| Compound ID |
Compound Name |
Compound Formula |
|
CP0085178
|
5-methyl-4-(4-nitrophenyl)-2-pyridin-2-yl-1H-pyrazol-3-one
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|
C15H12N4O3
|
1
|
| 1 |
IC50 = 60 nM
|
|
|
|
CP0350317
|
5-methyl-2-pyridin-2-yl-4-[4-(trifluoromethyl)phenyl]-1H-pyrazol-3-one
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|
C16H12F3N3O
|
1
|
| 1 |
IC50 = 150 nM
|
|
|
|
CP0758470
|
2-(6-methylbenzo[d]thiazol-2-yl)-4,5-dihydro-2H-benzo[e]indazol-1-ol
Show/Hide
|
C19H15N3OS
|
1
|
| 1 |
IC50 = 150 nM
|
|
|
|
CP0354787
|
5-methyl-3-oxo-2-pyridin-2-yl-N-[3-(trifluoromethyl)phenyl]-1H-pyrazole-4-carboxamide
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|
C17H13F3N4O2
|
1
|
| 1 |
IC50 = 170 nM
|
|
|
|
CP0065981
|
5-methyl-N-(4-nitrophenyl)-3-oxo-2-pyridin-2-yl-1H-pyrazole-4-carboxamide
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|
C16H13N5O4
|
1
|
| 1 |
IC50 = 200 nM
|
|
|
|
CP0831459
|
7-(4-methoxyphenyl)-2-(pyridin-2-yl)-4,5-dihydro-2H-benzo[e]indazol-1-ol
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|
C23H19N3O2
|
1
|
| 1 |
IC50 = 210 nM
|
|
|
|
CP0145497
|
N-(3-fluoro-4-methoxyphenyl)-5-methyl-3-oxo-2-pyridin-2-yl-1H-pyrazole-4-carboxamide
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|
C17H15FN4O3
|
1
|
| 1 |
IC50 = 260 nM
|
|
|
|
CP0762328
|
7-phenyl-2-(pyridin-2-yl)-4,5-dihydro-2H-benzo[e]indazol-1-ol
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|
C22H17N3O
|
1
|
| 1 |
IC50 = 260 nM
|
|
|
|
CP0743892
|
2-(pyridin-2-yl)-7-p-tolyl-4,5-dihydro-2H-benzo[e]indazol-1-ol
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|
C23H19N3O
|
1
|
| 1 |
IC50 = 270 nM
|
|
|
|
CP0095380
|
5-methyl-3-oxo-2-pyridin-2-yl-N-[4-(trifluoromethyl)phenyl]-1H-pyrazole-4-carboxamide
Show/Hide
|
C17H13F3N4O2
|
1
|
| 1 |
IC50 = 290 nM
|
|
|
|
CP0831460
|
7-bromo-2-(pyridin-2-yl)-4,5-dihydro-2H-benzo[e]indazol-1-ol
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|
C16H12BrN3O
|
1
|
| 1 |
IC50 = 310 nM
|
|
|
|
CP0241746
|
5-methyl-2-pyridin-2-yl-4-[3-(trifluoromethyl)phenyl]-1H-pyrazol-3-one
Show/Hide
|
C16H12F3N3O
|
1
|
| 1 |
IC50 = 320 nM
|
|
|
|
CP0780846
|
2-(6-methoxybenzo[d]thiazol-2-yl)-4,5-dihydro-2H-benzo[e]indazol-1-ol
Show/Hide
|
C19H15N3O2S
|
1
|
| 1 |
IC50 = 330 nM
|
|
|
|
CP0197135
|
4-(5-methyl-3-oxo-2-pyridin-2-yl-1H-pyrazol-4-yl)benzonitrile
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|
C16H12N4O
|
1
|
| 1 |
IC50 = 360 nM
|
|
|
|
CP0197136
|
2-(6-fluoro-1,3-benzothiazol-2-yl)-5-methyl-4-phenyl-1H-pyrazol-3-one
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|
C17H12FN3OS
|
1
|
| 1 |
IC50 = 390 nM
|
|
|
|
CP0780847
|
2-(6-fluorobenzo[d]thiazol-2-yl)-4,5-dihydro-2H-benzo[e]indazol-1-ol
Show/Hide
|
C18H12FN3OS
|
1
|
| 1 |
IC50 = 400 nM
|
|
|
|
CP0170206
|
5-methyl-N-(3-methylphenyl)-3-oxo-2-pyridin-2-yl-1H-pyrazole-4-carboxamide
Show/Hide
|
C17H16N4O2
|
1
|
| 1 |
IC50 = 410 nM
|
|
|
|
CP0170208
|
2-(1,3-benzothiazol-2-yl)-5-methyl-4-phenyl-1H-pyrazol-3-one
Show/Hide
|
C17H13N3OS
|
1
|
| 1 |
IC50 = 430 nM
|
|
|
|
CP0248111
|
2-(1H-benzimidazol-2-yl)-5-methyl-4-phenyl-1H-pyrazol-3-one
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|
C17H14N4O
|
1
|
| 1 |
IC50 = 520 nM
|
|
|
|
CP0762329
|
1-hydroxy-2-(pyridin-2-yl)-4,5-dihydro-2H-benzo[e]indazole-7-carbonitrile
Show/Hide
|
C17H12N4O
|
1
|
| 1 |
IC50 = 520 nM
|
|
|
|
CP0739794
|
2-(1-hydroxy-4,5-dihydro-2H-benzo[e]indazol-2-yl)benzo[d]thiazole-6-carboxylic acid
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|
C19H13N3O3S
|
1
|
| 1 |
IC50 = 560 nM
|
|
|
|
CP0079266
|
5-methyl-3-oxo-N-phenyl-2-pyridin-2-yl-1H-pyrazole-4-carboxamide
Show/Hide
|
C16H14N4O2
|
1
|
| 1 |
IC50 = 640 nM
|
|
|
|
CP0335612
|
N-(3-methoxyphenyl)-5-methyl-3-oxo-2-pyridin-2-yl-1H-pyrazole-4-carboxamide
Show/Hide
|
C17H16N4O3
|
1
|
| 1 |
IC50 = 660 nM
|
|
|
|
CP0335613
|
5-methyl-N-(4-methylphenyl)-3-oxo-2-pyridin-2-yl-1H-pyrazole-4-carboxamide
Show/Hide
|
C17H16N4O2
|
1
|
| 1 |
IC50 = 690 nM
|
|
|
|
CP0170147
|
5-methyl-N-(2-nitrophenyl)-3-oxo-2-pyridin-2-yl-1H-pyrazole-4-carboxamide
Show/Hide
|
C16H13N5O4
|
1
|
| 1 |
IC50 = 710 nM
|
|
|
|
CP0704279
|
2-(benzo[d]thiazol-2-yl)-4,5-dihydro-2H-benzo[e]indazol-1-ol
Show/Hide
|
C18H13N3OS
|
1
|
| 1 |
IC50 = 720 nM
|
|
|
|
CP0065982
|
ethyl 4-(5-methyl-3-oxo-2-pyridin-2-yl-1H-pyrazol-4-yl)benzoate
Show/Hide
|
C18H17N3O3
|
1
|
| 1 |
IC50 = 770 nM
|
|
|
|
CP0797806
|
2-(pyridin-2-yl)-4,5-dihydro-2H-benzo[e]indazol-1-ol
Show/Hide
|
C16H13N3O
|
1
|
| 1 |
IC50 = 830 nM
|
|
|
|
CP0335615
|
4-(4-fluorophenyl)-5-methyl-2-pyridin-2-yl-1H-pyrazol-3-one
Show/Hide
|
C15H12FN3O
|
1
|
| 1 |
IC50 = 910 nM
|
|
|
|
CP0335614
|
5-methyl-3-oxo-2-pyridin-2-yl-N-[2-(trifluoromethyl)phenyl]-1H-pyrazole-4-carboxamide
Show/Hide
|
C17H13F3N4O2
|
1
|
| 1 |
IC50 = 1000 nM
|
|
|
|
CP0241747
|
2-(6-methoxy-1,3-benzothiazol-2-yl)-5-methyl-4-phenyl-1H-pyrazol-3-one
Show/Hide
|
C18H15N3O2S
|
1
|
| 1 |
IC50 = 1040 nM
|
|
|
|
CP0145498
|
N-(1,3-benzodioxol-5-yl)-5-methyl-3-oxo-2-pyridin-2-yl-1H-pyrazole-4-carboxamide
Show/Hide
|
C17H14N4O4
|
1
|
| 1 |
IC50 = 1220 nM
|
|
|
|
CP0669868
|
4-(4-(diethylamino)benzylidene)-3-methyl-1-(pyridin-2-yl)-1H-pyrazol-5(4H)-one
Show/Hide
|
C20H22N4O
|
1
|
| 1 |
IC50 = 1530 nM
|
|
|
|
CP0085179
|
5-methyl-4-phenyl-2-pyridin-2-yl-1H-pyrazol-3-one
Show/Hide
|
C15H13N3O
|
1
|
| 1 |
IC50 = 1700 nM
|
|
|
|
CP0739795
|
2-(1H-benzo[d]imidazol-2-yl)-4,5-dihydro-2H-benzo[e]indazol-1-ol
Show/Hide
|
C18H14N4O
|
1
|
| 1 |
IC50 = 1760 nM
|
|
|
|
CP0248112
|
5-methyl-4-phenyl-2-(1,3-thiazol-2-yl)-1H-pyrazol-3-one
Show/Hide
|
C13H11N3OS
|
1
|
| 1 |
IC50 = 2190 nM
|
|
|
|
CP0689873
|
3-(4-(4-(diethylamino)benzylidene)-3-methyl-5-oxo-4,5-dihydro-1H-pyrazol-1-yl)-6-methyl-1,2,4-triazin-5(4H)-one
Show/Hide
|
C19H22N6O2
|
1
|
| 1 |
IC50 = 2570 nM
|
|
|
|
CP0739550
|
7-methoxy-2-(pyridin-2-yl)-4,5-dihydro-2H-benzo[e]indazol-1-ol
Show/Hide
|
C17H15N3O2
|
1
|
| 1 |
IC50 = 2770 nM
|
|
|
|
CP0218649
|
4-(4-methoxyphenyl)-5-methyl-2-pyridin-2-yl-1H-pyrazol-3-one
Show/Hide
|
C16H15N3O2
|
1
|
| 1 |
IC50 = 2820 nM
|
|
|
|
CP0075130
|
5-methyl-4-phenyl-2-pyrimidin-2-yl-1H-pyrazol-3-one
Show/Hide
|
C14H12N4O
|
1
|
| 1 |
IC50 > 5000 nM
|
|
|
|
CP0077664
|
5-methyl-3-oxo-N,2-diphenyl-1H-pyrazole-4-carboxamide
Show/Hide
|
C17H15N3O2
|
1
|
| 1 |
IC50 > 5000 nM
|
|
|
|
CP0085180
|
4-[4-(diethylamino)phenyl]-5-methyl-2-pyridin-2-yl-1H-pyrazol-3-one
Show/Hide
|
C19H22N4O
|
1
|
| 1 |
IC50 > 5000 nM
|
|
|
|
CP0130129
|
5-methyl-4-phenyl-2-(pyridin-2-ylmethyl)-1H-pyrazol-3-one
Show/Hide
|
C16H15N3O
|
1
|
| 1 |
IC50 > 5000 nM
|
|
|
|
CP0145499
|
4-(4-aminophenyl)-5-methyl-2-pyridin-2-yl-1H-pyrazol-3-one
Show/Hide
|
C15H14N4O
|
1
|
| 1 |
IC50 > 5000 nM
|
|
|
|
CP0220586
|
2-(3H-isoquinolin-2-yl)-5-methyl-4-phenyl-1H-pyrazol-3-one
Show/Hide
|
C19H17N3O
|
1
|
| 1 |
IC50 > 5000 nM
|
|
|
|
CP0248113
|
6-(5-methyl-3-oxo-4-phenyl-1H-pyrazol-2-yl)-1H-pyridazin-4-one
Show/Hide
|
C14H12N4O2
|
1
|
| 1 |
IC50 > 5000 nM
|
|
|
|
CP0704281
|
2-(4-methylbenzo[d]thiazol-2-yl)-4,5-dihydro-2H-benzo[e]indazol-1-ol
Show/Hide
|
C19H15N3OS
|
1
|
| 1 |
IC50 > 5000 nM
|
|
|
|
CP0831458
|
2-(1-hydroxy-4,5-dihydro-2H-benzo[e]indazol-2-yl)pyridine 1-oxide
Show/Hide
|
C16H13N3O2
|
1
|
| 1 |
IC50 > 5000 nM
|
|
|
