 |
Ki = 10.2 nM
|
|
|
|
CP0546690
|
US8791272, 9.28
Show/Hide
|
C26H26FN3O4
|
1
|
| 1 |
Ki = 10.4 nM
|
|
|
|
CP0418100
|
US9206164, 2
Show/Hide
|
C23H20F3N3O2
|
1
|
| 1 |
Ki = 11.3 nM
|
|
|
|
CP0466594
|
US8791272, 2.35
Show/Hide
|
C26H29N3O3
|
1
|
| 1 |
Ki = 11.6 nM
|
|
|
|
CP0575484
|
US8791272, 19.2
Show/Hide
|
C21H20Cl2N2O3S
|
1
|
| 1 |
Ki = 12 nM
|
|
|
|
CP0476990
|
US8791272, 19.3
Show/Hide
|
C23H24Cl2N2O3S
|
1
|
| 1 |
Ki = 12.2 nM
|
|
|
|
CP0426623
|
US8791272, 12.3
Show/Hide
|
C24H25ClN2O2
|
1
|
| 1 |
Ki = 12.3 nM
|
|
|
|
CP0565192
|
US8791272, 1.28
Show/Hide
|
C21H19BrClN3O3
|
1
|
| 1 |
Ki = 12.4 nM
|
|
|
|
CP0418102
|
US9206164, 40
Show/Hide
|
C20H18ClN5O2
|
1
|
| 1 |
Ki = 12.4 nM
|
|
|
|
CP0475776
|
US9206164, 93
Show/Hide
|
C22H21FN4O2
|
1
|
| 1 |
Ki = 12.8 nM
|
|
|
|
CP0410545
|
US8791272, 1.12
Show/Hide
|
C23H25N3O3
|
1
|
| 1 |
Ki = 12.9 nM
|
|
|
|
CP0463968
|
US8791272, 1.5
Show/Hide
|
C22H23N3O4
|
1
|
| 1 |
Ki = 12.9 nM
|
|
|
|
CP0488400
|
US8791272, 2.7
Show/Hide
|
C27H28F3N3O3
|
1
|
| 1 |
Ki = 12.9 nM
|
|
|
|
CP0514979
|
US9206164, 48
Show/Hide
|
C22H23N5O2
|
1
|
| 1 |
Ki = 12.9 nM
|
|
|
|
CP0441621
|
US9206164, 14
Show/Hide
|
C21H20N4O2
|
1
|
| 1 |
Ki = 13.4 nM
|
|
|
|
CP0563980
|
US8791272, 7.3
Show/Hide
|
C23H22F3N3O3
|
1
|
| 1 |
Ki = 13.5 nM
|
|
|
|
CP0415282
|
US8791272, 9.5
Show/Hide
|
C22H20F3N3O3
|
1
|
| 1 |
Ki = 13.7 nM
|
|
|
|
CP0443135
|
US8791272, 2.20
Show/Hide
|
C23H23Cl2N3O3
|
1
|
| 1 |
Ki = 13.9 nM
|
|
|
|
CP0383804
|
US8791272, 1.30
Show/Hide
|
C25H22BrN3O3
|
1
|
| 1 |
Ki = 14.6 nM
|
|
|
|
CP0488402
|
US8791272, 3.6
Show/Hide
|
C22H22BrN3O4
|
1
|
| 1 |
Ki = 14.9 nM
|
|
|
|
CP0410552
|
US8791272, 13.8
Show/Hide
|
C23H24Cl2N2O3
|
1
|
| 1 |
Ki = 15.5 nM
|
|
|
|
CP0415284
|
US8791272, 9.22
Show/Hide
|
C29H35N3O3
|
1
|
| 1 |
Ki = 15.6 nM
|
|
|
|
CP0546692
|
US8791272, 10.3
Show/Hide
|
C23H26ClN3O4S
|
1
|
| 1 |
Ki = 16.1 nM
|
|
|
|
CP0443037
|
US8791272, 1.19
Show/Hide
|
C21H19ClFN3O3
|
1
|
| 1 |
Ki = 16.2 nM
|
|
|
|
CP0475235
|
US9206164, 13
Show/Hide
|
C22H22FN5O2
|
1
|
| 1 |
Ki = 16.2 nM
|
|
|
|
CP0450125
|
US8791272, 1.2
Show/Hide
|
C22H22ClN3O3
|
1
|
| 1 |
Ki = 16.3 nM
|
|
|
|
CP0390248
|
US8791272, 3.5
Show/Hide
|
C22H22ClN3O4
|
1
|
| 1 |
Ki = 16.8 nM
|
|
|
|
CP0476980
|
US8791272, 4.1
Show/Hide
|
C22H24N4O3
|
1
|
| 1 |
Ki = 16.8 nM
|
|
|
|
CP0546519
|
US8791272, 2.28
Show/Hide
|
C28H35N3O3
|
1
|
| 1 |
Ki = 17.1 nM
|
|
|
|
CP0463986
|
US8791272, 2.59
Show/Hide
|
C25H23N3O3
|
1
|
| 1 |
Ki = 17.4 nM
|
|
|
|
CP0506871
|
US8791272, 2.43
Show/Hide
|
C31H24ClN3O3
|
1
|
| 1 |
Ki = 17.4 nM
|
|
|
|
CP0550365
|
US8791272, 1.18
Show/Hide
|
C21H19Cl2N3O3
|
1
|
| 1 |
Ki = 17.9 nM
|
|
|
|
CP0508930
|
US9206164, 62
Show/Hide
|
C22H19N5O2
|
1
|
| 1 |
Ki = 18.4 nM
|
|
|
|
CP0418109
|
US9206164, 100
Show/Hide
|
C20H17ClFN5O2
|
1
|
| 1 |
Ki = 18.5 nM
|
|
|
|
CP0546824
|
US8791272, 9.4
Show/Hide
|
C21H19ClFN3O3
|
1
|
| 1 |
Ki = 18.6 nM
|
|
|
|
CP0426554
|
US8791272, 1.31
Show/Hide
|
C22H22BrN3O3
|
1
|
| 1 |
Ki = 18.9 nM
|
|
|
|
CP0462661
|
US8791272, 2.57
Show/Hide
|
C24H21N3O3
|
1
|
| 1 |
Ki = 19.3 nM
|
|
|
|
CP0415283
|
US8791272, 9.9
Show/Hide
|
C21H19BrFN3O3
|
1
|
| 1 |
Ki = 19.4 nM
|
|
|
|
CP0480733
|
US8791272, 13.10
Show/Hide
|
C24H25F3N2O3
|
1
|
| 1 |
Ki = 19.6 nM
|
|
|
|
CP0443144
|
US8791272, 10.4
Show/Hide
|
C22H23Cl2N3O4S
|
1
|
| 1 |
Ki = 21.6 nM
|
|
|
|
CP0549870
|
US9206164, 78
Show/Hide
|
C22H18FN5O2
|
1
|
| 1 |
Ki = 21.7 nM
|
|
|
|
CP0493226
|
US9206164, 22
Show/Hide
|
C22H22N4O2
|
1
|
| 1 |
Ki = 21.9 nM
|
|
|
|
CP0488397
|
US8791272, 2.16
Show/Hide
|
C24H30F3N3O3
|
1
|
| 1 |
Ki = 23.9 nM
|
|
|
|
CP0450081
|
US8791272, 9.2
Show/Hide
|
C21H19ClFN3O3
|
1
|
| 1 |
Ki = 24.5 nM
|
|
|
|
CP0492613
|
US8791272, 9.18
Show/Hide
|
C24H25Cl2N3O3
|
1
|
| 1 |
Ki = 24.9 nM
|
|
|
|
CP0425127
|
US8791272, 8.4
Show/Hide
|
C26H31N3O3
|
1
|
| 1 |
Ki = 26.1 nM
|
|
|
|
CP0425134
|
US8791272, 10.5
Show/Hide
|
C22H23ClFN3O4S
|
1
|
| 1 |
Ki = 27.8 nM
|
|
|
|
CP0461542
|
US8791272, 2.56
Show/Hide
|
C20H17Cl2N3O3
|
1
|
| 1 |
Ki = 27.8 nM
|
|
|
|
CP0532386
|
US8791272, 1.9
Show/Hide
|
C24H22N4O3
|
1
|
| 1 |
Ki = 28.3 nM
|
|
|
|
CP0415277
|
US8791272, 3.8
Show/Hide
|
C19H25N3O4
|
1
|
| 1 |
Ki = 28.6 nM
|
|
|
|
CP0492504
|
US8791272, 13.6
Show/Hide
|
C23H23F3N2O4
|
1
|
| 1 |
Ki = 28.9 nM
|
|
|
|
CP0560354
|
US8791272, 14.4
Show/Hide
|
C22H22Cl2N2O3
|
1
|
| 1 |
Ki = 29 nM
|
|
|
|
CP0426620
|
US8791272, 1.20
Show/Hide
|
C22H22FN3O3
|
1
|
| 1 |
Ki = 29.3 nM
|
|
|
|
CP0410551
|
US8791272, 11.1
Show/Hide
|
C26H29F3N4O4S
|
1
|
| 1 |
Ki = 29.4 nM
|
|
|
|
CP0410655
|
US8791272, 1.33
Show/Hide
|
C21H27N3O3
|
1
|
| 1 |
Ki = 29.8 nM
|
|
|
|
CP0476985
|
US8791272, 13.1
Show/Hide
|
C21H20Cl2N2O3
|
1
|
| 1 |
Ki = 30 nM
|
|
|
|
CP0476984
|
US8791272, 9.19
Show/Hide
|
C25H25ClF3N3O3
|
1
|
| 1 |
Ki = 30.5 nM
|
|
|
|
CP0443139
|
US8791272, 5.3
Show/Hide
|
C20H19Cl2N3O4S
|
1
|
| 1 |
Ki = 30.6 nM
|
|
|
|
CP0450127
|
US8791272, 1.3
Show/Hide
|
C21H21N3O3
|
1
|
| 1 |
Ki = 30.8 nM
|
|
|
|
CP0555705
|
US8791272, 9.8
Show/Hide
|
C21H19Cl2N3O3
|
1
|
| 1 |
Ki = 31 nM
|
|
|
|
CP0443050
|
US8791272, 9.15
Show/Hide
|
C27H31ClFN3O3
|
1
|
| 1 |
Ki = 32 nM
|
|
|
|
CP0443051
|
US8791272, 9.25
Show/Hide
|
C27H37N3O3
|
1
|
| 1 |
Ki = 32.1 nM
|
|
|
|
CP0546517
|
US8791272, 1.32
Show/Hide
|
C18H23N3O3
|
1
|
| 1 |
Ki = 32.5 nM
|
|
|
|
CP0546815
|
US8791272, 5.2
Show/Hide
|
C20H20ClN3O4S
|
1
|
| 1 |
Ki = 33.7 nM
|
|
|
|
CP0426622
|
US8791272, 9.17
Show/Hide
|
C28H29N3O3
|
1
|
| 1 |
Ki = 34.9 nM
|
|
|
|
CP0476986
|
US8791272, 13.5
Show/Hide
|
C22H20ClF3N2O3
|
1
|
| 1 |
Ki = 36 nM
|
|
|
|
CP0546516
|
US8791272, 1.26
Show/Hide
|
C26H25N3O3
|
1
|
| 1 |
Ki = 36 nM
|
|
|
|
CP0546827
|
US8791272, 9.20
Show/Hide
|
C25H26F3N3O3
|
1
|
| 1 |
Ki = 38 nM
|
|
|
|
CP0476987
|
US8791272, 13.9
Show/Hide
|
C23H25ClN2O3
|
1
|
| 1 |
Ki = 39.1 nM
|
|
|
|
CP0555706
|
US8791272, 9.10
Show/Hide
|
C23H24FN3O3
|
1
|
| 1 |
Ki = 39.1 nM
|
|
|
|
CP0480731
|
US8791272, 9.26
Show/Hide
|
C27H39N3O3
|
1
|
| 1 |
Ki = 39.4 nM
|
|
|
|
CP0557880
|
US9206164, 23
Show/Hide
|
C24H22Cl2N4O2
|
1
|
| 1 |
Ki = 41.1 nM
|
|
|
|
CP0426624
|
US8791272, 14.2
Show/Hide
|
C21H20Cl2N2O3
|
1
|
| 1 |
Ki = 43 nM
|
|
|
|
CP0546693
|
US8791272, 19.1
Show/Hide
|
C25H24N2O3S
|
1
|
| 1 |
Ki = 43.5 nM
|
|
|
|
CP0546684
|
US8791272, 5.1
Show/Hide
|
C20H21N3O4S
|
1
|
| 1 |
Ki = 43.9 nM
|
|
|
|
CP0563976
|
US8791272, 1.35
Show/Hide
|
C19H23N3O3
|
1
|
| 1 |
Ki = 44.6 nM
|
|
|
|
CP0463972
|
US8791272, 2.25
Show/Hide
|
C24H26BrN3O3
|
1
|
| 1 |
Ki = 46.6 nM
|
|
|
|
CP0426625
|
US8791272, 19.4
Show/Hide
|
C23H26N2O3S
|
1
|
| 1 |
Ki = 48.8 nM
|
|
|
|
CP0480734
|
US8791272, 13.11
Show/Hide
|
C24H24ClF3N2O4
|
1
|
| 1 |
Ki = 48.8 nM
|
|
|
|
CP0466693
|
US8791272, 9.24
Show/Hide
|
C25H35N3O3
|
1
|
| 1 |
Ki = 49.1 nM
|
|
|
|
CP0571081
|
US8791272, 13.13
Show/Hide
|
C24H28N2O3
|
1
|
| 1 |
Ki = 49.9 nM
|
|
|
|
CP0569649
|
US8791272, 12.2
Show/Hide
|
C23H21F3N2O2
|
1
|
| 1 |
Ki = 56.3 nM
|
|
|
|
CP0413239
|
US9206164, 61
Show/Hide
|
C22H23N5O2
|
1
|
| 1 |
Ki = 56.4 nM
|
|
|
|
CP0413243
|
US9206164, 90
Show/Hide
|
C22H22FN5O2
|
1
|
| 1 |
Ki = 60.9 nM
|
|
|
|
CP0475774
|
US9206164, 69
Show/Hide
|
C24H25ClN4O2
|
1
|
| 1 |
Ki = 61.2 nM
|
|
|
|
CP0464839
|
US9206164, 35
Show/Hide
|
C24H24Cl2N4O2
|
1
|
| 1 |
Ki = 66.7 nM
|
|
|
|
CP0410652
|
US8791272, 1.21
Show/Hide
|
C23H22F3N3O3
|
1
|
| 1 |
Ki = 80.2 nM
|
|
|
|
CP0464840
|
US9206164, 37
Show/Hide
|
C21H22N6O2
|
1
|
| 1 |
Ki = 85.4 nM
|
|
|
|
CP0470647
|
US9206164, 107
Show/Hide
|
C20H18FN5O2
|
1
|
| 1 |
Ki = 87.4 nM
|
|
|
|
CP0475234
|
US9206164, 9
Show/Hide
|
C23H20F3N3O2
|
1
|
| 1 |
Ki = 97.8 nM
|
|
|
|
CP0488697
|
US9206164, 31
Show/Hide
|
C20H19N5O2
|
1
|
| 1 |
Ki = 118.5 nM
|
|
|
|
CP0555369
|
US8791272, 8.2
Show/Hide
|
C23H22F3N3O3
|
1
|
| 1 |
Ki = 124.7 nM
|
|
|
|
CP0565680
|
US8791272, 8.6
Show/Hide
|
C22H21Cl2N3O3
|
1
|
| 1 |
Ki = 125.5 nM
|
|
|
|
CP0550109
|
US8791272, 12.1
Show/Hide
|
C23H19F3N2O2
|
1
|
| 1 |
Ki = 127 nM
|
|
|
|
CP0419324
|
US9206164, 12
Show/Hide
|
C21H19FN4O2
|
1
|
| 1 |
Ki = 154.9 nM
|
|
|
|
CP0463989
|
US8791272, 7.2
Show/Hide
|
C22H22ClN3O3
|
1
|
| 1 |
Ki = 161.6 nM
|
|
|
|
CP0464838
|
US9206164, 25
Show/Hide
|
C22H21ClN4O2
|
1
|
| 1 |
Ki = 175.5 nM
|
|
|
|
CP0546686
|
US8791272, 5.4
Show/Hide
|
C21H20F3N3O4S
|
1
|
| 1 |
Ki = 230.2 nM
|
|
|
|
CP0464159
|
US8791272, 14.5
Show/Hide
|
C23H23F3N2O3
|
1
|
| 1 |
Ki = 253 nM
|
|
|
|
CP0426617
|
US8791272, 6.3
Show/Hide
|
C22H22F3N3O2
|
1
|
| 1 |
Ki = 261.1 nM
|
|
|
|
CP0464852
|
US9206164, 110
Show/Hide
|
C22H19F3N4O2
|
1
|
| 1 |
Ki = 287.2 nM
|
|
|
|
CP0508929
|
US9206164, 60
Show/Hide
|
C20H19N5O2
|
1
|
| 1 |
Ki = 298.7 nM
|
|
|
|
CP0463913
|
US9206164, 10
Show/Hide
|
C21H20N4O2
|
1
|
| 1 |
Ki = 308.2 nM
|
|
|
|
CP0443141
|
US8791272, 6.2
Show/Hide
|
C21H23N3O2
|
1
|
| 1 |
Ki = 311.4 nM
|
|
|
|
CP0466694
|
US8791272, 16.2
Show/Hide
|
C22H21F3N2O3S
|
1
|
| 1 |
Ki = 324 nM
|
|
|
|
CP0412330
|
US8791272, 16.5
Show/Hide
|
C21H20Cl2N2O3S
|
1
|
| 1 |
Ki = 325 nM
|
|
|
|
CP0546831
|
US8791272, 13.4
Show/Hide
|
C21H22N2O3
|
1
|
| 1 |
Ki = 325 nM
|
|
|
|
CP0518174
|
US9206164, 46
Show/Hide
|
C24H26N4O2
|
1
|
| 1 |
Ki = 339.8 nM
|
|
|
|
CP0488849
|
US9206164, 8
Show/Hide
|
C22H20ClN3O2
|
1
|
| 1 |
Ki = 394.1 nM
|
|
|
|
CP0464833
|
US9206164, 7
Show/Hide
|
C22H20ClN3O2
|
1
|
| 1 |
Ki = 397.4 nM
|
|
|
|
CP0383806
|
US8791272, 7.1
Show/Hide
|
C22H23N3O3
|
1
|
| 1 |
Ki = 406.6 nM
|
|
|
|
CP0569643
|
US8791272, 8.5
Show/Hide
|
C24H27N3O3
|
1
|
| 1 |
Ki = 427.1 nM
|
|
|
|
CP0565681
|
US8791272, 14.6
Show/Hide
|
C22H24N2O3
|
1
|
| 1 |
Ki = 428 nM
|
|
|
|
CP0546816
|
US8791272, 6.1
Show/Hide
|
C21H22ClN3O2
|
1
|
| 1 |
Ki = 437.8 nM
|
|
|
|
CP0532388
|
US8791272, 15.2
Show/Hide
|
C22H22N2O3
|
1
|
| 1 |
Ki = 552 nM
|
|
|
|
CP0546812
|
US8791272, 1.24
Show/Hide
|
C24H27N3O3
|
1
|
| 1 |
Ki = 553 nM
|
|
|
|
CP0563535
|
US8791272, 13.3
Show/Hide
|
C22H23ClN2O3
|
1
|
| 1 |
Ki = 619 nM
|
|
|
|
CP0549869
|
US9206164, 72
Show/Hide
|
C20H18FN5O2
|
1
|
| 1 |
Ki = 636 nM
|
|
|
|
CP0546521
|
US8791272, 8.7
Show/Hide
|
C24H24F3N3O3
|
1
|
| 1 |
Ki = 668.6 nM
|
|
|
|
CP0413242
|
US9206164, 85
Show/Hide
|
C21H20FN5O2
|
1
|
| 1 |
Ki = 683.1 nM
|
|
|
|
CP0488294
|
US8791272, 10.2
Show/Hide
|
C24H29N3O6S
|
1
|
| 1 |
Ki = 742 nM
|
|
|
|
CP0569635
|
US8791272, 14.3
Show/Hide
|
C21H22N2O3
|
1
|
| 1 |
Ki = 742 nM
|
|
|
|
CP0406807
|
US9206164, 30
Show/Hide
|
C22H22N4O2
|
1
|
| 1 |
Ki = 752.7 nM
|
|
|
|
CP0476988
|
US8791272, 15.1
Show/Hide
|
C22H24N2O3
|
1
|
| 1 |
Ki = 785 nM
|
|
|
|
CP0402733
|
US8791272, 3.2
Show/Hide
|
C23H25N3O4
|
1
|
| 1 |
Ki = 785.7 nM
|
|
|
|
CP0555641
|
US8791272, 16.6
Show/Hide
|
C21H20Cl2N2O4S
|
1
|
| 1 |
Ki = 853 nM
|
|
|
|
CP0476989
|
US8791272, 16.4
Show/Hide
|
C21H20Cl2N2O2S
|
1
|
| 1 |
Ki = 875 nM
|
|
|
|
CP0565682
|
US8791272, 16.1
Show/Hide
|
C22H21F3N2O2S
|
1
|
| 1 |
Ki = 992 nM
|
|
|
|
CP0571117
|
US8791272, 13.2
Show/Hide
|
C22H21F3N2O3
|
1
|
| 1 |
Ki = 1070 nM
|
|
|
|
CP0426621
|
US8791272, 9.1
Show/Hide
|
C21H20FN3O3
|
1
|
| 1 |
Ki = 1480.3 nM
|
|
|
|
CP0410553
|
US8791272, 14.1
Show/Hide
|
C22H21F3N2O3
|
1
|
| 1 |
Ki = 1532 nM
|
|
|
|
CP0466597
|
US8791272, 8.1
Show/Hide
|
C23H24ClN3O3
|
1
|
| 1 |
Ki = 1664.4 nM
|
|
|
|
CP0560355
|
US8791272, 16.3
Show/Hide
|
C22H21F3N2O4S
|
1
|
| 1 |
Ki = 2288 nM
|
|
|
|
CP0544503
|
US8791272, 1.22
Show/Hide
|
C22H19F4N3O3
|
1
|
| 1 |
Ki = 3319 nM
|
|
|
|
CP0561774
|
US8791272, 8.3
Show/Hide
|
C22H23N3O3
|
1
|
| 1 |
Ki = 3760.8 nM
|
|
|
