| Compound ID |
Compound Name |
Compound Formula |
|
CP0412420
|
(2S)-1-(7-ethylfuro[2,3-g]indazol-1-yl)propan-2-amine
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|
C14H17N3O
|
2
|
| 1 |
EC50 = 1 nM
|
|
|
| 2 |
Ki = 0.89 nM
|
|
|
|
CP0001238
|
14C-5-hydroxy tryptamine creatinine disulfate
Show/Hide
|
C10H12N2O
|
7
|
| 1 |
EC50 = 1.63 nM
|
|
|
| 2 |
EC50 = 1.7 nM
|
|
|
| 3 |
EC50 = 24 nM
|
|
|
| 4 |
EC50 = 25 nM
|
|
|
| 5 |
Ki = 8.3 nM
|
|
|
| 6 |
Ki = 214 nM
|
|
|
| 7 |
Ki = 445 nM
|
|
|
|
CP0172895
|
(S)-1-(1H-pyrrolo[2,3-f]quinolin-1-yl)propan-2-amine
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|
C14H15N3
|
1
|
| 1 |
EC50 = 2.9 nM
|
|
|
|
CP0451296
|
(S)-1-Methyl-2-(2,3,7,8-tetrahydro-furo[2,3-g]indol-1-yl)-ethylamine
Show/Hide
|
C13H18N2O
|
1
|
| 1 |
EC50 = 4.5 nM
|
|
|
|
CP0374738
|
(S)-2-(5-Fluoro-6-methylsulfanyl-2,3-dihydro-indol-1-yl)-1-methyl-ethylamine
Show/Hide
|
C12H17FN2S
|
1
|
| 1 |
EC50 = 6.7 nM
|
|
|
|
CP0216157
|
(S)-1-(5-chloro-1H-pyrrolo[2,3-f]quinolin-1-yl)propan-2-amine
Show/Hide
|
C14H14ClN3
|
1
|
| 1 |
EC50 = 6.9 nM
|
|
|
|
CP0409693
|
8,9-Dichloro-2,3,4,4a,5,6-hexahydro-1H-pyrazino[1,2-a]quinoxaline
Show/Hide
|
C11H13Cl2N3
|
1
|
| 1 |
EC50 = 7.6 nM
|
|
|
|
CP0196718
|
(R)-8,9-Dichloro-2,3,4,4a-tetrahydro-1H,6H-pyrazino[1,2-a]quinoxalin-5-one
Show/Hide
|
C11H11Cl2N3O
|
1
|
| 1 |
EC50 = 8 nM
|
|
|
|
CP0418829
|
8,9-Dichloro-2,3,4,4a-tetrahydro-1H,6H-pyrazino[1,2-a]quinoxalin-5-one
Show/Hide
|
C11H11Cl2N3O
|
1
|
| 1 |
EC50 = 12 nM
|
|
|
|
CP0059838
|
(4R,9aR)-6-Cyclopropylmethoxymethyl-4-methyl-1,2,3,4,9,9a-hexahydro-2,4a,5-triaza-fluorene
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|
C16H23N3O
|
2
|
| 1 |
EC50 = 15 nM
|
|
|
| 2 |
Ki = 3.6 nM
|
|
|
|
CP0193993
|
(S)-1-(6-chloro-5-fluoro-1H-indol-1-yl)propan-2-amine
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|
C11H12ClFN2
|
3
|
| 1 |
EC50 = 18 nM
|
|
|
| 2 |
EC50 = 52 nM
|
|
|
| 3 |
Ki = 26 nM
|
|
|
|
CP0380471
|
(R)-9-Chloro-8-trifluoromethyl-2,3,4,4a,5,6-hexahydro-1H-pyrazino[1,2-a]quinoxaline
Show/Hide
|
C12H13ClF3N3
|
1
|
| 1 |
EC50 = 19 nM
|
|
|
|
CP0467130
|
(R)-9-Chloro-8-trifluoromethyl-2,3,4,4a-tetrahydro-1H,6H-pyrazino[1,2-a]quinoxalin-5-one
Show/Hide
|
C12H11ClF3N3O
|
1
|
| 1 |
EC50 = 19 nM
|
|
|
|
CP0383093
|
(S)-2-(6-Ethylsulfanyl-5-fluoro-2,3-dihydro-indol-1-yl)-1-methyl-ethylamine
Show/Hide
|
C13H19FN2S
|
1
|
| 1 |
EC50 = 21 nM
|
|
|
|
CP0374112
|
(R)-2-(2-chlorophenethyl)-3-methyl-6-(2-methylpiperazin-1-yl)pyrimidin-4(3H)-one
Show/Hide
|
C18H23ClN4O
|
1
|
| 1 |
EC50 = 21 nM
|
|
|
|
CP0397150
|
2-(2-chlorophenethyl)-3-ethyl-6-(piperazin-1-yl)pyrimidin-4(3H)-one
Show/Hide
|
C18H23ClN4O
|
1
|
| 1 |
EC50 = 21 nM
|
|
|
|
CP0046618
|
1-(3-chlorophenyl)piperazine
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|
C10H13ClN2
|
2
|
| 1 |
EC50 = 26 nM
|
|
|
| 2 |
EC50 = 170 nM
|
|
|
|
CP0403844
|
(S)-1-Methyl-2-(6-methylsulfanyl-2,3-dihydro-indol-1-yl)-ethylamine
Show/Hide
|
C12H18N2S
|
1
|
| 1 |
EC50 = 26 nM
|
|
|
|
CP0498876
|
2-(4-cyclopropylbenzyl)-6,7,8,9-tetrahydro-2H-pyridazino[4,3-d]azepin-3(5H)-one
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|
C18H21N3O
|
1
|
| 1 |
EC50 = 26 nM
|
|
|
|
CP0447556
|
(R)-3-methyl-2-(2-methylphenethyl)-6-(2-methylpiperazin-1-yl)pyrimidin-4(3H)-one
Show/Hide
|
C19H26N4O
|
1
|
| 1 |
EC50 = 26 nM
|
|
|
|
CP0452589
|
(R)-2-(3-chlorophenethyl)-3-methyl-6-(2-methylpiperazin-1-yl)pyrimidin-4(3H)-one
Show/Hide
|
C18H23ClN4O
|
1
|
| 1 |
EC50 = 26 nM
|
|
|
|
CP0378061
|
(S)-1-Methyl-2-(2,3,8,9-tetrahydro-7H-pyrano[2,3-g]indol-1-yl)-ethylamine
Show/Hide
|
C14H20N2O
|
1
|
| 1 |
EC50 = 28 nM
|
|
|
|
CP0485399
|
2-(3-chlorobenzyl)-6,7,8,9-tetrahydro-2H-pyridazino[4,3-d]azepin-3(5H)-one
Show/Hide
|
C15H16ClN3O
|
1
|
| 1 |
EC50 = 30 nM
|
|
|
|
CP0452587
|
3-methyl-6-(piperazin-1-yl)-2-((2-(trifluoromethyl)phenoxy)methyl)pyrimidin-4(3H)-one
Show/Hide
|
C17H19F3N4O2
|
1
|
| 1 |
EC50 = 30 nM
|
|
|
|
CP0495879
|
(S)-2-(6-Chloro-5-fluoro-2,3-dihydro-indol-1-yl)-1-methyl-ethylamine
Show/Hide
|
C11H14ClFN2
|
1
|
| 1 |
EC50 = 31 nM
|
|
|
|
CP0421550
|
2-benzyl-6,7,8,9-tetrahydro-2H-pyridazino[4,3-d]azepin-3(5H)-one
Show/Hide
|
C15H17N3O
|
1
|
| 1 |
EC50 = 31 nM
|
|
|
|
CP0430980
|
2-(4-chlorobenzyl)-6,7,8,9-tetrahydro-2H-pyridazino[4,3-d]azepin-3(5H)-one
Show/Hide
|
C15H16ClN3O
|
1
|
| 1 |
EC50 = 31 nM
|
|
|
|
CP0520516
|
2-(2-chlorobenzyl)-6,7,8,9-tetrahydro-2H-pyridazino[4,3-d]azepin-3(5H)-one
Show/Hide
|
C15H16ClN3O
|
1
|
| 1 |
EC50 = 33 nM
|
|
|
|
CP0432833
|
(S)-2-(6-Ethylsulfanyl-2,3-dihydro-indol-1-yl)-1-methyl-ethylamine
Show/Hide
|
C13H20N2S
|
1
|
| 1 |
EC50 = 40 nM
|
|
|
|
CP0104535
|
(S)-N-(benzo[d][1,3]dioxol-5-ylmethyl)-1-(1H-pyrrolo[2,3-f]quinolin-1-yl)propan-2-amine
Show/Hide
|
C22H21N3O2
|
1
|
| 1 |
EC50 = 42 nM
|
|
|
|
CP0081902
|
(S)-2-(6-Bromo-2,3-dihydro-indol-1-yl)-1-methyl-ethylamine
Show/Hide
|
C11H15BrN2
|
1
|
| 1 |
EC50 = 44 nM
|
|
|
|
CP0403843
|
(S)-2-(6-Chloro-2,3-dihydro-indol-1-yl)-1-methyl-ethylamine
Show/Hide
|
C11H15ClN2
|
1
|
| 1 |
EC50 = 44 nM
|
|
|
|
CP0408598
|
(S)-8,9-Dichloro-2,3,4,4a,5,6-hexahydro-1H-pyrazino[1,2-a]quinoxaline
Show/Hide
|
C11H13Cl2N3
|
1
|
| 1 |
EC50 = 45 nM
|
|
|
|
CP0452588
|
2-((5-fluoro-2-methylphenoxy)methyl)-3-methyl-6-(piperazin-1-yl)pyrimidin-4(3H)-one
Show/Hide
|
C17H21FN4O2
|
1
|
| 1 |
EC50 = 46 nM
|
|
|
|
CP0156756
|
(R)-6-(2-methylpiperazin-1-yl)-2-(2-(2-(trifluoromethyl)phenoxy)ethyl)pyridazin-3(2H)-one
Show/Hide
|
C18H21F3N4O2
|
1
|
| 1 |
EC50 = 47 nM
|
|
|
|
CP0457521
|
2-(4-(trifluoromethoxy)benzyl)-6,7,8,9-tetrahydro-2H-pyridazino[4,3-d]azepin-3(5H)-one
Show/Hide
|
C16H16F3N3O2
|
1
|
| 1 |
EC50 = 48 nM
|
|
|
|
CP0511112
|
(R)-8,9-Dichloro-2,3,4,4a,5,6-hexahydro-1H-pyrazino[1,2-a]quinoxaline
Show/Hide
|
C11H13Cl2N3
|
1
|
| 1 |
EC50 = 49 nM
|
|
|
|
CP0172896
|
(S)-N-(naphthalen-2-ylmethyl)-1-(1H-pyrrolo[2,3-f]quinolin-1-yl)propan-2-amine
Show/Hide
|
C25H23N3
|
1
|
| 1 |
EC50 = 52 nM
|
|
|
|
CP0447561
|
3-(3-(2-chlorophenoxy)propyl)-6-methyl-2-(piperazin-1-yl)pyrimidin-4(1H)-one
Show/Hide
|
C18H23ClN4O2
|
1
|
| 1 |
EC50 = 56 nM
|
|
|
|
CP0397104
|
2-isopentyl-6,7,8,9-tetrahydro-2H-pyridazino[4,3-d]azepin-3(5H)-one
Show/Hide
|
C13H21N3O
|
1
|
| 1 |
EC50 = 62 nM
|
|
|
|
CP0377332
|
(S)-2-(5-Fluoro-6-iodo-2,3-dihydro-indol-1-yl)-1-methyl-ethylamine
Show/Hide
|
C11H14FIN2
|
1
|
| 1 |
EC50 = 64 nM
|
|
|
|
CP0485270
|
(R)-3-methyl-6-(2-methylpiperazin-1-yl)-2-(2-(trifluoromethyl)phenethyl)pyrimidin-4(3H)-one
Show/Hide
|
C19H23F3N4O
|
1
|
| 1 |
EC50 = 64 nM
|
|
|
|
CP0849995
|
4-(3-Chlorophenyl)-1,2,3,6-tetrahydropyridinium chloride
Show/Hide
|
C11H13Cl2N
|
3
|
| 1 |
EC50 = 72.3 nM
|
|
|
| 2 |
Ki = 280 nM
|
|
|
| 3 |
Ki = 318 nM
|
|
|
|
CP0034922
|
(S)-1-(1H-pyrrolo[3,2-h]isoquinolin-1-yl)propan-2-amine
Show/Hide
|
C14H15N3
|
1
|
| 1 |
EC50 = 73 nM
|
|
|
|
CP0510615
|
2-((2-chlorophenoxy)methyl)-3-methyl-6-(piperazin-1-yl)pyrimidin-4(3H)-one
Show/Hide
|
C16H19ClN4O2
|
1
|
| 1 |
EC50 = 73 nM
|
|
|
|
CP0034918
|
(S)-N-(2-chlorobenzyl)-1-(1H-pyrrolo[2,3-f]quinolin-1-yl)propan-2-amine
Show/Hide
|
C21H20ClN3
|
1
|
| 1 |
EC50 = 74 nM
|
|
|
|
CP0457541
|
3-(3-(2-fluorophenoxy)propyl)-6-methyl-2-(piperazin-1-yl)pyrimidin-4(3H)-one
Show/Hide
|
C18H23FN4O2
|
1
|
| 1 |
EC50 = 77 nM
|
|
|
|
CP0424572
|
(R)-9-Chloro-2,3,4,4a-tetrahydro-1H,6H-pyrazino[1,2-a]quinoxalin-5-one
Show/Hide
|
C11H12ClN3O
|
1
|
| 1 |
EC50 = 86 nM
|
|
|
|
CP0447559
|
2-(3-chlorophenethyl)-3-methyl-6-(piperazin-1-yl)pyrimidin-4(3H)-one
Show/Hide
|
C17H21ClN4O
|
1
|
| 1 |
EC50 = 96 nM
|
|
|
|
CP0034920
|
(S)-1-(1H-pyrrolo[3,2-h]quinolin-1-yl)propan-2-amine
Show/Hide
|
C14H15N3
|
1
|
| 1 |
EC50 = 97 nM
|
|
|
|
CP0452592
|
2-((2-chloro-5-fluorophenoxy)methyl)-3-ethyl-6-(piperazin-1-yl)pyrimidin-4(3H)-one
Show/Hide
|
C17H20ClFN4O2
|
1
|
| 1 |
EC50 = 103 nM
|
|
|
|
CP0535219
|
2-(2-(trifluoromethoxy)benzyl)-6,7,8,9-tetrahydro-2H-pyridazino[4,3-d]azepin-3(5H)-one
Show/Hide
|
C16H16F3N3O2
|
1
|
| 1 |
EC50 = 107 nM
|
|
|
|
CP0452591
|
3-((1-ethyl-6-oxo-4-(piperazin-1-yl)-1,6-dihydropyrimidin-2-yl)methoxy)benzonitrile
Show/Hide
|
C18H21N5O2
|
1
|
| 1 |
EC50 = 112 nM
|
|
|
|
CP0394571
|
2-(4-chloro-2-methylphenoxy)propanoic acid
Show/Hide
|
C10H11ClO3
|
1
|
| 1 |
EC50 = 120 nM
|
|
|
|
CP0494718
|
2-(4-(trifluoromethyl)benzyl)-6,7,8,9-tetrahydro-2H-pyridazino[4,3-d]azepin-3(5H)-one
Show/Hide
|
C16H16F3N3O
|
1
|
| 1 |
EC50 = 125 nM
|
|
|
|
CP0875251
|
4-(1H-Indol-3-yl)piperidinium chloride
Show/Hide
|
C13H17ClN2
|
3
|
| 1 |
EC50 = 128 nM
|
|
|
| 2 |
Ki = 366 nM
|
|
|
| 3 |
Ki = 612 nM
|
|
|
|
CP0383092
|
(S)-2-(5-Fluoro-6-trifluoromethyl-2,3-dihydro-indol-1-yl)-1-methyl-ethylamine
Show/Hide
|
C12H14F4N2
|
1
|
| 1 |
EC50 = 130 nM
|
|
|
|
CP0515912
|
9-Chloro-8-trifluoromethyl-2,3,4,4a-tetrahydro-1H,6H-pyrazino[1,2-a]quinoxalin-5-one
Show/Hide
|
C12H11ClF3N3O
|
1
|
| 1 |
EC50 = 136 nM
|
|
|
|
CP0870789
|
4-(3-Trifluoromethylphenyl)-1,2,3,6-tetrahydropyridinium chloride
Show/Hide
|
C12H13ClF3N
|
3
|
| 1 |
EC50 = 158 nM
|
|
|
| 2 |
Ki = 298 nM
|
|
|
| 3 |
Ki = 365 nM
|
|
|
|
CP0452590
|
2-((5-chloro-2-methylphenoxy)methyl)-3-methyl-6-(piperazin-1-yl)pyrimidin-4(3H)-one
Show/Hide
|
C17H21ClN4O2
|
1
|
| 1 |
EC50 = 160 nM
|
|
|
|
CP0447555
|
6-methyl-2-((R)-2-methylpiperazin-1-yl)-3-(3-phenoxypropyl)pyrimidin-4(1H)-one
Show/Hide
|
C19H26N4O2
|
1
|
| 1 |
EC50 = 163 nM
|
|
|
|
CP0915711
|
4-(1H-indol-3-yl)-1,2,3,6-tetrahydropyridinium chloride
Show/Hide
|
C13H15ClN2
|
3
|
| 1 |
EC50 = 163 nM
|
|
|
| 2 |
Ki = 296 nM
|
|
|
| 3 |
Ki = 632 nM
|
|
|
|
CP0524028
|
3-(benzyloxy)-1,4,5,6,7,8-hexahydropyrazolo[4,3-d]azepine
Show/Hide
|
C14H17N3O
|
1
|
| 1 |
EC50 = 176 nM
|
|
|
|
CP0216287
|
(S)-N-benzyl-1-(1H-pyrrolo[2,3-f]quinolin-1-yl)propan-2-amine
Show/Hide
|
C21H21N3
|
1
|
| 1 |
EC50 = 200 nM
|
|
|
|
CP0272372
|
(2-methyl-benzyl)-((S)-1-methyl-2-pyrrolo[2,3-f]quinolin-1-yl-ethyl)-amine
Show/Hide
|
C22H23N3
|
1
|
| 1 |
EC50 = 219 nM
|
|
|
|
CP0374110
|
3-methyl-6-(piperazin-1-yl)-2-(o-tolyloxymethyl)pyrimidin-4(3H)-one
Show/Hide
|
C17H22N4O2
|
1
|
| 1 |
EC50 = 228 nM
|
|
|
|
CP0034925
|
(S)-N-(1-(1H-pyrrolo[2,3-f]quinolin-1-yl)propan-2-yl)prop-2-en-1-amine
Show/Hide
|
C17H19N3
|
1
|
| 1 |
EC50 = 257 nM
|
|
|
|
CP0373280
|
3-(3-(3-chlorophenoxy)propyl)-6-methyl-2-(piperazin-1-yl)pyrimidin-4(1H)-one
Show/Hide
|
C18H23ClN4O2
|
1
|
| 1 |
EC50 = 262 nM
|
|
|
|
CP0397149
|
(R)-3-methyl-6-(2-methylpiperazin-1-yl)-2-phenethylpyrimidin-4(3H)-one
Show/Hide
|
C18H24N4O
|
1
|
| 1 |
EC50 = 262 nM
|
|
|
|
CP0452593
|
3-methyl-2-phenethyl-6-(piperazin-1-yl)pyrimidin-4(3H)-one
Show/Hide
|
C17H22N4O
|
1
|
| 1 |
EC50 = 275 nM
|
|
|
|
CP0439313
|
(S)-8,9-Dichloro-2,3,4,4a-tetrahydro-1H,6H-pyrazino[1,2-a]quinoxalin-5-one
Show/Hide
|
C11H11Cl2N3O
|
1
|
| 1 |
EC50 = 290 nM
|
|
|
|
CP0034919
|
(S)-1-(1H-pyrrolo[2,3-f]isoquinolin-1-yl)propan-2-amine
Show/Hide
|
C14H15N3
|
1
|
| 1 |
EC50 = 297 nM
|
|
|
|
CP0415695
|
3-((1-methyl-6-oxo-4-(piperazin-1-yl)-1,6-dihydropyrimidin-2-yl)methoxy)benzonitrile
Show/Hide
|
C17H19N5O2
|
1
|
| 1 |
EC50 = 319 nM
|
|
|
|
CP0520515
|
2-methyl-6,7,8,9-tetrahydro-2H-pyridazino[4,3-d]azepin-3(5H)-one
Show/Hide
|
C9H13N3O
|
1
|
| 1 |
EC50 = 338 nM
|
|
|
|
CP0255556
|
(S)-N-(cyclohexylmethyl)-1-(1H-pyrrolo[2,3-f]quinolin-1-yl)propan-2-amine
Show/Hide
|
C21H27N3
|
1
|
| 1 |
EC50 = 348 nM
|
|
|
|
CP0388336
|
2-((2-chloro-5-fluorophenoxy)methyl)-3-methyl-6-(piperazin-1-yl)pyrimidin-4(3H)-one
Show/Hide
|
C16H18ClFN4O2
|
1
|
| 1 |
EC50 = 361 nM
|
|
|
|
CP0535404
|
3-methyl-6-(piperazin-1-yl)-2-((3-(trifluoromethyl)phenoxy)methyl)pyrimidin-4(3H)-one
Show/Hide
|
C17H19F3N4O2
|
1
|
| 1 |
EC50 = 487 nM
|
|
|
|
CP0447560
|
2-((3-chlorophenoxy)methyl)-3-methyl-6-(piperazin-1-yl)pyrimidin-4(3H)-one
Show/Hide
|
C16H19ClN4O2
|
1
|
| 1 |
EC50 = 493 nM
|
|
|
|
CP0034921
|
(S)-N-(2-methoxybenzyl)-1-(1H-pyrrolo[2,3-f]quinolin-1-yl)propan-2-amine
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C22H23N3O
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1
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| 1 |
EC50 = 551 nM
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CP0867391
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4-(3-Chlorophenyl)piperidinium trifluoroacetate
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C13H15ClF3NO2
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3
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| 1 |
EC50 = 790 nM
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| 2 |
Ki = 931 nM
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| 3 |
Ki = 1430 nM
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CP0498721
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3-(3-(4-chlorophenoxy)propyl)-6-methyl-2-(piperazin-1-yl)pyrimidin-4(1H)-one
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C18H23ClN4O2
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1
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| 1 |
EC50 = 899 nM
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CP0469882
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6-methyl-3-(3-phenoxypropyl)-2-(piperazin-1-yl)pyrimidin-4(3H)-one
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C18H24N4O2
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1
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| 1 |
EC50 = 1020 nM
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CP0875255
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4-(3-Trifluoromethylphenyl)piperidinium chloride
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C12H15ClF3N
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2
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| 1 |
EC50 = 1260 nM
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| 2 |
Ki = 1550 nM
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CP0915713
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4-(4-Chlorophenyl)-1,2,3,6-tetrahydropyridinium chloride
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C11H13Cl2N
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2
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| 1 |
EC50 = 1760 nM
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| 2 |
Ki = 3100 nM
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CP0877858
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4-(3-Methylphenyl)piperidinium chloride
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C12H18ClN
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2
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| 1 |
EC50 = 1995 nM
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| 2 |
Ki = 3130 nM
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CP0887579
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SID26659403
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C11H14ClN
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2
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| 1 |
EC50 = 2450 nM
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| 2 |
Ki = 7180 nM
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CP0503510
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(S)-9-Chloro-8-trifluoromethyl-2,3,4,4a-tetrahydro-1H,6H-pyrazino[1,2-a]quinoxalin-5-one
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C12H11ClF3N3O
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1
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| 1 |
EC50 = 2600 nM
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CP0494719
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2-benzyl-1-methyl-1,2,5,6,7,8-hexahydropyrazolo[4,3-d]azepin-3(4H)-one
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C15H19N3O
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1
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| 1 |
EC50 = 2930 nM
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CP0875257
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4-(4-Bromophenyl)-1,2,3,6-tetrahydropyridinium chloride
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C11H13BrClN
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2
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| 1 |
EC50 = 3520 nM
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| 2 |
Ki = 2540 nM
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CP0477779
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2-benzyl-2,4,5,6,7,8-hexahydropyrazolo[4,3-d]azepine
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C14H17N3
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1
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| 1 |
EC50 = 4980 nM
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CP0494731
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4-((3-oxo-3,5,6,7,8,9-hexahydro-2H-pyridazino[4,3-d]azepin-2-yl)methyl)benzonitrile
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C16H16N4O
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1
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| 1 |
EC50 = 6630 nM
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CP0439985
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1-benzyl-1,2,5,6,7,8-hexahydropyrazolo[4,3-d]azepin-3(4H)-one
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C14H17N3O
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1
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| 1 |
EC50 > 10000 nM
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CP0469839
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2-benzyl-1,2,5,6,7,8-hexahydropyrazolo[4,3-d]azepin-3(4H)-one
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C14H17N3O
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1
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| 1 |
EC50 > 10000 nM
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CP0477780
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1-benzyl-1,4,5,6,7,8-hexahydropyrazolo[4,3-d]azepine
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C14H17N3
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1
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| 1 |
EC50 > 10000 nM
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CP0524025
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2-(2-phenoxyethyl)-6,7,8,9-tetrahydro-2H-pyridazino[4,3-d]azepin-3(5H)-one
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C16H19N3O2
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1
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| 1 |
EC50 > 10000 nM
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CP0535393
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2-phenyl-6,7,8,9-tetrahydro-2H-pyridazino[4,3-d]azepin-3(5H)-one
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C14H15N3O
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1
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| 1 |
EC50 > 10000 nM
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CP0447554
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3-(3-(4-fluorophenoxy)propyl)-6-methyl-2-(piperazin-1-yl)pyrimidin-4(1H)-one
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C18H23FN4O2
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1
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| 1 |
EC50 > 10000 nM
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CP0469885
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6-methyl-3-(3-phenylpropyl)-2-(piperazin-1-yl)pyrimidin-4(3H)-one
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C18H24N4O
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1
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| 1 |
EC50 > 10000 nM
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CP0469886
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3-(3-(benzyloxy)propyl)-6-methyl-2-(piperazin-1-yl)pyrimidin-4(3H)-one
Show/Hide
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C19H26N4O2
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1
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| 1 |
EC50 > 10000 nM
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CP0469887
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2-((4-chlorophenoxy)methyl)-3-methyl-6-(piperazin-1-yl)pyrimidin-4(3H)-one
Show/Hide
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C16H19ClN4O2
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1
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| 1 |
EC50 > 10000 nM
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CP0526909
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3-(3-(3-fluorophenoxy)propyl)-6-methyl-2-(piperazin-1-yl)pyrimidin-4(1H)-one
Show/Hide
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C18H23FN4O2
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1
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| 1 |
EC50 > 10000 nM
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CP0535388
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6-(3-chlorophenethyl)-3-methyl-2-(piperazin-1-yl)pyrimidin-4(3H)-one
Show/Hide
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C17H21ClN4O
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1
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| 1 |
EC50 > 10000 nM
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CP0535405
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3-methyl-6-(piperazin-1-yl)-2-((4-(trifluoromethyl)phenoxy)methyl)pyrimidin-4(3H)-one
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C17H19F3N4O2
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1
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| 1 |
EC50 > 10000 nM
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CP0006743
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4-methoxy-N-(2,4,6-trimethylphenyl)benzenesulfonamide
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C16H19NO3S
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2
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| 1 |
EC50 > 39810.72 nM
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| 2 |
IC50 > 39810.72 nM
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CP0428326
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4-(4-fluorophenyl)-N-[6-(pyrrolidin-1-ylmethyl)-7,8-dihydronaphthalen-2-yl]benzamide
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C28H27FN2O
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1
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| 1 |
IC50 = 0.53 nM
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CP0105756
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1-(17-chloro-3-oxa-2-azatetracyclo[12.4.0.02,6.07,12]octadeca-1(14),7,9,11,15,17-hexaen-4-yl)-N,N-dimethylmethanamine
Show/Hide
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C19H21ClN2O
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1
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| 1 |
IC50 = 1.047 nM
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CP0134845
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1-(17-fluoro-3-oxa-2-azatetracyclo[12.4.0.02,6.07,12]octadeca-1(14),7,9,11,15,17-hexaen-4-yl)-N,N-dimethylmethanamine
Show/Hide
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C19H21FN2O
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1
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| 1 |
IC50 = 1.148 nM
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CP0123725
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N,N-dimethyl-1-(17-methyl-3-oxa-2-azatetracyclo[12.4.0.02,6.07,12]octadeca-1(14),7,9,11,15,17-hexaen-4-yl)methanamine
Show/Hide
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C20H24N2O
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1
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| 1 |
IC50 = 3.02 nM
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CP0423539
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4-(4-fluorophenyl)-N-[3-(pyrrolidin-1-ylmethyl)-2H-chromen-7-yl]benzamide
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C27H25FN2O2
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1
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| 1 |
IC50 = 3.1 nM
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CP0400980
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1-(17-chloro-3,13-dioxa-2-azatetracyclo[12.4.0.02,6.07,12]octadeca-1(14),7,9,11,15,17-hexaen-4-yl)-N,N-dimethylmethanamine
Show/Hide
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C18H19ClN2O2
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1
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| 1 |
IC50 = 3.802 nM
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CP0464885
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N,N-dimethyl-1-(15-methyl-3-oxa-2-azatetracyclo[12.4.0.02,6.07,12]octadeca-1(18),7,9,11,14,16-hexaen-4-yl)methanamine
Show/Hide
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C20H24N2O
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1
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| 1 |
IC50 = 3.89 nM
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CP0393174
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1-(16-fluoro-3-oxa-2-azatetracyclo[12.4.0.02,6.07,12]octadeca-1(14),7,9,11,15,17-hexaen-4-yl)-N,N-dimethylmethanamine
Show/Hide
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C19H21FN2O
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1
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| 1 |
IC50 = 4.677 nM
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CP0453941
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1-(15-fluoro-3-oxa-2-azatetracyclo[12.4.0.02,6.07,12]octadeca-1(14),7,9,11,15,17-hexaen-4-yl)-N,N-dimethylmethanamine
Show/Hide
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C19H21FN2O
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1
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| 1 |
IC50 = 5.012 nM
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CP0467988
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3-oxa-2-azatetracyclo[12.4.0.02,6.07,12]octadeca-1(18),7,9,11,14,16-hexaen-4-ylmethanamine
Show/Hide
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C17H18N2O
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1
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| 1 |
IC50 = 5.623 nM
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CP0091879
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1-(9,17-difluoro-3-oxa-2-azatetracyclo[12.4.0.02,6.07,12]octadeca-1(14),7(12),8,10,15,17-hexaen-4-yl)-N,N-dimethylmethanamine
Show/Hide
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C19H20F2N2O
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1
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| 1 |
IC50 = 6.166 nM
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CP0497647
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N,N-dimethyl-1-(10-methyl-3-oxa-2-azatetracyclo[12.4.0.02,6.07,12]octadeca-1(18),7(12),8,10,14,16-hexaen-4-yl)methanamine
Show/Hide
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C20H24N2O
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1
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| 1 |
IC50 = 6.31 nM
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CP0183894
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N-methyl-1-(3-oxa-2-azatetracyclo[12.4.0.02,6.07,12]octadeca-1(18),7,9,11,14,16-hexaen-4-yl)methanamine
Show/Hide
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C18H20N2O
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1
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| 1 |
IC50 = 7.079 nM
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CP0416915
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4-(4-fluorophenyl)-N-[6-methyl-3-(pyrrolidin-1-ylmethyl)quinolin-7-yl]benzamide
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C28H26FN3O
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1
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| 1 |
IC50 = 7.4 nM
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CP0026495
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CHEBI:51137
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C18H20N2
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1
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| 1 |
IC50 = 7.413 nM
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CP0392920
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N,N-dimethyl-1-[8-(trifluoromethyl)-3-oxa-2-azatetracyclo[12.4.0.02,6.07,12]octadeca-1(18),7(12),8,10,14,16-hexaen-4-yl]methanamine
Show/Hide
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C20H21F3N2O
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1
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| 1 |
IC50 = 7.586 nM
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CP0497667
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1-(18-chloro-3-oxa-2-azatetracyclo[12.4.0.02,6.07,12]octadeca-1(14),7,9,11,15,17-hexaen-4-yl)-N,N-dimethylmethanamine
Show/Hide
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C19H21ClN2O
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1
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| 1 |
IC50 = 10.23 nM
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CP0464753
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1-(9-fluoro-3-oxa-2-azatetracyclo[12.4.0.02,6.07,12]octadeca-1(18),7(12),8,10,14,16-hexaen-4-yl)-N,N-dimethylmethanamine
Show/Hide
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C19H21FN2O
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1
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| 1 |
IC50 = 10.72 nM
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CP0431008
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N,N-dimethyl-1-(17-phenyl-3-oxa-2-azatetracyclo[12.4.0.02,6.07,12]octadeca-1(14),7,9,11,15,17-hexaen-4-yl)methanamine
Show/Hide
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C25H26N2O
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1
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| 1 |
IC50 = 11.22 nM
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CP0405608
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1-(11-fluoro-3-oxa-2-azatetracyclo[12.4.0.02,6.07,12]octadeca-1(18),7(12),8,10,14,16-hexaen-4-yl)-N,N-dimethylmethanamine
Show/Hide
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C19H21FN2O
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1
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| 1 |
IC50 = 11.75 nM
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CP0734983
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Dimethyl-(2,3,3a,8-tetrahydro-1-oxa-12b-aza-dibenzo[e,h]azulen-2-ylmethyl)-amine
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C19H22N2O
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1
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| 1 |
IC50 = 12.3 nM
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CP0402198
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N-ethyl-N-(3-oxa-2-azatetracyclo[12.4.0.02,6.07,12]octadeca-1(18),7,9,11,14,16-hexaen-4-ylmethyl)ethanamine
Show/Hide
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C21H26N2O
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1
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| 1 |
IC50 = 14.45 nM
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CP0384022
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4-(pyrrolidin-1-ylmethyl)-3-oxa-2-azatetracyclo[12.4.0.02,6.07,12]octadeca-1(18),7,9,11,14,16-hexaene
Show/Hide
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C21H24N2O
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1
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| 1 |
IC50 = 16.22 nM
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CP0438133
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N,N-dimethyl-3-(3-oxa-2-azatetracyclo[12.4.0.02,6.07,12]octadeca-1(18),7,9,11,14,16-hexaen-4-yl)propan-1-amine
Show/Hide
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C21H26N2O
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1
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| 1 |
IC50 = 18.62 nM
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CP0372936
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1-(9-methoxy-3-oxa-2-azatetracyclo[12.4.0.02,6.07,12]octadeca-1(18),7(12),8,10,14,16-hexaen-4-yl)-N,N-dimethylmethanamine
Show/Hide
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C20H24N2O2
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1
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| 1 |
IC50 = 19.5 nM
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CP0435998
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N,N-dimethyl-1-(8-methyl-3-oxa-2-azatetracyclo[12.4.0.02,6.07,12]octadeca-1(18),7,9,11,14,16-hexaen-4-yl)methanamine
Show/Hide
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C20H24N2O
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1
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| 1 |
IC50 = 30.2 nM
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CP0417492
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4-(4-fluorophenyl)-N-[2-(pyrrolidin-1-ylmethyl)quinolin-6-yl]benzamide
Show/Hide
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C27H24FN3O
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1
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| 1 |
IC50 = 36 nM
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CP0094561
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N,N-dimethyl-2-(3-oxa-2-azatetracyclo[12.4.0.02,6.07,12]octadeca-1(18),7,9,11,14,16-hexaen-4-yl)ethanamine
Show/Hide
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C20H24N2O
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1
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| 1 |
IC50 = 37.15 nM
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CP0439248
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2-{3-[(3-Chlorophenyl)sulfonyl]-1H-pyrrolo[2,3-b]pyridin-1-yl}ethylamine
Show/Hide
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C15H14ClN3O2S
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1
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| 1 |
IC50 = 44 nM
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CP0462673
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4-(4-chlorophenyl)-N-[3-(pyrrolidin-1-ylmethyl)quinolin-7-yl]piperidine-1-carboxamide
Show/Hide
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C26H29ClN4O
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1
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| 1 |
IC50 = 55 nM
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CP0417495
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4-(4-fluorophenyl)-N-[8-fluoro-3-(pyrrolidin-1-ylmethyl)quinolin-7-yl]benzamide
Show/Hide
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C27H23F2N3O
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1
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| 1 |
IC50 = 78 nM
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CP0417491
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4-(4-fluorophenyl)-N-[6-(pyrrolidin-1-ylmethyl)naphthalen-2-yl]benzamide
Show/Hide
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C28H25FN2O
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1
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| 1 |
IC50 = 120 nM
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CP0461934
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4-(4-fluorophenyl)-N-[3-(pyrrolidin-1-ylmethyl)quinolin-7-yl]benzamide
Show/Hide
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C27H24FN3O
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1
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| 1 |
IC50 = 160 nM
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CP0416914
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N-[6-chloro-3-(pyrrolidin-1-ylmethyl)quinolin-7-yl]-4-(4-fluorophenyl)benzamide
Show/Hide
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C27H23ClFN3O
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1
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| 1 |
IC50 = 240 nM
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CP0460839
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4-(4-fluorophenyl)-N-[6-fluoro-3-(pyrrolidin-1-ylmethyl)quinolin-7-yl]benzamide
Show/Hide
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C27H23F2N3O
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1
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| 1 |
IC50 = 280 nM
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CP0417493
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4-phenyl-N-[3-(pyrrolidin-1-ylmethyl)quinolin-7-yl]benzamide
Show/Hide
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C27H25N3O
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1
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| 1 |
IC50 = 310 nM
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CP0392599
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N-(3-oxa-2-azatetracyclo[12.4.0.02,6.07,12]octadeca-1(18),7,9,11,14,16-hexaen-4-ylmethyl)-N-propan-2-ylpropan-2-amine
Show/Hide
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C23H30N2O
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1
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| 1 |
IC50 = 323.59 nM
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CP0404509
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N,N-dimethyl-1-[11-(trifluoromethyl)-3-oxa-2-azatetracyclo[12.4.0.02,6.07,12]octadeca-1(18),7(12),8,10,14,16-hexaen-4-yl]methanamine
Show/Hide
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C20H21F3N2O
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1
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| 1 |
IC50 = 436.52 nM
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CP0405688
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2-[3-(3-chlorophenyl)sulfonylpyrrolo[2,3-b]pyridin-1-yl]-N,N-dimethylethanamine
Show/Hide
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C17H18ClN3O2S
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1
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| 1 |
IC50 = 477 nM
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CP0458174
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4-(4-methylphenyl)-N-[8-methyl-3-(pyrrolidin-1-ylmethyl)quinolin-7-yl]benzamide
Show/Hide
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C29H29N3O
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1
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| 1 |
IC50 = 540 nM
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CP0489268
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6-(4-methylphenyl)-N-[3-(pyrrolidin-1-ylmethyl)quinolin-7-yl]pyridine-3-carboxamide
Show/Hide
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C27H26N4O
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1
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| 1 |
IC50 = 570 nM
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CP0211700
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1H-indole-3-carboxylic acid[6-(2-chloro-pyridin-3-yloxy)-pyridin-3-yl]-amide
Show/Hide
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C19H13ClN4O2
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1
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| 1 |
IC50 = 590 nM
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CP0417494
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4-(4-chlorophenyl)-N-[3-(pyrrolidin-1-ylmethyl)quinolin-7-yl]benzamide
Show/Hide
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C27H24ClN3O
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1
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| 1 |
IC50 = 630 nM
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CP0380100
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2-(3-(3-fluorophenylsulfonyl)-1H-pyrrolo[2,3-b]pyridin-1-yl)-N,N-dimethylethanamine
Show/Hide
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C17H18FN3O2S
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1
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| 1 |
IC50 = 644 nM
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CP0432922
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4-(4-methylphenyl)-N-[3-(pyrrolidin-1-ylmethyl)quinolin-7-yl]benzamide
Show/Hide
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C28H27N3O
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1
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| 1 |
IC50 = 660 nM
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CP0437491
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2,2,2-trifluoro-N-methyl-N-(3-oxa-2-azatetracyclo[12.4.0.02,6.07,12]octadeca-1(18),7,9,11,14,16-hexaen-4-ylmethyl)acetamide
Show/Hide
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C20H19F3N2O2
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1
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| 1 |
IC50 = 691.83 nM
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CP0458237
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N-[8-methyl-3-(pyrrolidin-1-ylmethyl)quinolin-7-yl]-4-phenylbenzamide
Show/Hide
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C28H27N3O
|
1
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| 1 |
IC50 = 760 nM
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CP0460837
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6-(4-fluorophenyl)-N-[3-(pyrrolidin-1-ylmethyl)quinolin-7-yl]pyridine-3-carboxamide
Show/Hide
|
C26H23FN4O
|
1
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| 1 |
IC50 = 830 nM
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CP0423540
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6-(4-chlorophenyl)-N-[3-(pyrrolidin-1-ylmethyl)quinolin-7-yl]pyridine-3-carboxamide
Show/Hide
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C26H23ClN4O
|
1
|
| 1 |
IC50 = 930 nM
|
|
|
|
CP0419036
|
N,N-dimethyl-2-(3-naphthalen-1-ylsulfonylpyrrolo[2,3-b]pyridin-1-yl)ethanamine
Show/Hide
|
C21H21N3O2S
|
1
|
| 1 |
IC50 = 1135 nM
|
|
|
|
CP0421446
|
4-[(4-methylpiperazin-1-yl)methyl]-3-oxa-2-azatetracyclo[12.4.0.02,6.07,12]octadeca-1(18),7,9,11,14,16-hexaene
Show/Hide
|
C22H27N3O
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0422415
|
4-[[4-(3-chlorophenyl)piperazin-1-yl]methyl]-3-oxa-2-azatetracyclo[12.4.0.02,6.07,12]octadeca-1(18),7,9,11,14,16-hexaene
Show/Hide
|
C27H28ClN3O
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0460072
|
N,N-dimethyl-3-oxa-2-azatetracyclo[12.4.0.02,6.07,12]octadeca-1(18),7,9,11,14,16-hexaene-4-carboxamide
Show/Hide
|
C19H20N2O2
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0461043
|
4-[(4-phenylpiperazin-1-yl)methyl]-3-oxa-2-azatetracyclo[12.4.0.02,6.07,12]octadeca-1(18),7,9,11,14,16-hexaene
Show/Hide
|
C27H29N3O
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0461320
|
2-(3-oxa-2-azatetracyclo[12.4.0.02,6.07,12]octadeca-1(18),7,9,11,14,16-hexaen-4-ylmethyl)isoindole-1,3-dione
Show/Hide
|
C25H20N2O3
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0463614
|
N,N-dimethyl-4-(3-oxa-2-azatetracyclo[12.4.0.02,6.07,12]octadeca-1(18),7,9,11,14,16-hexaen-4-yl)butan-1-amine
Show/Hide
|
C22H28N2O
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0464735
|
4-(piperazin-1-ylmethyl)-3-oxa-2-azatetracyclo[12.4.0.02,6.07,12]octadeca-1(18),7,9,11,14,16-hexaene
Show/Hide
|
C21H25N3O
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0475727
|
4-(morpholin-4-ylmethyl)-3-oxa-2-azatetracyclo[12.4.0.02,6.07,12]octadeca-1(18),7,9,11,14,16-hexaene
Show/Hide
|
C21H24N2O2
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0476618
|
4-(1,3-dihydroisoindol-2-ylmethyl)-3-oxa-2-azatetracyclo[12.4.0.02,6.07,12]octadeca-1(18),7,9,11,14,16-hexaene
Show/Hide
|
C25H24N2O
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0383066
|
1-(11-chloro-3-oxa-2-azatetracyclo[12.4.0.02,6.07,12]octadeca-1(18),7(12),8,10,14,16-hexaen-4-yl)-N,N-dimethylmethanamine
Show/Hide
|
C19H21ClN2O
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0508933
|
1-(8-fluoro-3-oxa-2-azatetracyclo[12.4.0.02,6.07,12]octadeca-1(18),7(12),8,10,14,16-hexaen-4-yl)-N,N-dimethylmethanamine
Show/Hide
|
C19H21FN2O
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0515871
|
N,N-dimethyl-1-[9-(trifluoromethyl)-3-oxa-2-azatetracyclo[12.4.0.02,6.07,12]octadeca-1(18),7(12),8,10,14,16-hexaen-4-yl]methanamine
Show/Hide
|
C20H21F3N2O
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0383206
|
4-(4-fluorophenyl)-N-[8-methyl-3-(pyrrolidin-1-ylmethyl)quinolin-7-yl]benzamide
Show/Hide
|
C28H26FN3O
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0417496
|
4-(4-chlorophenyl)-N-[8-methyl-3-(pyrrolidin-1-ylmethyl)quinolin-7-yl]benzamide
Show/Hide
|
C28H26ClN3O
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0417497
|
4-(4-methoxyphenyl)-N-[8-methyl-3-(pyrrolidin-1-ylmethyl)quinolin-7-yl]benzamide
Show/Hide
|
C29H29N3O2
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0458176
|
4-(4-methoxyphenyl)-N-[3-(pyrrolidin-1-ylmethyl)quinolin-7-yl]benzamide
Show/Hide
|
C28H27N3O2
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0487250
|
N-[8-ethyl-3-(pyrrolidin-1-ylmethyl)quinolin-7-yl]-4-(4-fluorophenyl)benzamide
Show/Hide
|
C29H28FN3O
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0424416
|
2-[3-(Phenylsulfonyl)-1H-pyrrolo[2,3-b]pyridin-1-yl]ethylamine
Show/Hide
|
C15H15N3O2S
|
1
|
| 1 |
IC50 > 5000 nM
|
|
|
|
CP0529512
|
(2S)-1-furo[2,3-g]indazol-1-ylpropan-2-amine
Show/Hide
|
C12H13N3O
|
1
|
| 1 |
Ki = 0.2 nM
|
|
|
|
CP0554015
|
(2S)-1-(7-methylfuro[2,3-g]indazol-1-yl)propan-2-amine
Show/Hide
|
C13H15N3O
|
1
|
| 1 |
Ki = 0.2 nM
|
|
|
|
CP0046703
|
1-(2-{4-[5-chloro-1-(4-fluorophenyl)-1H-indol-3-yl]piperidin-1-yl}ethyl)imidazolidin-2-one
Show/Hide
|
C24H26ClFN4O
|
1
|
| 1 |
Ki = 0.2 nM
|
|
|
|
CP0161466
|
(4R,10aR)-7-Chloro-4,6-dimethyl-1,2,3,4,10,10a-hexahydro-pyrazino[1,2-a]indole
Show/Hide
|
C13H17ClN2
|
1
|
| 1 |
Ki = 0.3 nM
|
|
|
|
CP0373361
|
(2S)-1-(3-methoxyfuro[2,3-g]indazol-1-yl)propan-2-amine
Show/Hide
|
C13H15N3O2
|
1
|
| 1 |
Ki = 0.51 nM
|
|
|
|
CP0080536
|
1-(3-chloro-5,6-dihydrobenzo[b][1]benzothiepin-5-yl)-4-methyl-piperazine;maleate
Show/Hide
|
C19H21ClN2S
|
1
|
| 1 |
Ki = 0.57 nM
|
|
|
|
CP0376381
|
(4R,9aR)-6-bromo-4-methyl-1,2,3,4,9,9a-hexahydro-2,4a,5-triaza-fluorene
Show/Hide
|
C11H14BrN3
|
1
|
| 1 |
Ki = 0.8 nM
|
|
|
|
CP0031743
|
1H-imidazo[4,5-c]pyridine derivative
Show/Hide
|
C18H26N4O2S
|
1
|
| 1 |
Ki = 0.92 nM
|
|
|
|
CP0050128
|
N,N-dimethyl-1-[(2S,4R,6R)-3-oxatetracyclo[12.4.0.02,6.07,12]octadeca-1(18),7,9,11,14,16-hexaen-4-yl]methanamine
Show/Hide
|
C20H23NO
|
1
|
| 1 |
Ki = 0.93 nM
|
|
|
|
CP0094782
|
2-{3-[4-(4-Fluoro-phenyl)-piperazin-1-yl]-propyl}-2H-naphtho[1,8-cd]isothiazole 1,1-dioxide
Show/Hide
|
C23H24FN3O2S
|
1
|
| 1 |
Ki = 1 nM
|
|
|
|
CP0372474
|
1-((S)-2-aminopropyl)-7-fluoro-1H-indazol-6-ol
Show/Hide
|
C10H12FN3O
|
1
|
| 1 |
Ki = 1 nM
|
|
|
|
CP0530334
|
N,N-dimethyl-1-[(4S,6R)-3-oxa-2-azatetracyclo[12.4.0.02,6.07,12]octadeca-1(18),7,9,11,14,16-hexaen-4-yl]methanamine
Show/Hide
|
C19H22N2O
|
1
|
| 1 |
Ki = 1 nM
|
|
|
|
CP0422213
|
1-((S)-2-aminopropyl)-7-chloro-1H-indazol-6-ol
Show/Hide
|
C10H12ClN3O
|
1
|
| 1 |
Ki = 1.2 nM
|
|
|
|
CP0056386
|
5-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-6-chloroindolin-2-one
Show/Hide
|
C21H21ClN4OS
|
1
|
| 1 |
Ki = 1.259 nM
|
|
|
|
CP0386220
|
(2S)-1-thieno[2,3-g]indazol-1-ylpropan-2-amine
Show/Hide
|
C12H13N3S
|
1
|
| 1 |
Ki = 1.4 nM
|
|
|
|
CP0386221
|
(2S)-1-(6-methoxy-1H-indazol-1-yl)propan-2-amine
Show/Hide
|
C11H15N3O
|
2
|
| 1 |
Ki = 1.5 nM
|
|
|
| 2 |
Ki = 16 nM
|
|
|
|
CP0436958
|
(4R,9aR)-6-chloro-4-methyl-1,2,3,4,9,9a-hexahydro-2,4a,5-triaza-fluorene
Show/Hide
|
C11H14ClN3
|
1
|
| 1 |
Ki = 1.6 nM
|
|
|
|
CP0074886
|
(4R,10aS)-7-Chloro-4,6-dimethyl-1,2,3,4,10,10a-hexahydro-pyrazino[1,2-a]indole
Show/Hide
|
C13H17ClN2
|
1
|
| 1 |
Ki = 1.9 nM
|
|
|
|
CP0439530
|
(4R,9aR)-6-[1-((S)-ethoxy)-ethyl]-4-methyl-1,2,3,4,9,9a-hexahydro-2,4a,5-triaza-fluorene
Show/Hide
|
C15H23N3O
|
1
|
| 1 |
Ki = 2.3 nM
|
|
|
|
CP0382359
|
7-bromo-6-chloro-2,3,4,5-tetrahydro-1H-3-benzazepine
Show/Hide
|
C10H11BrClN
|
1
|
| 1 |
Ki = 2.4 nM
|
|
|
|
CP0373360
|
(2S)-1-(3-ethylfuro[2,3-g]indazol-1-yl)propan-2-amine
Show/Hide
|
C14H17N3O
|
1
|
| 1 |
Ki = 2.5 nM
|
|
|
|
CP0496060
|
(4R,9aR)-4,6-dimethyl-1,2,3,4,9,9a-hexahydro-2,4a,5-triaza-fluorene
Show/Hide
|
C12H17N3
|
1
|
| 1 |
Ki = 2.7 nM
|
|
|
|
CP0440946
|
(2S)-1-(3,7-diethylfuro[2,3-g]indazol-1-yl)propan-2-amine
Show/Hide
|
C16H21N3O
|
1
|
| 1 |
Ki = 2.7 nM
|
|
|
|
CP0112004
|
1-((S)-8-Chloro-10,11-dihydro-dibenzo[b,f]thiepin-10-yl)-4-methyl-piperazine
Show/Hide
|
C19H21ClN2S
|
1
|
| 1 |
Ki = 2.9 nM
|
|
|
|
CP0044585
|
1-((S)-2-aminopropyl)-1H-indazol-6-ol
Show/Hide
|
C10H13N3O
|
1
|
| 1 |
Ki = 3 nM
|
|
|
|
CP0205856
|
(R)-N-((11-(4-methylpiperazin-1-yl)-10,11-dihydrodibenzo[b,f]thiepin-2-yl)methyl)acetamide
Show/Hide
|
C22H27N3OS
|
1
|
| 1 |
Ki = 3.1 nM
|
|
|
|
CP0422236
|
N,N-dimethyl-1-[(2S,4S,6R)-3-oxatetracyclo[12.4.0.02,6.07,12]octadeca-1(18),7,9,11,14,16-hexaen-4-yl]methanamine
Show/Hide
|
C20H23NO
|
1
|
| 1 |
Ki = 3.25 nM
|
|
|
|
CP0431212
|
1-((S)-2-aminopropyl)-7-methyl-1H-indazol-6-ol
Show/Hide
|
C11H15N3O
|
1
|
| 1 |
Ki = 3.6 nM
|
|
|
|
CP0526503
|
(2S)-1-(6,7-dichloroindazol-1-yl)propan-2-amine
Show/Hide
|
C10H11Cl2N3
|
1
|
| 1 |
Ki = 4 nM
|
|
|
|
CP0057042
|
(R)-1-(4-iodo-2,5-dimethoxyphenyl)propan-2-amine
Show/Hide
|
C11H16INO2
|
1
|
| 1 |
Ki = 4 nM
|
|
|
|
CP0466886
|
1-((S)-2-aminopropyl)-7-iodo-1H-indazol-6-ol
Show/Hide
|
C10H12IN3O
|
1
|
| 1 |
Ki = 4.8 nM
|
|
|
|
CP0647511
|
2-Cyclohexyl-3-(4-fluoro-piperidin-3-yl)-1H-indole
Show/Hide
|
C19H24F2N2
|
1
|
| 1 |
Ki = 5 nM
|
|
|
|
CP0454034
|
(2S)-1-(7-ethyl-3-methylfuro[2,3-g]indazol-1-yl)propan-2-amine
Show/Hide
|
C15H19N3O
|
1
|
| 1 |
Ki = 5 nM
|
|
|
|
CP0045063
|
2-methyl-4-(4-methylpiperazin-1-yl)-10H-thieno[2,3-b][1,5]benzodiazepine
Show/Hide
|
C17H20N4S
|
1
|
| 1 |
Ki = 5.012 nM
|
|
|
|
CP0373307
|
6-chloro-2,3,4,5-tetrahydro-1H-3-benzazepine-7-carbonitrile
Show/Hide
|
C11H11ClN2
|
1
|
| 1 |
Ki = 5.1 nM
|
|
|
|
CP0319460
|
((2S,3aS,12bS)-11-Bromo-2,3,3a,12b-tetrahydro-1,8-dioxa-dibenzo[e,h]azulen-2-ylmethyl)-dimethyl-amine
Show/Hide
|
C19H20BrNO2
|
1
|
| 1 |
Ki = 6 nM
|
|
|
|
CP0478245
|
N,N-dimethyl-1-[(2S,6R)-3-oxatetracyclo[12.4.0.02,6.07,12]octadeca-1(18),7,9,11,14,16-hexaen-4-yl]methanamine
Show/Hide
|
C20H23NO
|
1
|
| 1 |
Ki = 6.7 nM
|
|
|
|
CP0057346
|
3-(2-aminopropyl)-1H-indol-5-ol
Show/Hide
|
C11H14N2O
|
1
|
| 1 |
Ki = 7 nM
|
|
|
|
CP0383416
|
(E)-1-(2-(4-(4-fluorostyryl)phenylsulfonyl)phenyl)ethanol
Show/Hide
|
C22H19FO3S
|
1
|
| 1 |
Ki = 7 nM
|
|
|
|
CP0513632
|
(2S)-1-(5,6-dichloroindazol-1-yl)propan-2-amine
Show/Hide
|
C10H11Cl2N3
|
1
|
| 1 |
Ki = 7.5 nM
|
|
|
|
CP0025667
|
2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-(2-methyl-2,3-dihydro-indol-1-yl)-ethanone
Show/Hide
|
C18H19ClN4
|
1
|
| 1 |
Ki = 7.943 nM
|
|
|
|
CP0167141
|
(R)-N-((11-(4-methylpiperazin-1-yl)-10,11-dihydrodibenzo[b,f]thiepin-2-yl)methyl)isobutyramide
Show/Hide
|
C24H31N3OS
|
1
|
| 1 |
Ki = 8 nM
|
|
|
|
CP0405082
|
1-ethyl-3-[(8-methoxy-2,3-dihydro-1H-cyclopenta[a]naphthalen-1-yl)methyl]thiourea
Show/Hide
|
C18H22N2OS
|
1
|
| 1 |
Ki = 8 nM
|
|
|
|
CP0099665
|
2-(5-Methoxy-1H-indol-3-yl)-1-methyl-ethylamine
Show/Hide
|
C12H16N2O
|
1
|
| 1 |
Ki = 8.3 nM
|
|
|
|
CP0492372
|
N-ethyl-2-[2-(3-fluorophenyl)-1H-indol-3-yl]-N-methylethanamine
Show/Hide
|
C19H21FN2
|
1
|
| 1 |
Ki = 8.4 nM
|
|
|
|
CP0373309
|
6,7-dichloro-2,3,4,5-tetrahydro-1H-3-benzazepine
Show/Hide
|
C10H11Cl2N
|
1
|
| 1 |
Ki = 8.8 nM
|
|
|
|
CP0431209
|
1-(2-aminoethyl)-1H-indazol-6-ol
Show/Hide
|
C9H11N3O
|
1
|
| 1 |
Ki = 9.6 nM
|
|
|
|
CP0448928
|
N-methyl-1-[(2S,6R)-3-oxatetracyclo[12.4.0.02,6.07,12]octadeca-1(18),7,9,11,14,16-hexaen-4-yl]methanamine
Show/Hide
|
C19H21NO
|
1
|
| 1 |
Ki = 9.7 nM
|
|
|
|
CP0802170
|
6-Fluoro-3-(4-fluoro-piperidin-3-yl)-2-phenyl-1H-indole
Show/Hide
|
C19H18F2N2
|
1
|
| 1 |
Ki = 10 nM
|
|
|
|
CP0461094
|
N-ethyl-N-methyl-2-(2-phenyl-1H-indol-3-yl)ethanamine
Show/Hide
|
C19H22N2
|
1
|
| 1 |
Ki = 11 nM
|
|
|
|
CP0126974
|
N-[[1-(4-fluorophenyl)-3-[1-[2-(2-oxoimidazolidin-1-yl)ethyl]piperidin-4-yl]indol-5-yl]methyl]acetamide
Show/Hide
|
C27H32FN5O2
|
1
|
| 1 |
Ki = 11 nM
|
|
|
|
CP0406335
|
N-ethyl-N-methyl-2-[2-[3-(trifluoromethyl)phenyl]-1H-indol-3-yl]ethanamine
Show/Hide
|
C20H21F3N2
|
1
|
| 1 |
Ki = 12 nM
|
|
|
|
CP0311945
|
((2S,3aS,12bS)-11-Chloro-2,3,3a,12b-tetrahydro-1,8-dioxa-dibenzo[e,h]azulen-2-ylmethyl)-dimethyl-amine
Show/Hide
|
C19H20ClNO2
|
1
|
| 1 |
Ki = 12 nM
|
|
|
|
CP0454033
|
(2S)-1-(7-ethyl-3-methoxyfuro[2,3-g]indazol-1-yl)propan-2-amine
Show/Hide
|
C15H19N3O2
|
1
|
| 1 |
Ki = 12 nM
|
|
|
|
CP0039958
|
(risperidone)3-{2-[4-(6-Fluoro-benzo[d]isoxazol-3-yl)-piperidin-1-yl]-ethyl}-2-methyl-6,7,8,9-tetrahydro-pyrido[1,2-a]pyrimidin-4-one
Show/Hide
|
C23H27FN4O2
|
1
|
| 1 |
Ki = 12.59 nM
|
|
|
|
CP0438192
|
N,N-dimethyl-1-[(2S,6R)-13-methyl-3-oxa-13-azatetracyclo[12.4.0.02,6.07,12]octadeca-1(18),7,9,11,14,16-hexaen-4-yl]methanamine
Show/Hide
|
C20H24N2O
|
1
|
| 1 |
Ki = 12.9 nM
|
|
|
|
CP0075436
|
(2,3-Dimethoxy-phenyl)-{1-[2-(4-fluoro-phenyl)-ethyl]-piperidin-4-yl}-methanol
Show/Hide
|
C22H28FNO3
|
1
|
| 1 |
Ki = 13 nM
|
|
|
|
CP0440947
|
(2S)-1-(3-methylfuro[2,3-g]indazol-1-yl)propan-2-amine
Show/Hide
|
C13H15N3O
|
1
|
| 1 |
Ki = 13 nM
|
|
|
|
CP0059927
|
1,2,3,4,8,9,10,11,12,13-decahydrocycloocta[b][1,4]diazepino[6,7,1-hi]indole
Show/Hide
|
C17H22N2
|
1
|
| 1 |
Ki = 13 nM
|
|
|
|
CP0468547
|
(4R,9aR)-4-methyl-6-trifluoromethyl-1,2,3,4,9,9a-hexahydro-2,4a,5-triaza-fluorene
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C12H14F3N3
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1
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| 1 |
Ki = 14 nM
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CP0412421
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6-chloro-7-nitro-2,3,4,5-tetrahydro-1H-3-benzazepine
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C10H11ClN2O2
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1
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| 1 |
Ki = 14 nM
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CP0403988
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2-[2-[3,5-bis(trifluoromethyl)phenyl]-1H-indol-3-yl]-N-ethyl-N-methylethanamine
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C21H20F6N2
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1
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| 1 |
Ki = 15 nM
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CP0394016
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2-benzyl-4-(4-methylphenyl)-6,7,8,9-tetrahydro-5H-pyrimido[4,5-d]azepine
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C22H23N3
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1
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| 1 |
Ki = 15 nM
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CP0453367
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N-methyl-1-[(2R,4S,6S)-3-oxatetracyclo[12.4.0.02,6.07,12]octadeca-1(18),7,9,11,14,16-hexaen-4-yl]methanamine
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C19H21NO
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1
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| 1 |
Ki = 15.9 nM
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CP0311380
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6-Fluoro-2-(4-fluoro-phenyl)-3-piperidin-3-yl-1H-indole
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C19H18F2N2
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1
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| 1 |
Ki = 16 nM
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CP0441912
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(4R,9aR)-6-methoxymethyl-4-methyl-1,2,3,4,9,9a-hexahydro-2,4a,5-triaza-fluorene
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C13H19N3O
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1
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| 1 |
Ki = 16 nM
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CP0403652
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(4-Fluoro-phenyl)-{1-[(3aR,12bS)-1-(3,3a,8,12b-tetrahydro-2H-1-oxa-dibenzo[e,h]azulen-2-yl)methyl]-piperidin-4-yl}-methanone
Show/Hide
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C30H30FNO2
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1
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| 1 |
Ki = 17 nM
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CP0345222
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3-[[1-(2-(2,4-Difluorophenyl)ethyl)-4-piperidinyl]sulfonyl]benzamide
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C20H22F2N2O3S
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1
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| 1 |
Ki = 18 nM
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CP0746305
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3-((3R,4R)-4-fluoropiperidin-3-yl)-2-phenyl-1H-indole
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C19H19FN2
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1
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| 1 |
Ki = 19 nM
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CP0844291
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(3R,4R)-6-Fluoro-2-(4-fluorophenyl)-3-(4-fluoropiperidin-3-yl)-1H-indole
Show/Hide
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C19H17F3N2
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1
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| 1 |
Ki = 19 nM
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CP0428084
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(E)-5-fluoro-2-(2-(5-(2-fluorophenylsulfonyl)pyridin-2-yl)vinyl)benzonitrile
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C20H12F2N2O2S
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1
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| 1 |
Ki = 19 nM
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CP0371841
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2-benzyl-4-(4-fluorophenyl)-6,7,8,9-tetrahydro-5H-pyrimido[4,5-d]azepine
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C21H20FN3
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1
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| 1 |
Ki = 20 nM
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CP0526502
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(2S)-1-(7-propan-2-ylfuro[2,3-g]indazol-1-yl)propan-2-amine
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C15H19N3O
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1
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| 1 |
Ki = 20 nM
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CP0412415
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7,8,9,10-tetrahydro-6H-furo[2,3-i][3]benzazepine
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C12H13NO
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1
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| 1 |
Ki = 20 nM
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CP0412422
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6-chloro-7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepine
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C11H14ClNO
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1
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| 1 |
Ki = 20 nM
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CP0251195
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((2R,3aS,12bS)-11-Chloro-2,3,3a,12b-tetrahydro-1,8-dioxa-dibenzo[e,h]azulen-2-ylmethyl)-dimethyl-amine
Show/Hide
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C19H20ClNO2
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1
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| 1 |
Ki = 21 nM
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CP0475230
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(4R,9aS)-6-bromo-4-methyl-1,2,3,4,9,9a-hexahydro-2,4a,5-triaza-fluorene
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C11H14BrN3
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1
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| 1 |
Ki = 21 nM
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CP0417691
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(E)-3-(4-(2,4-difluorostyryl)phenylsulfonyl)benzamide
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C21H15F2NO3S
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1
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| 1 |
Ki = 21 nM
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CP0195465
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1-(2-(4-(5-(aminomethyl)-1-(4-fluorophenyl)-1H-indol-3-yl)piperidin-1-yl)ethyl)imidazolidin-2-one
Show/Hide
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C25H30FN5O
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1
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| 1 |
Ki = 22 nM
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CP0392942
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2-cyclopentyl-4-(4-methylphenyl)-6,7,8,9-tetrahydro-5H-pyrimido[4,5-d]azepine
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C20H25N3
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1
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| 1 |
Ki = 23 nM
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CP0373308
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7,8,9,10-tetrahydro-6H-furo[3,2-i][3]benzazepine
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C12H13NO
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1
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| 1 |
Ki = 23 nM
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CP0454651
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N,N-dimethyl-1-[(2S,6R)-3-oxa-13-thiatetracyclo[12.4.0.02,6.07,12]octadeca-1(18),7,9,11,14,16-hexaen-4-yl]methanamine
Show/Hide
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C19H21NOS
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1
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| 1 |
Ki = 24.7 nM
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CP0040626
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1-(2,4-difluorophenethyl)-4-(phenylsulfonyl)piperidine
Show/Hide
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C19H21F2NO2S
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1
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| 1 |
Ki = 25 nM
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CP0373359
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(2S)-1-(3-propylfuro[2,3-g]indazol-1-yl)propan-2-amine
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C15H19N3O
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1
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| 1 |
Ki = 25 nM
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CP0240469
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(S)-N-((11-(4-methylpiperazin-1-yl)-10,11-dihydrodibenzo[b,f]thiepin-2-yl)methyl)acetamide
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C22H27N3OS
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1
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| 1 |
Ki = 26 nM
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CP0383041
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4-[(3aR,12bS)-1-(3,3a,8,12b-Tetrahydro-2H-1-oxa-dibenzo[e,h]azulen-2-yl)methyl]-morpholine
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C22H25NO2
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1
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| 1 |
Ki = 27 nM
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CP0376926
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1-(4-fluorophenyl)-4-[6-methoxyspiro[3,4-dihydro-2H-chromene-2,4'-(hexahydropyridine)]-1-yl]-1-butanone
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C24H28FNO3
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1
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| 1 |
Ki = 28 nM
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CP0420430
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N,N-dimethyl-1-[(2R,4S,6S)-3-oxatetracyclo[12.4.0.02,6.07,12]octadeca-1(18),7,9,11,14,16-hexaen-4-yl]methanamine
Show/Hide
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C20H23NO
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1
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| 1 |
Ki = 28 nM
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CP0453498
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3-[2-((S)-2-Methoxymethyl-pyrrolidin-1-yl)-ethyl]-2-phenyl-1H-indole
Show/Hide
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C22H26N2O
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1
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| 1 |
Ki = 29 nM
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CP0453441
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N-ethyl-2-[2-(2-fluorophenyl)-1H-indol-3-yl]-N-methylethanamine
Show/Hide
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C19H21FN2
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1
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| 1 |
Ki = 30 nM
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CP0439673
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N-ethyl-2-[2-(4-fluorophenyl)-1H-indol-3-yl]-N-methylethanamine
Show/Hide
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C19H21FN2
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1
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| 1 |
Ki = 31 nM
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CP0454625
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1-[(2S,6R)-3,13-dioxatetracyclo[12.4.0.02,6.07,12]octadeca-1(18),7,9,11,14,16-hexaen-4-yl]-N,N-dimethylmethanamine
Show/Hide
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C19H21NO2
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1
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| 1 |
Ki = 31 nM
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CP0500615
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(2S)-1-(6-fluoroindazol-1-yl)propan-2-amine
Show/Hide
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C10H12FN3
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1
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| 1 |
Ki = 32 nM
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CP0438554
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1-[(2S,6R)-3,13-dioxatetracyclo[13.4.0.02,6.07,12]nonadeca-1(19),7,9,11,15,17-hexaen-4-yl]-N,N-dimethylmethanamine
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C20H23NO2
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1
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| 1 |
Ki = 32.5 nM
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CP0372472
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1-((R)-2-aminopropyl)-1H-indazol-6-ol
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C10H13N3O
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1
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| 1 |
Ki = 34 nM
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CP0420816
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N-ethyl-N-methyl-2-[2-(3-nitrophenyl)-1H-indol-3-yl]ethanamine
Show/Hide
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C19H21N3O2
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1
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| 1 |
Ki = 36 nM
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CP0467124
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3-[2-((R)-2-Methyl-piperidin-1-yl)-ethyl]-2-phenyl-1H-indole
Show/Hide
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C22H26N2
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1
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| 1 |
Ki = 36 nM
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CP0506837
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2-[2-(4-chlorophenyl)-1H-indol-3-yl]-N-ethyl-N-methylethanamine
Show/Hide
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C19H21ClN2
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1
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| 1 |
Ki = 36 nM
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CP0441076
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2-benzyl-4-[4-(trifluoromethyl)phenyl]-6,7,8,9-tetrahydro-5H-pyrimido[4,5-d]azepine
Show/Hide
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C22H20F3N3
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1
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| 1 |
Ki = 38 nM
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CP0483639
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4,5,6,7,9,10,11,12-Octahydro-8H-5,7a-diaza-benzo[cd]cyclohepta[a]azulene
Show/Hide
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C16H20N2
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1
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| 1 |
Ki = 38 nM
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CP0430154
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3-[[1-(2-(2,4-Difluorophenyl)ethyl)-4-piperidinyl]sulfonyl]benzonitrile
Show/Hide
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C20H20F2N2O2S
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1
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| 1 |
Ki = 39 nM
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CP0420527
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1-((4R,9aR)-4-methyl-1,2,3,4,9,9a-hexahydro-2,4a,5-triaza-fluoren-6-yl)-ethanol
Show/Hide
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C13H19N3O
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1
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| 1 |
Ki = 39 nM
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CP0044329
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1-(2,4-difluorophenethyl)-4-(4-fluorophenylsulfonyl)piperidine
Show/Hide
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C19H20F3NO2S
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2
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| 1 |
Ki = 39 nM
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| 2 |
Ki = 92 nM
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CP0033479
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(chloropromazine) [3-(2-Chloro-phenothiazin-10-yl)-propyl]-dimethyl-amine
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C17H19ClN2S
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1
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| 1 |
Ki = 39.81 nM
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CP0466838
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2-(4-(4-(5-fluoro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)butyl)isoindoline-1,3-dione
Show/Hide
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C25H24FN3O2
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1
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| 1 |
Ki = 39.81 nM
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CP0345192
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1'-[2-(2,4-Difluorophenyl)ethyl]-3,4-dihydrospiro[2H-1-benzothiopyran-2,4'-piperidine]-1,1-dioxide
Show/Hide
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C21H23F2NO2S
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1
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| 1 |
Ki = 41 nM
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CP0250615
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((2S,3aS,12bS)-11-Fluoro-2,3,3a,12b-tetrahydro-1,8-dioxa-dibenzo[e,h]azulen-2-ylmethyl)-dimethyl-amine
Show/Hide
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C19H20FNO2
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1
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| 1 |
Ki = 41 nM
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CP0435135
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(E)-4-(4-(2,4-difluorostyryl)phenylsulfonyl)benzamide
Show/Hide
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C21H15F2NO3S
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1
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| 1 |
Ki = 41 nM
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CP0071154
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2-(5-methoxy-1H-indol-3-yl)-N,N-dimethyl-ethanamine
Show/Hide
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C13H18N2O
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1
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| 1 |
Ki = 42 nM
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CP0393387
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1-[(8-methoxy-2,3-dihydro-1H-cyclopenta[a]naphthalen-1-yl)methyl]-3-propylthiourea
Show/Hide
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C19H24N2OS
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1
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| 1 |
Ki = 42 nM
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CP0480878
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4-Phenyl-1-[(3aR,12bS)-1-(3,3a,8,12b-tetrahydro-2H-1-oxa-dibenzo[e,h]azulen-2-yl)methyl]-piperidine
Show/Hide
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C29H31NO
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1
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| 1 |
Ki = 42.7 nM
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CP0528118
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(E)-2-(2,4-difluorostyryl)-5-(2-fluorophenylsulfinyl)pyridine
Show/Hide
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C19H12F3NOS
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1
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| 1 |
Ki = 43 nM
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CP0386222
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(2S)-1-(5-fluoroindazol-1-yl)propan-2-amine
Show/Hide
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C10H12FN3
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1
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| 1 |
Ki = 43 nM
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CP0373312
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6-chloro-7-fluoro-2,3,4,5-tetrahydro-1H-3-benzazepine
Show/Hide
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C10H11ClFN
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1
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| 1 |
Ki = 43 nM
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CP0870788
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4-(5,6,7,8-tetrahydronaphthalen-1-yl)piperidinium trifluoroacetate
Show/Hide
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C17H22F3NO2
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2
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| 1 |
Ki = 43 nM
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| 2 |
Ki = 55 nM
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CP0039099
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1-(2-Phenylethyl)-4-(phenylsulfonyl)piperidine
Show/Hide
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C19H23NO2S
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1
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| 1 |
Ki = 46 nM
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CP0373311
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6-chloro-N-methyl-2,3,4,5-tetrahydro-1H-3-benzazepin-7-amine
Show/Hide
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C11H15ClN2
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1
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| 1 |
Ki = 46 nM
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CP0039100
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2-[[1-(2-(2,4-Difluorophenyl)ethyl)-4-piperidinyl]sulfonyl]benzonitrile
Show/Hide
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C20H20F2N2O2S
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1
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| 1 |
Ki = 47 nM
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CP0191221
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(S,E)-1-(2-(4-(4-fluorostyryl)phenylsulfonyl)phenyl)ethanol
Show/Hide
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C22H19FO3S
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1
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| 1 |
Ki = 47 nM
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CP0701507
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(3R,4R)-6-Fluoro-3-(4-fluoropiperidin-3-yl)-1H-indole-2-carboxylic acid phenylamide
Show/Hide
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C20H19F2N3O
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1
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| 1 |
Ki = 48 nM
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CP0829638
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(3R,4R)-6-Fluoro-3-(4-fluoropiperidin-3-yl)-2-thiophen-3-yl-1H-indole
Show/Hide
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C17H16F2N2S
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1
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| 1 |
Ki = 50 nM
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CP0372249
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4-(4-fluorophenyl)-2-[(4-fluorophenyl)methyl]-6,7,8,9-tetrahydro-5H-pyrimido[4,5-d]azepine
Show/Hide
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C21H19F2N3
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1
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| 1 |
Ki = 50 nM
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CP0042927
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7-{4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butoxy}-3,4-dihydroquinolin-2(1H)-one
Show/Hide
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C23H27Cl2N3O2
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1
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| 1 |
Ki = 50.12 nM
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CP0424952
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(4R,9aS)-6-chloro-4-methyl-1,2,3,4,9,9a-hexahydro-2,4a,5-triaza-fluorene
Show/Hide
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C11H14ClN3
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1
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| 1 |
Ki = 52 nM
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CP0420529
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((4R,9aR)-4-methyl-1,2,3,4,9,9a-hexahydro-2,4a,5-triaza-fluoren-6-yl)-methanol
Show/Hide
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C12H17N3O
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1
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| 1 |
Ki = 54 nM
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CP0511470
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4-(4-Chloro-benzenesulfonyl)-1-[2-(2,4-difluoro-phenyl)-ethyl]-piperidine
Show/Hide
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C19H20ClF2NO2S
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1
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| 1 |
Ki = 58 nM
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CP0275194
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8-((2S,3aS,12bS)-11-Bromo-2,3,3a,12b-tetrahydro-1,8-dioxa-dibenzo[e,h]azulen-2-ylmethyl)-3-methyl-7-oxa-8-aza-bicyclo[4.2.0]octa-1(6),2,4-triene
Show/Hide
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C24H20BrNO3
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1
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| 1 |
Ki = 58 nM
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CP0500622
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(2S)-1-pyrazolo[3,4-e][1,3]benzoxazol-1-ylpropan-2-amine
Show/Hide
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C11H12N4O
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1
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| 1 |
Ki = 59 nM
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CP0420528
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(4R,9aR)-4-methyl-1,2,3,4,9,9a-hexahydro-2,4a,5-triaza-fluorene-6-carbonitrile
Show/Hide
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C12H14N4
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1
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| 1 |
Ki = 60 nM
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CP0228798
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1-(2-{4-[1-(4-Fluoro-phenyl)-5-(2-methyl-2H-tetrazol-5-yl)-1H-indol-3-yl]-piperidin-1-yl}-ethyl)-imidazolidin-2-one
Show/Hide
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C26H29FN8O
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1
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| 1 |
Ki = 60 nM
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CP0875253
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4-(1-Naphthyl)piperidinium trifluoroacetate
Show/Hide
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C17H18F3NO2
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2
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| 1 |
Ki = 60 nM
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| 2 |
Ki = 72 nM
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CP0416460
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1-ethyl-3-[(8-methoxy-2,3-dihydro-1H-cyclopenta[a]naphthalen-1-yl)methyl]urea
Show/Hide
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C18H22N2O2
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1
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| 1 |
Ki = 60 nM
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CP0459154
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N-[(8-methoxy-2,3-dihydro-1H-cyclopenta[a]naphthalen-1-yl)methyl]acetamide
Show/Hide
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C17H19NO2
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1
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| 1 |
Ki = 61 nM
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CP0146501
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((2R,3aS,12bS)-11-Fluoro-2,3,3a,12b-tetrahydro-1,8-dioxa-dibenzo[e,h]azulen-2-ylmethyl)-dimethyl-amine
Show/Hide
|
C19H20FNO2
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1
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| 1 |
Ki = 63 nM
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CP0428086
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(E)-2-(2-chloro-4-fluorostyryl)-5-(2-fluorophenylsulfonyl)pyridine
Show/Hide
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C19H12ClF2NO2S
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1
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| 1 |
Ki = 64 nM
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CP0376933
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(E)-2,4-difluoro-1-(4-(phenylsulfonyl)styryl)benzene
Show/Hide
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C20H14F2O2S
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1
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| 1 |
Ki = 65 nM
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CP0373310
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6-chloro-3-methyl-7-nitro-1,2,4,5-tetrahydro-3-benzazepine
Show/Hide
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C11H13ClN2O2
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1
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| 1 |
Ki = 66 nM
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CP0152373
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1-(2,4-difluorophenethyl)-4-fluoro-4-(4-fluorophenylsulfonyl)piperidine
Show/Hide
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C19H19F4NO2S
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2
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| 1 |
Ki = 69 nM
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| 2 |
Ki = 180 nM
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CP0366089
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((2S,3aS,12bS)-11-Methoxy-2,3,3a,12b-tetrahydro-1,8-dioxa-dibenzo[e,h]azulen-2-ylmethyl)-dimethyl-amine
Show/Hide
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C20H23NO3
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1
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| 1 |
Ki = 72 nM
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CP0429925
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(8-methoxy-2,3-dihydro-1H-cyclopenta[a]naphthalen-1-yl)methylthiourea
Show/Hide
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C16H18N2OS
|
1
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| 1 |
Ki = 72 nM
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CP0490292
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2-benzyl-4-(4-fluorophenyl)-5,6,7,8-tetrahydropyrido[3,4-d]pyrimidine
Show/Hide
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C20H18FN3
|
1
|
| 1 |
Ki = 75 nM
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CP0345223
|
3-(1-Phenethyl-piperidin-4-yl)-2-phenyl-1H-indole
Show/Hide
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C27H28N2
|
1
|
| 1 |
Ki = 79 nM
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CP0492300
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8,8,10,10-Tetramethyl-1,2,3,4,8,9,10,11-octahydro-[1,4]diazepino[6,7,1-jk]carbazole
Show/Hide
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C19H26N2
|
1
|
| 1 |
Ki = 79 nM
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CP0371842
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4-(4-fluorophenyl)-2-propan-2-yl-6,7,8,9-tetrahydro-5H-pyrimido[4,5-d]azepine
Show/Hide
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C17H20FN3
|
1
|
| 1 |
Ki = 80 nM
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CP0916293
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(3R,4R)-6-Fluoro-3-(4-fluoro-piperidin-3-yl)-2-pyridin-3-yl-1H-indole
Show/Hide
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C18H17F2N3
|
1
|
| 1 |
Ki = 85 nM
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CP0077877
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((2R,3aS,12bS)-11-Bromo-2,3,3a,12b-tetrahydro-1,8-dioxa-dibenzo[e,h]azulen-2-ylmethyl)-dimethyl-amine
Show/Hide
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C19H20BrNO2
|
1
|
| 1 |
Ki = 87 nM
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CP0270573
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2-Phenyl-3-piperidin-3-yl-1H-indole
Show/Hide
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C19H20N2
|
1
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| 1 |
Ki = 89 nM
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CP0436549
|
(4R,9aR)-6-[1-((R)-ethoxy)-ethyl]-4-methyl-1,2,3,4,9,9a-hexahydro-2,4a,5-triaza-fluorene
Show/Hide
|
C15H23N3O
|
1
|
| 1 |
Ki = 93 nM
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CP0260914
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(S)-N-((11-(4-methylpiperazin-1-yl)-10,11-dihydrodibenzo[b,f]thiepin-2-yl)methyl)isobutyramide
Show/Hide
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C24H31N3OS
|
1
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| 1 |
Ki = 93 nM
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CP0382988
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4,5,6,7,9,10-Hexahydro-8H-5,7a-diaza-benzo[cd]cyclopenta[a]azulene
Show/Hide
|
C14H16N2
|
1
|
| 1 |
Ki = 97 nM
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CP0371096
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4-[[1-(2-(2,4-Difluorophenyl)ethyl)-4-piperidinyl]sulfonyl]benzamide
Show/Hide
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C20H22F2N2O3S
|
1
|
| 1 |
Ki = 100 nM
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CP0371839
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2-tert-butyl-4-(4-fluorophenyl)-5,6,7,8-tetrahydropyrido[4,3-d]pyrimidine
Show/Hide
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C17H20FN3
|
1
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| 1 |
Ki = 100 nM
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CP0099167
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(4-(2,4-difluorophenethyl)piperidin-1-yl)(2-fluorophenyl)methanone
Show/Hide
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C20H20F3NO
|
1
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| 1 |
Ki = 100 nM
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CP0429929
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methyl N-[(8-methoxy-2,3-dihydro-1H-cyclopenta[a]naphthalen-1-yl)methyl]carbamate
Show/Hide
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C17H19NO3
|
1
|
| 1 |
Ki = 100 nM
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CP0428406
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(4R,9aR)-6-methoxy-4-methyl-1,2,3,4,9,9a-hexahydro-2,4a,5-triaza-fluorene
Show/Hide
|
C12H17N3O
|
1
|
| 1 |
Ki = 104 nM
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CP0470578
|
1-(3-Chloro-phenyl)-4-[(3aR,12bS)-1-(3,3a,8,12b-tetrahydro-2H-1-oxa-dibenzo[e,h]azulen-2-yl)methyl]-piperazine
Show/Hide
|
C28H29ClN2O
|
1
|
| 1 |
Ki = 107.4 nM
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CP0379567
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2-cyclopentyl-4-(4-fluorophenyl)-5,6,7,8-tetrahydropyrido[4,3-d]pyrimidine
Show/Hide
|
C18H20FN3
|
1
|
| 1 |
Ki = 110 nM
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CP0126860
|
1-(2-{4-[1-(4-Fluoro-phenyl)-5-(1-methyl-1H-[1,2,3]triazol-4-yl)-1H-indol-3-yl]-piperidin-1-yl}-ethyl)-imidazolidin-2-one
Show/Hide
|
C27H30FN7O
|
1
|
| 1 |
Ki = 110 nM
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|
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CP0453215
|
7-Fluoro-1,2,3,4,8,9,10,11-octahydro-[1,4]diazepino[6,7,1-jk]carbazole
Show/Hide
|
C15H17FN2
|
1
|
| 1 |
Ki = 111 nM
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CP0442228
|
N-ethyl-N-methyl-2-(2-thiophen-2-yl-1H-indol-3-yl)ethanamine
Show/Hide
|
C17H20N2S
|
1
|
| 1 |
Ki = 120 nM
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CP0379565
|
2-cyclopentyl-4-(4-methoxyphenyl)-6,7,8,9-tetrahydro-5H-pyrimido[4,5-d]azepine
Show/Hide
|
C20H25N3O
|
1
|
| 1 |
Ki = 120 nM
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CP0461357
|
1-Methyl-4-[(3aR,12bS)-1-(2,3,3a,12b-tetrahydro-1-oxa-8-thia-dibenzo[e,h]azulen-2-yl)methyl]-piperazine
Show/Hide
|
C22H26N2OS
|
1
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| 1 |
Ki = 120 nM
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CP0461004
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1-[(2S,6R)-3,14-dioxatetracyclo[13.4.0.02,6.07,12]nonadeca-1(19),7,9,11,15,17-hexaen-4-yl]-N,N-dimethylmethanamine
Show/Hide
|
C20H23NO2
|
1
|
| 1 |
Ki = 123.5 nM
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CP0144949
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2-[1-({6-chloroimidazo[2,1-b][1,3]thiazole-5-}sulfonyl)-1H-indol-3-yl]ethan-1-amine
Show/Hide
|
C15H13ClN4O2S2
|
1
|
| 1 |
Ki = 124 nM
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CP0373055
|
(E)-2-(4-(2,4-difluorostyryl)phenylsulfonyl)benzamide
Show/Hide
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C21H15F2NO3S
|
1
|
| 1 |
Ki = 127 nM
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CP0245024
|
1-(4-Fluorophenyl)-2-[4-(phenylsulfonyl)-1-piperidinyl]-ethanone
Show/Hide
|
C19H20FNO3S
|
1
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| 1 |
Ki = 130 nM
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CP0420526
|
6-chloro-1,2,3,4,9,9a-hexahydro-2,4a,5-triaza-fluorene
Show/Hide
|
C10H12ClN3
|
1
|
| 1 |
Ki = 131 nM
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CP0907832
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(3R,4R)-7-Fluoro-3-(4-fluoropiperidin-3-yl)-2-phenyl-1H-indole
Show/Hide
|
C19H18F2N2
|
1
|
| 1 |
Ki = 132 nM
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|
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CP0533140
|
(2S)-1-(7-chloro-6-methoxyindazol-1-yl)propan-2-amine
Show/Hide
|
C11H14ClN3O
|
1
|
| 1 |
Ki = 140 nM
|
|
|
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CP0410497
|
(8-methoxy-2,3-dihydro-1H-cyclopenta[a]naphthalen-1-yl)methylurea
Show/Hide
|
C16H18N2O2
|
1
|
| 1 |
Ki = 145 nM
|
|
|
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CP0371098
|
3-(1-Methyl-piperidin-3-yl)-2-phenyl-1H-indole
Show/Hide
|
C20H22N2
|
1
|
| 1 |
Ki = 150 nM
|
|
|
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CP0371094
|
1'-(2,4-difluorophenethyl)-6-methoxyspiro[3,4-dihydro-2H-chromene-2,4'-(hexahydropyridine)]
Show/Hide
|
C22H25F2NO2
|
1
|
| 1 |
Ki = 150 nM
|
|
|
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CP0383998
|
2-benzyl-4-(4-fluorophenyl)-6,7,8,9-tetrahydro-5H-pyrimido[4,5-c]azepine
Show/Hide
|
C21H20FN3
|
1
|
| 1 |
Ki = 150 nM
|
|
|
|
CP0826952
|
(3R,4R)-7-Chloro-3-(4-fluoropiperidin-3-yl)-2-phenyl-1H-indole
Show/Hide
|
C19H18ClFN2
|
1
|
| 1 |
Ki = 154 nM
|
|
|
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CP0312008
|
8-[[(2S,4S,6S)-17-bromo-3,13-dioxatetracyclo[12.4.0.02,6.07,12]octadeca-1(14),7,9,11,15,17-hexaen-4-yl]methyl]-N,N-dimethyl-7-oxa-8-azabicyclo[4.2.0]octa-1(6),2,4-trien-3-amine
Show/Hide
|
C25H23BrN2O3
|
1
|
| 1 |
Ki = 157 nM
|
|
|
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CP0374269
|
4-{3-[2-(Ethyl-methyl-amino)-ethyl]-1H-indol-2-yl}-benzonitrile
Show/Hide
|
C20H21N3
|
1
|
| 1 |
Ki = 160 nM
|
|
|
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CP0424511
|
N,N-diethyl-2-(2-phenyl-1H-indol-3-yl)ethanamine
Show/Hide
|
C20H24N2
|
1
|
| 1 |
Ki = 160 nM
|
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|
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CP0427025
|
(E)-2-(4-fluorostyryl)-5-(2-fluorophenylsulfinyl)pyridine
Show/Hide
|
C19H13F2NOS
|
1
|
| 1 |
Ki = 160 nM
|
|
|
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CP0429924
|
N-[(2-methoxy-8,9-dihydro-7H-cyclopenta[h]quinolin-9-yl)methyl]acetamide
Show/Hide
|
C16H18N2O2
|
1
|
| 1 |
Ki = 160 nM
|
|
|
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CP0877970
|
rac-2-fluoro-N-(3-hydroxy-2-(7-methoxynaphthalen-1-yl)propyl)acetamide
Show/Hide
|
C16H18FNO3
|
1
|
| 1 |
Ki = 165.96 nM
|
|
|
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CP0448518
|
N,N-dimethyl-1-[(2S,6S)-3-oxatetracyclo[12.4.0.02,6.07,12]octadeca-1(18),7,9,11,14,16-hexaen-4-yl]methanamine
Show/Hide
|
C20H23NO
|
1
|
| 1 |
Ki = 166 nM
|
|
|
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CP0457342
|
2-{4-[(3aR,12bS)-1-(3,3a,8,12b-Tetrahydro-2H-1-oxa-dibenzo[e,h]azulen-2-yl)methyl]-piperazin-1-yl}-ethanol
Show/Hide
|
C24H30N2O2
|
1
|
| 1 |
Ki = 170 nM
|
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|
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CP0716967
|
Dimethyl-[(2R,3aR,12bS)-1-(2,3,3a,12b-tetrahydro-1,8-dioxa-dibenzo[e,h]azulen-2-yl)methyl]-amine
Show/Hide
|
C19H21NO2
|
1
|
| 1 |
Ki = 179 nM
|
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|
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CP0439696
|
N,N-dimethyl-2-(2-phenyl-1H-indol-3-yl)ethanamine
Show/Hide
|
C18H20N2
|
1
|
| 1 |
Ki = 180 nM
|
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CP0432490
|
N-[2-(8-methoxy-2,3-dihydro-1H-cyclopenta[a]naphthalen-1-yl)ethyl]acetamide
Show/Hide
|
C18H21NO2
|
1
|
| 1 |
Ki = 180 nM
|
|
|
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CP0035139
|
1-[(2R,4R,6S)-3,13-dioxatetracyclo[12.4.0.02,6.07,12]octadeca-1(18),7,9,11,14,16-hexaen-4-yl]-N,N-dimethylmethanamine
Show/Hide
|
C19H21NO2
|
1
|
| 1 |
Ki = 183 nM
|
|
|
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CP0160384
|
8-((2S,3aS,12bS)-11-Bromo-2,3,3a,12b-tetrahydro-1,8-dioxa-dibenzo[e,h]azulen-2-ylmethyl)-3-phenyl-7-oxa-8-aza-bicyclo[4.2.0]octa-1(6),2,4-triene
Show/Hide
|
C29H22BrNO3
|
1
|
| 1 |
Ki = 183 nM
|
|
|
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CP0237838
|
8-((2S,3aS,12bS)-11-Bromo-2,3,3a,12b-tetrahydro-1,8-dioxa-dibenzo[e,h]azulen-2-ylmethyl)-7-oxa-8-aza-bicyclo[4.2.0]octa-1(6),2,4-triene-3-carbonitrile
Show/Hide
|
C24H17BrN2O3
|
1
|
| 1 |
Ki = 183 nM
|
|
|
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CP0463465
|
1-[(2S,6S)-3,13-dioxatetracyclo[12.4.0.02,6.07,12]octadeca-1(18),7,9,11,14,16-hexaen-4-yl]-N,N-dimethylmethanamine
Show/Hide
|
C19H21NO2
|
1
|
| 1 |
Ki = 183 nM
|
|
|
|
CP0435136
|
8-(4-(2,4-difluorophenethyl)piperidin-1-ylsulfonyl)quinoline
Show/Hide
|
C22H22F2N2O2S
|
1
|
| 1 |
Ki = 184 nM
|
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|
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CP0847771
|
(R)-2-fluoro-N-(3-hydroxy-2-(7-methoxynaphthalen-1-yl)propyl)acetamide
Show/Hide
|
C16H18FNO3
|
1
|
| 1 |
Ki = 186.21 nM
|
|
|
|
CP0474630
|
(R)-2-Methyl-1,2,3,4,8,9,10,11-octahydro-[1,4]diazepino[6,7,1-jk]carbazole
Show/Hide
|
C16H20N2
|
1
|
| 1 |
Ki = 189 nM
|
|
|
|
CP0376936
|
1'-(2,4-difluorophenethyl)-8-fluorospiro[3,4-dihydro-2H-chromene-2,4'-(hexahydropyridine)]
Show/Hide
|
C21H22F3NO
|
1
|
| 1 |
Ki = 190 nM
|
|
|
|
CP0391337
|
1-[(8-methoxy-2,3-dihydro-1H-cyclopenta[a]naphthalen-1-yl)methyl]-3-propylurea
Show/Hide
|
C19H24N2O2
|
1
|
| 1 |
Ki = 190 nM
|
|
|
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CP0407867
|
(R)-8-(4-(3-(5-fluoro-1H-indol-3-yl)propyl)piperazin-1-yl)-2-methyl-2H-benzo[b][1,4]oxazin-3(4H)-one
Show/Hide
|
C24H27FN4O2
|
1
|
| 1 |
Ki = 199.53 nM
|
|
|
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CP0434496
|
(E)-2-(4-fluorostyryl)-5-(phenylsulfinyl)pyridine
Show/Hide
|
C19H14FNOS
|
1
|
| 1 |
Ki = 200 nM
|
|
|
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CP0372250
|
2-cyclopentyl-4-(4-fluorophenyl)-6,7,8,9-tetrahydro-5H-pyrimido[4,5-d]azepine
Show/Hide
|
C19H22FN3
|
1
|
| 1 |
Ki = 200 nM
|
|
|
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CP0429916
|
2-methoxy-N-[(8-methoxy-2,3-dihydro-1H-cyclopenta[a]naphthalen-1-yl)methyl]acetamide
Show/Hide
|
C18H21NO3
|
1
|
| 1 |
Ki = 200 nM
|
|
|
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CP0458483
|
(E)-2-(4-fluoro-2-methylstyryl)-5-(2-fluorophenylsulfonyl)pyridine
Show/Hide
|
C20H15F2NO2S
|
1
|
| 1 |
Ki = 220 nM
|
|
|
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CP0378677
|
N-[3-hydroxy-2-(7-methoxynaphthalen-1-yl)propyl]acetamide
Show/Hide
|
C16H19NO3
|
1
|
| 1 |
Ki = 229.09 nM
|
|
|
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CP0380594
|
3-[2-((S)-2-Methyl-piperidin-1-yl)-ethyl]-2-phenyl-1H-indole
Show/Hide
|
C22H26N2
|
1
|
| 1 |
Ki = 230 nM
|
|
|
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CP0371095
|
1'-phenethylspiro[1,2,3,4-tetrahydronaphthalene-2,4'-(hexahydropyridine)]-1-ol; hydrochloride
Show/Hide
|
C22H27NO
|
1
|
| 1 |
Ki = 230 nM
|
|
|
|
CP0860616
|
3-Chloro-N-[3-((R)-1-methyl-pyrrolidin-2-ylmethyl)-1H-indol-5-yl]-benzenesulfonamide
Show/Hide
|
C20H22ClN3O2S
|
1
|
| 1 |
Ki = 231 nM
|
|
|
|
CP0319461
|
((2R,3aS,12bS)-11-Methoxy-2,3,3a,12b-tetrahydro-1,8-dioxa-dibenzo[e,h]azulen-2-ylmethyl)-dimethyl-amine
Show/Hide
|
C20H23NO3
|
1
|
| 1 |
Ki = 235 nM
|
|
|
|
CP0777252
|
2-Iodo-N-(3-(R)-1-pyrrolidin-2-ylmethyl-1H-indol-5-yl)-benzenesulfonamide
Show/Hide
|
C20H22IN3O2S
|
1
|
| 1 |
Ki = 235 nM
|
|
|
|
CP0438782
|
4-Phenyl-1-[(3aR,12bS)-1-(2,3,3a,12b-tetrahydro-1-oxa-8-thia-dibenzo[e,h]azulen-2-yl)methyl]-piperidine
Show/Hide
|
C28H29NOS
|
1
|
| 1 |
Ki = 239 nM
|
|
|
|
CP0463855
|
9,9-Dimethyl-1,2,3,4,8,9,10,11-octahydro-[1,4]diazepino[6,7,1-jk]carbazole
Show/Hide
|
C17H22N2
|
1
|
| 1 |
Ki = 243 nM
|
|
|
|
CP0077886
|
8-((2S,3aS,12bS)-11-Bromo-2,3,3a,12b-tetrahydro-1,8-dioxa-dibenzo[e,h]azulen-2-ylmethyl)-7-oxa-8-aza-bicyclo[4.2.0]octa-1(6),2,4-triene-3-carboxylic acid ethyl ester
Show/Hide
|
C26H22BrNO5
|
1
|
| 1 |
Ki = 246 nM
|
|
|
|
CP0525463
|
2-Phenyl-3-(2-pyrrolidin-1-yl-ethyl)-1H-indole
Show/Hide
|
C20H22N2
|
1
|
| 1 |
Ki = 260 nM
|
|
|
|
CP0375784
|
2-Phenyl-3-(2-piperidin-1-yl-ethyl)-1H-indole
Show/Hide
|
C21H24N2
|
1
|
| 1 |
Ki = 268 nM
|
|
|
|
CP0092119
|
8-((2S,3aS,12bS)-11-Bromo-2,3,3a,12b-tetrahydro-1,8-dioxa-dibenzo[e,h]azulen-2-ylmethyl)-7-oxa-8-aza-bicyclo[4.2.0]octa-1(6),2,4-trien-3-ylamine
Show/Hide
|
C23H19BrN2O3
|
1
|
| 1 |
Ki = 270 nM
|
|
|
|
CP0429922
|
1-[(2-methoxy-8,9-dihydro-7H-cyclopenta[h]quinolin-9-yl)methyl]-3-propylurea
Show/Hide
|
C18H23N3O2
|
1
|
| 1 |
Ki = 285 nM
|
|
|
|
CP0873359
|
2-Chloro-N-[3-((R)-1-methyl-pyrrolidin-2-ylmethyl)-1H-indol-5-yl]-benzenesulfonamide
Show/Hide
|
C20H22ClN3O2S
|
1
|
| 1 |
Ki = 289 nM
|
|
|
|
CP0447444
|
1'-(2,4-difluorophenethyl)spiro[1,2,3,4-tetrahydronaphthalene-2,4'-(hexahydropyridine)]
Show/Hide
|
C22H25F2N
|
1
|
| 1 |
Ki = 320 nM
|
|
|
|
CP0393386
|
1-[(2-methoxy-8,9-dihydro-7H-cyclopenta[h]quinolin-9-yl)methyl]-3-methylurea
Show/Hide
|
C16H19N3O2
|
1
|
| 1 |
Ki = 340 nM
|
|
|
|
CP0077915
|
1-[8-((2S,3aS,12bS)-11-Bromo-2,3,3a,12b-tetrahydro-1,8-dioxa-dibenzo[e,h]azulen-2-ylmethyl)-7-oxa-8-aza-bicyclo[4.2.0]octa-1(6),2,4-trien-3-yl]-azetidin-2-one
Show/Hide
|
C26H21BrN2O4
|
1
|
| 1 |
Ki = 356 nM
|
|
|
|
CP0490453
|
6-Chloro-1,2,3,4,8,9,10,11-octahydro-[1,4]diazepino[6,7,1-jk]carbazole
Show/Hide
|
C15H17ClN2
|
1
|
| 1 |
Ki = 358 nM
|
|
|
|
CP0409239
|
1-(2-Chloro-benzenesulfonyl)-3-(1,2,3,6-tetrahydro-pyridin-4-yl)-1H-indole
Show/Hide
|
C19H17ClN2O2S
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1
|
| 1 |
Ki = 383 nM
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CP0245025
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2-Phenyl-3-piperidin-4-yl-1H-indole
Show/Hide
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C19H20N2
|
1
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| 1 |
Ki = 400 nM
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CP0415634
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2-phenyl-3-[(1S,5R)-8-(2-phenylethyl)-8-azabicyclo[3.2.1]octan-3-yl]-1H-indole
Show/Hide
|
C29H30N2
|
1
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| 1 |
Ki = 400 nM
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CP0371840
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2-benzyl-4-(4-fluorophenyl)-5,6,7,8-tetrahydropyrido[4,3-d]pyrimidine
Show/Hide
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C20H18FN3
|
1
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| 1 |
Ki = 400 nM
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CP0432491
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N-[(8-methoxy-2,3-dihydro-1H-cyclopenta[a]naphthalen-1-yl)methyl]ethanesulfonamide
Show/Hide
|
C17H21NO3S
|
1
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| 1 |
Ki = 400 nM
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CP0490433
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(E)-2-(2,4-difluorostyryl)-5-(2-fluorophenylsulfonyl)pyridine
Show/Hide
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C19H12F3NO2S
|
1
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| 1 |
Ki = 410 nM
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CP0384002
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2-cyclobutyl-4-(4-fluorophenyl)-5,6,7,8-tetrahydropyrido[4,3-d]pyrimidine
Show/Hide
|
C17H18FN3
|
1
|
| 1 |
Ki = 410 nM
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CP0267173
|
3-(2-{4-[1-(4-Fluoro-phenyl)-5-(2-methyl-2H-tetrazol-5-yl)-1H-indol-3-yl]-piperidin-1-yl}-ethyl)-oxazolidin-2-one
Show/Hide
|
C26H28FN7O2
|
1
|
| 1 |
Ki = 410 nM
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CP0847773
|
(R)-N-(3-hydroxy-2-(7-methoxynaphthalen-1-yl)propyl)propionamide
Show/Hide
|
C17H21NO3
|
1
|
| 1 |
Ki = 416.87 nM
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CP0448560
|
1'-(2,4-difluorophenethyl)-5-fluorospiro[3,4-dihydro-2H-chromene-2,4'-(hexahydropyridine)]
Show/Hide
|
C21H22F3NO
|
1
|
| 1 |
Ki = 440 nM
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CP0039097
|
1'-(2,4-difluorophenethyl)spiro[3,4-dihydro-2H-chromene-2,4'-(hexahydropyridine)]
Show/Hide
|
C21H23F2NO
|
1
|
| 1 |
Ki = 450 nM
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CP0457420
|
(S)-2-Methyl-1,2,3,4,8,9,10,11-octahydro-[1,4]diazepino[6,7,1-jk]carbazole
Show/Hide
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C16H20N2
|
1
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| 1 |
Ki = 452 nM
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CP0441080
|
4-(2-cyclopentyl-6,7,8,9-tetrahydro-5H-pyrimido[4,5-d]azepin-4-yl)benzonitrile
Show/Hide
|
C20H22N4
|
1
|
| 1 |
Ki = 460 nM
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CP0816404
|
(3R,4R)-5-Fluoro-3-(4-fluoropiperidin-3-yl)-2-phenyl-1H-indole
Show/Hide
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C19H18F2N2
|
1
|
| 1 |
Ki = 500 nM
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CP0294233
|
4-(4-Chloro-benzyl)-2-(1-methyl-azepan-4-yl)-2H-phthalazin-1-one
Show/Hide
|
C22H24ClN3O
|
1
|
| 1 |
Ki = 501.19 nM
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CP0376934
|
2,4-difluoro-1-(4-(phenylsulfonyl)phenethyl)benzene
Show/Hide
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C20H16F2O2S
|
1
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| 1 |
Ki = 526 nM
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CP0853639
|
2-Chloro-N-(3-(R)-1-pyrrolidin-2-ylmethyl-1H-indol-5-yl)-benzenesulfonamide
Show/Hide
|
C19H20ClN3O2S
|
1
|
| 1 |
Ki = 566 nM
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CP0428082
|
(E)-5-fluoro-2-(2-(5-(2-fluorophenylsulfonyl)pyridin-2-yl)vinyl)phenol
Show/Hide
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C19H13F2NO3S
|
1
|
| 1 |
Ki = 580 nM
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CP0405073
|
N-[(8-methoxy-2,3-dihydro-1H-cyclopenta[a]naphthalen-1-yl)methyl]methanesulfonamide
Show/Hide
|
C16H19NO3S
|
1
|
| 1 |
Ki = 580 nM
|
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CP0402050
|
6-Methyl-1,2,3,4,8,9,10,11-octahydro-[1,4]diazepino[6,7,1-jk]carbazole
Show/Hide
|
C16H20N2
|
1
|
| 1 |
Ki = 599 nM
|
|
|
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CP0437526
|
1'-(2,4-difluorophenethyl)-7-fluorospiro[3,4-dihydro-2H-chromene-2,4'-(hexahydropyridine)]
Show/Hide
|
C21H22F3NO
|
1
|
| 1 |
Ki = 600 nM
|
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|
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CP0347888
|
4-[[1-(2-(2,4-Difluorophenyl)ethyl)-4-piperidinyl]sulfonyl]benzonitrile
Show/Hide
|
C20H20F2N2O2S
|
1
|
| 1 |
Ki = 640 nM
|
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CP0401076
|
1-Methyl-4-[(3aR,12bS)-1-(3,3a,8,12b-tetrahydro-2H-1-oxa-dibenzo[e,h]azulen-2-yl)methyl]-piperazine
Show/Hide
|
C23H28N2O
|
1
|
| 1 |
Ki = 677 nM
|
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|
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CP0847772
|
2,2-difluoro-N-(3-hydroxy-2-(7-methoxynaphthalen-1-yl)propyl)acetamide
Show/Hide
|
C16H17F2NO3
|
1
|
| 1 |
Ki = 691.83 nM
|
|
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CP0178199
|
Agomelatine
Show/Hide
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C15H17NO2
|
2
|
| 1 |
Ki = 707.95 nM
|
|
|
| 2 |
Ki = 708 nM
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|
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CP0877971
|
rac-N-(1-hydroxy-3-(7-methoxynaphthalen-1-yl)propan-2-yl)propionamide
Show/Hide
|
C17H21NO3
|
1
|
| 1 |
Ki = 707.95 nM
|
|
|
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CP0394268
|
(E)-2-(2-(5-(2-fluorophenylsulfonyl)pyridin-2-yl)vinyl)phenol
Show/Hide
|
C19H14FNO3S
|
1
|
| 1 |
Ki = 810 nM
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CP0915712
|
4-(2-Trifluoromethylphenyl)piperidinium chloride
Show/Hide
|
C12H15ClF3N
|
1
|
| 1 |
Ki = 826 nM
|
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CP0376502
|
6-chloro-1'-phenethylspiro[1,2,3,4-tetrahydronaphthalene-2,4'-(hexahydropyridine)]-1-one
Show/Hide
|
C22H24ClNO
|
1
|
| 1 |
Ki = 850 nM
|
|
|
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CP0382448
|
2-Methyl-4,5,6,7,9,10-hexahydro-8H-5,7a-diaza-benzo[cd]cyclopenta[a]azulene
Show/Hide
|
C15H18N2
|
1
|
| 1 |
Ki = 985 nM
|
|
|
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CP0392941
|
4-(4-fluorophenyl)-2-(2-methylpropyl)-5,6,7,8-tetrahydropyrido[4,3-d]pyrimidine
Show/Hide
|
C17H20FN3
|
1
|
| 1 |
Ki = 1000 nM
|
|
|
|
CP0441078
|
4-(4-fluorophenyl)-2-[(4-fluorophenyl)methyl]-5,6,7,8-tetrahydropyrido[4,3-d]pyrimidine
Show/Hide
|
C20H17F2N3
|
1
|
| 1 |
Ki = 1000 nM
|
|
|
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CP0371837
|
2-butan-2-yl-4-(4-fluorophenyl)-5,6,7,8-tetrahydropyrido[4,3-d]pyrimidine
Show/Hide
|
C17H20FN3
|
1
|
| 1 |
Ki = 1020 nM
|
|
|
|
CP0333143
|
3-(2-{4-[1-(4-Fluoro-phenyl)-5-(1-methyl-1H-[1,2,4]triazol-3-yl)-1H-indol-3-yl]-piperidin-1-yl}-ethyl)-1H-quinazoline-2,4-dione
Show/Hide
|
C32H30FN7O2
|
1
|
| 1 |
Ki = 1100 nM
|
|
|
|
CP0867388
|
4-(2,3-Dimethylphenyl)piperidinium chloride
Show/Hide
|
C13H20ClN
|
1
|
| 1 |
Ki = 1160 nM
|
|
|
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CP0458482
|
(E)-2-(4-fluoro-2-methoxystyryl)-5-(2-fluorophenylsulfonyl)pyridine
Show/Hide
|
C20H15F2NO3S
|
1
|
| 1 |
Ki = 1400 nM
|
|
|
|
CP0448533
|
1-[6-fluorospiro[3,4-dihydro-2H-chromene-2,4'-(hexahydropyridine)]-1-yl]-4-phenyl-2-butanol
Show/Hide
|
C23H28FNO2
|
1
|
| 1 |
Ki = 1500 nM
|
|
|
|
CP0416462
|
N-[2-(2-methoxy-8,9-dihydro-7H-cyclopenta[h]quinolin-9-yl)ethyl]acetamide
Show/Hide
|
C17H20N2O2
|
1
|
| 1 |
Ki = 1600 nM
|
|
|
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CP0875254
|
4-(2-Methoxyphenyl)piperidinium chloride
Show/Hide
|
C12H18ClNO
|
1
|
| 1 |
Ki = 1800 nM
|
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|
|
CP0702373
|
N-(4-{4-[(6-Butyl-8-quinolinyl)oxy]-1-piperidinyl}butyl)ethanesulfonamide dihydrochloride
Show/Hide
|
C24H39Cl2N3O3S
|
1
|
| 1 |
Ki = 1995.26 nM
|
|
|
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CP0262775
|
3-(1-Benzyl-piperidin-3-yl)-2-phenyl-1H-indole
Show/Hide
|
C26H26N2
|
1
|
| 1 |
Ki = 2000 nM
|
|
|
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CP0311378
|
3-(1-Methyl-piperidin-2-yl)-2-phenyl-1H-indole
Show/Hide
|
C20H22N2
|
1
|
| 1 |
Ki = 2000 nM
|
|
|
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CP0347876
|
3-(1-(2-Phenylethyl)piperidin-3-yl)-2-phenyl-1H-indole
Show/Hide
|
C27H28N2
|
1
|
| 1 |
Ki = 2400 nM
|
|
|
|
CP0417789
|
3-(phenylsulfonyl)-1H-indole, 18i
Show/Hide
|
C21H24N2O2S
|
1
|
| 1 |
Ki = 2400 nM
|
|
|
|
CP0490205
|
1-{2-[3-(2-Phenyl-1H-indol-3-yl)-piperidin-1-yl]-ethyl}-imidazolidin-2-one
Show/Hide
|
C24H28N4O
|
1
|
| 1 |
Ki = 2500 nM
|
|
|
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CP0427030
|
2-(4-fluorophenethyl)-5-(4-fluorophenylsulfonyl)pyridine
Show/Hide
|
C19H15F2NO2S
|
1
|
| 1 |
Ki = 2700 nM
|
|
|
|
CP0403987
|
3-{2-[2-((R)-Methoxymethyl)-pyrrolidin-1-yl]-ethyl}-2-phenyl-1H-indole
Show/Hide
|
C22H26N2O
|
1
|
| 1 |
Ki = 3000 nM
|
|
|
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CP0877856
|
4-(2-Methylphenyl)piperidinium chloride
Show/Hide
|
C12H18ClN
|
1
|
| 1 |
Ki = 3170 nM
|
|
|
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CP0371838
|
4-(4-fluorophenyl)-2-phenyl-5,6,7,8-tetrahydropyrido[4,3-d]pyrimidine
Show/Hide
|
C19H16FN3
|
1
|
| 1 |
Ki = 4000 nM
|
|
|
|
CP0254576
|
8-((2S,3aS,12bS)-11-Bromo-2,3,3a,12b-tetrahydro-1,8-dioxa-dibenzo[e,h]azulen-2-ylmethyl)-3-morpholin-4-ylmethyl-7-oxa-8-aza-bicyclo[4.2.0]octa-1(6),2,4-triene
Show/Hide
|
C28H27BrN2O4
|
1
|
| 1 |
Ki = 4105 nM
|
|
|
|
CP0504966
|
2-benzyl-4-(4-fluorophenyl)-6,7,8,9-tetrahydro-5H-pyrimido[5,4-c]azepine
Show/Hide
|
C21H20FN3
|
1
|
| 1 |
Ki = 5000 nM
|
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|
|
CP0511384
|
2-cyclopropyl-4-(4-fluorophenyl)-5,6,7,8-tetrahydropyrido[4,3-d]pyrimidine
Show/Hide
|
C16H16FN3
|
1
|
| 1 |
Ki = 5000 nM
|
|
|
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CP0516500
|
4-(4-chlorophenyl)-2-methyl-6,7,8,9-tetrahydro-5H-pyrimido[4,5-d]azepine
Show/Hide
|
C15H16ClN3
|
1
|
| 1 |
Ki = 5000 nM
|
|
|
|
CP0915714
|
4-(3-Methoxyphenyl)piperidinium chloride
Show/Hide
|
C12H18ClNO
|
1
|
| 1 |
Ki = 6190 nM
|
|
|
|
CP0870812
|
4-(4-Trifluoromethylphenyl)piperidinium chloride
Show/Hide
|
C12H15ClF3N
|
1
|
| 1 |
Ki = 8320 nM
|
|
|
|
CP0849996
|
4-Phenylpiperidinium chloride
Show/Hide
|
C11H16ClN
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0875252
|
4-(4-Fluorophenyl)piperidinium chloride
Show/Hide
|
C11H15ClFN
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0877852
|
4-(4-Methylphenyl)piperidinium chloride
Show/Hide
|
C12H18ClN
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0877857
|
4-(4-(dimethylamino)phenyl)piperidinium chloride
Show/Hide
|
C13H21ClN2
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0915715
|
4-(4-Chlorophenyl)piperidinium chloride
Show/Hide
|
C11H15Cl2N
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0945744
|
4-(4-Methoxyphenyl)piperidinium chloride
Show/Hide
|
C12H18ClNO
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0953625
|
4-(3-Hydroxyphenyl)piperidinium chloride
Show/Hide
|
C11H16ClNO
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
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CP0847750
|
(S)-N-(1-hydroxy-3-(7-methoxynaphthalen-1-yl)propan-2-yl)propionamide
Show/Hide
|
C17H21NO3
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0877969
|
(S)-2-fluoro-N-(3-hydroxy-2-(7-methoxynaphthalen-1-yl)propyl)acetamide
Show/Hide
|
C16H18FNO3
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0405083
|
1-[(8-methoxy-1-methyl-2,3-dihydrocyclopenta[a]naphthalen-1-yl)methyl]-3-propylthiourea
Show/Hide
|
C20H26N2OS
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0414939
|
1-[(8-methoxy-1-methyl-2,3-dihydrocyclopenta[a]naphthalen-1-yl)methyl]-3-propylurea
Show/Hide
|
C20H26N2O2
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0429915
|
N-[(8-methoxy-1-methyl-2,3-dihydrocyclopenta[a]naphthalen-1-yl)methyl]acetamide
Show/Hide
|
C18H21NO2
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0429921
|
1-[(8-methoxy-1-methyl-2,3-dihydrocyclopenta[a]naphthalen-1-yl)methyl]-3-methylthiourea
Show/Hide
|
C18H22N2OS
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
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CP0469375
|
1-ethyl-3-[(8-methoxy-1-methyl-2,3-dihydrocyclopenta[a]naphthalen-1-yl)methyl]thiourea
Show/Hide
|
C19H24N2OS
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0485368
|
1-ethyl-3-[(8-methoxy-1-methyl-2,3-dihydrocyclopenta[a]naphthalen-1-yl)methyl]urea
Show/Hide
|
C19H24N2O2
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0508414
|
N-[(8-methoxy-1-methyl-2,3-dihydrocyclopenta[a]naphthalen-1-yl)methyl]methanesulfonamide
Show/Hide
|
C17H21NO3S
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0493922
|
3-(2-Azetidin-1-yl-ethyl)-2-phenyl-1H-indole
Show/Hide
|
C19H20N2
|
1
|
| 1 |
Ki > 1000 nM
|
|
|
|
CP0508569
|
N-ethyl-2-[2-(furan-2-yl)-1H-indol-3-yl]-N-methylethanamine
Show/Hide
|
C17H20N2O
|
1
|
| 1 |
Ki > 1000 nM
|
|
|
|
CP0844290
|
(3R,4R)-6-Fluoro-3-(4-fluoropiperidin-3-yl)-1H-indole-2-carboxylic Acid Methyl Ester
Show/Hide
|
C15H16F2N2O2
|
1
|
| 1 |
Ki > 2000 nM
|
|
|
|
CP0427027
|
(E)-2-(4-fluorostyryl)-5-(phenylsulfonyl)pyridine
Show/Hide
|
C19H14FNO2S
|
1
|
| 1 |
Ki > 4000 nM
|
|
|
|
CP0427028
|
(E)-2-(4-fluorostyryl)-5-(3-fluorophenylsulfonyl)pyridine
Show/Hide
|
C19H13F2NO2S
|
1
|
| 1 |
Ki > 4000 nM
|
|
|
|
CP0427032
|
5-(benzenesulfonyl)-2-[(E)-2-(2,4-difluorophenyl)ethenyl]pyridine
Show/Hide
|
C19H13F2NO2S
|
1
|
| 1 |
Ki > 4000 nM
|
|
|
|
CP0428085
|
(E)-2-(4-fluorostyryl)-5-(2-fluorophenylsulfonyl)pyridine
Show/Hide
|
C19H13F2NO2S
|
1
|
| 1 |
Ki > 4000 nM
|
|
|
|
CP0428088
|
(E)-2-(2-fluorostyryl)-5-(2-fluorophenylsulfonyl)pyridine
Show/Hide
|
C19H13F2NO2S
|
1
|
| 1 |
Ki > 4000 nM
|
|
|
|
CP0428089
|
(E)-5-(4-fluorostyryl)-2-(4-fluorophenylsulfonyl)pyridine
Show/Hide
|
C19H13F2NO2S
|
1
|
| 1 |
Ki > 4000 nM
|
|
|
|
CP0434500
|
(E)-5-(2-fluorophenylsulfonyl)-2-(2-(pyridin-4-yl)vinyl)pyridine
Show/Hide
|
C18H13FN2O2S
|
1
|
| 1 |
Ki > 4000 nM
|
|
|
|
CP0445062
|
(E)-2-(3-fluorostyryl)-5-(2-fluorophenylsulfonyl)pyridine
Show/Hide
|
C19H13F2NO2S
|
1
|
| 1 |
Ki > 4000 nM
|
|
|
|
CP0458021
|
5-(4-fluorophenethyl)-2-(4-fluorophenylsulfonyl)pyridine
Show/Hide
|
C19H15F2NO2S
|
1
|
| 1 |
Ki > 4000 nM
|
|
|
|
CP0516363
|
(E)-2-(4-fluorostyryl)-5-(4-fluorophenylsulfonyl)pyridine
Show/Hide
|
C19H13F2NO2S
|
1
|
| 1 |
Ki > 4000 nM
|
|
|
|
CP0105167
|
3-{4-[1-(4-Fluoro-phenyl)-5-pyrimidin-2-yl-1H-indol-3-yl]-piperidin-1-yl}-propionitrile
Show/Hide
|
C26H24FN5
|
1
|
| 1 |
Ki > 4200 nM
|
|
|
|
CP0134581
|
3-(2-{4-[1-(4-Fluoro-phenyl)-5-pyrimidin-2-yl-1H-indol-3-yl]-piperidin-1-yl}-ethyl)-oxazolidin-2-one
Show/Hide
|
C28H28FN5O2
|
1
|
| 1 |
Ki > 4200 nM
|
|
|
|
CP0163622
|
3-{4-[1-(4-Fluoro-phenyl)-5-(1-methyl-1H-[1,2,4]triazol-3-yl)-1H-indol-3-yl]-piperidin-1-yl}-propionitrile
Show/Hide
|
C25H25FN6
|
1
|
| 1 |
Ki > 4200 nM
|
|
|
|
CP0320413
|
3-(2-{4-[1-(4-Fluoro-phenyl)-5-(1-methyl-1H-[1,2,4]triazol-3-yl)-1H-indol-3-yl]-piperidin-1-yl}-ethyl)-1-methyl-pyrrolidin-2-one
Show/Hide
|
C29H33FN6O
|
1
|
| 1 |
Ki > 4200 nM
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CP0343878
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3-(2-{4-[1-(4-Fluoro-phenyl)-5-(1-methyl-1H-[1,2,4]triazol-3-yl)-1H-indol-3-yl]-piperidin-1-yl}-ethyl)-oxazolidin-2-one
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C27H29FN6O2
|
1
|
| 1 |
Ki > 4200 nM
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CP0408686
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8-((2S,3aS,12bS)-11-Bromo-2,3,3a,12b-tetrahydro-1,8-dioxa-dibenzo[e,h]azulen-2-ylmethyl)-3-morpholin-4-yl-7-oxa-8-aza-bicyclo[4.2.0]octa-1(6),2,4-triene
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C27H25BrN2O4
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1
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| 1 |
Ki > 5454 nM
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