| Compound ID |
Compound Name |
Compound Formula |
|
CP0846140
|
3-({5-[4-(Ethylsulfonyl)phenoxy]-2-(pyridin-2-yl)-1Hbenzimidazol-6-yl}methyl)-1,3-oxazolidine-2,4-dione
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|
C24H20N4O6S
|
2
|
| 1 |
EC50 = 20 nM
|
|
|
| 2 |
EC50 = 90 nM
|
|
|
|
CP0375578
|
1-({5-[4-(Ethylsulfonyl)phenoxy]-2-(pyridin-2-yl)-1Hbenzimidazol-6-yl}methyl)pyrrolidine-2,5-dione
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|
C25H22N4O5S
|
2
|
| 1 |
EC50 = 40 nM
|
|
|
| 2 |
EC50 = 160 nM
|
|
|
|
CP0428948
|
1-({5-[4-(Ethylsulfonyl)phenoxy]-2-(pyridin-2-yl)-1Hbenzimidazol-6-yl}methyl)pyrrolidin-2-one
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|
C25H24N4O4S
|
2
|
| 1 |
EC50 = 60 nM
|
|
|
| 2 |
EC50 = 350 nM
|
|
|
|
CP0428949
|
3-({5-[4-(Ethylsulfonyl)phenoxy]-2-(pyridin-2-yl)-1Hbenzimidazol-6-yl}methyl)-1,3-oxazolidin-2-one
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|
C24H22N4O5S
|
2
|
| 1 |
EC50 = 60 nM
|
|
|
| 2 |
EC50 = 250 nM
|
|
|
|
CP0860857
|
3-({5-[4-(Ethylsulfonyl)phenoxy]-2-(pyridin-2-yl)-1Hbenzimidazol-6-yl}methyl)-1-methylimidazolidine-2,4-dione
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|
C25H23N5O5S
|
2
|
| 1 |
EC50 = 60 nM
|
|
|
| 2 |
EC50 = 180 nM
|
|
|
|
CP0381151
|
5-(4-(ethylsulfonyl)phenoxy)-6-((1-methyl-1H-tetrazol-5-yl)methyl)-2-(pyridin-2-yl)-1H-benzo[d]imidazole
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|
C23H21N7O3S
|
2
|
| 1 |
EC50 = 70 nM
|
|
|
| 2 |
EC50 = 410 nM
|
|
|
|
CP0470279
|
N-[[6-(4-ethylsulfonylphenoxy)-2-pyridin-2-yl-3H-benzimidazol-5-yl]methyl]-N-methylacetamide
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|
C24H24N4O4S
|
2
|
| 1 |
EC50 = 70 nM
|
|
|
| 2 |
EC50 = 300 nM
|
|
|
|
CP0507293
|
1-({5-[4-(Ethylsulfonyl)phenoxy]-2-(pyridin-2-yl)-1Hbenzimidazol-6-yl}methyl)-3-methylimidazolidin-2-one
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|
C25H25N5O4S
|
2
|
| 1 |
EC50 = 80 nM
|
|
|
| 2 |
EC50 = 320 nM
|
|
|
|
CP0428952
|
6-[(1,1-Dioxidoisothiazolidin-2-yl)methyl]-5-[4-(ethylsulfonyl)phenoxy]-2-(pyridin-2-yl)-1H-benzimidazole
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|
C24H24N4O5S2
|
2
|
| 1 |
EC50 = 90 nM
|
|
|
| 2 |
EC50 = 460 nM
|
|
|
|
CP0375572
|
4-({5-[4-(Ethylsulfonyl)phenoxy]-2-(pyridin-2-yl)-1Hbenzimidazol-6-yl}methyl)morpholin-3-one
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|
C25H24N4O5S
|
2
|
| 1 |
EC50 = 100 nM
|
|
|
| 2 |
EC50 = 280 nM
|
|
|
|
CP0430706
|
N-ethyl-N-[[6-(4-ethylsulfonylphenoxy)-2-pyridin-2-yl-3H-benzimidazol-5-yl]methyl]acetamide
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|
C25H26N4O4S
|
2
|
| 1 |
EC50 = 110 nM
|
|
|
| 2 |
EC50 = 500 nM
|
|
|
|
CP0375580
|
5-[4-(Ethylsulfonyl)phenoxy]-6-(1H-imidazol-1-ylmethyl)-2-(pyridin-2-yl)-1H-benzimidazole
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|
C24H21N5O3S
|
2
|
| 1 |
EC50 = 120 nM
|
|
|
| 2 |
EC50 = 430 nM
|
|
|
|
CP0405514
|
3-(5-(4-(ethylsulfonyl)phenoxy)-2-(pyridin-2-yl)-1H-benzo[d]imidazol-6-yl)-N,N-dimethylpropanamide
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|
C25H26N4O4S
|
2
|
| 1 |
EC50 = 120 nM
|
|
|
| 2 |
EC50 = 620 nM
|
|
|
|
CP0470280
|
N-[[6-(4-ethylsulfonylphenoxy)-2-pyridin-2-yl-3H-benzimidazol-5-yl]methyl]acetamide
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|
C23H22N4O4S
|
2
|
| 1 |
EC50 = 220 nM
|
|
|
| 2 |
EC50 = 1410 nM
|
|
|
|
CP0375579
|
5-[4-(Ethylsulfonyl)phenoxy]-2-(pyridin-2-yl)-6-(pyrrolidin-1-ylmethyl)-1H-benzimidazole
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|
C25H26N4O3S
|
1
|
| 1 |
EC50 > 5000 nM
|
|
|
|
CP0428951
|
1-({5-[4-(Ethylsulfonyl)phenoxy]-2-(pyridin-2-yl)-1Hbenzimidazol-6-yl}methyl)imidazolidin-2-one
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|
C24H23N5O4S
|
1
|
| 1 |
EC50 > 5000 nM
|
|
|
